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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

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Halaman 234 / 236
Zetomipzomib DB16070
small molecule | CAS: 1629677-75-3

Zetomipzomib is under investigation in clinical trial NCT04033926 (A Phase 2 Study of KZR-616 to Evaluate Safety and Efficacy in Patients With Active Polymyositis or Dermatomyositis).

Kategori:
Oxazines
Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech

Deskripsi belum tersedia.

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Zibotentan DB06629
small molecule | CAS: 186497-07-4

Deskripsi belum tersedia.

Target Protein:
Endothelin-1 receptor
Waktu Paruh-
Vol. Distribusi-
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Ziconotide Approved DB06283
biotech | CAS: 107452-89-1

Ziconotide (also known as SNX-111) is a neurotoxic peptide derived from the cone snail _Conus magus_ comprising 25 amino acids with three disulphide bonds.[A202835, L13389] Other such peptides, collectively termed conotoxins, exist, and some have shown effica…

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAntiarrhythmic agents +22
Target Protein:
Voltage-dependent N-type calcium channel subunit alpha-1BVoltage-dependent P/Q-type calcium channel subunit alpha-1A
Waktu ParuhIn patients adminis…
Vol. DistribusiIn patients adminis…
KlirensZiconotide CSF clea…
Genetik -
Zicronapine DB12188
small molecule | CAS: 170381-16-5

Zicronapine has been used in trials studying the treatment of Schizophrenia.

Target Protein:
D(2) dopamine receptorD(1A) dopamine receptor5-hydroxytryptamine receptor 2A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zidebactam DB13090
small molecule | CAS: 1436861-97-0

Zidebactam is under investigation in clinical trial NCT02674347 (MAD Study to Evaluate the Safety, Tolerability and Pharmacokinetics of Intravenous Zidebactam in Healthy Adults).

Kategori:
Aza CompoundsCycloparaffins
Waktu Paruh-
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Zidovudine Approved DB00495
small molecule | CAS: 30516-87-1

A dideoxynucleoside compound in which the 3'-hydroxy group on the sugar moiety has been replaced by an azido group. This modification prevents the formation of phosphodiester linkages which are needed for the completion of nucleic acid chains. The compoun…

Kategori:
Agents Causing Muscle ToxicityAnti-HIV AgentsAnti-Infective Agents +37
Target Protein:
Receptor-type tyrosine-protein kinase FLT3Reverse transcriptase/RNaseHGag-Pol polyprotein +1
Waktu ParuhElimination half li…
Vol. DistribusiApparent volume of …
Klirens* 0.65 +/- 0.29 L/h…
Genetik -
small molecule | CAS: 29706-85-2

Deskripsi belum tersedia.

Kategori:
DeoxyribonucleosidesDeoxyribonucleotidesDideoxynucleosides +6
Target Protein:
Thymidylate kinaseThymidylate kinase
Waktu Paruh-
Vol. Distribusi-
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Zifibancimig DB19332
biotech | CAS: 2517939-46-5

Zifibancimig is under investigation in clinical trial NCT04567303, focusing on participants with neovascular age-related macular degeneration.

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Ziftomenib DB17171
small molecule | CAS: 2134675-36-6

Deskripsi belum tersedia.

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Zigakibart DB18892
biotech | CAS: 2642175-46-8

Zigakibart is under investigation in clinical trial NCT05852938 (A Study of BION-1301 in Adults With Iga Nephropathy).

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Genetik -
biotech | CAS: 2220231-04-7

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
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Zilebesiran DB18929
biotech | CAS: 2380166-33-4

Zilebesiran is under investigation in clinical trial NCT06272487 (Zilebesiran as Add-on Therapy in Patients With High Cardiovascular Risk and Hypertension Not Adequately Controlled by Standard of Care Antihypertensive Medications (KARDIA-3)).

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Zileuton Approved DB00744
small molecule | CAS: 111406-87-2

Leukotrienes are substances that induce numerous biological effects including augmentation of neutrophil and eosinophil migration, neutrophil and monocyte aggregation, leukocyte adhesion, increased capillary permeability, and smooth muscle contraction. These …

Kategori:
Agents to Treat Airway DiseaseAmidesAnalgesics +19
Target Protein:
Polyunsaturated fatty acid 5-lipoxygenase
Waktu Paruh2.5 hours
Vol. Distribusi* 1.2 L/kg
Klirens* Apparent oral cl=…
Genetik -
Zilovertamab DB18403
biotech | CAS: 2485779-13-1

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2376463-48-6

Zilovertamab vedotin is an Antibody-drug conjugate (ADC) comprising an anti-ROR1 monoclonal antibody (UC-961), a proteolytically cleavable maleimidocaproyl-valine-citrulline-para-aminobenzoate linker (mc-vc-PAB), and a monomethyl auristatin E (MMAE) cytotoxin.

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Zilpaterol DB11479
small molecule | CAS: 119520-05-7

Zilpaterol is a ?2 adrenergic agonist sold under the trade name, Zilmax, produced by Intervet, a subsidiary of Merck & Co. Zilpaterol is typically fed to cattle in the last three to six weeks of life with a brief washout period to clear the drug from the tiss…

Kategori:
Heterocyclic Compounds, Fused-RingOrganosilicon CompoundsReceptors, Adrenergic, beta
Waktu Paruh-
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Ziltivekimab DB18836
biotech | CAS: 2226654-05-1

Ziltivekimab is under investigation in clinical trial NCT06200207 (A Research Study Looking Into How Ziltivekimab Works Compared to Placebo in Participants With Heart Failure and Inflammation).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
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Zilucoplan Approved DB15636
small molecule | CAS: 1841136-73-9

Zilucoplan is a 15 amino-acid, synthetic macrocyclic peptide. It is a complement inhibitor that works to prevent the activation of C5, which is a complement protein involved in the innate immune system to initiate inflammatory responses.[A261841] On October 1…

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating AgentsBlood Proteins +5
Target Protein:
Complement C5
Waktu ParuhThe mean plasma ter…
Vol. DistribusiThe mean volume of …
KlirensNo information is a…
Genetik -
Zilurgisertib DB18152
small molecule | CAS: 2173389-57-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Zimberelimab DB17505
biotech | CAS: 2259860-24-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zimelidine Approved DB04832
small molecule | CAS: 56775-88-3

Zimelidine has been banned worldwide due to serious, sometimes fatal, cases of central and/or peripheral neuropathy known as Guillain-Barré syndrome and due to a peculiar hypersensitivity reaction involving many organs including skin exanthema, flu-like sympt…

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsCytochrome P-450 CYP3A Inhibitors +16
Target Protein:
Sodium-dependent serotonin transporterAmine oxidase [flavin-containing] BAmine oxidase [flavin-containing] A
Waktu Paruh8.4 +/- 2.0 hours f…
Vol. Distribusi-
Klirens-
Genetik -
Zinc Approved DB01593
small molecule | CAS: 7440-66-6

A metallic element of atomic number 30 and atomic weight 65.38. It is a necessary trace element in the diet, forming an essential part of many enzymes, and playing an important role in protein synthesis and in cell division. Zinc deficiency is associated with…

Kategori:
Agents for Treatment of Hemorrhoids and Anal Fissures for Topical UseDiet, Food, and NutritionElements +12
Target Protein:
B1 bradykinin receptorMethylated-DNA--protein-cysteine methyltransferaseFructose-bisphosphate aldolase A +121
Waktu ParuhThe half-life of zi…
Vol. DistribusiA pharmacokinetic s…
KlirensIn one study of hea…
Genetik -
Zinc acetate Approved DB14487
small molecule | CAS: 557-34-6

Deskripsi belum tersedia.

Kategori:
AcetatesAcids, AcyclicAgents for Treatment of Hemorrhoids and Anal Fissures for Topical Use +7
Target Protein:
B1 bradykinin receptorMethylated-DNA--protein-cysteine methyltransferaseFructose-bisphosphate aldolase A +121
Waktu ParuhThe half-life of zi…
Vol. DistribusiA pharmacokinetic s…
KlirensIn one study of hea…
Genetik -
Zinc ascorbate Approved DB14485
small molecule | CAS: 331242-75-2

Deskripsi belum tersedia.

Kategori:
Agents for Treatment of Hemorrhoids and Anal Fissures for Topical UseMetal cationsMetal divalent cations +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zinc cation DB14532
small molecule | CAS: 23713-49-7

Deskripsi belum tersedia.

Kategori:
Copper Absorption InhibitorDecreased Copper Ion AbsorptionMetal cations +3
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Zinc chloride Approved DB14533
small molecule | CAS: 7646-85-7

Zinc chloride is a solution of ions indicated for use in total parenteral nutrition to maintain zinc levels and prevent deficiency syndromes.[L14189] Zinc chloride was granted FDA approval before 26 June 1986.[L14189]

Kategori:
AcidsAcids, NoncarboxylicAgents for Treatment of Hemorrhoids and Anal Fissures for Topical Use +20
Target Protein:
B1 bradykinin receptorMethylated-DNA--protein-cysteine methyltransferaseFructose-bisphosphate aldolase A +94
Waktu ParuhUsing a two compart…
Vol. Distribusi-
KlirensIn one study of hea…
Genetik -
Zinc citrate DB11154
small molecule | CAS: 546-46-3

Zinc citrate is a zinc salt of citric acid. It is available as dietary supplements as a treatment of zinc deficiency and source of zinc, which is an essential trace element. Zinc citrate demonstrates effective absorption following oral administration [A27280].

Kategori:
Metal cationsMetal divalent cationsZinc Compounds
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Zinc gluconate Approved DB11248
small molecule | CAS: 4468-02-4

Zinc gluconate is a zinc salt of gluconic acid comprised of two gluconic acid molecules for each zinc cation (2+). Zinc gluconate is a generally recognized as safe (GRAS) substance by FDA [L2081]. It is available as a trace mineral supplement and over the cou…

Kategori:
Acids, AcyclicAgents for Treatment of Hemorrhoids and Anal Fissures for Topical UseAlimentary Tract and Metabolism +8
Waktu Paruh280 days [L2091]
Vol. DistribusiStored primarily in…
KlirensPlease refer to Dru…
Genetik -
Zinc iodide DB15961
small molecule | CAS: 10139-47-6

Deskripsi belum tersedia.

Kategori:
AnionsElectrolytesIodine Compounds +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 14354-67-7

Deskripsi belum tersedia.

Kategori:
Biological FactorsCoordination ComplexesHeterocyclic Compounds, Fused-Ring +5
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Zinc orotate DB15720
small molecule | CAS: 60388-02-5

Deskripsi belum tersedia.

Kategori:
PyrimidinesPyrimidinones
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Zinc phenolsulfonate Approved DB15793
small molecule | CAS: 127-82-2

Deskripsi belum tersedia.

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Zinc picolinate DB11175
small molecule | CAS: 17949-65-4

Zinc picolinate is a zinc salt of picolinic acid. It is available as OTC dietary supplements as a source of zinc to treat and prevent zinc deficiency. The absorption of zinc after oral administration of zinc picolinate is shown to be effective.

Kategori:
Compounds used in a research, industrial, or household settingMetal cationsMetal divalent cations +3
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Zinc sulfate Approved DB09322
small molecule | CAS: 7733-02-0

Zinc sulfate is the inorganic compound with the formula ZnSO4 and historically known as "white vitriol". It is on the World Health Organization's List of Essential Medicines, a list of the most important medication needed in a basic health system.

Kategori:
Agents for Treatment of Hemorrhoids and Anal Fissures for Topical UseAlimentary Tract and MetabolismAstringents +17
Waktu Paruh3 hours
Vol. DistribusiAfter absorption zi…
Klirens-
Genetik -
Zinlirvimab DB18867
biotech | CAS: 2417213-75-1

Zinlirvimab is under investigation in clinical trial NCT03707977 (Dual Bnab Treatment in Children).

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biotech | CAS: 1387453-03-3

Zinpentraxin alfa is a recombinant form of PTX-2, a naturally circulating human protein. It is under investigation in clinical trial NCT01981850 (A Phase 2 Study Of PRM-151 In Subjects With Myelofibrosis).

Kategori:
Acute-Phase ProteinsAmino Acids, Peptides, and ProteinsAmyloid +7
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Zipalertinib DB18763
small molecule | CAS: 1661854-97-2

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
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Zipeprol DB13564
small molecule | CAS: 34758-83-3

Deskripsi belum tersedia.

Kategori:
Antitussive AgentsCentral Nervous System AgentsCough and Cold Preparations +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ziprasidone Approved DB00246
small molecule | CAS: 146939-27-7

Disorders such as schizophrenia and bipolar disorder can significantly impair mood, cognition, and behavior.[A190525] These mental illnesses can often be accompanied by comorbidities such as depression and substance abuse, and can significantly impact the qua…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +45
Target Protein:
D(2) dopamine receptorNeuronal acetylcholine receptor subunit alpha-75-hydroxytryptamine receptor 2A +24
Waktu ParuhThe half life of zi…
Vol. DistribusiThe mean apparent v…
KlirensThe mean apparent s…
Genetik -
biotech | CAS: 2377668-38-5

Deskripsi belum tersedia.

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Zirconium chloride hydroxide Approved DB15479
small molecule | CAS: 10119-31-0

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
biotech

Zirconium panitumumab Zr-89 is under investigation in clinical trial NCT05423197 (Study Evaluating Zr-panitumumab for Assessment of Suspected Metastatic Lesions on 18F-FDG-PET/CT in Head and Neck Squamous Cell Carcinoma).

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Ziritaxestat DB15403
small molecule | CAS: 1628260-79-6

Ziritaxestat is under investigation in clinical trial NCT03798366 (A Clinical Study to Test How Effective and Safe GLPG1690 is for Patients With Systemic Sclerosis).

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ZK-806711 DB03373
small molecule

Deskripsi belum tersedia.

Target Protein:
Serine protease 1
Waktu Paruh-
Vol. Distribusi-
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ZK-93423 DB17063
small molecule | CAS: 83910-44-5

ZK-93423 is a beta-carboline with muscle relaxant activity with agonistic properties at the benzodiazepine receptor.[A253172]

Kategori:
Anti-Anxiety AgentsAnticonvulsantsCentral Nervous System Agents +7
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1Gamma-aminobutyric acid receptor subunit beta-2Gamma-aminobutyric acid receptor subunit gamma-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
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ZM-39923 DB17064
small molecule | CAS: 273727-89-2

ZM-39923 is a small molecule that inhibits Janus kinase and human tissue transglutaminase (TGM2).[A253177]

Target Protein:
Tyrosine-protein kinase JAK1Tyrosine-protein kinase JAK3
Waktu Paruh-
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Zofenopril Approved DB13166
small molecule | CAS: 81872-10-8

Zofenopril is employed as both a cardioprotective and anti-hypertensive agent. It is an angiotensin-converting enzyme (ACE) inhibitor.

Kategori:
ACE Inhibitors and DiureticsAgents Acting on the Renin-Angiotensin SystemAgents causing angioedema +10
Target Protein:
Angiotensin-converting enzyme
Waktu Paruh-
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Zofenoprilat DB08766
small molecule | CAS: 75176-37-3

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, CyclicAmino Acids, Peptides, and Proteins +1
Target Protein:
Cytosol aminopeptidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1323976-37-9

Deskripsi belum tersedia.

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