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16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

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Hasil Pencarian (16004)

Halaman 233 / 321
Omadacycline Approved DB12455
small molecule | CAS: 389139-89-3

Omadacycline has been used in trials studying the treatment of Bacterial Pneumonia, Bacterial Infections, Community-Acquired Infections, and Skin Structures and Soft Tissue Infections. Omadacycline represents a significant advance over the well-known tetracyc…

Kategori:
Anti-Bacterial AgentsAntibacterials for Systemic UseAntiinfectives for Systemic Use +3
Target Protein:
30S ribosomal protein S330S ribosomal protein S730S ribosomal protein S8 +3
Waktu ParuhOmadacycline has a …
Vol. DistribusiOmadacycline has a …
KlirensOmadacycline has a …
Genetik -
Omalizumab Approved DB00043
biotech | CAS: 242138-07-4

Omalizumab is a recombinant DNA-derived humanized monoclonal antibody directed against human immunoglobulin E (IgE).[L50482] IgE promotes the release of inflammatory mediators from mast cells and basophils during allergic and inflammatory reactions. By bindin…

Kategori:
Agents to Treat Airway DiseaseAmino Acids, Peptides, and ProteinsAnti-Allergic Agents +17
Target Protein:
Immunoglobulin heavy constant epsilon
Waktu ParuhIn asthma patients,…
Vol. DistribusiIn patients with as…
KlirensIn pharmacokinetic …
Genetik -
Omapatrilat DB00886
small molecule | CAS: 167305-00-2

Omapatrilat is an investigational drug that inhibits both neutral endopeptidase (NEP) and angiotensin converting enzyme (ACE). The inhibition of NEP elevates natriuretic peptide levels, increasing excretion of sodium in urine, dilating blood vessels, and redu…

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing angioedemaAgents causing hyperkalemia +11
Target Protein:
NeprilysinAngiotensin-converting enzyme
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Omarigliptin DB11992
small molecule | CAS: 1226781-44-7

Omarigliptin has been used in trials studying the treatment of Type 2 Diabetes Mellitus and Chronic Renal Insufficiency.

Kategori:
Agents causing angioedemaBlood Glucose Lowering AgentsDPP-IV Inhibitors +1
Target Protein:
Dipeptidyl peptidase 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Omaveloxolone Approved DB12513
small molecule | CAS: 1474034-05-3

Omaveloxolone (RTA-408) is a semisynthetic oleanane triterpenoid with antioxidant and anti-inflammatory properties.[A257534,A257539] Omaveloxolone acts as an activator of nuclear factor (erythroid-derived 2)-like 2 (Nrf2), a transcription factor that mitigate…

Kategori:
Anti-Inflammatory AgentsAntioxidantsCytochrome P-450 CYP2C8 Inducers +13
Target Protein:
Nuclear factor erythroid 2-related factor 2Kelch-like ECH-associated protein 1
Waktu ParuhOmaveloxolone has a…
Vol. DistribusiOmaveloxolone has a…
KlirensOmaveloxolone has a…
Genetik -
Ombitasvir Approved DB09296
small molecule | CAS: 1258226-87-7

Ombitasvir is a direct acting antiviral medication used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV). HCV is a single-stranded RNA virus that is categorized into nine…

Kategori:
AmidesAminesAmino Acids +18
Target Protein:
Nonstructural protein 5AGenome polyprotein
Waktu ParuhOmbitasvir has a ha…
Vol. DistribusiOmbitasvir has a vo…
KlirensClearance of Ombita…
Genetik -
Ombrabulin DB12882
small molecule | CAS: 181816-48-8

Ombrabulin has been used in trials studying the treatment of Sarcoma, Neoplasms, Solid Tumor, Neoplasms, Malignant, and Advanced Solid Tumors, among others.

Kategori:
Amino AcidsAmino Acids, NeutralAmino Acids, Peptides, and Proteins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Omburtamab DB15635
biotech | CAS: 1895083-75-6

CD276 (B7-H3) is a B7/CD28 immunoglobulin superfamily member frequently expressed among solid human tumours.[A242487, A242492] Omburtamab, formerly the murine anti-B7-H3 antibody 8H9, and its humanized forms are currently under clinical development for use in…

Target Protein:
CD276 antigen
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 873697-71-3

Omecamtiv Mecarbil has been used in trials studying the treatment and basic science of Heart Failure, Echocardiogram, Pharmacokinetics, Chronic Heart Failure, and History of Chronic Heart Failure, among others.

Kategori:
AmidesCardiac Stimulants Excl. Cardiac GlycosidesCardiac Therapy
Target Protein:
Myosin-binding protein C, cardiac-type
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Omega-3 fatty acids Approved DB11133
small molecule | CAS: 329042-31-1

Omega-3 fatty acids are polyunsaturated fatty acids (PUFAs) with a double bond at the third carbon atom from the end of the carbon chain. The three types of omega-3 fatty acids involved in human physiology are ?-linolenic acid (ALA) (found in plant oils), eic…

Kategori:
Alimentary Tract and MetabolismBile and Liver TherapyDietary Fats +12
Target Protein:
Peroxisome proliferator-activated receptor gammaPeroxisome proliferator-activated receptor alphaSterol regulatory element-binding protein 1
Waktu ParuhApproximate half-li…
Vol. DistribusiVd of EPA is aproxi…
KlirensClearance of EPA is…
Genetik -
Omega-3-acid ethyl esters Approved DB09539
small molecule | CAS: 308081-97-2

Omega-3-acid ethyl esters are prescription drugs that contain eicosapentaenoic acid-ethyl ester (EPA) and docosahexaenoic acid-ethyl ester (DHA) that are used in combination with changes in diet to lower triglyceride levels in adults with severe (? 500 mg/dL)…

Kategori:
AutacoidsBiological FactorsDiet, Food, and Nutrition +15
Target Protein:
Sterol regulatory element-binding protein 1
Waktu Paruh79 hours ± 47 hours…
Vol. Distribusi82 ± 56L[A18890]
Klirens757 mL/h ± 283mL/h[…
Genetik -
Omega-3-carboxylic acids Approved DB09568
small molecule

The omega-3 carboxylic acid (OM3-CA) is a new formulation of omega-3 fatty acids that present an enhanced bioavailability in the treatment of dyslipidemia. The increased bioavailability is explained because OM3-CA is found in a form of polyunsaturated free f…

Kategori:
Fatty Acids, Omega-3
Target Protein:
Diacylglycerol O-acyltransferase 23-hydroxyacyl-CoA dehydrogenase type-2Enoyl-CoA hydratase, mitochondrial +3
Waktu ParuhThe half-life of OM…
Vol. DistribusiThis pharmacokineti…
KlirensThe registered clea…
Genetik -
small molecule

Omega-6 fatty acids are polyunsaturated fatty acids with a final carbon-carbon double bond in the n-6 position, that is, the sixth bond, counting from the methyl end. They are a family of fatty acid molecules that act as precursors to potent lipid mediator si…

Kategori:
Fatty AcidsFatty Acids, UnsaturatedLipids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Omeprazole Approved DB00338
small molecule | CAS: 73590-58-6

Originally approved by the FDA in 1989, omeprazole is a _proton-pump inhibitor_, used to treat gastric acid-related disorders. These disorders may include gastroesophageal reflux disease (GERD), peptic ulcer disease, and other diseases characterized by the ov…

Kategori:
2-PyridinylmethylsulfinylbenzimidazolesAcid ReducersAlimentary Tract and Metabolism +37
Target Protein:
Potassium-transporting ATPase alpha chain 1Potassium-transporting ATPase subunit betaAryl hydrocarbon receptor
Gen Terkait:
CYP2C19 CYP2C19
Waktu Paruh0.5-1 hour (healthy…
Vol. DistribusiApproximately 0.3 L…
KlirensHealthy subject (de…
Genetik 2 Varian
biotech | CAS: 2249927-58-8

Omfiloctocog alfa is under investigation in clinical trial NCT03947567 (Safety and Efficacy of Long-term Treatment With SCT800 in Previously Treated Hemophilia a Patients.).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Omidenepag isopropyl Approved DB15071
small molecule | CAS: 1187451-19-9

Omidenepag isopropyl is a topical ocular hypotensive agent used to reduce intraocular pressure (IOP) in patients with glaucoma and ocular hypertension.[L43503] Omidenepag isopropyl is quickly metabolized to its active metabolite, omidenepag, a molecule with h…

Kategori:
Antiglaucoma AgentsHypotensive AgentsOphthalmic Solutions +6
Target Protein:
Prostaglandin E2 receptor EP2 subtypeProstaglandin E2 receptor EP1 subtype
Waktu ParuhThe half-life of om…
Vol. DistribusiNot available.
KlirensNot available.
Genetik -
Omidubicel Approved DB17132
biotech

Omidubicel is a nicotinamide-modified allogeneic hematopoietic progenitor cell therapy derived from cord blood used as an allogeneic stem cell donor source. Umbilical blood cord cells are expanded _ex-vivo_ and [nicotinamide] (a form of vitamin B3) is used as…

Kategori:
Allogeneic Cord Blood Hematopoietic Progenitor Cell TherapyCells, AllogeneicCells, Cultured, Allogeneic +1
Waktu ParuhThere is limited ph…
Vol. DistribusiThere is limited ph…
KlirensThere is limited ph…
Genetik -
Omiganan DB06610
small molecule | CAS: 204248-78-2

Omiganan has been investigated for the treatment of Mupirocin-resistant MRSA skin infections.

Kategori:
Amino Acids, Peptides, and ProteinsAntimicrobial PeptidesMembrane Proteins +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Omigapil DB12879
small molecule | CAS: 181296-84-4

Omigapil has been used in trials studying the treatment of Congenital Muscular Dystrophy.

Kategori:
EthersEthers, Cyclic
Target Protein:
Glyceraldehyde-3-phosphate dehydrogenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Omilancor DB19277
small molecule | CAS: 1912399-75-7

Deskripsi belum tersedia.

Target Protein:
LanC-like protein 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Omipalisib DB12703
small molecule | CAS: 1086062-66-9

Omipalisib has been used in trials studying the treatment of CANCER, Solid Tumours, and Idiopathic Pulmonary Fibrosis.

Kategori:
AmidesBenzene DerivativesHeterocyclic Compounds, Fused-Ring +4
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Omoconazole DB13684
small molecule | CAS: 74512-12-2

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAntifungal AgentsAntifungals for Dermatological Use +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ompenaclid DB18819
small molecule | CAS: 353-09-3

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAmidinesFatty Acids +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OMS-103HP DB05303
small molecule

OMS103HP is the first drug being developed to improve joint function following arthroscopic surgery, one of the most common procedures performed today by orthopedic surgeons.

Kategori:
Acids, CarbocyclicBenzocycloheptenesDibenzocycloheptenes +3
Target Protein:
Tumor necrosis factorInterleukin-1 receptor type 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OMS-824 DB17874
small molecule | CAS: 1207549-69-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OMS906 DB17722
biotech

OMS906 is a humanized Igg4 monoclonal antibody against mannan-binding lectin-associated serine protease-3 (MASP-3) currently being developed by Omeros.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Onalespib DB06306
small molecule | CAS: 912999-49-6

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +3
Target Protein:
Heat shock protein HSP 90-alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Onamelatucel-L DB17330
biotech

Deskripsi belum tersedia.

Kategori:
Biological ProductsComplex MixturesMelanoma +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Onapristone DB12637
small molecule | CAS: 96346-61-1

Onapristone has been used in trials studying the treatment of Prostate Cancer, Recurrent Prostate Cancer, Metastatic Prostate Cancer, Androgen-independent Prostate Cancer, and Progesterone Receptor Positive Tumor: Max 1 Line of Prior Chemotherapy, no Prior Ho…

Kategori:
Antineoplastic AgentsFertility AgentsFertility Agents, Female +5
Target Protein:
Progesterone receptorGlucocorticoid receptorAdhesion G-protein coupled receptor D1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Onartuzumab DB11746
biotech | CAS: 1133766-06-9

Onartuzumab has been used in trials studying the treatment of Neoplasms, Lung Cancer, Glioblastoma, Gastric Cancer, and Colorectal Cancer, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Onasemnogene abeparvovec Approved DB15528
biotech | CAS: 1922968-73-7

Onasemnogene abeparvovec is an adeno-associated virus vector-based gene therapy that has been approved by the FDA in May 2019 for the treatment of infant patients (less than 2 years of age) with spinal muscular atrophy (SMA) and a specific mutation in the sur…

Kategori:
Adeno-associated Viral Vector TherapiesAmino Acids, Peptides, and ProteinsBiological Products +7
Waktu ParuhThere is limited ph…
Vol. DistribusiThere is limited ph…
KlirensThere is limited ph…
Genetik -
Onatasertib DB12570
small molecule | CAS: 1228013-30-6

Onatasertib (CC-223) has been used in trials studying the treatment and basic science of Multiple Myeloma, Glioblastoma Multiforme, HepatoCellular Carcinoma, Non-small Cell Lung Cancer, and Diffuse Large B-Cell Lymphoma, among others.

Target Protein:
Serine/threonine-protein kinase mTOR
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ONCOS-102 DB17274
biotech | CAS: 1802359-98-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ONCOS?102 DB17173
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ondansetron Approved DB00904
small molecule | CAS: 99614-02-5

A competitive serotonin type 3 receptor antagonist. It is effective in the treatment of nausea and vomiting caused by cytotoxic chemotherapy drugs, including cisplatin, and has reported anxiolytic and neuroleptic properties. Having been developed in the 19…

Kategori:
Anti-Anxiety AgentsAntidepressive AgentsAntiemetic Serotonin 5-HT3 Receptor Antagonists +29
Target Protein:
5-hydroxytryptamine receptor 3A5-hydroxytryptamine receptor 4Mu-type opioid receptor +2
Gen Terkait:
CYP2D6 CYP2D6
Waktu ParuhThe half-life of on…
Vol. DistribusiThe volume of distr…
KlirensThe clearance value…
Genetik 2 Varian
Ondelopran DB12585
small molecule | CAS: 676501-25-0

Ondelopran has been used in trials studying the treatment of Alcohol Dependence.

Kategori:
AminesBenzene DerivativesBenzyl Compounds +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Onercept DB06495
biotech | CAS: 199685-57-9

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsMembrane ProteinsPolyethylene Glycols +3
Target Protein:
Tumor necrosis factor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Onfekafusp alfa DB16269
biotech | CAS: 1957239-88-1

Onfekafusp alfa is under investigation in clinical trial NCT02938299 (Neoadjuvant L19IL2/L19TNF- Pivotal Study).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ongericimab DB18949
biotech | CAS: 2145096-91-7

Ongericimab is under investigation in clinical trial NCT05325203 (A Study to Evaluate the Efficacy and Safety of JS002 in Patients With Heterozygous Familial Hypercholesterolemia (Hefh).).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ONL-1204 DB18239
biotech | CAS: 2040964-58-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and Proteins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ONO-2952 DB14802
small molecule | CAS: 895169-20-7

ONO-2952 is under investigation in clinical trial NCT01887002 (Study to Evaluate the Effects of ONO-2952 on Pain Perception Produced by Rectal Distention in Female Subjects With Diarrhea-Predominant Irritable Bowel Syndrome (IBS-D)).

Kategori:
CycloparaffinsHeterocyclic Compounds, Fused-Ring
Target Protein:
Translocator protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ONO-5334 DB19206
small molecule | CAS: 620614-15-5

ONO-5334 is under investigation in clinical trial NCT00532337 (Controlled Study of ONO-5334 in Postmenopausal Women With Osteopenia or Osteoporosis).

Kategori:
Osteoporosis, Postmenopausal, drug therapySulfur CompoundsThiazoles
Target Protein:
Cathepsin K
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ONO-7579 DB17236
small molecule | CAS: 1622212-25-2

Deskripsi belum tersedia.

Kategori:
Enzyme InhibitorsProtein Kinase Inhibitors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ONO-8539 DB15325
small molecule | CAS: 459842-29-6

ONO-8539 is under investigation in clinical trial NCT01707901 (A Study of the Effect of ONO-8539 on Oesophageal Pain Hypersensitivity in Patients With Non-erosive Reflux Disease).

Kategori:
Acids, CarbocyclicBenzene DerivativesReceptors, Prostaglandin E, EP1 Subtype, antagonists & inhibitors +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ONT-093 DB14069
small molecule | CAS: 216227-54-2

ONT-093 is an orally bioavailable inhibitor of P-glycoprotein (P-gp). In pre-clinical studies, ONT-093 could inhibit P-gp and reverse multidrug resistance at nM concentrations with no effect on paclitaxel pharmacokinetics.

Kategori:
Drug Resistance, MultipleP-glycoprotein inhibitors
Target Protein:
ATP-dependent translocase ABCB1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ontamalimab DB15298
biotech | CAS: 2098790-40-8

Ontamalimab is under investigation in clinical trial NCT03627091 (Efficacy and Safety Study of SHP647 as Maintenance Treatment in Participants With Moderate to Severe Crohn's Disease (CARMEN CD 307)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Onternabez DB18076
small molecule | CAS: 256934-39-1

Deskripsi belum tersedia.

Kategori:
Cannabinoid Receptor AgonistsCannabinoids and similarsHormones +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ontorpacept DB17116
biotech | CAS: 2131089-46-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ontuxizumab DB16270
biotech | CAS: 946415-62-9

Ontuxizumab is a humanized monoclonal antibody that targets endosialin or tumour endothelial marker 1 (TEM-1). It is under investigation in clinical trial NCT01574716 (Sarcoma Study of Morab-004 Utilization: Research and Clinical Evaluation).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 11601–11650 dari 16004
Sebelumnya Halaman 233 / 321 Berikutnya