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13591

Total database: 17430
Struktur (SMILES)
10177 (74.9%)
Target
7625 (56.1%)
Genomik
104 (0.8%)
Referensi
13591 (100.0%)

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Hasil Pencarian (13591)

Halaman 231 / 272
small molecule | CAS: 1039726-31-2

Deskripsi belum tersedia.

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small molecule | CAS: 1638746-88-9

Deskripsi belum tersedia.

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Satralizumab Approved DB15762
biotech | CAS: 1535963-91-7

Satralizumab is a recombinant humanized monoclonal antibody targeted against human interleukin-6 (IL-6) receptors, similar to [tocilizumab], which is produced in Chinese hamster ovary cells and based on an IgG2 framework.[L15536] Satralizumab is used in the t…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +11
Target Protein:
Interleukin-6 receptor subunit alpha
Waktu ParuhThe terminal half-l…
Vol. DistribusiSatralizumab is sub…
KlirensThe total clearance…
Genetik -
Satraplatin DB04996
small molecule | CAS: 129580-63-8

Satraplatin is a platinum compound that is currently under investigation as one treatment of patients with advanced prostate cancer who have failed previous chemotherapy. As an investigation drug, it has not yet received U.S. Food and Drug Administration (FDA…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsOrganometallic Compounds +1
Target Protein:
DNA
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Savolitinib DB12048
small molecule | CAS: 1313725-88-0

Savolitinib has been used in trials studying the treatment and health services research of Tumor, Food Effect, Gastric Cancer, Health Subjects, and Colorectal Cancer, among others.

Kategori:
Tyrosine Kinase Inhibitors
Target Protein:
Hepatocyte growth factor receptor
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Saw palmetto Approved DB14360
biotech

Saw palmetto is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
AngiospermsArecaceaeBiological Products +12
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Saxagliptin Approved DB06335
small molecule | CAS: 361442-04-8

Saxagliptin (rINN) is an orally active hypoglycemic (anti-diabetic drug) of the new dipeptidyl peptidase-4 (DPP-4) inhibitor class of drugs. FDA approved on July 31, 2009.

Kategori:
Agents causing angioedemaAlimentary Tract and MetabolismAmino Acids, Peptides, and Proteins +20
Target Protein:
Dipeptidyl peptidase 4
Waktu ParuhSaxagliptin = 2.5 h…
Vol. Distribusi151 L
KlirensRenal clearance, si…
Genetik -
SB 11285 DB17511
small molecule

SB 11285 is a second-generation Stimulator of Interferon Genes (STING) agonist.[L45123] SB 11285 is under investigation in clinical trial NCT04096638 (Evaluating Safety and Efficacy of SB 11285 Alone and in Combination With Atezolizumab in Patients With Advan…

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SB 224289 DB17052
small molecule | CAS: 180083-23-2

SB-224289 is a small molecule with a high affinity for human 5-HT1B receptors.[A253122]

Kategori:
Piperidines
Target Protein:
5-hydroxytryptamine receptor 1B
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SB-1578 DB15294
small molecule | CAS: 937273-04-6

SB-1578 is under investigation in clinical trial NCT01235871 (A Single and Multiple-Dose Study of SB1578).

Kategori:
fms-Like Tyrosine Kinase 3, antagonists & inhibitorsHeterocyclic Compounds, Fused-RingJanus Kinase 2, antagonists & inhibitors +1
Target Protein:
Tyrosine-protein kinase JAK2
Waktu Paruh-
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SB-218078 DB17051
small molecule | CAS: 135897-06-2

SB-218078 is a specific inhibitor of CHK1.[A253117]

Target Protein:
Serine/threonine-protein kinase Chk1
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SB-249553 DB05285
small molecule

SB-249553 is a vaccine that has MAGE-3 cancer antigen and the Adjuvant SBAS-2. It is also under by GlaxoSmithKline to treat melanoma and lung cancer.

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SB-269970 DB13988
small molecule | CAS: 201038-74-6

SB-269970 is an experimental drug developed by GlaxoSmithKline. In the studies performed with this agent, it has been suggested that SB-269970 acts either as a selective antagonist or inverse agonist of the serotonin receptor 7 (5-HT7).[A31816,A31817]

Kategori:
AmidesBenzene DerivativesSulfones +1
Target Protein:
5-hydroxytryptamine receptor 7
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SB-409513 DB01793
small molecule

Deskripsi belum tersedia.

Target Protein:
Glycogen synthase kinase-3 beta
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SB-559448 DB05930
small molecule

SB-559448 is a small-molecule drug that mimics the activity of thrombopoietin (TPO), a protein factor that promotes growth and production of blood platelets. This drug is developed by GlaxoSmithKline and used to treat Thrombocytopenia.Thrombocytopenia (decrea…

Target Protein:
Thrombopoietin receptor
Waktu Paruh-
Vol. Distribusi-
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SB-649868 DB14822
small molecule | CAS: 380899-24-1

SB-649868 is under investigation in clinical trial NCT01030939 (Study to Investigate Safety, Tolerability, Pharmacokinetics and Cardiac Function After Repeat Doses of SB-649868 in Healthy-volunteers).

Kategori:
Carbon RadioisotopesHeterocyclic Compounds, Fused-RingSulfur Compounds
Target Protein:
Orexin/Hypocretin receptor type 1
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SB-705498 DB11883
small molecule | CAS: 501951-42-4

SB-705498 has been investigated for the treatment of Rhinitis, Chronic Cough, and Non-allergic Rhinitis.

Kategori:
AmidesTRPV Cation Channels, antagonists & inhibitors
Target Protein:
Transient receptor potential cation channel subfamily V member 1
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SB-743921 DB05546
small molecule | CAS: 618430-39-0

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +4
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SB-773812 DB16042
small molecule | CAS: 630407-66-8

SB-773812 is under investigation in clinical trial NCT00259870 (SB-773812 Administered in Adults With Schizophrenia).

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SB220025 DB04338
small molecule

Deskripsi belum tersedia.

Kategori:
Calcium-Calmodulin-Dependent Protein Kinases, antagonists & inhibitors
Target Protein:
Mitogen-activated protein kinase 14Mitogen-activated protein kinase 1
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SB719125 DB16753
biotech

Deskripsi belum tersedia.

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SBT-100 DB17215
biotech

SBT-100 is an anti-signal transducer and activator of transcription 3 (STAT3) B VHH13 single-domain antibody (sdAb). It was granted orphan drug designation by the FDA for the treatment of pancreatic cancer and osteosarcoma.[L44131,L44136]

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SBT-272 DB18037
small molecule | CAS: 2356106-71-1

Deskripsi belum tersedia.

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SBT101 DB18139
biotech

SBT101 is a non-replicating recombinant adeno-associated virus serotype 9 (AAV9) gene therapy vector containing the human adenosine triphosphate (ATP)-binding cassette (ABC) sub-family D member 1 (ABCD1) gene.

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SC 41930 DB17101
small molecule | CAS: 120072-59-5

Deskripsi belum tersedia.

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAnti-Inflammatory Agents +9
Target Protein:
Leukotriene B4 receptor 1Leukotriene B4 receptor 2
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SC-236 DB14059
small molecule | CAS: 170569-86-5

SC-236 is a potent, selective, orally active inhibitor of cyclooxygenase-2 (COX-2) [L2964] that has been studied in cancer therapy [A33375], lower back pain [A33376], and inflammation [A33373], [A33374],[L2962], [A33377].

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAmides +14
Target Protein:
Cyclooxygenase 2Prostaglandin G/H synthase 2Nuclear factor NF-kappa-B complex
Waktu ParuhLong plasma half-li…
Vol. Distribusi-
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SC-74020 DB01630
small molecule

Deskripsi belum tersedia.

Kategori:
AmidesAminesHydroxy Acids +3
Target Protein:
72 kDa type IV collagenase
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Scallop Approved DB10623
biotech

Scallop allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
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Scarlet red Approved DB19136
small molecule | CAS: 85-83-6

Scarlet red is under investigation in clinical trial NCT00591916 (New Treatment for Donor Sites).

Kategori:
Coloring AgentsCompounds used in a research, industrial, or household setting
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SCH-58500 DB17416
biotech

SCH-58500 is a recombinant replication-deficient adenovirus vector carrying the human p53 gene.

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SCH-900271 DB12433
small molecule | CAS: 915210-50-3

Sch 900271 has been used in trials studying the treatment of Mixed Hyperlipidemia and Primary Hypercholesterolemia.

Target Protein:
Hydroxycarboxylic acid receptor 2
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Schinus molle pollen Approved DB10483
biotech

Schinus molle pollen is the pollen of the Schinus molle plant. Schinus molle pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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biotech

Schisandra chinensis fruit is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

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SCIB1 DB18439
biotech

SCIB1 is an investigational cancer vaccine being developed by Scancell Ltd. It is being investigated for the treatment of melanoma. It consists of plasmid DNA molecules that express a modified antibody in human cells, working to stimulate the patient's T cell…

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Scopolamine Approved DB00747
small molecule | CAS: 51-34-3

Scopolamine is a tropane alkaloid isolated from members of the _Solanaceae_ family of plants, similar to [atropine] and [hyoscyamine], all of which structurally mimic the natural neurotransmitter [acetylcholine].[A228423, A228763] Scopolamine was first synthe…

Kategori:
AdjuvantsAdjuvants, AnesthesiaAgents producing tachycardia +30
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M3 +5
Waktu ParuhThe half-life of sc…
Vol. DistribusiThe volume of distr…
KlirensIV infusion of 0.5 …
Genetik -
biotech

Centruroides (scorpion) Immune F(ab')2 (equine) is a purified preparation of immune globulin F(ab’)2 fragments that are derived from plasma of the horses immunized with venom of *C. noxius*, *C. l. limpidus*, *C. l. tecomanus*, and *C. s. suffusus*. It is int…

Kategori:
AntiveninsPassively Acquired ImmunityVenom Neutralization
Waktu Paruh159 ± 57 h [FDA lab…
Vol. DistribusiSteady state: 13.6 …
Klirens83.5 ± 38.4 ml/Hr […
Genetik -
Scriptaid DB17053
small molecule | CAS: 287383-59-9

Scriptaid is a histone deacetylase (HDAC) inhibitor researched for its anti-tumor properties.[A253127]

Kategori:
AminesAntineoplastic AgentsEnzyme Inhibitors +2
Target Protein:
Histone deacetylase 1
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biotech

Scutellaria baicalensis root is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
AngiospermsBiological ProductsComplex Mixtures +10
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Scutellaria lateriflora Approved DB14339
biotech

Scutellaria lateriflora is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

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SCY-635 DB12451
small molecule | CAS: 210759-10-7

SCY-635 has been investigated for the treatment of Chronic Hepatitis C and Hepatitis C Infection.

Kategori:
Amino Acids, Peptides, and ProteinsPeptidesPeptides, Cyclic
Target Protein:
Guided entry of tail-anchored proteins factor CAMLG
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scyllo-inositol DB03106
small molecule | CAS: 488-59-5

An isomer of glucose that has traditionally been considered to be a B vitamin although it has an uncertain status as a vitamin and a deficiency syndrome has not been identified in man. (From Martindale, The Extra Pharmacopoeia, 30th ed, p1379) Inositol phosph…

Kategori:
AlcoholsCarbohydratesStereoisomerism +1
Target Protein:
Lysosomal acid glucosylceramidase1-phosphatidylinositol phosphodiesteraseCDP-diacylglycerol--inositol 3-phosphatidyltransferase +1
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SD-0006 DB07943
small molecule | CAS: 271576-80-8

Deskripsi belum tersedia.

Target Protein:
Mitogen-activated protein kinase 14
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Vol. Distribusi-
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SD146 DB02729
small molecule | CAS: 183854-21-9

Deskripsi belum tersedia.

Target Protein:
Gag-Pol polyprotein
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Vol. Distribusi-
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Sea scallop Approved DB15538
biotech

Sea scallop allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
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SEA-BCMA DB18309
biotech | CAS: 2115084-53-0

Deskripsi belum tersedia.

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Sebelipase alfa Approved DB11563
biotech | CAS: 1276027-63-4

The lysosomal acid lipase (LAL) enzyme is found in lysosomes and is primarily responsible for the metabolism of lipids, and its absence or deficiency results in the accumulation of lipids in various organs. This lipid accumulation can lead to end-organ damage…

Kategori:
Alimentary Tract and MetabolismCarboxylic Ester HydrolasesCholesterol Ester Storage Disease, drug therapy +7
Waktu ParuhThe mean half-life …
Vol. DistribusiIn patients 4-11 ye…
KlirensAcross all age grou…
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Sebetralstat DB18305
small molecule | CAS: 1933514-13-6

Deskripsi belum tersedia.

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Secalciferol DB18406
small molecule | CAS: 55721-11-4

Deskripsi belum tersedia.

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Seclidemstat DB17117
small molecule | CAS: 1423715-37-0

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +1
Target Protein:
Lysine-specific histone demethylase 1A
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Secnidazole Approved DB12834
small molecule | CAS: 3366-95-8

Secnidazole is a second-generation 5-nitroimidazole antimicrobial agent. It is structurally related to other 5-nitroimidazoles, including [DB00916] and [DB00911], but displays improved oral absorption and a longer terminal elimination half-life than other dru…

Kategori:
Anti-Infective AgentsAntibacterials for Systemic UseAntiinfectives for Systemic Use +18
Waktu ParuhThe plasma eliminat…
Vol. DistribusiThe apparent volume…
KlirensThe total body clea…
Genetik -
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