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13591

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10177 (74.9%)
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7625 (56.1%)
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Halaman 230 / 272
Salix nigra pollen Approved DB10398
biotech

Salix nigra pollen is the pollen of the Salix nigra plant. Salix nigra pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
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Genetik -
Salmeterol Approved DB00938
small molecule | CAS: 89365-50-4

Salmeterol is a long-acting beta-2 adrenergic receptor agonist drug that is currently prescribed for the treatment of asthma and chronic obstructive pulmonary disease COPD.[L11545,L11548,L11551,L11554,L11557] It has a longer duration of action than the short-…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic beta-2 Receptor Agonists +35
Target Protein:
Beta-2 adrenergic receptorBeta-1 adrenergic receptorBeta-3 adrenergic receptor
Waktu ParuhThe half life of sa…
Vol. DistribusiIn asthmatic patien…
KlirensThe average clearan…
Genetik -
Salmon calcitonin Approved DB00017
biotech | CAS: 47931-85-1

Synthetic peptide, 32 residues long formulated as a nasal spray.

Kategori:
Amino Acids, Peptides, and ProteinsBone Density Conservation AgentsBone Density, drug effects +15
Target Protein:
Calcitonin receptor
Waktu ParuhHalf-life eliminati…
Vol. Distribusi0.15 to 0.3 L/kg
Klirens-
Genetik -
Salsalate Approved DB01399
small molecule | CAS: 552-94-3

Salsalate is a nonsteroidal anti-inflammatory agent for oral administration. Salsalate's mode of action as an anti-inflammatory and antirheumatic agent may be due to inhibition of synthesis and release of prostaglandins. The usefulness of salicylic acid, the …

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +17
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu ParuhThe parent compound…
Vol. Distribusi-
Klirens-
Genetik -
Salsola kali pollen Approved DB10388
biotech

Salsola kali pollen is the pollen of the Salsola kali plant. Salsola kali pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Salvia miltiorrhiza root is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
AngiospermsBiological ProductsComplex Mixtures +15
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 96574-01-5

Salvianolic acid A is under investigation in clinical trial NCT03908242 (Phase I Study of Continuous Administration of Salvianolic Acid A Tablet).

Kategori:
Acids, CarbocyclicAntineoplastic AgentsCinnamates +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 121521-90-2

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAldehyde ReductaseAldehyde Reductase, antagonists & inhibitors +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Salvinorin A DB12327
small molecule | CAS: 83729-01-5

Salvinorin A has been investigated for the basic science of Pharmaceutical Preparations.

Kategori:
AlkaloidsCentral Nervous System AgentsCentral Nervous System Depressants +6
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorKappa-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Samalizumab DB12636
biotech | CAS: 1073059-33-2

Samalizumab has been used in trials studying the treatment of Multiple Myeloma and B-cell Chronic Lymphocytic Leukemia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Samarium DB12403
small molecule | CAS: 7440-19-9

Samarium has been used in trials studying the treatment and prevention of Pain, Cancer, Metastasis, Prostate Cancer, and Metastatic Osteosarcoma, among others.

Kategori:
ElementsLanthanoid Series ElementsMetals +1
Waktu Paruh-
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Genetik -
Samarium (153Sm) lexidronam Approved DB05273
small molecule | CAS: 122575-21-7

Samarium Sm 153 lexidronam is a radioactive medication used to treat pain caused by cancer that has spread to the bone. It is a radiopharmaceutical. Radiopharmaceuticals are radioactive agents that may be used to diagnose some diseases by studying the functio…

Kategori:
AnalgesicsAnalgesics, Non-NarcoticCentral Nervous System Agents +7
Waktu Paruh-
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Genetik -
Samarium Sm-153 DB12905
small molecule | CAS: 15766-00-4

Samarium 153 has been used in trials studying the supportive care of Pain, Lung Cancer, Breast Cancer, Prostate Cancer, and Metastatic Cancer.

Kategori:
ElementsIsotopesLanthanoid Series Elements +2
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Samatasvir DB12660
small molecule | CAS: 1312547-19-5

Samatasvir has been used in trials studying the treatment of Hepatitis C, Chronic, Chronic Hepatitis C Virus, and Chronic Hepatitis C Infection.

Kategori:
Acids, AcyclicHeterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Samidorphan Approved DB12543
small molecule | CAS: 852626-89-2

[Olanzapine] is an effective atypical antipsychotic that, like other antipsychotics, is associated with weight gain, metabolic dysfunction, and increased risk of type II diabetes.[A235638, A235643] Samidorphan is a novel opioid antagonist structurally related…

Kategori:
AlkaloidsAntipsychotic AgentsCentral Nervous System Agents +17
Target Protein:
Mu-type opioid receptorKappa-type opioid receptorDelta-type opioid receptor
Waktu ParuhSamidorphan has a m…
Vol. DistribusiSamidorphan followi…
KlirensSamidorphan has a m…
Genetik -
Samuraciclib DB16061
small molecule | CAS: 1805833-75-3

Samuraciclib is under investigation in clinical trial NCT03363893 (Modular Study to Evaluate CT7001 Alone in Cancer Patients With Advanced Malignancies).

Target Protein:
Cyclin-dependent kinase 7
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 141646-08-4

Sanfetrinem cilexetil is under investigation in clinical trial NCT05388448 (EBA, Safety and Tolerability of Sanfetrinem Cilexetil).

Kategori:
Amides
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Sanglifehrin A DB03393
small molecule

Deskripsi belum tersedia.

Target Protein:
Peptidyl-prolyl cis-trans isomerase A
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Santonin DB19377
small molecule

Santonin is a anthelmintic drug that was previously approved in the US to treat certain parasitic infections.

Kategori:
AnthelminticsAnti-Infective AgentsAntinematodal Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sapablursen DB18608
biotech | CAS: 2273007-95-5

Sapablursen is a synthetic 2'-O-(2-methoxyethyl)-modified antisense oligonucleotide linked to a tri-antennary cluster of N-acetyl galactosamine (GalNAc3) sugars targeting transmembrane protease, serine 6 messenger ribonucleic acid

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Sapacitabine DB06365
small molecule | CAS: 151823-14-2

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsNucleic Acids, Nucleotides, and NucleosidesNucleosides +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sapanisertib DB11836
small molecule | CAS: 1224844-38-5

Sapanisertib has been used in trials studying the treatment of HCC, Solid Tumor, Gliosarcoma, Liver Cancer, and Glioblastoma, among others.

Kategori:
Heterocyclic Compounds, Fused-RingPurines
Target Protein:
Serine/threonine-protein kinase mTOR
Waktu Paruh-
Vol. Distribusi-
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Sapitinib DB12183
small molecule | CAS: 848942-61-0

Sapitinib has been used in trials studying the treatment and basic science of Neoplasms, Breast Cancer, Breast Neoplasms, Metastatic Cancer, and Metastatic Breast Cancer, among others.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Receptor tyrosine-protein kinase erbB-2
Waktu Paruh-
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Saposin C DB17380
biotech

Saposin C is a lysosomal protein. Recombinant, non-glycosylated Saposin C is an active ingredient of BXQ-350, which is a novel, investigational anti-neoplastic therapy. BXQ-350 consists of Saposin C and the phospholipid dioleoylphosphatidyl-serine (DOPS), a p…

Kategori:
CoenzymesEnzymes and CoenzymesSphingolipid Activator Proteins
Waktu Paruh-
Vol. Distribusi-
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Saprisartan DB01347
small molecule | CAS: 146623-69-0

Saprisartan is an AT1 receptor antagonist. It is based on medications of losartan's prototypical chemical structure. The mode of (functional) AT1 receptor antagonism has been characterized as insurmountable/noncompetitive for saprisartan. It is very likely t…

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing angioedemaAgents causing hyperkalemia +6
Target Protein:
Type-1 angiotensin II receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sapropterin Approved DB00360
small molecule | CAS: 62989-33-7

Sapropterin (tetrahydrobiopterin or BH4) is a cofactor in the synthesis of nitric oxide. It is also essential in the conversion of phenylalanine to tyrosine by the enzyme phenylalanine-4-hydroxylase; the conversion of tyrosine to L-dopa by the enzyme tyrosine…

Kategori:
Alimentary Tract and MetabolismAminesBCRP/ABCG2 Inhibitors +15
Target Protein:
Phenylalanine-4-hydroxylaseNitric oxide synthase 3Tyrosine 3-monooxygenase +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Saquinavir Approved DB01232
small molecule | CAS: 127779-20-8

Saquinavir is an HIV-1 protease inhibitor used in combination with [ritonavir] and other antiretrovirals for the treatment of human immunodeficiency virus-1 (HIV-1) infection. In 1995 it became the first protease inhibitor approved by the FDA, followed shortl…

Kategori:
Agents Causing Muscle ToxicityAnti-HIV AgentsAnti-Infective Agents +44
Target Protein:
Gag-Pol polyproteinPol polyprotein
Waktu Paruh-
Vol. DistribusiThe steady-state vo…
KlirensThe systemic cleara…
Genetik -
SAR-125844 DB15382
small molecule | CAS: 1116743-46-4

SAR-125844 is under investigation in clinical trial NCT01391533 (Study of SAR125844 Single Agent Administered as Slow Intravenous Infusion in Adult Patients With Advanced Malignant Solid Tumors).

Kategori:
AmidesHeterocyclic Compounds, Fused-RingSulfur Compounds +1
Target Protein:
Hepatocyte growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SAR-405838 DB12541
small molecule | CAS: 1303607-60-4

SAR405838 has been used in trials studying the treatment of Neoplasm Malignant.

Kategori:
Heterocyclic Compounds, Fused-RingP-glycoprotein substrates
Target Protein:
Cellular tumor antigen p53
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SAR-439459 DB17864
biotech | CAS: 2114339-57-8

SAR-439459 is a pan-transforming Growth Factor-beta (TGF?) neutralizing antibody.[A259862] Developed by Sanofi, it is being investigated for the treatment of cancers and Osteogenesis Imperfecta.

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SAR443122 DB16492
small molecule | CAS: 2125450-76-0

SAR443122, was investigated in several clinical trials to evaluate its safety and efficacy. NCT04469621 was studied in severe COVID-19 patients, while NCT05588843 is currently recruiting participants with ulcerative colitis. Additionally, NCT04781816, which w…

Kategori:
Experimental Unapproved Treatments for COVID-19
Target Protein:
Receptor-interacting serine/threonine-protein kinase 1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
SAR445136 DB17708
biotech

SAR445136 is an investigational zinc finger nuclease gene-edited cell therapy. It consists of autologous CD34+ hematopoietic stem precursor cells (HSPC) modified ex vivo by zinc finger nucleases (ZFN) that target the BCL11A gene erythroid-specific enhancer (E…

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Vol. Distribusi-
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Genetik -
Saracatinib DB11805
small molecule | CAS: 379231-04-6

Saracatinib has been investigated for the treatment of Cancer, Osteosarcoma, Ovarian Cancer, Fallopian Tube Cancer, and Primary Peritoneal Cancer.

Kategori:
Antineoplastic AgentsCytochrome P-450 CYP3A InhibitorsCytochrome P-450 CYP3A4 Inhibitors +6
Target Protein:
Proto-oncogene tyrosine-protein kinase SrcTyrosine-protein kinase ABL1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Saralasin DB06763
small molecule | CAS: 34273-10-4

Deskripsi belum tersedia.

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing hyperkalemiaAgents that produce hypertension +8
Target Protein:
Type-2 angiotensin II receptorType-1 angiotensin II receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sarecycline Approved DB12035
small molecule | CAS: 1035654-66-0

Sarecycline is a semi-synthetic derivative of tetracycline that was initially discovered by Paratek Pharmaceuticals from Boston, MA but then licensed to Warner Chilcott of Rockaway, NJ in July of 2007 [A40005]. After completing various phase-II and phase-III …

Kategori:
Anti-Acne PreparationsAnti-Acne Preparations for Systemic UseAnti-Bacterial Agents +7
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe mean apparent v…
KlirensThe mean apparent o…
Genetik -
Saredutant DB06660
small molecule | CAS: 142001-63-6

Saredutant (SR 48968) is a neurokinin-2 antagonist drug being developed as an antidepressant and anxiolytic by Sanofi-Aventis.

Kategori:
Acids, CarbocyclicAmidesAntidepressive Agents +4
Target Protein:
Substance-K receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sargramostim Approved DB00020
biotech | CAS: 123774-72-1

Sargramostim is a human recombinant granulocyte macrophage colony-stimulating factor (GM-CSF) expressed in yeast. It is a glycoprotein that is 127 residues. Substitution of Leu23 leads to a difference from native protein.

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating Agents +14
Target Protein:
Granulocyte-macrophage colony-stimulating factor receptor subunit alphaInterleukin-3 receptor subunit alphaCytokine receptor common subunit beta +2
Waktu Paruh-
Vol. Distribusi-
Klirens* 420 mL/min/m2 [No…
Genetik -
Sarilumab Approved DB11767
biotech | CAS: 1189541-98-7

Sarilumab is a fully human anti-interleukin 6 (IL-6) receptor monoclonal IgG1 antibody that binds to both membrane-bound and soluble IL-6 receptor forms, thus blocking the cis- and trans-inflammatory signalling cascades of IL-6.[A27262] Sarilumab was develope…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +22
Target Protein:
Interleukin-6 receptor subunit alphaHigh affinity immunoglobulin gamma Fc receptor ILow affinity immunoglobulin gamma Fc region receptor II-a +3
Waktu ParuhThe half-life will …
Vol. DistribusiIn patients with rh…
KlirensSarilumab is not el…
Genetik -
Sarizotan DB06454
small molecule | CAS: 351862-32-3

Deskripsi belum tersedia.

Target Protein:
5-hydroxytryptamine receptor 1AD(2) dopamine receptorD(3) dopamine receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sarocladium strictum Approved DB14168
biotech

Sarocladium strictum allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +2
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Saroglitazar DB13115
small molecule | CAS: 495399-09-2

Saroglitazar has been investigated for the treatment of Fatty Liver.

Kategori:
Acids, Carbocyclic
Waktu Paruh-
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Genetik -
Sarpogrelate DB12163
small molecule | CAS: 125926-17-2

Sarpogrelate has been investigated for the treatment of Diabetes Mellitus, Diabetic Nephropathy, Coronary Artery Disease, and Renal Insufficiency, Chronic.

Kategori:
Acids, AcyclicAntidepressive AgentsAntiplatelet agents +8
Target Protein:
5-hydroxytryptamine receptor 2C5-hydroxytryptamine receptor 2A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sarracenia Purpurea Approved DB13965
biotech

_Sarracenia purpurea_, commonly known as the purple pitcher plant, northern pitcher plant, turtle socks, or side-saddle flower, is a perennial carnivorous plant in the family _Sarraceniaceae_. _Sarracenia purpurea_ attract and trap insects within their pitche…

Kategori:
Miscellaneous Analgesics and Antipyretics
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
biotech

SARS-CoV-2 mRNA vaccine (ARCoV) is a novel mRNA coronavirus vaccine that consists of a lipid nanoparticle-encapsulated mRNA encoding the receptor binding domain of SARS-CoV-2[A220048]. It is the first COVID-19 mRNA vaccine to be approved for clinical trials …

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Genetik -
biotech

The University of Queensland (UQ), in partnership with The Coalition for Epidemic Preparedeness Inovations (CEPI) and CSL has developed a COVID-19 candidate, SARS-CoV-2 Sclamp. The vaccine was developed using UQ’s rapid response ‘molecular clamp’ vaccine plat…

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Genetik -
biotech

Bimervax is an adjuvanted non-mRNA COVID-19 vaccine utilizing a SARS-CoV-2 recombinant spike (S) protein receptor binding domain (RBD) fusion heterodimer.[L48902] It is intended to elicit protection against Omicron XBB.1.5, one of the dominant circulating SAR…

Kategori:
COVID-19 VaccinesVaccinesViral Vaccines
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Sarsagenin DB16928
small molecule | CAS: 126-19-2

Deskripsi belum tersedia.

Kategori:
CholestanesDrugs, Chinese HerbalFused-Ring Compounds +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Saruparib DB18982
small molecule | CAS: 2589531-76-8

Saruparib is under investigation in clinical trial NCT06380751 (Saruparib (AZD5305) Plus Camizestrant Compared With CDK4/6 Inhibitor Plus Endocrine Therapy or Plus Camizestrant in Hr-positive, Her2-negative (IHC 0, 1+, 2+/ ISH Non-amplified), BRCA1, BRCA2, or…

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
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Saruplase DB13646
biotech | CAS: 99149-95-8

Deskripsi belum tersedia.

Kategori:
Agents causing angioedemaAmino Acids, Peptides, and ProteinsAnticoagulants +16
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Satavaptan DB14923
small molecule | CAS: 185913-78-4

Satavaptan is under investigation in clinical trial NCT00359437 (Satavaptan in the Prevention of Ascites Recurrence in Patients With Ascites Due to Cirrhosis of the Liver).

Kategori:
Antidiuretic Hormone Receptor AntagonistsNatriuretic AgentsOxazines
Target Protein:
Vasopressin V2 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 11451–11500 dari 13591
Sebelumnya Halaman 230 / 272 Berikutnya