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11778

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Halaman 233 / 236
biotech | CAS: 943976-23-6

Yttrium Y-90 clivatuzumab tetraxetan is under investigation in clinical trial NCT00603863 (Safety and Efficacy Study of Different Doses of 90Y-hPAM4 Combined With Gemcitabine in Pancreatic Cancer).

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biotech | CAS: 501423-27-4

Deskripsi belum tersedia.

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Z-160 DB12743
small molecule | CAS: 41332-24-5

Z160 has been used in trials studying the treatment of Postherpetic Neuralgia and Lumbosacral Radiculopathy.

Kategori:
Antiarrhythmic agentsBenzene DerivativesCalcium Channel Blockers +3
Target Protein:
Voltage-dependent calcium channel subunit alpha-2/delta-1
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small molecule | CAS: 161401-82-7

Non-methylated, competitive, and irreversible inhibitor of caspase 1, as well as other caspases,1 which can be used directly with purified enzymes. It does not require an esterase to hydrolyze the O-methyl ester like the cell-permeable form, Z-Val-Ala-Asp(O-M…

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsCaspase Inhibitors +7
Target Protein:
Caspase-1
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Zabedosertib DB18767
small molecule | CAS: 1931994-81-8

Deskripsi belum tersedia.

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingProtein Kinase Inhibitors +1
Target Protein:
Interleukin-1 receptor-associated kinase 4
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Zabofloxacin DB12479
small molecule | CAS: 219680-11-2

Zabofloxacin has been used in trials studying the treatment of Community Acquired Pneumonia and Chronic Obstructive Pulmonary Disease.

Kategori:
4-QuinolonesHeterocyclic Compounds, Fused-RingQuinolines +1
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Zafiride DB18371
biotech

Zafiride is a human tumor necrosis factor coupled to the C terminus of CNGRCG peptide.

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Zafirlukast Approved DB00549
small molecule | CAS: 107753-78-6

Zafirlukast is an oral leukotriene receptor antagonist (LTRA) for the maintenance treatment of asthma, often used in conjunction with an inhaled steroid and/or long-acting bronchodilator. It is available as a tablet and is usually dosed twice daily. Another l…

Kategori:
Acids, AcyclicAgents to Treat Airway DiseaseAmides +37
Target Protein:
Cysteinyl leukotriene receptor 1
Waktu Paruh10 hours
Vol. Distribusi* 70 L
Klirens* apparent oral CL=…
Genetik -
biotech | CAS: 2567881-78-9

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
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Zagotenemab DB16674
biotech | CAS: 2019133-28-7

Zagotenemab is under investigation in clinical trial NCT03518073 (A Study of LY3303560 in Participants With Early Symptomatic Alzheimer's Disease).

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Zalcitabine Approved DB00943
small molecule | CAS: 7481-89-2

A dideoxynucleoside compound in which the 3'-hydroxyl group on the sugar moiety has been replaced by a hydrogen. This modification prevents the formation of 5' to 3' phosphodiester linkages, which are needed for the elongation of DNA chains, thus resulting in…

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +20
Target Protein:
Gag-Pol polyproteinReverse transcriptase/RNaseH
Waktu Paruh2 hours
Vol. Distribusi* 0.304 to 0.734 L/…
Klirens* 285 mL/min [HIV-i…
Genetik -
Zaleplon Approved DB00962
small molecule | CAS: 151319-34-5

Zaleplon is a sedative/hypnotic, mainly used for insomnia. It is known as a nonbenzodiazepine hypnotic. Zaleplon interacts with the GABA receptor complex and shares some of the pharmacological properties of the benzodiazepines. Zaleplon is a schedule IV drug …

Kategori:
AcetatesAcids, AcyclicAmides +22
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1
Waktu ParuhApproximately 1 hour
Vol. Distribusi* 1.4 L/kg
Klirens* 1 L/h/kg
Genetik -
small molecule

Deskripsi belum tersedia.

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Zaltoprofen DB06737
small molecule | CAS: 74711-43-6

A non-steroidal anti-inflammatory drug approved for use in Japan in 1993.

Kategori:
Acids, AcyclicAgents causing hyperkalemiaAgents that produce hypertension +19
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Zalunfiban DB18766
small molecule | CAS: 1448313-27-6

Deskripsi belum tersedia.

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Zalutumumab DB12202
biotech | CAS: 667901-13-5

Zalutumumab is a fully human IgG1 monoclonal antibody designed to bind with selectivity to the epidermal growth factor receptor (EGFR). Zalutumumab has been investigated for the treatment of Squamous Cell Cancer and Head and Neck Cancer.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Target Protein:
Epidermal growth factor receptor
Waktu Paruh-
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Zalypsis DB12454
small molecule | CAS: 308359-57-1

Zalypsis has been used in trials studying the treatment of Lymphoma, Solid Tumors, Ewing's Sarcoma, Endometrial Cancer, and Uterine Cervical Cancer, among others.

Kategori:
AlkaloidsHeterocyclic Compounds, Fused-RingIsoquinolines
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Zamaporvint DB18765
small molecule | CAS: 1900754-56-4

Deskripsi belum tersedia.

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Zamerovimab DB17766
biotech | CAS: 2419087-87-7

Deskripsi belum tersedia.

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Zampilimab DB16381
biotech | CAS: 2098280-42-1

Zampilimab is under investigation in clinical trial NCT04335578 (A Study to Evaluate Safety, Tolerability, Pharmacokinetics, and Efficacy of UCB7858 in Adult Kidney Transplant Recipients With Chronic Allograft Injury).

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biotech

Deskripsi belum tersedia.

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Zanapezil DB04859
small molecule | CAS: 142852-50-4

Zanapezil (TAK-147) is a selective acetylcholine (ACh) esterase inhibitor under investigation as a drug for Alzheimer's disease (AD) treatment.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Acetylcholinesterase
Waktu Paruh-
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Zandatrigine DB19051
small molecule | CAS: 2154406-04-7

Zandatrigine is under investigation in clinical trial NCT05226780 (Extension Study to Evaluate How Safe and Tolerable NBI-921352 Is as an Adjunctive Therapy for Participants With SCN8A-DEE).

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Zanidatamab Approved DB15471
biotech | CAS: 2169946-15-8

Zanidatamab is a bispecific antibody that binds two non-overlapping sites of HER2 (ERBB2).[A264718] It has been investigated for the treatment of HER2-positive solid tumors, including gastroesophageal, colorectal, and biliary tract cancers.[A264718] In No…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
Target Protein:
Receptor tyrosine-protein kinase erbB-2
Waktu ParuhBased on population…
Vol. DistribusiBased on population…
KlirensBased on population…
Genetik -
biotech | CAS: 2329698-82-8

According to Zymeworks, "ZW49 (zanidatamab zovodotin) is a bispecific anti-HER2 ADC that is based on the same antibody framework as [ZW25] but armed with a cytotoxic payload."[L8234] It is being investigated for several indications characterized by HER2 expre…

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Zanolimumab DB17376
biotech | CAS: 652153-01-0

Zanolimumab is a fully human monoclonal antibody directed against CD4.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
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Zansecimab DB16389
biotech | CAS: 2415205-37-5

Zansecimab is under investigation in clinical trial NCT04342897 (A Study of LY3127804 in Participants With COVID-19).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntibodies +9
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biotech

Zanthoxylum clava-herculis bark is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

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Zanubrutinib Approved DB15035
small molecule | CAS: 1691249-45-2

Zanubrutinib is a novel Bruton's tyrosine kinase (BTK) inhibitor used for the treatment of adult patients with mantle cell lymphoma (MCL) who have received at least one prior therapy.[L10163] Mantle cell lymphoma is an aggressive mature B-cell non-Hodgkin lym…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBruton's tyrosine kinase (BTK) inhibitors +19
Target Protein:
Tyrosine-protein kinase BTKEpidermal growth factor receptorReceptor tyrosine-protein kinase erbB-2 +12
Waktu ParuhFollowing administr…
Vol. DistribusiThe geometric mean …
KlirensThe mean (%CV) appa…
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Zanzalintinib DB17525
small molecule | CAS: 2367004-54-2

Deskripsi belum tersedia.

Target Protein:
Hepatocyte growth factor receptor
Waktu Paruh-
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Zapnometinib DB18244
small molecule | CAS: 303175-44-2

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAminesAminobenzoates +4
Waktu Paruh-
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Zardaverine DB02918
small molecule | CAS: 101975-10-4

Deskripsi belum tersedia.

Kategori:
Anti-Asthmatic AgentsAutonomic AgentsBronchodilator Agents +4
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4D
Waktu Paruh-
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Zasocitinib DB19278
small molecule | CAS: 2272904-53-5

Deskripsi belum tersedia.

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Zastumotide DB14926
biotech | CAS: 949885-73-8

Zastumotide is a recombinant MAGE-A3 Antigen-Specific Cancer Immunotherapeutic (MAGE-A3 ASCI) also known as astuprotimut-R. It is under investigation in clinical trial NCT00257738 (0804 GCC: MAGE-A3/HPV 16 Vaccine for Squamous Cell Carcinoma of the Head and N…

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Zatolmilast DB14790
small molecule | CAS: 1606974-33-7

BPN-14770 is under investigation in clinical trial NCT02840279 (A Multiple Ascending Dose Study of BPN14770 in Healthy Young and Elderly Male or Female Subjects).

Kategori:
Acids, AcyclicEnzyme InhibitorsFatty Acids +5
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4D
Waktu Paruh-
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Zavegepant Approved DB15688
small molecule | CAS: 1337918-83-8

Zavegepant (BHV-3500) is a calcitonin gene-related peptide (CGRP) receptor antagonist.[L45505] CGRP is released from sensory nerves and acts as a strong vasodilator, and thanks to these properties, it is involved in pain pathways. CGRP receptors are expressed…

Kategori:
Antimigraine PreparationsCalcitonin Gene-Related Peptide (CGRP) AntagonistsCalcitonin Gene-Related Peptide Receptor Antagonists +14
Target Protein:
Calcitonin gene-related peptide type 1 receptor
Waktu ParuhFollowing a 10 mg d…
Vol. DistribusiIntranasal zavegepa…
KlirensIntranasal zavegepa…
Genetik -
ZB131 DB17164
biotech

ZB131 is a monoclonal antibody with a high affinity and specificity for cancer-specific plectin (CSP), a cell surface protein identified in a wide range of cancers that correlates with poor prognosis and aggressive tumors.[L44081]

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ZD-6126 DB11872
small molecule | CAS: 219923-05-4

ZD6126 has been used in trials studying the treatment of Kidney Neoplasms, Colorectal Neoplasms, Metastases, Neoplasm, and Carcinoma, Renal Cell.

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ZD4407 DB06539
small molecule | CAS: 166882-70-8

The drug ZD4407, an antiasthmatic developed by AstraZeneca, functions as a 5-lipoxygenase inhibitor. It entered Phase 1 clinical trials for chronic obstructive pulmonary disease (COPD) in the United Kingdom but was discontinued during this phase in March 2003

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Zea mays pollen Approved DB10357
biotech

Zea mays pollen is the pollen of the Zea mays plant. Zea mays pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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Zeatin DB11337
small molecule | CAS: 1637-39-4

An aminopurine factor in plant extracts that induces cell division. (Grant & Hackh's Chemical Dict, 5th ed)

Kategori:
CytokininsGrowth SubstancesHeterocyclic Compounds, Fused-Ring +2
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Zeaxanthin Approved DB11176
small molecule | CAS: 144-68-3

Zeaxanthin is a most common carotenoid alcohols found in nature that is involved in the xanthophyll cycle. As a coexistent isomer of lutein, zeaxanthin is synthesized in plants and some micro-organisms. It gives the distinct yellow color to many vegetables an…

Kategori:
AlkenesBiological FactorsCarotenoids +8
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ZED-1227 DB19208
small molecule | CAS: 1542132-88-6

ZED-1227 is under investigation in clinical trial NCT05305599 (Different Doses of ZED1227 vs. Placebo in NAFLD).

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Zelavespib DB12638
small molecule | CAS: 873436-91-0

Zelavespib (PU-H71) has been used in trials studying the treatment of LYMPHOMA, Solid Tumors, Metastatic Solid Tumor, and Myeloproliferative Neoplasms (MPN).

Kategori:
Antineoplastic AgentsDioxolesHeterocyclic Compounds, Fused-Ring
Target Protein:
Heat shock protein HSP 90-beta
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Zelpultide alfa DB18587
biotech | CAS: 2245003-06-7

Zelpultide alfa is a recombinant human surfactant protein D.

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Zelquistinel DB19336
small molecule | CAS: 2151842-64-5

Zelquistinel is under investigation in clinical trial NCT06547489 (GATE-251 or Placebo for the Reduction of Symptoms of Major Depressive Disorder).

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Zeluvalimab DB18868
biotech | CAS: 2315361-37-4

Zeluvalimab is under investigation in clinical trial NCT04631601 (Safety and Efficacy of Therapies for Metastatic Castration-resistant Prostate Cancer (Mcrpc)).

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Zemirciclib DB18823
small molecule | CAS: 2057509-72-3

Deskripsi belum tersedia.

Target Protein:
Cyclin-dependent kinase 9
Waktu Paruh-
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Zenarestat DB02132
small molecule | CAS: 112733-06-9

Deskripsi belum tersedia.

Kategori:
Aldehyde Reductase, antagonists & inhibitorsEnzyme InhibitorsHeterocyclic Compounds, Fused-Ring
Target Protein:
Aldo-keto reductase family 1 member B1
Waktu Paruh-
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Zeranol DB11478
small molecule | CAS: 26538-44-3

Zeranol is a non-steroidal estrogen agonist. It is a mycotoxin, derived from fungi in the Fusarium family, and may be found as a contaminant in fungus-infected crops. It is 3-4x more potent as an estrogen agonist than the related compound zearalenone.

Kategori:
Benzene DerivativesEstrogensEstrogens, Non-Steroidal +6
Target Protein:
Estrogen receptorSex hormone-binding globulin
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