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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
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11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 231 / 236
Vosaroxin DB11999
small molecule | CAS: 175414-77-4

Vosaroxin is under investigation for the treatment of Leukemia, Myeloid, Acute.

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsHeterocyclic Compounds, Fused-Ring +1
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-beta
Waktu Paruh-
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Vosoritide Approved DB11928
biotech | CAS: 1480724-61-5

Achondroplasia is an autosomal dominant genetic disease and the most common cause of dwarfism in humans.[A242277] It results from a gain-of-function missense mutation in _FGFR3_ that results in a dramatic suppression of bone growth, both in volume and in leng…

Kategori:
Amino Acids, Peptides, and ProteinsC-type Natriuretic Peptide AnalogDrugs Affecting Bone Structure and Mineralization +7
Target Protein:
Atrial natriuretic peptide receptor 2
Waktu ParuhThe mean half-life …
Vol. DistribusiThe mean apparent v…
KlirensThe mean apparent c…
Genetik -
Voxelotor Approved DB14975
small molecule | CAS: 1446321-46-5

Voxelotor is a novel hemoglobin S polymerization inhibitor for the treatment of sickle cell disease. This is a genetically inherited condition most prevalent in the Middle East, Africa, and certain parts of India. Sickle cell disease can lead to excruciating …

Kategori:
AldehydesBlood and Blood Forming OrgansCytochrome P-450 CYP2B6 Substrates +7
Target Protein:
Hemoglobin subunit alpha
Waktu ParuhThe plasma eliminat…
Vol. DistribusiThe apparent volume…
KlirensThe apparent oral c…
Genetik -
Voxilaprevir Approved DB12026
small molecule | CAS: 1535212-07-7

Voxilaprevir is a Direct-Acting Antiviral (DAA) medication used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV). HCV is a single-stranded RNA virus that is categorized i…

Kategori:
Acids, AcyclicAmidesAmino Acids +36
Target Protein:
Genome polyproteinGenome polyprotein
Waktu Paruh33 hr [FDA Label]
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Voxtalisib DB12400
small molecule | CAS: 934493-76-2

Voxtalisib has been used in trials studying the treatment of Cancer, Melanoma, Lymphoma, Glioblastoma, and Breast Cancer, among others.

Kategori:
AmidesHeterocyclic Compounds, Fused-RingPhosphatidylinositol 3-Kinases, antagonists & inhibitors +2
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoformSerine/threonine-protein kinase mTOR
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VP-14637 DB12195
small molecule | CAS: 235106-62-4

MDT-637 has been investigated for the treatment of Drug Safety.

Kategori:
Benzene DerivativesHydrazines
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VPO-227 DB18004
small molecule | CAS: 1314873-02-3

Deskripsi belum tersedia.

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VS-4718 DB15273
small molecule | CAS: 1061353-68-1

VS-4718 is under investigation in clinical trial NCT02215629 (Dose Escalation Study in Acute Myeloid or B-Cell Acute Lymphoblastic Leukemia).

Kategori:
AminesFocal Adhesion Protein-Tyrosine Kinases, antagonists & inhibitorsPyridines
Target Protein:
Focal adhesion kinase 1
Waktu Paruh-
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VS-5584 DB12986
small molecule | CAS: 1246560-33-7

VS-5584 has been used in trials studying the treatment of Lymphoma, Metastatic Cancer, and Non Hematologic Cancers.

Kategori:
Heterocyclic Compounds, Fused-RingOxazines
Target Protein:
Target of rapamycin complex 2 subunit MAPKAP1Serine/threonine-protein kinase mTORPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
Waktu Paruh-
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VSF-173 DB05753
small molecule

VSF-173 is an oral small molecule. It is an oral compound that has demonstrated effects on animal sleep/wake patterns and gene expression patterns suggestive of a stimulant effect. It is developed for the treatment of excessive sleepiness. Study shows that VS…

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VT-1598 DB17757
small molecule | CAS: 2089320-99-8

Deskripsi belum tersedia.

Target Protein:
Lanosterol 14-alpha demethylase
Waktu Paruh-
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VTP-194204 DB11806
small molecule | CAS: 220619-73-8

Nrx194204 has been used in trials studying the treatment of Parkinson's Disease and Non-small Cell Lung Cancer.

Kategori:
Fatty AcidsLigandsLipids +1
Target Protein:
Retinoic acid receptor RXR-gamma
Waktu Paruh-
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VTP-201227 DB05652
small molecule

VTP-201227 has a novel mechanism of action and is being developed as a topical agent for the treatment of psoriasis with potential extensions into other dermatological indications. It is being developed by Vitae Pharmaceuticals.

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VTP-27999 DB12416
small molecule | CAS: 942142-51-0

VTP-27999 has been used in trials studying the basic science of Renal Function.

Kategori:
Acids, AcyclicAgents Acting on the Renin-Angiotensin SystemRenin Inhibitors
Target Protein:
Renin
Waktu Paruh-
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VTX-801 DB17646
biotech

VTX-801 is a replication-deficient recombinant adeno-associated viral vector (rAAV) consisting of an AAV liver tropic capsid containing a single-stranded DNA genome carrying a shortened version of the ATP7B gene (ATP7B-minigene). It is being investigated in W…

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VTX-803 DB18271
biotech

Deskripsi belum tersedia.

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Vudalimab DB18833
biotech | CAS: 2329669-72-7

Vudalimab is under investigation in clinical trial NCT05005728 (Xmab®20717 (Vudalimab) Alone or in Combination With Chemotherapy or Targeted Therapy in Patients With Metastatic Castration-resistant Prostate Cancer).

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Vunakizumab DB15154
biotech | CAS: 1792181-33-9

Vunakizumab is under investigation in clinical trial NCT03463187 (Multi-Dose Study of SHR-1314 in Subjects With Moderate-to-severe Plaque Psoriasis).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
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Vutiglabridin DB18781
small molecule | CAS: 1800188-47-9

Deskripsi belum tersedia.

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Vutrisiran Approved DB16699
biotech | CAS: 1867157-35-4

Vutrisiran is a double-stranded small interfering ribonucleic acid (siRNA) that targets wild-type and mutant transthyretin (TTR) messenger RNA (mRNA).[L42065] This siRNA therapeutic is indicated for the treatment of neuropathies associated with hereditary tra…

Kategori:
Antisense OligonucleotidesNervous SystemNucleic Acids, Nucleotides, and Nucleosides +4
Target Protein:
Transthyretin mRNA
Waktu ParuhThe median half-lif…
Vol. DistribusiBased on a populati…
KlirensThe apparent cleara…
Genetik -
VX-702 DB05470
small molecule | CAS: 745833-23-2

VX-702 is a small molecule investigational oral anti-cytokine therapy for treatment of inflammatory diseases, specifically rheumatoid arthritis (RA). It acts as a p38 MAP kinase inhibitor. In the future, VX-702 may be investigated for combination with methotr…

Kategori:
AmidesBenzene Derivatives
Target Protein:
Mitogen-activated protein kinase 14Tumor necrosis factorInterleukin-1 beta +1
Waktu Paruh-
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VX-765 DB05507
small molecule

VX-765 is the orally available prodrug of a potent and selective competitive inhibitor of ICE/caspase-1 (VRT-043198). VX-765 is currently under clinical development for the treatment of inflammatory and autoimmune conditions, as it blocks the hypersensitive r…

Kategori:
Acids, CarbocyclicAmino Acids, Peptides, and ProteinsAminobenzoates +4
Target Protein:
Caspase-1Interleukin-1 beta
Waktu Paruh-
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VXM01 DB17420
biotech

Deskripsi belum tersedia.

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biotech

Fecal microbiota transplantation (FMT) is effective in enhancing the gut microbiota of patients experiencing a high range of disease states, including Clostridioides difficile (C. diff) infection, Crohn’s disease, and ulcerative colitis. Washed microbiota pre…

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Water Approved DB09145
small molecule | CAS: 7732-18-5

Water (chemical formula: H2O) is a transparent fluid which forms the world's streams, lakes, oceans and rain, and is the major constituent of the fluids of organisms. As a chemical compound, a water molecule contains one oxygen and two hydrogen atoms that are…

Kategori:
DiluentsEENT Drugs, MiscellaneousIrrigating Solutions +2
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Watermelon Approved DB10578
biotech

Watermelon allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
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WAY-151693 DB02071
small molecule

Deskripsi belum tersedia.

Kategori:
AmidesAminesHydroxy Acids +3
Target Protein:
Collagenase 3
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Genetik -
biotech

Deskripsi belum tersedia.

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Wheat Approved DB10579
biotech

Wheat allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
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Wheat germ oil DB16570
biotech | CAS: 313258-61-6

Deskripsi belum tersedia.

Kategori:
Biological ProductsComplex MixturesLipids +4
Waktu Paruh-
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White fish Approved DB10627
biotech

White fish allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
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Genetik -
White pepper Approved DB10679
biotech

White pepper allergenic extract is used in allergenic testing.

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WIN-54954 DB08723
small molecule | CAS: 107355-45-3

WIN-54954 is a broad-spectrum antipicornavirus drug.

Target Protein:
Genome polyproteinGenome polyprotein
Waktu Paruh-
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WL-1002 DB05346
small molecule

WL-1002 is developed by Winston Laboratories which is a topical cream formulation of 075% zucapaicin (also known as civamide), for the treatment of pain due to osteoarthritis.

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WNT-974 DB12561
small molecule | CAS: 1243244-14-5

WNT974 has been used in trials studying the treatment of Metastatic Colorectal Cancer and Squamous Cell Carcinoma, Head And Neck.

Kategori:
Enzyme Inhibitors
Target Protein:
Protein-serine O-palmitoleoyltransferase porcupine
Waktu Paruh-
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Wood creosote DB13271
small molecule | CAS: 8021-39-4

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesCough and Cold PreparationsCresols +2
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Wortmannin DB08059
small molecule | CAS: 19545-26-7

Wortmannin is a steroid metabolite of _Penicillium funiculosum_ and _Talaromyces wortmannii_ fungi. This drug acts as a nonspecific, covalent inhibitor of phosphoinositide 3-kinase enzymes (PI3Ks).

Kategori:
AndrostadienesAndrostanesAndrostenes +16
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoformPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoformSerine/threonine-protein kinase PLK1 +2
Waktu Paruh-
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WP-1066 DB12679
small molecule | CAS: 857064-38-1

WP1066 has been used in trials studying the treatment of Melanoma, Brain Cancer, Solid Tumors, and Central Nervous System Neoplasms.

Kategori:
Benzene DerivativesBenzylidene CompoundsHeterocyclic Compounds, Fused-Ring +2
Target Protein:
Signal transducer and activator of transcription 3
Waktu Paruh-
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WP-1122 DB17192
small molecule

WP-1122 is a prodrug of 2-deoxy-D-glucose (2-DG). It was granted FDA orphan designation for the treatment of glioblastoma multiforme.[L47361]

Kategori:
CarbohydratesDeoxy Sugars
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WP-1301 DB17702
biotech | CAS: 1609460-62-9

WP1301 is a synthetic peptide derived from hFVIII. It binds to an MHC class II molecule and is recognized by a Factor VIII-specific T cell.[L46138]

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WRR-99 DB03573
small molecule

Deskripsi belum tersedia.

Target Protein:
Cathepsin FCruzipain
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WSD-0922 DB17170
small molecule | CAS: 2226552-64-1

Deskripsi belum tersedia.

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WT-1 122 long DB17353
biotech | CAS: 952720-86-4

Deskripsi belum tersedia.

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WT-1 331 long DB17355
biotech | CAS: 935395-34-9

Deskripsi belum tersedia.

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WT-1 427 long DB17354
biotech | CAS: 935395-33-8

Deskripsi belum tersedia.

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WT-1 A1 DB17352
small molecule | CAS: 852243-39-1

Deskripsi belum tersedia.

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WTx-Bortezomib DB17389
biotech

Deskripsi belum tersedia.

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WU-CART-007 DB18617
biotech

WU-CART-007 consists of allogeneic, fratricide-resistant genetically modified T cells transduced with a 2nd generation 4-1BB-CD3z chimeric antigen receptor targeting human CD7.

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WVE-003 DB17870
biotech

WVE-003 is an allele-selective antisense oligonucleotide that works to selectively reduce the toxic mutant huntingtin (mHTT) protein.[L46787]

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WVE-N531 DB17848
biotech

Deskripsi belum tersedia.

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