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12560

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9109 (72.5%)
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6912 (55.0%)
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12560 (100.0%)

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Halaman 227 / 252
TC-2216 DB06044
small molecule | CAS: 1159824-71-1

TC-2216 is an investigational novel small molecule that is being developed as an oral treatment for depression and anxiety disorders. TC-2216 showed greater potency than and anti-depressant effects comparable to selective serotonin reuptake inhibitors and tri…

Target Protein:
Neuronal acetylcholine receptor subunit alpha-4Neuronal acetylcholine receptor subunit beta-2
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TC-2696 DB05576
small molecule | CAS: 552302-36-0

Deskripsi belum tersedia.

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TC-5231 DB05333
small molecule

TC-5231 is a small molecule that has been under investigation as an oral treatment for ADHD (Attention Deficit/Hyperactivity Disorder). TC-5231 is mecamylamine hydrochloride, the active ingredient in FDA-approved product, Inversine, but in a lower dose than I…

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TC-6987 DB14854
small molecule | CAS: 1196701-27-5

TC-6987 is under investigation in clinical trial NCT01296087 (TC-6987 for the Treatment of Mild to Moderate Asthma).

Target Protein:
Neuronal acetylcholine receptor subunit alpha-7
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TCB-008 DB18352
biotech

TCB-008 is an Allogeneic CD3+ T lymphocyte ex vivo expanded expressing the gamma delta T-cell receptor.

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TD-0903 DB16463
small molecule | CAS: 2412496-23-0

TD-0903 was investigated in clinical trials for its potential to treat acute lung injury (ALI) associated with COVID-19, including NCT04350736, NCT05091723 (a pharmacokinetics study in healthy participants with supplemental oxygenation), and NCT04402866 (focu…

Kategori:
AzetinesExperimental Unapproved Treatments for COVID-19Heterocyclic Compounds, Fused-Ring +1
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TD-2749 DB05905
small molecule | CAS: 863248-59-3

TD-2749 is selective 5-HT4 agonists discovered by Theravance through the application of multivalent drug design in a drug discovery program dedicated to finding new medicines for GI motility disorders such as chronic constipation, constipation-predominant irr…

Target Protein:
5-hydroxytryptamine receptor 4
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TD101 DB06596
small molecule

TD101, a small interfering RNA (siRNA) designed for the treatment of pachyonychia congenita

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TDI-01 DB19450
small molecule

TDI-01 is a small molecule is being developed by Beijing Tide Pharmaceutical.

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Tea leaf Approved DB10580
biotech

Tea leaf allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract +1
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Tebapivat DB19338
small molecule

Tebapivat is under investigation in clinical trial NCT05490446 (A Study of Tebapivat (AG-946) in Participants With Anemia Due to Lower-risk Myelodysplastic Syndromes (LR-MDS)).

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Tebentafusp Approved DB15283
biotech | CAS: 1874157-95-5

Tebentafusp is a gp100 peptide-HLA-directed CD3 T cell engager.[L39995] It is a bispecific, fusion protein and first-in-class drug of immune-mobilizing monoclonal T cell receptors against cancer (ImmTACs), a recently developed cancer immunotherapy with a nove…

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +6
Target Protein:
Melanocyte protein PMEL
Waktu ParuhThe median terminal…
Vol. DistribusiThe geometric mean …
KlirensThe geometric mean …
Genetik -
small molecule | CAS: 161715-24-8

Deskripsi belum tersedia.

Kategori:
AmidesAnti-Bacterial AgentsAntibacterials for Systemic Use +5
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Tebotelimab DB16685
biotech | CAS: 2245725-04-4

Tebotelimab is under investigation in clinical trial NCT04082364 (Combination Margetuximab, INCMGA00012, MGD013, and Chemotherapy Phase 2/3 Trial in HER2+ Gastric/gej Cancer (MAHOGANY)).

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Tecadenoson DB04954
small molecule | CAS: 204512-90-3

Tecadenoson is a novel selective A1 adenosine receptor agonist that is currently being evaluated for the conversion of paroxysmal supraventricular tachycardia (PSVT) to sinus rhythm. It is being developed by CV Therapeutics, Inc.

Kategori:
Heterocyclic Compounds, Fused-RingNeurotransmitter AgentsNucleic Acids, Nucleotides, and Nucleosides +7
Target Protein:
Adenosine receptor A1
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Tecarfarin DB12823
small molecule | CAS: 867257-26-9

Tecarfarin has been used in trials studying the prevention of Thrombosis and Thromboembolism.

Kategori:
Acids, CarbocyclicBenzene DerivativesBenzopyrans +5
Target Protein:
Vitamin K epoxide reductase complex subunit 1
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Tecastemizole DB06457
small molecule | CAS: 75970-99-9

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Histamine H1 receptorVoltage-gated inwardly rectifying potassium channel KCNH2
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Teceleukin DB15389
biotech | CAS: 136279-32-8

Teceleukin is under investigation in clinical trial NCT03610490 (Autologous Tumor Infiltrating Lymphocytes MDA-TIL in Treating Patients With Recurrent or Refractory Ovarian Cancer, Osteosarcoma, or Pancreatic Ductal Adenocarcinoma).

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsAnalgesics, Non-Narcotic +12
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Tecemotide DB12568
biotech | CAS: 221214-84-2

Tecemotide has been used in trials studying the treatment of Prostate Cancer and Carcinoma, Non-Small-Cell Lung.

Kategori:
Amino Acids, Peptides, and ProteinsBiological ProductsCarbohydrates +6
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biotech | CAS: 154361-49-6

Reduced Fab fragment of the murine IgG1 monoclonal antibody IMMU-4 (also called NP-4) with specificity for carcinoembryonic antigen (CEA) covalently labeled with Technitium 99. The molecule has a molecular weight of ~54,000 Daltons.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +9
Target Protein:
Cell adhesion molecule CEACAM1
Waktu ParuhApproximately 1 hour
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small molecule | CAS: 374107-43-4

99mTc-Ciprofloxacin is a new formulation of ciprofloxacin (INFECTON), being investigated as a radioimaging agent for the potential diagnosis of infection, including fever of unknown origin, osteomyelitis, wound infection, abdominal abscess, pneumonia, appendi…

Kategori:
4-QuinolonesAnti-Bacterial AgentsCytochrome P-450 CYP1A2 Inhibitors +9
Target Protein:
DNA gyrase subunit BDNA topoisomerase 2-beta
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biotech

Technetium Tc-99m epratuzumab is under investigation in clinical trial NCT00003337 (Radiolabeled Monoclonal Antibody in the Detection and Staging of Patients With Non-Hodgkin's Lymphoma).

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Technetium Tc-99m etidronate Approved DB09411
small molecule | CAS: 63347-65-9

Deskripsi belum tersedia.

Kategori:
Compounds used in a research, industrial, or household settingDiagnostic RadiopharmaceuticalsDiagnostic Uses of Chemicals +6
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small molecule | CAS: 72950-39-1

Deskripsi belum tersedia.

Kategori:
Diagnostic RadiopharmaceuticalsHepatic and Reticulo Endothelial SystemTechnetium (99Mtc) Compounds
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Technetium Tc-99m mebrofenin Approved DB09137
small molecule | CAS: 1415247-71-0

Technetium Tc 99m Mebrofenin is a diagnostic radiopharmaceutical composed of diisopropyl-iminodiacetic acid (DISIDA) attached to a technetium-99m ion. Following intravenous injection, single photon emission computer tomography (SPECT) imaging of the liver o…

Kategori:
AminesAmino AcidsAmino Acids, Peptides, and Proteins +14
Waktu ParuhTechnetium Tc 99m d…
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Technetium Tc-99m medronate Approved DB09138
small molecule | CAS: 121524-79-6

Technetium (99mTc) medronic acid is a pharmaceutical product used in nuclear medicine imaging. It is composed of a technetium ion complexed with medronic acid, a type of bisphosphonate. Like other bisphosphonates used in the treatment of osteoporosis, medroni…

Kategori:
Compounds used in a research, industrial, or household settingDiagnostic RadiopharmaceuticalsDiagnostic Uses of Chemicals +11
Waktu ParuhTechnetium Tc-99m d…
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small molecule | CAS: 165942-79-0

Technetium Tc-99m nofetumomab merpentan (Tc-99m nm) consists of a Fab fragment of an IgG2b of the pancarcinoma murine antibody NR-LU-10.[A32115] The NR-LU-10 antibody is directed against a 40 kDa glycoprotein antigen expressed in a variety of cancers and some…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Target Protein:
Epithelial cell adhesion moleculeB-lymphocyte antigen CD20
Waktu ParuhThe radioactive hal…
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Technetium Tc-99m oxidronate Approved DB09139
small molecule | CAS: 72945-61-0

Technetium Tc-99m oxidronate, also known as 99mTc-methylene diphosphonate, is a radiopharmaceutical agent. A radiopharmaceutical is defined as a medicinal formulation containing radioisotopes that are used in major clinical areas for diagnosis and/or therapy.…

Kategori:
Diagnostic RadiopharmaceuticalsDrugs that are Mainly Renally ExcretedOrganometallic Compounds +6
Waktu ParuhThe elimination of …
Vol. DistribusiThe distribution of…
KlirensDuring the first 24…
Genetik -
small molecule | CAS: 52997-54-3

A radionuclide imaging agent used primarily in scintigraphy or tomography of the heart to evaluate the extent of the necrotic myocardial process. It has also been used in noninvasive tests for the distribution of organ involvement in different types of amyloi…

Kategori:
AcidsAcids, NoncarboxylicCompounds used in a research, industrial, or household setting +17
Target Protein:
HydroxyapatiteAmorphous calcium phosphate
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Technetium Tc-99m sestamibi Approved DB09161
small molecule | CAS: 109581-73-9

Technetium Tc-99m sestamibi (commonly sestamibi) is a pharmaceutical agent used in nuclear medicine imaging. The drug is a coordination complex consisting of the radioisotope technetium-99m bound to six methoxyisobutylisonitrile (MIBI) ligands, hence the name…

Kategori:
Compounds used in a research, industrial, or household settingDiagnostic RadiopharmaceuticalsDiagnostic Uses of Chemicals +10
Waktu ParuhTechnetium Tc 99m d…
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KlirensThe effective half-…
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Technetium Tc-99m succimer Approved DB09436
small molecule | CAS: 65438-08-6

Technetium Tc-99m (<sup>99m</sup>Tc) succimer, also known as technetium Tc-99m dimercaptosuccinic acid (DMSA),[A245643] is a radioactive diagnostic agent used to evaluate functional renal tissue and tubular function in patients with renal parenchymal disorder…

Kategori:
Acids, AcyclicCompounds used in a research, industrial, or household settingDiagnostic Radiopharmaceuticals +14
Waktu ParuhTechnetium Tc-99m d…
Vol. DistribusiThere is no informa…
KlirensThere is no informa…
Genetik -
small molecule | CAS: 127455-27-0

Technetium Tc-99m tetrofosmin is a drug used in nuclear myocardial perfusion imaging. The radioisotope, technetium-99m, is chelated by two 1,2-bis[di-(2-ethoxyethyl)phosphino]ethane ligands which belong to the group of diphosphines and which are referred to a…

Kategori:
Compounds used in a research, industrial, or household settingDiagnostic RadiopharmaceuticalsDiagnostic Uses of Chemicals +7
Waktu ParuhTechnetium-99m tetr…
Vol. DistribusiReports have shown …
KlirensTechnetium-99m tetr…
Genetik -
small molecule | CAS: 1333204-77-5

Deskripsi belum tersedia.

Kategori:
Organometallic Compounds
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Teclistamab Approved DB16655
biotech | CAS: 2119595-80-9

Teclistamab is an IgG4-PAA bispecific antibody that targets the CD3 receptor expressed on the surface of T cells and B cell maturation antigen (BCMA) expressed on malignant multiple myeloma cells.[A253587] Teclistamab consists of an anti-BCMA arm and an anti-…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntineoplastic Agents +8
Target Protein:
T-cell surface glycoprotein CD3Tumor necrosis factor receptor superfamily member 17
Waktu ParuhBased on non-compar…
Vol. DistribusiThe mean (CV%) volu…
KlirensTeclistamab exhibit…
Genetik -
Teclozan DB13205
small molecule | CAS: 5560-78-1

Teclozan is an antiprotozoal agent employed typically as a therapy to treat protozoan infections.

Kategori:
AminesAntiparasitic Products, Insecticides and RepellentsAntiprotozoals +3
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Tecovirimat Approved DB12020
small molecule | CAS: 869572-92-9

The World Health Organization declared smallpox, a contagious and sometimes fatal infectious disease, eradicated in 1980. However, there have been longstanding concerns that smallpox may be used as a bioweapon.[A35133,L3614] Tecovirimat is an antiviral drug t…

Kategori:
Acids, CarbocyclicAmidesAnti-Infective Agents +27
Target Protein:
Envelope protein F13
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe clearance rate …
Genetik -
Tedatioxetine DB12641
small molecule | CAS: 508233-95-2

Tedatioxetine has been used in trials studying the treatment of Major Depressive Disorder.

Target Protein:
5-hydroxytryptamine receptor 2C
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Tedisamil DB06200
small molecule | CAS: 90961-53-8

Tedisamil (planned trade name Pulzium) is an investigational drug for atrial fibrillation and atrial flutter. It is currently being developed by Solvay and is currently under regulatory review by the United States Food and Drug Administration.

Kategori:
Antiarrhythmic agentsAntiarrhythmics, Class IIICardiac Therapy +7
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Tedizolid Approved DB14569
small molecule | CAS: 856866-72-3

Drug-resistant bacteria, such as methicillin-resistant _Staphylococcus aureus_, vancomycin-resistant _Enterococcus faecium_, and penicillin-resistant _Streptococcus penumoniae_, represent a massive public health threat.[A199086, A199131] Tedizolid is a member…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibacterials for Systemic Use +5
Target Protein:
23S ribosomal RNA
Waktu ParuhTedizolid has a hal…
Vol. DistribusiThe volume of distr…
KlirensTedizolid has an ap…
Genetik -
Tedizolid phosphate Approved DB09042
small molecule | CAS: 856867-55-5

Drug-resistant bacteria, such as methicillin-resistant _Staphylococcus aureus_, vancomycin-resistant _Enterococcus faecium_, and penicillin-resistant _Streptococcus penumoniae_, represent a massive public health threat.[A199086, A199131] Tedizolid is a member…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntidepressive Agents +10
Target Protein:
23S ribosomal RNA
Waktu ParuhTedizolid has a hal…
Vol. DistribusiThe volume of distr…
KlirensTedizolid has an ap…
Genetik -
Tefibazumab DB16378
biotech | CAS: 521079-87-8

Tefibazumab is under investigation in clinical trial NCT00198289 (Aurexis® in Cystic Fibrosis Subjects Chronically Colonized With Staphylococcus Aureus in Their Lungs).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
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biotech | CAS: 2143580-10-1

Tefidsogene civaparvovec, formerly known as SB-913, is an investigational therapy for genome editing. It consists of an adeno-associated virus (AAV) type 2/6 vector and a zinc finger nuclease (ZFN) system that inserts a correct copy of the Iduronate 2-Sulfata…

Kategori:
Adeno-associated Viral Vector Therapies
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Tefinostat DB15321
small molecule | CAS: 914382-60-8

Tefinostat is under investigation in clinical trial NCT02759601 (Dose Escalation Trial of Tefinostat for Cancer Associated Inflamation in Hepatocellular Carcinoma (HCC)).

Kategori:
AmidesAminesAniline Compounds +4
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Tegafur Approved DB09256
small molecule | CAS: 17902-23-7

Tegafur (INN, BAN, USAN) is a prodrug of [DB00544] (5-FU), an antineoplastic agent used as the treatment of various cancers such as advanced gastric and colorectal cancers. It is a pyrimidine analogue used in combination therapies as an active chemotherapeuti…

Kategori:
AntimetabolitesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +22
Target Protein:
Thymidylate synthase
Gen Terkait:
DPYD DPYD DPYD +4
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensNo pharmacokinetic …
Genetik 7 Varian
Tegafur-uracil Approved DB09327
small molecule | CAS: 74578-38-4

Tegafur-uracil is an anti-tumor compound containing tegafur (1-(2-tetrahydrofuryl)-5-fluorouracil) and uracil in a molar ratio of 1:4. It was developed as an anti-cancer therapy by Taiho Pharmaceutical Co Ltd.[A32073] It is approved in different countries but…

Kategori:
Cytochrome P-450 CYP2A6 SubstratesCytochrome P-450 Substrates
Target Protein:
Dihydropyrimidine dehydrogenase [NADP(+)]Thymidylate synthaseRNA +1
Waktu ParuhThe presence of ura…
Vol. DistribusiThe volume of distr…
KlirensThe reported cleara…
Genetik -
Tegaserod Approved DB01079
small molecule | CAS: 145158-71-0

Novartis' brand name Zelnorm (tegaserod) had originally received approval from the US FDA in 2002 for the treatment of irritable bowel syndrome with constipation (IBS-C).[L5918,F4229] It was, however, voluntarily withdrawn from widespread use in the US market…

Kategori:
Alimentary Tract and MetabolismAntidepressive AgentsBCRP/ABCG2 Substrates +25
Target Protein:
5-hydroxytryptamine receptor 45-hydroxytryptamine receptor 2C5-hydroxytryptamine receptor 2A +1
Waktu ParuhThe mean terminal e…
Vol. DistribusiAlthough tegaserod …
KlirensAlthough tegaserod …
Genetik -
Tegavivint DB17109
small molecule | CAS: 1227637-23-1

Deskripsi belum tersedia.

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Tegileridine DB18988
small molecule | CAS: 2095345-66-5

Tegileridine is under investigation in clinical trial NCT06458400 (To Evaluate the Efficacy and Safety of Tegileridine and Oliceridine Injections in the Treatment of Postoperative Pain).

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Tegobuvir DB11852
small molecule | CAS: 1000787-75-6

Tegobuvir has been investigated for the treatment of Hepatitis C, Chronic.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Genome polyprotein
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Tegoprazan DB16690
small molecule | CAS: 942195-55-3

Tegoprazan (also known as CJ-12420) is a novel therapeutic developed by CJ Healthcare Corp for treating acid-related gastrointestinal diseases.[A234215, A234220] This drug is a potent and high-selective potassium-competitive acid blocker (P-CAB) with a fast o…

Kategori:
Alimentary Tract and MetabolismDrugs for Acid Related DisordersDrugs for Peptic Ulcer and Gastro-Oesophageal Reflux Disease (Gord) +2
Target Protein:
Sodium/Potassium Transporting ATPase
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