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6694

Total database: 17430
Struktur (SMILES)
4518 (67.5%)
Target
3751 (56.0%)
Genomik
81 (1.2%)
Referensi
6694 (100.0%)

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Hasil Pencarian (6694)

Halaman 23 / 134
small molecule | CAS: 149301-79-1

Specific inhibitor of phospholipase A2.[A252972]

Kategori:
EicosanoidsEnzyme InhibitorsFatty Acids +3
Target Protein:
Cytosolic phospholipase A2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aranidipine DB09229
small molecule | CAS: 86780-90-7

Aranidipine is a novel dihydropyridine derivative that gives rise to two active metabolites (M-1? and M-1?) that exhibit hypotensive activity. It is a calcium antagonist with the formula methyl 2-oxopropyl 1,4-dihydro-2,6-dimethyl-4-(2-nitrophenyl)-3,5-pyridi…

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsBradycardia-Causing Agents +8
Target Protein:
Voltage-dependent L-type calcium channel subunit alpha-1CVoltage-dependent L-type calcium channel subunit alpha-1DVoltage-dependent L-type calcium channel subunit alpha-1F +3
Waktu ParuhThe elimination hal…
Vol. Distribusi-
Klirens-
Genetik -
Arbaclofen DB08891
small molecule | CAS: 69308-37-8

Arbaclofen, or STX209, is the R-enantiomer of baclofen. It is believed to be a selective gamma-amino butyric acid type B receptor agonist, and has been investigated as a treatment for autism spectrum disorder and fragile X syndrome in randomized, double blind…

Target Protein:
Gamma-aminobutyric acid type B receptor subunit 1Gamma-aminobutyric acid type B receptor subunit 2
Waktu Paruh-
Vol. Distribusi-
KlirensBlood clearance of …
Genetik -
small molecule | CAS: 847353-30-4

Arbaclofen Placerbil is a prodrug of Arbaclofen, which is a selective gamma-amino-butyric acid type B receptor agonist and the R-enantiomer of baclofen. It was discovered, and has been patented by XenoPort as a new chemical entity with an improved pharmacokin…

Kategori:
Acids, AcyclicAminobutyratesButyrates +10
Target Protein:
Gamma-aminobutyric acid type B receptor subunit 1Gamma-aminobutyric acid receptor subunit gamma-3Gamma-aminobutyric acid type B receptor subunit 2
Waktu ParuhIV bolus administra…
Vol. DistribusiRadioactive labelin…
KlirensBlood clearance of …
Genetik -
Arbekacin DB06696
small molecule | CAS: 51025-85-5

An semisynthetic aminoglycoside antibiotic. Often used for treatment of multi-resistant bacterial infection such as methicillin-resistant _Staphylococcus aureus_ (MRSA).

Kategori:
Agents that produce neuromuscular block (indirect)Aminoglycoside AntibacterialsAnti-Bacterial Agents +9
Target Protein:
30S ribosomal protein S12
Waktu Paruh3 hours
Vol. Distribusi-
Klirens-
Genetik -
Arbutamine Approved DB01102
small molecule | CAS: 128470-16-6

Arbutamine, administered through a closed-loop, computer-controlled drug-delivery system, is indicated to elicit acute cardiovascular responses, similar to those produced by exercise, in order to aid in diagnosing the presence or absence of coronary artery di…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic and Dopaminergic Agents +17
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptorBeta-3 adrenergic receptor
Waktu ParuhElimination half-li…
Vol. Distribusi-
Klirens-
Genetik -
ARC183 DB05124
biotech

ARC183 is a DNA aptamer, which is a single-stranded DNA molecule consisting of 15 deoxynucleotides that forms well-defined three-dimensional configuration, allowing it to bind to thrombin with high affinity and specificity. The key advantage of ARC183 compar…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Arcitumomab DB17201
biotech | CAS: 154361-48-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ardeparin Approved DB00407
small molecule | CAS: 9005-49-6

Ardeparin, marketed under the US trade name Normiflo, is a low molecular weight heparin (LMWH) anticoagulant used for the prevention of postoperative venous thrombosis. Ardeparin is derived via peroxide degradation of heparin extracted from porcine intestinal…

Kategori:
Agents causing hyperkalemiaAnticoagulantsCarbohydrates +7
Target Protein:
Antithrombin-IIIHeparin cofactor 2
Waktu ParuhElimination half-li…
Vol. Distribusi-
Klirens-
Genetik -
Arecoline DB04365
small molecule | CAS: 63-75-2

An alkaloid obtained from the betel nut (Areca catechu), fruit of a palm tree. It is an agonist at both muscarinic and nicotinic acetylcholine receptors. It is used in the form of various salts as a ganglionic stimulant, a parasympathomimetic, and a vermifuge…

Kategori:
AlkaloidsCholinergic AgentsCholinergic Agonists +3
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Argan oil DB14310
biotech

Argan oil is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
Biological ProductsComplex MixturesLipids +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Arginine DB00125
small molecule | CAS: 74-79-3

An essential amino acid that is physiologically active in the L-form.

Kategori:
Acids, AcyclicAmino AcidsAmino Acids, Basic +14
Target Protein:
Cationic amino acid transporter 3Antizyme inhibitor 2Argininosuccinate lyase +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 4320-30-3

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsBile and Liver Therapy +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Argininosuccinate lyaseArgininosuccinate synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ARGX-119 DB18133
biotech

ARGX-119 is a monoclonal antibody that targets and activates muscle-specific kinase (MuSK).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aripiprazole Approved DB01238
small molecule | CAS: 129722-12-9

Aripiprazole is an atypical antipsychotic orally indicated for the treatment of schizophrenia, bipolar I, major depressive disorder, irritability associated with autism, and Tourette's.[L45859] It is also indicated as an injection for agitation associated wit…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +48
Target Protein:
D(2) dopamine receptor5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 1A +35
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe steady-state vo…
KlirensThe clearance of ar…
Genetik -
Aripiprazole lauroxil Approved DB14185
small molecule | CAS: 1259305-29-7

Aripiprazole lauroxil is a long-acting injectable atypical antipsychotic drug used in the treatment of schizophrenia in adult patients. It is a prodrug of [aripiprazole], which acts as a partial agonist at the D2 and 5-HT1A receptors, and as an antagonist at …

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +29
Target Protein:
D(2) dopamine receptor5-hydroxytryptamine receptor 1A5-hydroxytryptamine receptor 2A +22
Waktu ParuhThe mean aripiprazo…
Vol. DistribusiBased on population…
KlirensIn rats, the cleara…
Genetik -
ARM-210 DB16944
small molecule | CAS: 1467605-57-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Armodafinil Approved DB06413
small molecule | CAS: 112111-43-0

Armodafinil is the enantiopure of the wakefulness-promoting agent modafinil (Provigil), and is indicated to improve wakefulness in adult patients with excessive sleepiness associated with obstructive sleep apnea (OSA), narcolepsy, or shift work disorder (SWD)…

Kategori:
Benzene DerivativesBenzhydryl CompoundsCentral Nervous System Agents +21
Target Protein:
Alpha-1D adrenergic receptorSodium-dependent dopamine transporter
Waktu ParuhTerminal half-life …
Vol. DistribusiApparent volume of …
KlirensThe oral clearance …
Genetik -
ARO-ANG3 DB17626
biotech

ARO-ANG3 is a subcutaneously administered RNA interference (RNAi)-based investigational medicine targeting angiopoietin-like protein 3 (ANGPTL3). It was granted an orphan drug designation for the treatment of homozygous familial hypercholesterolemia (HoFH).[L…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aroplatin DB17319
small molecule | CAS: 114488-24-3

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsOrganometallic Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Arotinoid acid DB02877
small molecule | CAS: 71441-28-6

Arotinoid acid is a retinoic acid analog which acts as a selective RAR agonist.

Kategori:
Acids, CarbocyclicAlkenesBenzene Derivatives +9
Target Protein:
Retinoic acid receptor beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Arsanilic acid DB03006
small molecule | CAS: 98-50-0

An arsenical which has been used as a feed additive for enteric conditions in pigs and poultry. It causes blindness and is ototoxic and nephrotoxic in animals. [PubChem]

Kategori:
Adjuvants, ImmunologicAlkenesAnti-Infective Agents +10
Target Protein:
Lysozyme C
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Arsenic trioxide Approved DB01169
small molecule | CAS: 1327-53-3

Arsenic trioxide is a chemotherapeutic agent of idiopathic function used to treat leukemia that is unresponsive to first line agents. It is suspected that arsenic trisulfide induces cancer cells to undergo apoptosis. In general, arsenic is known to be a natur…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsArsenicals +16
Target Protein:
Inhibitor of nuclear factor kappa-B kinase subunit betaThioredoxin reductase 1, cytoplasmicTranscription factor Jun +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Arsenous acid DB04456
small molecule | CAS: 13464-58-9

Deskripsi belum tersedia.

Kategori:
AnionsArsenicalsElectrolytes +1
Target Protein:
Arsenate reductaseArsenical pump-driving ATPase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Artemether Approved DB06697
small molecule | CAS: 71963-77-4

Artemether is an antimalarial agent used to treat acute uncomplicated malaria. It is administered in combination with lumefantrine for improved efficacy. This combination therapy exerts its effects against the erythrocytic stages of <i>Plasmodium spp.</i> and…

Kategori:
Anti-Infective AgentsAntimalarialsAntiparasitic Agents +25
Target Protein:
Sodium/potassium-transporting ATPase subunit alpha-1
Waktu ParuhArtemether, 1.6 +/-…
Vol. Distribusi-
Klirens-
Genetik -
Artemisia ludoviciana pollen Approved DB10762
biotech

Artemisia ludoviciana pollen is the pollen of the Artemisia ludoviciana plant. Artemisia ludoviciana pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Pollen Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Artemisia vulgaris root Approved DB14170
biotech

Artemisia vulgaris root allergenic extract is used in allergenic testing.

Kategori:
Non-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Artemisinin DB13132
small molecule | CAS: 63968-64-9

Artemisinin has been used in trials studying the treatment of Schizophrenia, Malaria, Falciparum, and Plasmodium Falciparum.

Kategori:
Anti-Infective AgentsAntimalarialsAntiparasitic Products, Insecticides and Repellents +13
Target Protein:
Dihydroorotate dehydrogenase (quinone), mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Artemisone DB16097
small molecule | CAS: 255730-18-8

Artemisone is under investigation in clinical trial NCT00936767 (Artemisone for the Treatment of Uncomplicated Falciparum Malaria in Western Cambodia).

Kategori:
Free RadicalsPeroxidesReactive Oxygen Species +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Artemotil Approved DB13851
small molecule | CAS: 75887-54-6

Artemotil, also known as ?-arteether, is a semi-synthetic derivative of artemisinin and a fast acting blood schizonticide specifically indicated for the treatment of chloroquine-resistant _Plasmodium falciparum_ malaria and cerebral malaria cases.

Kategori:
AmebicidesAnti-Infective AgentsAntimalarials +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Artenimol Approved DB11638
small molecule | CAS: 71939-50-9

Artenimol is an artemisinin derivative and antimalarial agent used in the treatment of uncomplicated *Plasmodium falciparum* infections [FDA Label]. It was first authorized for market by the European Medicines Agency in October 2011 in combination with [DB139…

Kategori:
Anti-Infective AgentsAntimalarialsAntiparasitic Agents +16
Target Protein:
Actin, cytoplasmic 2Alpha-aminoadipic semialdehyde dehydrogenaseAnnexin A2 +188
Waktu ParuhArtenimol was repor…
Vol. DistribusiArtenimol was obser…
KlirensArtenimol was obser…
Genetik -
Arterolane DB19027
small molecule | CAS: 664338-39-0

Arterolane is under investigation in clinical trial NCT03452475 (Comparison of Arterolane-piperaquine Versus Arterolane-piperaquine+mefloquine Versus Artemether-lumefantrine in Kenyan Children).

Kategori:
AnionsAntimalarialsAntiparasitic Products, Insecticides and Repellents +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Artesunate Approved DB09274
small molecule | CAS: 88495-63-0

Artesunate is indicated for the initial treatment of severe malaria.[L14099] The World Health Organization recommends artesunate as first line treatment for severe malaria.[L890] Artesunate was developed out of a need for a more hydrophilic derivative of [art…

Kategori:
Acids, AcyclicAnionsAnthelmintics +28
Target Protein:
Malaria protein EXP-1
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of ar…
Genetik -
Arundic acid DB05343
small molecule | CAS: 185517-21-9

Arundic acid has been investigated for the treatment of Amyotrophic Lateral Sclerosis (ALS).

Kategori:
Acids, AcyclicFatty AcidsLipids
Target Protein:
Beta-3 adrenergic receptorProtein S100-B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ARX201 DB05082
small molecule

ARX201 (PEG-ahGH) is a recombinant form of human growth hormone that has been modified using Ambrx’s patented ReCODE™ technology to achieve precise spatial positioning of the site of polyethylene glycol (PEG) attachment to human growth hormone, by biosyntheti…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Arylomycin A2 DB01934
small molecule

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Target Protein:
Signal peptidase I
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ASC-618 DB18423
biotech

ASC-618 is a recombinant adeno-associated virus serotype 8 (rAAV2/8) vector expressing bioengineered B domain deleted liver-codon-optimized human factor VIII.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Asciminib Approved DB12597
small molecule | CAS: 1492952-76-7

Asciminib is a tyrosine kinase inhibitor (TKI) used in the treatment of chronic-phase Philadelphia chromosome-positive chronic myeloid leukemia (Ph+ CML). More specifically, it is an inhibitor of the ABL1 kinase activity of the BCR-ABL1 fusion protein[L38995]…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBcr-Abl Tyrosine Kinase Inhibitors +26
Target Protein:
Tyrosine-protein kinase ABL1
Waktu ParuhThe terminal elimin…
Vol. DistribusiAt steady-state, th…
KlirensThe total apparent …
Genetik -
Ascorbic acid Approved DB00126
small molecule | CAS: 50-81-7

A six carbon compound related to glucose. It is found naturally in citrus fruits and many vegetables. Ascorbic acid is an essential nutrient in human diets, and necessary to maintain connective tissue and bone. Its biologically active form, vitamin C, functio…

Kategori:
Acids, AcyclicAlimentary Tract and MetabolismAntioxidants +20
Target Protein:
Solute carrier family 23 member 2Solute carrier family 23 member 1Hyaluronate lyase +23
Waktu Paruh16 days (3.4 hours …
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 129499-78-1

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicCarbohydratesHydroxy Acids +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ascrinvacumab DB12261
biotech | CAS: 1463459-96-2

Ascrinvacumab has been used in trials studying the treatment and basic science of Neoplasms, Advanced Solid Tumors, Carcinoma, Hepatocellular, and Malignant Pleural Mesothelioma.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Asenapine Approved DB06216
small molecule | CAS: 65576-45-6

Developed by Schering-Plough after its merger with Organon International, asenapine is a sublingually administered, atypical antipsychotic for treatment of schizophrenia and acute mania associated with bipolar disorder. Asenapine also belongs to the dibenzo-o…

Kategori:
Acid ReducersAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +41
Target Protein:
5-hydroxytryptamine receptor 2AD(2) dopamine receptor5-hydroxytryptamine receptor 1A +17
Waktu Paruh24 hours (range of …
Vol. Distribusi20-25 L/kg
Klirens-
Genetik -
Asfotase alfa Approved DB09105
biotech | CAS: 1174277-80-5

Asfotase alfa is a first-in-class bone-targeted enzyme replacement therapy designed to address the underlying cause of hypophosphatasia (HPP)—deficient alkaline phosphatase (ALP). Hypophosphatasia is almost always fatal when severe skeletal disease is obvious…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsAntibodies +16
Target Protein:
Pyrophosphate
Waktu ParuhApproximately 5 day…
Vol. Distribusi-
Klirens-
Genetik -
ASI402 DB06373
biotech | CAS: 372075-37-1

ASI402 is a monoclonal antibody that targets an aberrantly glycosylated antigen Mucin 1. It is being investigated in cancers.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Target Protein:
Mucin-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Asiatic acid DB14054
small molecule | CAS: 464-92-6

From Centella asiatica and other plants; shows a variety of bioactivities.

Kategori:
TerpenesTriterpenes
Target Protein:
Glycogen phosphorylase, muscle form
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ASP-2138 DB18473
biotech

ASP-2138 is a bispecific antibody directed against CLDN18.2 and T cell receptor complex CD3

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ASP-3026 DB12729
small molecule | CAS: 1097917-15-1

ASP3026 has been used in trials studying the treatment of Solid Tumor, B-Cell Lymphoma, Advanced Malignancies, Positive for Anaplastic Lymphoma Kinase, and Positive for Proto-Oncogene Tyrosine-Protein Kinase ROS.

Kategori:
Sulfur Compounds
Target Protein:
ALK tyrosine kinase receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1349719-22-7

Asparaginase _Erwinia chrysanthemi_ is an asparaginase-specific enzyme derived from _Erwinia_ _chrysanthemi_ used as an anticancer agent. It works by depleting the stores of an important amino acid called asparagine, which is involved in DNA synthesis and cel…

Kategori:
AmidohydrolasesAntineoplastic AgentsAsparaginase +7
Waktu ParuhThe apparent half-l…
Vol. DistribusiThe volume of distr…
KlirensThe geometric mean …
Genetik -
biotech | CAS: 9015-68-3

Asparaginase derived from _Escherichia coli_ (L-asparagine amidohydrolase, EC 3.5.1.1) is an enzyme responsible for the metabolism of L-asparagine, by catalyzing L-asparagine into L-aspartic acid and ammonia. It also facilitates the production of oxaloacetate…

Kategori:
AmidohydrolasesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +7
Target Protein:
L-asparagine
Waktu ParuhPlasma half life of…
Vol. DistribusiApparent volume of …
Klirens-
Genetik -
Menampilkan 1101–1150 dari 6694
Sebelumnya Halaman 23 / 134 Berikutnya