Hasil Filter

16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (16004)

Halaman 229 / 321
NPI 32101 DB05264
small molecule

NPI 32101 possesses both anti-inflammatory and broad spectrum antimicrobial activities. This combination of pharmacological properties may have additional therapeutic uses beyond dermatology.

Target Protein:
Cytokine receptor common subunit beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NPS-2143 DB05695
small molecule | CAS: 284035-33-2

Deskripsi belum tersedia.

Target Protein:
Extracellular calcium-sensing receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NPT520-34 DB17920
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NRC-AN-019 DB17110
small molecule | CAS: 879507-25-2

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesAntineoplastic Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NRP-2945 DB18150
biotech

NRP-2945 is a 11-mer peptidomimetic.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NRX-1074 DB11784
small molecule | CAS: 1421866-48-9

NRX-1074 has been used in trials studying the treatment of Schizophrenia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NS-2359 DB05805
small molecule | CAS: 195875-68-4

NS2359 is a triple monoamine re-uptake inhibitor with a new, unique drug profile expected to yield important benefits compared to existing treatments of depression. Enhancing the function of the three neurotransmitters serotonin, noradrenalin and dopamine, NS…

Kategori:
AlkaloidsAza CompoundsAzabicyclo Compounds +1
Target Protein:
Sodium-dependent dopamine transporterSodium-dependent noradrenaline transporterSodium-dependent serotonin transporter
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NS-3728 DB05835
small molecule | CAS: 265646-85-3

NS3728 is an orally active chloride channel blocker for the treatment of cancer.

Kategori:
AmidesAminesAnilides +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NS-398 DB14060
small molecule | CAS: 123653-11-2

NS-398 is a COX-2 inhibitor. It was developed as part of the mechanistic study of the cyclooxygenases.

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAmides +14
Target Protein:
Prostaglandin G/H synthase 2Cyclooxygenase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NS-8593 DB16897
small molecule | CAS: 875755-39-8

Deskripsi belum tersedia.

Kategori:
AminesNaphthalenes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NS13001 DB16898
small molecule | CAS: 1063331-94-1

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingPurines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NSC-663284 DB17038
small molecule | CAS: 383907-43-5

NSC-663284 is a potent quinolinedione Cdc25 phosphatase inhibitor.[A253052]

Kategori:
cdc25 Phosphatases, antagonists & inhibitorsHeterocyclic Compounds, Fused-RingQuinolines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NSI-189 DB16230
small molecule | CAS: 1270138-40-3

NSI-189 is under investigation in clinical trial NCT02695472 (Study of NSI-189 for Major Depressive Disorder).

Kategori:
AminesPyridines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NSI-566 DB17954
biotech

NSI-566 is a stem cell therapy consisting of human spinal cord-derived neural stem cells. Developed by Seneca Biopharma, it is being investigated for the treatment of amyotrophic lateral sclerosis (ALS), stroke, and chronic spinal cord injury (cSCI).[L47097]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NT 13 DB16953
small molecule | CAS: 117928-93-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NT-102 DB18112
small molecule | CAS: 1607447-79-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NT-219 DB17490
small molecule | CAS: 1198078-60-2

Deskripsi belum tersedia.

Target Protein:
Insulin receptor substrate 2Insulin receptor substrate 1Signal transducer and activator of transcription 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NTLA-2001 DB18525
biotech

NTLA-2001 is a clustered regularly interspaced short palindromic repeats CRISPR/ Cas9-based gene therapy consisting of a single guide RNA targeting the human TTR gene and a messenger RNA encoding Cas9.

Kategori:
Biomimetic MaterialsDrug CarriersMembranes, Artificial +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NTLA-2002 DB17597
biotech

NTLA-2002 is a lipid nanoparticle encapsulating single guide RNA (G012267) targeting the human KLKB1 gene and messenger RNA (mRNA000042) encoding Cas9. It is an investigational therapy designed to knock out the target gene kallikrein B1 (KLKB1) to reduce plas…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NTP-42 DB18302
small molecule | CAS: 2055599-51-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NTx-265 DB05649
biotech

NTx-265 is a combination of two currently marketed large molecules designed to stimulate the growth and differentiation of neural stem cells in adults who have suffered a stroke – the second leading cause of death worldwide. In May 2006, biotechnology company…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NU1025 DB02690
small molecule | CAS: 90417-38-2

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Poly [ADP-ribose] polymerase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NUC B1000 DB05242
biotech

NUC B1000 is an expressed interfering RNA (eiRNA)- based product consisting of a plasmid DNA construct designed to produce four short interfering RNA (siRNA) molecules, formulated with a proprietary cationic-lipid delivery system. [F3910] eiRNA is an approach…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NUC-7738 DB19148
small molecule | CAS: 2348493-39-8

NUC-7738 is under investigation in clinical trial NCT03829254 (A Safety, Pharmacokinetic and Clinical Activity Study of NUC-7738 in Patients With Advanced Solid Tumours and Lymphoma).

Kategori:
Benzene DerivativesHeterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nurulimab DB18946
biotech | CAS: 2168561-20-2

Nurulimab is under investigation in clinical trial NCT05732805 (A Clinical Study of BCD-217 (Nurulimab + Prolgolimab) Followed by Anti-pd-1 Compared to Anti-pd-1 Monotherapy as First-line Treatment in Subjects With Unresectable/metastatic Melanoma).

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsMonoclonal antibodies and antibody drug conjugates
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nusinersen Approved DB13161
small molecule | CAS: 1258984-36-9

An antisense oligonucleotide that induces survival motor neuron (SMN) protein expression, it was approved by the U.S. FDA in December, 2016 as Spinraza for the treatment of children and adults with spinal muscular atrophy (SMA). It is adminstrated as direct i…

Kategori:
Antisense OligonucleotidesIncreased Protein SynthesisMusculo-Skeletal System +4
Target Protein:
Survival motor neuron protein
Waktu ParuhThe mean terminal e…
Vol. DistribusiCSF: 0.4 L Plasma…
KlirensSlow clearance is o…
Genetik -
Nutlin-3 DB17039
small molecule | CAS: 548472-68-0

Nutlin-3 is a small molecule inhibitor that targets p53-Mdm2 interaction.[A253057]

Kategori:
Stereoisomerism
Target Protein:
Cellular tumor antigen p53
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nutmeg oil DB15996
biotech | CAS: 8008-45-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nuvaxovid Approved DB15810
biotech

SARS-CoV-2, the causative agent of COVID-19, relies on the interaction between its trimeric spike (S) glycoprotein and angiotensin-converting enzyme 2 (hACE2) expressed on host cells in order to establish a productive infection in humans.[A243789] Antibodies …

Kategori:
Biological ProductsComplex MixturesCOVID-19 Vaccines +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 8046-97-7

Deskripsi belum tersedia.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NV-07a DB05845
small molecule

NV-07a is topical skin repair compound protecting skin from sun-induced immunosuppression and UV-induced damage.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NV-18 DB05886
small molecule

NV-18 is a product of the Novogen diphenolic synthetic analogue program that is creating drugs with diverse activities against specific types of cancer. Like phenoxodiol, NV-18 is broadly effective in the laboratory against almost all human cancer types, but …

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NV-354 DB18392
small molecule | CAS: 866465-21-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NV-5138 DB19180
small molecule | CAS: 2095886-80-7

NV-5138 is under investigation in clinical trial NCT06235905 (Open-label of SPN-820 in Adults With Major Depressive Disorder).

Kategori:
Amino AcidsAmino Acids, Branched-ChainAmino Acids, Essential +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NV-52 DB05673
small molecule

NV-52 is an investigational synthetic flavonoid thromboxane synthase (TXS) inhibitor developed for the maintenance of remission in inflammatory bowel disease.

Target Protein:
Thromboxane-A synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NVD-001 DB18459
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NVL-655 DB18682
small molecule

NVL-655 is an orally bioavailable, brain-penetrant anaplastic lymphoma kinase (ALK) inhibitor inhibitor being investigated for the treatment of non-small cell lung cancer.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NVP-LEQ-506 DB12857
small molecule | CAS: 1204975-42-7

LEQ506 has been used in trials studying the treatment of Advanced Solid Tumors, Recurrent or Refractory Medulloblastoma, and Locally Advanced or Metastatic Basal Cell Carcinoma.

Target Protein:
Protein smoothened
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NX-1207 DB05493
small molecule

NX-1207 is an investigational new drug for BPH, whose chemical entity and mechanism of action remain undisclosed. Nymox Pharmaceutical Corporation recently completed studies of NX-1207 for treatment of benign prostatic hyperplasia (BPH).

Kategori:
Amino Acids, Peptides, and Proteins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NX-210c DB18209
biotech | CAS: 216682-41-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NXN-188 DB06096
small molecule

NXN-188 is a first-in-class, dual-action small molecule incorporating both neuronal nitric oxide synthase (nNOS) inhibition and 5-HT agonism that is being developed for the treatment of acute migraine.

Target Protein:
Nitric oxide synthase 15-hydroxytryptamine receptor 1B5-hydroxytryptamine receptor 1D
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

NY-ESO-1 peptide vaccine is an investigational cancer immunotherapy. It contains a peptide derived from the cancer-testis antigen (NY-ESO-1).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nylidrin Approved DB06152
small molecule | CAS: 447-41-6

Nylidrin, also known as _buphenine_ belongs to the category of drugs called _vasodilators_, which relax blood vessels and increase blood flow. Nylidrin is a peripheral vasodilator. Some studies show the evidence of improving cognitive impairment in selected i…

Kategori:
2-Amino-1-Phenylethanol DerivativesAdrenergic AgentsAdrenergic Agonists +29
Target Protein:
Interferon alpha/beta receptor 2Voltage-dependent T-type calcium channel subunit alpha-1I
Waktu ParuhDuration of action …
Vol. Distribusi-
Klirens-
Genetik -
Nystatin Approved DB00646
small molecule | CAS: 1400-61-9

Nystatin is a polyene antifungal drug that has broad-spectrum fungicidal and fungistatic activity against a number of yeasts and fungi, most notably _Candida_ species.[L10686] It is one of the most effective antifungal agents synthesized by bacteria, in this …

Kategori:
Alimentary Tract and MetabolismAnti-Infective AgentsAntidiarrheals, Intestinal Antiinflammatory/antiinfective Agents +17
Target Protein:
Ergosterol
Waktu Paruh-
Vol. DistribusiNystatin is not abs…
Klirens-
Genetik -
NYX-2925 DB19149
small molecule | CAS: 2012536-16-0

NYX-2925 is under investigation in clinical trial NCT04146896 (Efficacy and Safety of NYX-2925 in Subjects With Neuropathic Pain Associated With Diabetic Peripheral Neuropathy (DPN)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
4-hydroxy-tetrahydrodipicolinate synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Transaldolase B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NZ-1002 DB17688
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Poly [ADP-ribose] polymerase 1Exotoxin AElongation factor 2 +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Stromelysin-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 11401–11450 dari 16004
Sebelumnya Halaman 229 / 321 Berikutnya