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13591

Total database: 17430
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10177 (74.9%)
Target
7625 (56.1%)
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104 (0.8%)
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13591 (100.0%)

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Hasil Pencarian (13591)

Halaman 237 / 272
Somatrem Approved DB09098
biotech | CAS: 82030-87-3

Despite the ability of almost all contemporary recombinant growth hormones to cause definite and demonstrable increases in growth rate in patients who are administered the drug, the use of these agents continues to be mired in persistent bioethical debate [A3…

Kategori:
Amino Acids, Peptides, and ProteinsAnterior Pituitary Lobe Hormones and AnaloguesGrowth Hormone +9
Target Protein:
Growth hormone receptorInsulin-like growth factor 1 receptor
Waktu ParuhThe mean terminal h…
Vol. DistribusiAnimal studies with…
KlirensThe clearance of so…
Genetik -
Somatrogon Approved DB14960
biotech | CAS: 1663481-09-1

Somatrogon is a long-acting recombinant human growth hormone. Growth hormone is a peptide hormone secreted by the pituitary gland that plays a crucial role in promoting longitudinal growth during childhood and adolescence and regulating metabolic function in …

Kategori:
Amino Acids, Peptides, and ProteinsAnterior Pituitary Lobe Hormones and AnaloguesGrowth Hormone +10
Target Protein:
Growth hormone receptor
Waktu ParuhFollowing subcutane…
Vol. DistribusiFollowing subcutane…
KlirensFollowing subcutane…
Genetik -
biotech | CAS: 1088845-67-3

Somatropin pegol is under investigation in clinical trial NCT00715689 (Dose Study in Growth Hormone Deficient Adults Investigating Safety, Pharmacokinetics and Pharmacodynamics of NNC126-0083).

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsEthylene Glycols +10
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Somavaratan DB12421
biotech | CAS: 1448335-08-7

Somavaratan has been used in trials studying the treatment of Growth Disorders and Adult Growth Hormone Deficiency.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Soneclosan DB04393
small molecule | CAS: 3380-30-1

Deskripsi belum tersedia.

Target Protein:
Enoyl-[acyl-carrier-protein] reductase [NADH]Enoyl-[acyl-carrier-protein] reductase [NADH] FabI
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sonedenoson DB12443
small molecule | CAS: 131865-88-8

Sonedenoson has been used in trials studying the treatment of Foot Ulcer, Diabetic and Diabetes Complications.

Kategori:
Heterocyclic Compounds, Fused-RingNucleic Acids, Nucleotides, and NucleosidesNucleosides +3
Target Protein:
Adenosine receptor A2a
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sonelokimab DB18843
biotech | CAS: 1414386-05-2

Sonelokimab is under investigation in clinical trial NCT06411379 (Study to Evaluate the Efficacy and Safety of Subcutaneous Sonelokimab Compared With Placebo in Adult Participants With Moderate to Severe Hidradenitis Suppurativa).

Kategori:
Amino Acids, Peptides, and ProteinsBlood ProteinsGlobulins +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sonepcizumab DB06305
biotech | CAS: 1031360-18-5

A humanized monoclonal antibody directed against sphingosine 1-phosphate (S1P) with potential antiangiogenic and antineoplastic activities. Upon administration, sonepcizumab binds S1P, which may result in the inhibition of tumor angiogenesis. S1P is the extra…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sonidegib Approved DB09143
small molecule | CAS: 956697-53-3

Sonidegib is a Hedgehog signaling pathway inhibitor (via smoothened antagonism) developed as an anticancer agent by Novartis. It was FDA approved in 2015 for the treatment of basal cell carcinoma.

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBenzene Derivatives +8
Target Protein:
Protein smoothened
Waktu ParuhHalf-life ~ 28 days…
Vol. DistribusiEstimated volume of…
Klirens-
Genetik -
Sonlicromanol DB16333
small molecule | CAS: 1541170-75-5

Sonlicromanol is under investigation in clinical trial NCT04165239 (The KHENERGYZE Study).

Kategori:
AntioxidantsBenzopyransBiological Factors +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sonolisib DB12601
small molecule | CAS: 502632-66-8

Sonolisib has been used in trials studying the treatment of Glioblastoma, Prostate Cancer, Advanced Solid Tumors, Advanced BRAF-mutant Cancers, and Non Small Cell Lung Cancer (NSCLC), among others.

Kategori:
Fused-Ring CompoundsSteroids
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sonrotoclax DB18753
small molecule | CAS: 2383086-06-2

Deskripsi belum tersedia.

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Genetik -
Soquelitinib DB18749
small molecule | CAS: 2226636-04-8

Deskripsi belum tersedia.

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SOR-C13 DB15366
biotech | CAS: 1187852-48-7

SOR-C13 is under investigation in clinical trial NCT01578564 (Safety and Tolerability Study of SOR-C13 in Subjects With Advanced Cancers Commonly Known to Express the TRPV6 Channel).

Kategori:
Amino Acids, Peptides, and ProteinsAntiarrhythmic agentsAntineoplastic Agents +9
Target Protein:
Transient receptor potential cation channel subfamily V member 6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sorafenib Approved DB00398
small molecule | CAS: 284461-73-0

Sorafenib is a bi-aryl urea and an oral multikinase inhibitor. It targets cell surface tyrosine kinase receptors and downstream intracellular kinases that are implicated in tumour cell proliferation and tumour angiogenesis.[A255852] First approved by the FDA …

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +51
Target Protein:
Serine/threonine-protein kinase B-rafEpidermal growth factor receptorRAF proto-oncogene serine/threonine-protein kinase +8
Waktu ParuhThe mean eliminatio…
Vol. DistribusiSorafenib is widely…
Klirens-
Genetik -
Soraprazan DB17856
small molecule | CAS: 261944-46-1

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Potassium-transporting ATPase alpha chain 1Potassium-transporting ATPase subunit beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sorbinil DB02712
small molecule | CAS: 68367-52-2

Deskripsi belum tersedia.

Kategori:
Aldehyde Reductase, antagonists & inhibitorsImidazoles
Target Protein:
Aldo-keto reductase family 1 member B1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sorbitol Approved DB01638
small molecule | CAS: 50-70-4

A polyhydric alcohol with about half the sweetness of sucrose. Sorbitol occurs naturally and is also produced synthetically from glucose. It was formerly used as a diuretic and may still be used as a laxative and in irrigating solutions for some surgical proc…

Kategori:
AlcoholsAlimentary Tract and MetabolismBlood and Blood Forming Organs +22
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sorghum halepense pollen Approved DB10365
biotech

Sorghum halepense pollen is the pollen of the Sorghum halepense plant. Sorghum halepense pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityGrass Pollen Allergen ExtractsIncreased Histamine Release +2
Waktu Paruh-
Vol. Distribusi-
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Genetik -
SOT-107 DB05337
biotech

SOT-107 is a drug that is a combination of a protein called transferrin and a poison called diphtheria toxin. This drug treat for a type of brain cancer called a high grade glioma brain tumour. About half of all brain tumours are gliomas.

Kategori:
ADP Ribose TransferasesBacterial ToxinsBiological Factors +6
Target Protein:
Glioma pathogenesis-related protein 1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Sotagliflozin Approved DB12713
small molecule | CAS: 1018899-04-1

Sotagliflozin is a dual inhibitor of SGLT1 and SGLT2, the first of its kind,[A244499] which is approved for use in the EU, in combination with insulin, to improve glycemic control in patients with type 1 diabetes mellitus (T1DM) and a BMI ?27 kg/m<sup>2</sup>…

Kategori:
Alimentary Tract and MetabolismBCRP/ABCG2 InhibitorsBlood Glucose Lowering Agents +24
Target Protein:
Sodium/glucose cotransporter 2Sodium/glucose cotransporter 1
Waktu ParuhThe mean terminal h…
Vol. DistribusiSotagliflozin has a…
KlirensIn healthy voluntee…
Genetik -
Sotalol Approved DB00489
small molecule | CAS: 3930-20-9

Sotalol is a methanesulfonanilide developed in 1960.[A178579] It was the first of the class III anti arrhythmic drugs.[A178579] Sotalol was first approved as an oral tablet on 30 October 1992.[L6334] A racemic mixture of sotalol is currently formulated as a t…

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-Antagonists +23
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptorVoltage-gated inwardly rectifying potassium channel KCNH2
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe apparent volume…
KlirensIn patients with a …
Genetik -
Sotatercept Approved DB12118
biotech | CAS: 1001080-50-7

Sotatercept is an activin signalling inhibitor. It is a homodimeric recombinant fusion protein consisting of the extracellular domain of the human activin receptor type IIA (ActRIIA) linked to the human IgG1 Fc domain.[L50351] On March 26, 2024, sotatercep…

Kategori:
Amino Acids, Peptides, and ProteinsBlood ProteinsImmunoglobulin G +5
Target Protein:
Activin receptor type-2AActivin receptor type-1BGrowth/differentiation factor 8 +1
Waktu ParuhThe effective half-…
Vol. DistribusiThe population PK m…
KlirensClearance is approx…
Genetik -
Sotevtamab DB19120
biotech | CAS: 2411526-47-9

Sotevtamab is under investigation in clinical trial NCT06225843 (Sotevtamab (AB-16B5) Combined With FOLFOX as Neoadjuvant Treatment Prior to Resection of Colorectal Cancer Liver Metastasis).

Waktu Paruh-
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Genetik -
Soticlestat DB16987
small molecule | CAS: 1429505-03-2

Deskripsi belum tersedia.

Kategori:
Cholesterol 24S-Hydroxylase Inhibitor
Target Protein:
Cholesterol 24-hydroxylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sotigalimab DB16413
biotech | CAS: 2305607-45-6

Sotigalimab is under investigation in clinical trial NCT03123783 (CD40 Agonistic Antibody APX005M in Combination With Nivolumab).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sotirimod DB05680
small molecule | CAS: 227318-75-4

Deskripsi belum tersedia.

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Sotorasib Approved DB15569
small molecule | CAS: 2252403-56-6

Sotorasib, also known as AMG-510, is an acrylamide-derived KRAS inhibitor developed by Amgen.[A187547,A187556] It is indicated in the treatment of adult patients with KRAS G12C mutant non-small cell lung cancer.[L34288] This mutation makes up >50% of all KRAS…

Kategori:
Antineoplastic AgentsAntineoplastic Agents, ImmunologicalAntineoplastic and Immunomodulating Agents +13
Target Protein:
GTPase KRas
Waktu ParuhSotorasib has a ter…
Vol. DistribusiThe volume of distr…
KlirensSotorasib has an ap…
Genetik -
Sotrastaurin DB12369
small molecule | CAS: 425637-18-9

Sotrastaurin has been used in trials studying the basic science and treatment of Uveal Melanoma, Richter Syndrome, Prolymphocytic Leukemia, Recurrent Mantle Cell Lymphoma, and Recurrent Small Lymphocytic Lymphoma, among others.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Protein kinase C theta typeProtein kinase C beta typeProtein kinase C alpha type
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sotrovimab Approved DB16355
biotech | CAS: 2423014-07-5

Sotrovimab (VIR-7831), also known as GSK4182136, is a monoclonal antibody that can neutralize the SARS-CoV-2 virus.[L34440] Sotrovimab was initially been granted emergency use authorization (EUA) to treat mild-to-moderate COVID-19 on May 26, 2021, based on in…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntibodies +13
Target Protein:
Spike glycoprotein
Waktu ParuhThis antibody has u…
Vol. DistribusiSotrovimab is an Fc…
Klirens-
Genetik -
Sour cherry Approved DB10630
biotech

Sour cherry allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sovaprevir DB12069
small molecule | CAS: 1001667-23-7

Sovaprevir has been investigated for the treatment of Hepatitis C, Chronic.

Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sovesudil DB18812
small molecule | CAS: 1333400-14-8

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicBenzene Derivatives
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sovleplenib DB17557
small molecule | CAS: 1415792-84-5

Sovleplenib is a novel, investigational, selective small molecule inhibitor for oral administration targeting spleen tyrosine kinase (Syk). It is under investigation in clinical trial NCT03483948 (Phase I Study of Hmpl-523+azacitidine in Elderly Patients With…

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Soy sterol DB11325
biotech | CAS: 129311-52-0

Deskripsi belum tersedia.

Kategori:
Biological FactorsCholestanesFused-Ring Compounds +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Soybean oil Approved DB09422
biotech | CAS: 8001-22-7

Derived from soybeans, soybean oil is a common vegetable oil and a source of polyunsaturated and saturated fatty acids. It is a complex mixture of triglycerides where per 100 g, soybean oil has 16 g of saturated fat, 23 g of monounsaturated fat, and 58 g of p…

Kategori:
Biological ProductsCaloric AgentsComplex Mixtures +12
Target Protein:
Peroxisome proliferator-activated receptor alpha
Waktu Paruh-
Vol. DistribusiAfter triglycerides…
KlirensThe elimination rat…
Genetik -
SP-420 DB16069
small molecule | CAS: 911714-45-9

SP-420 is under investigation in clinical trial NCT03801889 (SP-420 in Subjects With Transfusion-dependent Beta-thalassemia or Other Rare Anemias).

Kategori:
CyclohexanesCycloparaffinsKetones +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sp-722 DB04503
small molecule

Deskripsi belum tersedia.

Target Protein:
Thymidylate synthaseThymidylate synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SP-8203 DB11670
small molecule | CAS: 1176758-04-5

SP-8203 has been used in trials studying the treatment of Ischemic Stroke.

Kategori:
AcetatesAcids, AcyclicAmides +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SP-876 DB03558
small molecule

Deskripsi belum tersedia.

Target Protein:
Thymidylate synthaseThymidylate synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SP2456 DB03957
small molecule

Deskripsi belum tersedia.

Target Protein:
Interleukin-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Spaglumic acid DB08835
small molecule | CAS: 4910-46-7

Spaglumic acid is the ?-aspartyl isoform of N-Acetyl-l-aspartylglutamate (isospaglumic Acid is N-(N-Acetyl-l-?-aspartyl)-l-glutamic acid). In eye drops, spaglumic acid is either a magnesium or sodium salt of N-Acetyl-l-aspartylglutamate. Spaglumic acid is a m…

Kategori:
Antiallergic Agents, Excl. CorticosteroidsDecongestants and AntiallergicsMast Cell Stabilizers +3
Target Protein:
Glutamate carboxypeptidase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

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Sparfloxacin Approved DB01208
small molecule | CAS: 110871-86-8

Sparfloxacin is a fluoroquinolone antibiotic indicated for bacterial infections. Sparfloxacin exerts its antibacterial activity by inhibiting DNA gyrase, a bacterial topoisomerase. DNA gyrase is an essential enzyme which controls DNA topology and assists in D…

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +16
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA gyrase subunit A +2
Waktu ParuhMean terminal elimi…
Vol. Distribusi-
Klirens-
Genetik -
Sparfosic acid DB03459
small molecule | CAS: 51321-79-0

Sparfosic acid is a solid. This compound belongs to the n-acyl-alpha amino acids. These are compounds containing an alpha amino acid which bears an acyl group at the terminal nitrogen atom. This substance is known to target aspartate carbamoyltransferase cata…

Kategori:
AcetatesAcids, AcyclicAmino Acids +12
Target Protein:
Aspartate carbamoyltransferase catalytic chainMultifunctional protein CAD
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sparsentan Approved DB12548
small molecule | CAS: 254740-64-2

Sparsentan is a dual antagonist of the endothelin type A receptor (ET<sub>A</sub>R) and the angiotensin II (Ang II) type 1 receptor (AT<sub>1</sub>R) with a similar affinity for both (9.3 nM for ET<sub>A</sub>R and 0.8 nM for AT<sub>1</sub>R).[A257330,L45300]…

Kategori:
Agents Acting on the Renin-Angiotensin SystemAmidesAngiotensin 2 Receptor Blocker +30
Target Protein:
Endothelin-1 receptorType-1 angiotensin II receptorType-2 angiotensin II receptor
Waktu ParuhSparsentan has an e…
Vol. DistribusiAt the approved rec…
KlirensSparsentan has a ti…
Genetik -
Spartalizumab DB14892
biotech | CAS: 1935694-88-4

Spartalizumab is under investigation in clinical trial NCT02605967 (Safety and Efficacy Study of PDR001 in Patients With Recurrent or Metastatic Nasopharyngeal Carcinoma).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Target Protein:
Programmed cell death protein 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sparteine DB06727
small molecule | CAS: 90-39-1

Sparteine is a plant alkaloid derived from _Cytisus scoparius_ and _Lupinus mutabilis_ which may chelate calcium and magnesium. It is a sodium channel blocker, so it falls in the category of class 1a antiarrhythmic agents. Sparteine is not currently FDA-appro…

Kategori:
AlkaloidsAntiarrhythmic agentsAntiarrhythmics, Class I +13
Waktu Paruh-
Vol. Distribusi-
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Genetik -
SPC2968 DB06351
biotech

SPC2968 is a synthetic antisense oligodeoxynucleotide targeting hypoxia-inducible factor-1alpha (HIF-1alpha). It was under investigation in clinical trial NCT02564614 (A Study of Hypoxia-inducible Factor 1a (HIF1A) Messenger Ribonucleic Acid (mRNA) Antagonist…

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Spearmint Approved DB10683
biotech

Spearmint allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 11801–11850 dari 13591
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