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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
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14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 233 / 282
Riltozinameran Approved DB17095
biotech | CAS: 2749948-25-0

The Omicron variant of SARS-CoV-2 is a variant of concern that was first reported in November 2021.[L43922] It tends to cause less severe disease but is significantly more virulent than both the original virus and earlier variants (e.g. Delta).[L43917] As of …

Kategori:
COVID-19 VaccinesmRNA VaccinesVaccines +1
Waktu Paruh-
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Riluzole Approved DB00740
small molecule | CAS: 1744-22-5

A glutamate antagonist (receptors, glutamate) used as an anticonvulsant (anticonvulsants) and to prolong the survival of patients with amyotrophic lateral sclerosis. Riluzole is marketed as Rilutek by Sanofi.

Kategori:
AnticonvulsantsBCRP/ABCG2 SubstratesBenzothiazoles +15
Target Protein:
Sodium channel protein type 5 subunit alphaSodium channel protein type 11 subunit alphaCystine/glutamate transporter
Waktu ParuhThe mean eliminatio…
Vol. Distribusi-
Klirens-
Genetik -
Rilvegostomig DB18991
biotech | CAS: 2640305-01-5

Rilvegostomig is under investigation in clinical trial NCT06109779 (Rilvegostomig + Chemotherapy as Adjuvant Therapy for Biliary Tract Cancer After Resection (Artemide-biliary01)).

Waktu Paruh-
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Rilzabrutinib DB17709
small molecule | CAS: 1575591-66-0

Rilzabrutinib is an oral, reversible covalent inhibitor of Bruton's tyrosine kinase being investigated for the treatment of immune disorders, such as immune thrombocytopenic purpura.[A259073, A259078]

Waktu Paruh-
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Rimacalib DB12571
small molecule | CAS: 215174-50-8

Rimacalib has been used in trials studying the treatment of Rheumatoid Arthritis (RA).

Kategori:
Enzyme InhibitorsOxazinesProtein Kinase Inhibitors
Target Protein:
Calcium/calmodulin-dependent protein kinase type II subunit alphaCalcium/calmodulin-dependent protein kinase type II subunit betaCalcium/calmodulin-dependent protein kinase type II subunit delta +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rimantadine Approved DB00478
small molecule | CAS: 13392-28-4

An RNA synthesis inhibitor that is used as an antiviral agent in the prophylaxis and treatment of influenza.

Kategori:
AdamantanesAnti-Infective AgentsAntiinfectives for Systemic Use +8
Target Protein:
Matrix protein 2
Waktu Paruh25 to 30 hours in y…
Vol. Distribusi-
Klirens-
Genetik -
Rimazolium DB13289
small molecule | CAS: 35615-72-6

Rimazolium is an experimental analgesic drug [A176186].

Kategori:
AnalgesicsNervous SystemPyrimidines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rimegepant Approved DB12457
small molecule | CAS: 1289023-67-1

Rimegepant is an oral antagonist of the CGRP receptor developed by Biohaven Pharmaceuticals.[L11028] It received FDA approval on February 27, 2020 for the acute treatment migraine headache,[L11974] and was subsequently approved by the European Commission in A…

Kategori:
AnalgesicsAntimigraine PreparationsBCRP/ABCG2 Substrates +19
Target Protein:
Calcitonin gene-related peptide type 1 receptor
Waktu ParuhThe elimination hal…
Vol. DistribusiAt steady state, th…
Klirens-
Genetik -
Rimeporide DB12861
small molecule | CAS: 187870-78-6

Rimeporide has been used in trials studying the treatment of Muscular Dystrophy, Duchenne.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Rimiducid DB04974
small molecule | CAS: 195514-63-7

Rimiducid is a lipid-permeable tacrolimus analogue and a protein dimerizer. It was designed to overcome limitations of current cellular immunotherapies used for cancer and other blood disorders by enhancing the control of the immune cell activity and function…

Kategori:
Cross-Linking Reagents
Target Protein:
Peptidyl-prolyl cis-trans isomerase FKBP1ASerine/threonine-protein kinase mTOR
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rimiterol DB13559
small molecule | CAS: 32953-89-2

Deskripsi belum tersedia.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic beta-Agonists +8
Target Protein:
Beta-3 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rimonabant Approved DB06155
small molecule | CAS: 168273-06-1

Rimonabant is an anorectic anti-obesity drug produced and marketed by Sanofi-Aventis. It is an inverse agonist for the cannabinoid receptor CB1. Its main avenue of effect is reduction in appetite. Rimonabant is the first selective CB1 receptor blocker to be a…

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAnti-Obesity Agents +12
Target Protein:
Cannabinoid receptor 1G-protein coupled receptor 55
Waktu Paruh6 to 9 days with no…
Vol. Distribusi-
Klirens-
Genetik -
Rimtuzalcap DB16733
small molecule | CAS: 2167246-24-2

Rimtuzalcap is a novel modulator of small-conductance calcium-activated potassium channels that is under investigation for the treatment of essential tremor.[L38414]

Target Protein:
Small conductance calcium-activated potassium channel protein 1Small conductance calcium-activated potassium channel protein 2Small conductance calcium-activated potassium channel protein 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rindopepimut DB05374
small molecule | CAS: 1108208-65-6

Rindopepimut (CDX-110) is an injectable peptide cancer vaccine which targets a mutant protein called EGFRvIII present in about 25% to 30% of glioblastoma cases. The vaccine consists of the EGFRv3-specific peptide (a 13-amino acid mutant vIII epitope) conjugat…

Kategori:
Antineoplastic AgentsAntineoplastic Agents, ImmunologicalBiological Products +2
Target Protein:
Epidermal growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rineterkib DB17560
small molecule | CAS: 1715025-32-3

Rineterkib is an inhibitor of extracellular signal-regulated kinase (ERK) being investigated in NCT04097821 (A Randomized, Open-label, Phase I/II Open Platform Study Evaluating Safety and Efficacy of Novel Ruxolitinib Combinations in Myelofibrosis Patients).

Waktu Paruh-
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Rintatolimod DB16425
biotech | CAS: 38640-92-5

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAntiviral AgentsBase Pair Mismatch +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rinucumab DB16313
biotech | CAS: 1569263-06-4

Rinucumab is under investigation in clinical trial NCT02418754 (Study of Intravitreal REGN2176-3 in Participants With Neovascular ("Wet") Age-related Macular Degeneration (AMD)).

Waktu Paruh-
Vol. Distribusi-
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Riociguat Approved DB08931
small molecule | CAS: 625115-55-1

Riociguat is a soluble guanylate cyclase (sGC) agonist approved in the USA, Europe and several other regions for patients with group I PAH (pulmonary arterial hypertension) in WHO FC II or III; and for the treatment of patients with inoperable CTEPH (chronic …

Kategori:
Antihypertensive AgentsAntihypertensives for Pulmonary Arterial HypertensionBCRP/ABCG2 Substrates +11
Target Protein:
Retinal guanylyl cyclase 1Guanylate cyclase soluble subunit alpha-2
Waktu ParuhAbout 12 hours in p…
Vol. DistribusiVolume of distribut…
Klirens-
Genetik -
Ripasudil DB13165
small molecule | CAS: 223645-67-8

Ripasudil, as hydrochloride hydrate (K-115), is a specifc Rho-associated coiled-coil containing protein kinase (ROCK) inhibitor used for the treatment of glaucoma and ocular hypertension. It was first approved for treatment in Japan in September 2014. This me…

Kategori:
AmidesAntiglaucoma Preparations and MioticsHeterocyclic Compounds, Fused-Ring +5
Target Protein:
Rho-associated protein kinase 1Rho-associated protein kinase 2
Waktu ParuhThe half life of Ri…
Vol. Distribusi-
KlirensRipasudil has a ren…
Genetik -
Ripertamab DB16314
biotech | CAS: 2249927-04-4

Ripertamab is under investigation in clinical trial NCT02772822 (A Study Comparing the Efficiency and Safety of S-chop(cyclophosphamide, Hydroxydaunomycin, Oncovin, and Prednisone) Versus R-CHOP in Untreated Cd20(cluster of Differentiation Antigen 20)-positiv…

Waktu Paruh-
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Genetik -
Ripretinib Approved DB14840
small molecule | CAS: 1442472-39-0

Ripretinib is a kinase inhibitor used for the treatment of advanced gastrointestinal stromal tumor (GIST) that has not adequately responded to other kinase inhibitors such as [sunitinib] and [imatinib]. Ripretinib, also known as Qinlock, is manufactured by De…

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +19
Target Protein:
Mast/stem cell growth factor receptor KitPlatelet-derived growth factor receptor betaAngiopoietin-1 receptor +3
Waktu ParuhThe average half-li…
Vol. DistribusiThe mean volume of …
KlirensThe mean apparent c…
Genetik -
Risankizumab Approved DB14762
biotech | CAS: 1612838-76-2

Risankizumab is a fully humanized IgG1 monoclonal antibody (mAb) directed against interleukin 23 (IL-23).[L39885] It gained its first global approval in Japan in March 2019, followed by approval in Canada, the US, and Europe in April 2019.[A254716] Risankizum…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +15
Target Protein:
Interleukin-23
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe estimated stead…
KlirensThe estimated syste…
Genetik -
Risdiplam Approved DB15305
small molecule | CAS: 1825352-65-5

Risdiplam is an orally bioavailable mRNA splicing modifier used for the treatment of spinal muscular atrophy (SMA).[L12615] It increases systemic SMN protein concentrations by improving the efficiency of _SMN2_ gene transcription. This mechanism of action is …

Kategori:
BCRP/ABCG2 SubstratesCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Substrates +11
Waktu ParuhThe terminal elimin…
Vol. DistribusiFollowing oral admi…
KlirensFor a 14.9kg patien…
Genetik -
Risedronic acid Approved DB00884
small molecule | CAS: 105462-24-6

Risedronic acid is a third generation bisphosphonate that is used for the treatment of some forms of osteoperosis and Paget's disease[FDA Label][A959,A203111]. It functions by preventing resorption of bone[FDA Label][A959].

Kategori:
Agents Causing Muscle ToxicityBisphosphonatesBone Density Conservation Agents +9
Target Protein:
HydroxylapatiteFarnesyl pyrophosphate synthase
Waktu ParuhThe initial half li…
Vol. Distribusi13.8 L/kg[FDA Label…
KlirensMean renal clearanc…
Genetik -
Risperidone Approved DB00734
small molecule | CAS: 106266-06-2

Risperidone is a second-generation antipsychotic (SGA) medication used in the treatment of a number of mood and mental health conditions including schizophrenia and bipolar disorder.[L12885] It is one of the most widely used SGAs. [Paliperidone], another comm…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +42
Target Protein:
5-hydroxytryptamine receptor 2AD(2) dopamine receptorAlpha-1B adrenergic receptor +9
Waktu Paruh3 hours in extensiv…
Vol. DistribusiThe volume of distr…
KlirensRisperidone is clea…
Genetik -
Risuteganib DB14911
small molecule | CAS: 1307293-62-4

Risuteganib is under investigation in clinical trial NCT02348918 (Phase 2 Randomized Clinical Trial of Luminate® as Compared to Avastin® in the Treatment of Diabetic Macular Edema).

Kategori:
Amino Acids, Peptides, and Proteins
Target Protein:
Vascular endothelial growth factor A, long formVascular endothelial growth factor BVascular endothelial growth factor C +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ritanserin DB12693
small molecule | CAS: 87051-43-2

Ritanserin has been used in trials studying the treatment of Cocaine-Related Disorders.

Kategori:
Anti-Anxiety AgentsAntidepressive AgentsAntidepressive Agents, Second-Generation +21
Target Protein:
5-hydroxytryptamine receptor 2B5-hydroxytryptamine receptor 2CVoltage-dependent N-type calcium channel subunit alpha-1B +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ritiometan Approved DB13267
small molecule | CAS: 34914-39-1

Ritiometan is a nasal spray which is marketed by the name Nécyrane in France. It is indicated for use in viral rhinitis/ the common cold.

Kategori:
Nasal Preparations
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ritivixibat DB18030
small molecule | CAS: 2460667-52-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ritlecitinib Approved DB14924
small molecule | CAS: 1792180-81-4

Ritlecitinib (PF-06651600) is a highly selective inhibitor of Janus kinase 3 (JAK3) and the tyrosine kinase expressed in hepatocellular carcinoma (TEC) kinase family. In June 2023, it was approved by the FDA for the treatment of severe alopecia areata in adul…

Kategori:
Antineoplastic and Immunomodulating AgentsCytochrome P-450 CYP1A2 InhibitorsCytochrome P-450 CYP1A2 Inhibitors (strength unknown) +16
Target Protein:
Tyrosine-protein kinase JAK3Tyrosine-protein kinase TecTyrosine-protein kinase ITK/TSK +3
Waktu ParuhRitlecitinib has a …
Vol. DistribusiRitlecitinib is pre…
KlirensRitlecitinib is pre…
Genetik -
Ritobegron DB12080
small molecule | CAS: 255734-04-4

Ritobegron is under investigation in clinical trial NCT02256735 (Study to Investigate the Effect of KUC 7483 CL on the QT/QTc Interval of the ECG in Comparison to Placebo and Moxifloxacin in Healthy Male and Female Volunteers).

Kategori:
Acids, AcyclicAdrenergic AgentsAdrenergic Agonists +15
Target Protein:
Beta-3 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ritodrine Approved DB00867
small molecule | CAS: 26652-09-5

Adrenergic beta-agonist used to control premature labor.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic beta-2 Receptor Agonists +18
Target Protein:
Beta-2 adrenergic receptorBeta adrenergic receptorATP-sensitive potassium channel +4
Waktu Paruh1.7-2.6 hours
Vol. Distribusi-
Klirens-
Genetik -
Ritonavir Approved DB00503
small molecule | CAS: 155213-67-5

Ritonavir is an HIV protease inhibitor that interferes with the reproductive cycle of HIV. Although it was initially developed as an independent antiviral agent, it has been shown to possess advantageous properties in combination regimens with low-dose ritona…

Kategori:
Acids, AcyclicAgents Causing Muscle ToxicityAnti-HIV Agents +69
Target Protein:
Gag-Pol polyproteinPol polyproteinNuclear receptor subfamily 1 group I member 2
Waktu ParuhThe approximate hal…
Vol. DistribusiThe estimated volum…
KlirensThe apparent oral c…
Genetik -
Rituximab Approved DB00073
biotech | CAS: 174722-31-7

Rituximab is a genetically engineered chimeric murine/human monoclonal antibody directed against the CD20 antigen found on the surface of normal and malignant B lymphocytes. The antibody is an IgG1 kappa immunoglobulin containing murine light and heavy-chain …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +21
Target Protein:
B-lymphocyte antigen CD20
Gen Terkait:
FCGR3A
Waktu ParuhIn patients with no…
Vol. DistribusiBased on a pharmaco…
KlirensIn patients with no…
Genetik 1 Varian
biotech | CAS: 1613506-32-3

Rivabazumab pegol is being investigated as a treatment of Pseudomonas aeruginosa lung infections in patients with cystic fibrosis.[A259457]

Waktu Paruh-
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Genetik -
Rivanicline DB05855
small molecule | CAS: 15585-43-0

Rivanicline (TC-2403, RJR-2403, (E)-metanicotine) is a partial agonist at neuronal nicotinic acetylcholine receptors, binding primarily to the ?4?2 subtype. It was originally developed as a potential treatment for Alzheimer's disease for its nootropic effects…

Kategori:
AlkaloidsPyridinesSolanaceous Alkaloids
Target Protein:
Neuronal acetylcholine receptor subunit beta-2Interleukin-8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rivaroxaban Approved DB06228
small molecule | CAS: 366789-02-8

Rivaroxaban is an anticoagulant and the first orally active direct factor Xa inhibitor. Unlike warfarin, routine lab monitoring of INR is not necessary. However there is no antidote available in the event of a major bleed. Only the 10 mg tablet can be taken w…

Kategori:
AnticoagulantsAntithrombinsBCRP/ABCG2 Substrates +17
Target Protein:
Coagulation factor X
Waktu ParuhThe terminal half l…
Vol. DistribusiThe steady state Vd…
KlirensSystemic clearance …
Genetik -
Rivastigmine Approved DB00989
small molecule | CAS: 123441-03-2

Rivastigmine is a parasympathomimetic or cholinergic agent for the treatment of mild to moderate dementia of the Alzheimer's type. Rivastigmine is a cholinesterase inhibitor that inhibits both butyrylcholinesterase and acetylcholinesterase.

Kategori:
Acids, AcyclicAnti-Dementia DrugsBradycardia-Causing Agents +13
Target Protein:
AcetylcholinesteraseCholinesterase
Waktu Paruh1.5 hours
Vol. Distribusi* 1.8 to 2.7 L/kg
Klirens* renal cl=2.1-2.8 …
Genetik -
Rivenprost DB16315
small molecule | CAS: 256382-08-8

Rivenprost is under investigation in clinical trial NCT00296556 (Therapeutic Study of ONO-4819CD for Ulcerative Colitis).

Kategori:
Fatty AcidsHeptanoic AcidsLipids
Target Protein:
Prostaglandin E2 receptor EP4 subtypeProstaglandin E2 Receptors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rivipansel DB12778
small molecule | CAS: 927881-99-0

Rivipansel has been used in trials studying the other, basic science, and treatment of Pain Crisis, Renal impairment, Anemia, Sickle Cell, Sickle Cell Disease, and Sickle Cell Disorders, among others.

Kategori:
CarbohydratesGlycoconjugatesLipids
Target Protein:
E-selectinL-selectinP-selectin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rivoceranib DB14765
small molecule | CAS: 811803-05-1

Rivoceranib is under investigation in clinical trial NCT02726854 (Apatinib as Second-line Treatment of Advanced Pancreatic Cancer).

Kategori:
Antineoplastic AgentsEnzyme InhibitorsProtein Kinase Inhibitors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rivoglitazone DB09200
small molecule | CAS: 185428-18-6

Rivoglitazone (INN) is a thiazolidinedione undergoing research for use in the treatment of type 2 diabetes. It is being developed by Daiichi Sankyo Co.

Kategori:
Blood Glucose Lowering AgentsCytochrome P-450 CYP2C8 InhibitorsCytochrome P-450 CYP2C8 Inhibitors (strength unknown) +8
Target Protein:
Peroxisome proliferator-activated receptor gamma
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rizatriptan Approved DB00953
small molecule | CAS: 144034-80-0

Rizatriptan is a second-generation triptan [A258918] and a selective 5-HT<sub>1B and 5-HT1D</sub> receptor agonist.[L46018] Used in the treatment of migraines, rizatriptan was first approved in the US in 1998.[L46018] Rizatriptan is available in oral tablets,…

Kategori:
Agents that produce hypertensionAminesAnalgesics +26
Target Protein:
5-hydroxytryptamine receptor 1B5-hydroxytryptamine receptor 1D5-hydroxytryptamine receptor 1A +3
Gen Terkait:
GNB3
Waktu ParuhThe plasma half-lif…
Vol. DistribusiThe mean volume of …
KlirensAn early study invo…
Genetik 1 Varian
RLY-2608 DB16751
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RLYB212 DB17727
biotech

RLYB212 is a human monoclonal antibody against Antigen-1A Immunoglobulin (HPA-1A). It is currently being developed by Rallybio for the prevention of fetal and neonatal alloimmune thrombocytopenia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Ro 12-7310 DB08455
small molecule | CAS: 65316-65-6

Deskripsi belum tersedia.

Kategori:
AlkenesBiological FactorsCarotenoids +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ro 24-7429 DB16062
small molecule | CAS: 139339-45-0

Ro 24-7429 is under investigation in clinical trial NCT00002314 (A Study of Ro 24-7429 in Patients With Hiv-related Kaposi's Sarcoma).

Kategori:
BenzazepinesHeterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RO-4584820 DB08094
small molecule | CAS: 741713-40-6

Deskripsi belum tersedia.

Target Protein:
Cyclin-dependent kinase 4Cyclin-dependent kinase 1Cyclin-dependent kinase 7 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RO-4987655 DB12933
small molecule | CAS: 874101-00-5

RO4987655 has been used in trials studying the treatment of Neoplasms.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RO-5028442 DB12721
small molecule | CAS: 920022-47-5

RO5028442 has been used in trials studying Autistic Disorder.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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