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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 230 / 236
Vitamin A Approved DB00162
small molecule | CAS: 68-26-8

Retinol and derivatives of retinol that play an essential role in metabolic functioning of the retina, the growth of and differentiation of epithelial tissue, the growth of bone, reproduction, and the immune response. Dietary vitamin A is derived from a varie…

Kategori:
Adjuvants, ImmunologicAlimentary Tract and MetabolismAlkenes +33
Target Protein:
Retinoic acid receptor RXR-gammaApolipoprotein DProstaglandin-H2 D-isomerase +13
Waktu Paruh1.9 hours
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 15713-12-9

Deskripsi belum tersedia.

Target Protein:
5-methyltetrahydrofolate--homocysteine S-methyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vitamin E Approved DB00163
small molecule | CAS: 59-02-9

In 1922, vitamin E was demonstrated to be an essential nutrient[A32448]. Vitamin E is a term used to describe 8 different fat soluble tocopherols and tocotrienols, alpha-tocopherol being the most biologically active[A176104]. Vitamin E acts as an antioxidant,…

Kategori:
AntioxidantsBasic Ointments and ProtectantsBenzopyrans +23
Target Protein:
SEC14-like protein 4SEC14-like protein 3SEC14-like protein 2 +7
Waktu Paruh44 hours in prematu…
Vol. Distribusi0.41L/kg in prematu…
Klirens6.5mL/hr/kg in prem…
Genetik -
Vitamin K7 DB15664
small molecule | CAS: 83-69-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vitespen DB06400
biotech | CAS: 492448-75-6

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsBiological ProductsComplex Mixtures +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vixarelimab DB16350
biotech | CAS: 2243320-83-2

Vixarelimab is under investigation in clinical trial NCT03816891 (A Study to Assess the Efficacy, Safety, and Tolerability of KPL-716 in Reducing Pruritus in Prurigo Nodularis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vixotrigine DB11706
small molecule | CAS: 934240-30-9

Vixotrigine has been investigated for the treatment of Bipolar Disorder and Bipolar Depression.

Kategori:
Amino AcidsAmino Acids, CyclicAmino Acids, Peptides, and Proteins +4
Target Protein:
Sodium channel protein type 9 subunit alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vixtimotamab DB17393
biotech | CAS: 2243775-32-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
VK-0214 DB17670
small molecule | CAS: 852949-30-5

Deskripsi belum tersedia.

Target Protein:
Thyroid hormone receptor beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
VK-2809 DB15137
small molecule | CAS: 852948-13-1

VK-2809 is under investigation in clinical trial NCT02927184 (Safety and Tolerability of VK2809 in Patients With Primary Hypercholesterolemia and Non-Alcoholic Fatty Liver Disease).

Kategori:
Organophosphorus Compounds
Target Protein:
Thyroid hormone receptor beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
VL-2397 DB17796
small molecule | CAS: 1186200-57-6

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntifungal Agents +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
VLTS-934 DB05597
small molecule

VLTS-934 was developed by Valentis inc. for the treatment of Peripheral Arterial Disease (PAD). It was under investigation in clinical trial NCT00113009 (Trial of VLTS-934 in Subjects With Intermittent Claudication Secondary to Peripheral Arterial Disease).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
VLX-1005 DB18307
small molecule | CAS: 1532593-30-8

Deskripsi belum tersedia.

Kategori:
AmidesBenzene DerivativesSulfonamides +2
Target Protein:
Arachidonate 12-lipoxygenase, 12R-type
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
VLX-1570 DB16030
small molecule | CAS: 1956378-23-6

VLX-1570 is under investigation in clinical trial NCT02372240 (A Study of VLX1570 and Dexamethasone in Myeloma Patients).

Kategori:
Benzene Derivatives
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
VM4-037 DB15319
small molecule | CAS: 1071470-72-8

VM4-037 is under investigation in clinical trial NCT00884520 (An Exploratory, Open Label, Multi-Center, Non-Randomized Study of [F-18]VM4-037).

Kategori:
AmidesAmino Acids, Peptides, and ProteinsFluorine Radioisotopes +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
VMD-928 DB18052
small molecule | CAS: 1802770-18-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
VO659 DB18160
biotech | CAS: 1479142-52-3

VO659 is an antisense oligonucleotide being investigated for the treatment of Huntington's disease.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Voacamine DB04877
small molecule | CAS: 3371-85-5

Voacamine is an alkaloid isolated from the bark of the _Pescheria fuchsiae folia_ tree. It is an antimalarial drug approved for use in several African countries. Voacamine is also under investigation for use in modulating multidrug-resistance in tumor cells.

Kategori:
AlkaloidsHeterocyclic Compounds, Fused-RingIndole Alkaloids +5
Target Protein:
ATP-dependent translocase ABCB1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vobarilizumab DB14891
biotech | CAS: 1628814-88-9

Vobarilizumab is under investigation in clinical trial NCT02101073 (ALX-0061 Phase I Bioavailability Study in Healthy Volunteers).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2490556-51-7

Vobramitamab duocarmazine is under investigation in clinical trial NCT05551117 (A Study of Vobramitamab Duocarmazine in Participants With Metastatic Castration Resistant Prostate Cancer and Other Solid Tumors).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vocacapsaicin DB17071
small molecule | CAS: 1931116-86-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1300724-82-6

Vocimagene amiretrorepvec is under investigation in clinical trial NCT02576665 (A Study of Toca 511, a Retroviral Replicating Vector, Combined With Toca FC in Patients With Solid Tumors or Lymphoma (Toca 6)).

Kategori:
Amino Acids, Peptides, and ProteinsAminohydrolasesEnzymes +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Voclosporin Approved DB11693
small molecule | CAS: 515814-01-4

Lupus nephritis (LN) is a type of glomerulonephritis occurring in patients with systemic lupus erythematosus (SLE). LN is a significant cause of renal failure, morbidity, and death in patients with SLE. Within 10 years of being diagnosed with SLE, 5-20% of …

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating AgentsCalcineurin Inhibitor Immunosuppressant +16
Target Protein:
Guided entry of tail-anchored proteins factor CAMLGProtein phosphatase 3 catalytic subunit alphaCalcineurin subunit B type 1 +1
Waktu ParuhThe average termina…
Vol. DistribusiThe apparent volume…
KlirensThe mean apparent s…
Genetik -
Vodobatinib DB17141
small molecule | CAS: 1388803-90-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vodudeutentan DB17410
small molecule | CAS: 2364365-83-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vofatamab DB14781
biotech | CAS: 1312305-12-6

Vofatamab is under investigation in clinical trial NCT02401542 (Dose Escalation, Expansion Study of Vofatamab (B-701) in Treatment of Locally Advanced or Metastatic Urothelial Cell Carcinoma).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Voglibose DB04878
small molecule | CAS: 83480-29-9

Voglibose is an alpha-glucosidase inhibitor used for lowering post-prandial blood glucose levels in people with diabetes mellitus. It is made in India by Ranbaxy Labs and sold under the trade name Volix.

Kategori:
AlcoholsAlimentary Tract and MetabolismBlood Glucose Lowering Agents +11
Target Protein:
Maltase-glucoamylase
Waktu ParuhThe half-life of vo…
Vol. Distribusi-
Klirens-
Genetik -
Volagidemab DB16421
biotech | CAS: 1233956-13-2

Volagidemab is under investigation in clinical trial NCT03117998 (Multiple Dose Study to Evaluate the Efficacy, Safety and Pharmacodynamics of REMD-477 in Subjects With Type 1 Diabetes Mellitus).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Volanesorsen Approved DB15067
biotech | CAS: 915430-78-3

Volanesorsen is an antisense oligonucleotide that binds to apoC-III mRNA to prevent its translation.[L16621] It is indicated to treat familial chylomicronemia, a genetic condition that prevents breakdown of triglycerides and chylomicrons.[L16621] This drug is…

Kategori:
CarbohydratesGlycosidesLipid Modifying Agents +4
Target Protein:
Apolipoprotein C-III
Waktu ParuhVolanesorsen has a …
Vol. DistribusiThe volume of distr…
KlirensThe exact rate of c…
Genetik -
Volasertib DB12062
small molecule | CAS: 755038-65-4

Volasertib has been used in trials studying the treatment of Leukemia, Neoplasms, Leukemia, Myeloid, Acute, Myelodysplastic Syndromes, and Leukemia, Monocytic, Acute, among others.

Kategori:
Antineoplastic AgentsHeterocyclic Compounds, Fused-Ring
Target Protein:
Serine/threonine-protein kinase PLK1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Volixibat DB13914
small molecule | CAS: 1025216-57-2

Volixibat, also known as SHP626 or LUM002, is an investigational drug that will potentially be used for the treatment of Non-Alcoholic Steatohepatitis (NASH). If approved for use, it will be the first available agent for the treatment of NASH. Volixibat is…

Kategori:
CarbohydratesHeterocyclic Compounds, Fused-RingLipid Regulating Agents +1
Target Protein:
Ileal sodium/bile acid cotransporter
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Volociximab DB06647
biotech | CAS: 558480-40-3

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAngiogenesis InhibitorsAngiogenesis Modulating Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2092457-20-8

Volrubigene ralaparvovec is under investigation in clinical trial NCT03223194 (Gene Transfer Clinical Study in Crigler-najjar Syndrome).

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Volrustomig DB18893
biotech | CAS: 2407760-40-9

Volrustomig is under investigation in clinical trial NCT06097728 (MEDI5752 in Combination With Carboplatin Plus Pemetrexed in Unresectable Pleural Mesothelioma).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Von Willebrand factor human Approved DB13133
biotech | CAS: 109319-16-6

The human von Willebrand factor (vWF) is a human plasma-derived vWF, an endogenous large multimeric plasma glycoprotein involved in hemostasis. It serves a dual role in hemostasis by mediating platelet adhesion and aggregation at the site of blood vessel inju…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood and Blood Forming Organs +8
Target Protein:
Coagulation factor VIIICollagen alpha-1(I) chainAsialoglycoprotein receptor 1 +1
Waktu ParuhIn patients with Ty…
Vol. DistribusiThe volume of distr…
KlirensIn patients with Ty…
Genetik -
Vonafexor DB18782
small molecule | CAS: 1192171-69-9

Deskripsi belum tersedia.

Target Protein:
Bile acid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vonicog alfa Approved DB12872
biotech

Vonicog alfa is a recombinant human von Willebrand factor (rVWF) produced from Chinese hamster ovary cells.[A264444] Used to treat von Willebrand Disease (vWD), it mimics the biological actions of endogenous VWF,[L51274] which is a critical plasma glycoprotei…

Kategori:
von Willebrand Factor
Target Protein:
Coagulation factor VIIICollagen alpha-1(I) chain
Waktu ParuhIn Study 071001, th…
Vol. Distribusi-
KlirensIn Study 071001, th…
Genetik -
Vonlerolizumab DB16352
biotech | CAS: 1638935-72-4

Vonlerolizumab is under investigation in clinical trial NCT03029832 (A Study of MOXR0916 in Combination With Atezolizumab Versus Atezolizumab Alone in Participants With Untreated Locally Advanced or Metastatic Urothelial Carcinoma Who Are Ineligible for Cispl…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vonoprazan Approved DB11739
small molecule | CAS: 881681-00-1

Vonoprazan is a potassium-competitive acid blocker (PCAB) that inhibits H<sup>+</sup>, K<sup>+</sup>-ATPase-mediated gastric acid secretion. PCABs represent an alternative to proton-pump inhibitors for the treatment of acid-related disorders. Unlike proton-pu…

Kategori:
Alimentary Tract and MetabolismAmidesCytochrome P-450 CYP2B6 Substrates +17
Target Protein:
Hydrogen potassium ATPase
Waktu ParuhVonoprazan has an e…
Vol. DistribusiVonoprazan has an a…
KlirensVonoprazan has an a…
Genetik -
Vopratelimab DB15378
biotech | CAS: 2039148-04-2

Vopratelimab is under investigation in clinical trial NCT02904226 (JTX-2011 Alone and in Combination With Anti-PD-1 or Anti-CTLA-4 in Subjects With Advanced and/or Refractory Solid Tumors).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vorapaxar Approved DB09030
small molecule | CAS: 618385-01-6

Vorapaxar is a tricyclic himbacine-derived selective inhibitor of protease activated receptor (PAR-1) indicated for reducing the incidence of thrombotic cardiovascular events in patients with a history of myocardial infarction (MI) or with peripheral arterial…

Kategori:
AnticoagulantsAntiplatelet agentsBlood and Blood Forming Organs +11
Target Protein:
Proteinase-activated receptor 1
Waktu ParuhVorapaxar has an ef…
Vol. Distribusi424 L
Klirens-
Genetik -
Vorasidenib Approved DB17097
small molecule | CAS: 1644545-52-7

Vorasidenib is a first-in-class dual isocitrate dehydrogenase-1 (IDH1) and isocitrate dehydrogenase-2 (IDH2) inhibitor.[A264209] It works by suppressing the levels of D-2-hydroxyglutarate (2-HG), an oncometabolite produced by mutant IDH1 and IDH2 isoforms.[L5…

Kategori:
AminesBCRP/ABCG2 InhibitorsCytochrome P-450 CYP1A2 Substrates +26
Target Protein:
Isocitrate dehydrogenase [NAD] subunit alpha, mitochondrialIsocitrate dehydrogenase [NAD] subunit beta, mitochondrialIsocitrate dehydrogenase [NAD] subunit gamma, mitochondrial +2
Waktu ParuhThe mean (CV%) stea…
Vol. DistribusiThe mean (CV%) volu…
KlirensThe mean (CV%) stea…
Genetik -
Voretigene neparvovec Approved DB13932
biotech | CAS: 1646819-03-5

Voretigene Neparvovec-rzyl (VN-rzyl) is an adeno-associated virus vector-based gene therapy.[L1094] An adeno-associated virus is a small virus that infects humans and other primates. It is not pathogenic and it causes a very mild immune response. This type of…

Kategori:
Adeno-associated Viral Vector TherapiesOphthalmologicalsSensory Organs
Target Protein:
Retinoid isomerohydrolase
Waktu ParuhBased on the pharma…
Vol. DistribusiVN-rzyl was shown t…
KlirensAccording to the ki…
Genetik -
Voriconazole Approved DB00582
small molecule | CAS: 137234-62-9

Voriconazole (Vfend, Pfizer) is a triazole antifungal medication used to treat serious fungal infections.[L15571] It is used to treat invasive fungal infections that are generally seen in patients who are immunocompromised. These include invasive candidiasis,…

Kategori:
14-alpha Demethylase InhibitorsAnti-Infective AgentsAntifungal Agents +35
Target Protein:
Lanosterol 14-alpha demethylase
Gen Terkait:
CYP2C19 CYP2C19 CYP2C19
Waktu ParuhVoriconazole follow…
Vol. DistribusiThe estimated volum…
KlirensThe clearance of vo…
Genetik 3 Varian
Vorinostat Approved DB02546
small molecule | CAS: 149647-78-9

Vorinostat (rINN) or suberoylanilide hydroxamic acid (SAHA), is a drug currently under investigation for the treatment of cutaneous T cell lymphoma (CTCL), a type of skin cancer, to be used when the disease persists, gets worse, or comes back during or after …

Kategori:
AmidesAminesAnilides +15
Target Protein:
Histone deacetylase 1Histone deacetylase 2Histone deacetylase 3 +4
Waktu Paruh2 hours
Vol. Distribusi-
Klirens-
Genetik -
Vorolanib DB15247
small molecule | CAS: 1013920-15-4

Vorolanib is under investigation in clinical trial NCT03904719 (CM082 and JS001 in Patients With Advanced Small-cell Lung Cancer (SCLC)).

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingProtein Kinase Inhibitors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vorozole DB13767
small molecule | CAS: 129731-10-8

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsAromatase Inhibitors +8
Target Protein:
Aromatase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1165741-01-4

Vorsetuzumab mafodotin is under investigation in clinical trial NCT01677390 (A Phase 1b Study of SGN-75 in Combination With Everolimus in Patients With Renal Cell Carcinoma).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vortioxetine Approved DB09068
small molecule | CAS: 508233-74-7

Vortioxetine is an antidepressant medication indicated for the treatment of major depressive disorder (MDD). It is classified as a serotonin modulator and stimulator (SMS) as it has a multimodal mechanism of action towards the serotonin neurotransmitter syste…

Kategori:
Agents that produce hypertensionAnti-Anxiety AgentsAntidepressive Agents +30
Target Protein:
Sodium-dependent serotonin transporter5-hydroxytryptamine receptor 3A5-hydroxytryptamine receptor 7 +4
Waktu ParuhMean terminal half­…
Vol. DistribusiThe apparent volume…
Klirens-
Genetik -
Voruciclib DB15157
small molecule | CAS: 1000023-04-0

Voruciclib is under investigation in clinical trial NCT03547115 (A Phase 1 Study of Voruciclib in Subjects With B-Cell Malignancies or AML).

Kategori:
Antineoplastic AgentsCarbohydratesEnzyme Inhibitors +6
Target Protein:
Cyclin-dependent kinase 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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