Hasil Filter

12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
Referensi
12560 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (12560)

Halaman 226 / 252
Tanfanercept DB19142
biotech | CAS: 2119738-70-2

Tanfanercept is under investigation in clinical trial NCT06400589 (A Study to Evaluate the Efficacy and Safety of Tanfanercept (HL036) in Dry Eye Disease).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Taniborbactam DB16338
small molecule | CAS: 1613267-49-4

Taniborbactam is under investigation in clinical trial NCT03840148 (Safety and Efficacy Study of Cefepime/vnrx-5133 in Patients With Complicated Urinary Tract Infections).

Kategori:
AcidsAcids, NoncarboxylicBoron Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Taniraleucel DB18311
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tannic acid Approved DB09372
small molecule | CAS: 1401-55-4

Tannic acid is a polyphenolic compound. It is a type of the commercially available tannins. It acts as a weak acid. Tannic acid is found in the nutgalls formed by insects on twigs of certain oak trees (Quercus infectoria and other Quercus species). It is remo…

Kategori:
Benzene DerivativesBiopolymersCompounds used in a research, industrial, or household setting +4
Target Protein:
Anoctamin-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tanomastat DB06276
small molecule | CAS: 179545-77-8

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAntineoplastic AgentsBenzene Derivatives +1
Target Protein:
72 kDa type IV collagenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tanshinone I DB16886
small molecule | CAS: 568-73-0

Deskripsi belum tersedia.

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAnti-Infective Agents +16
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tantalum DB12859
small molecule | CAS: 7440-25-7

Tantalum has been investigated for the treatment and prevention of Osteoarthritis, Knee Osteoarthritis, Intraoperative Bleeding, and Adolescent Idiopathic Scoliosis.

Kategori:
ElementsMetalsMetals, Heavy +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tanzisertib DB11798
small molecule | CAS: 899805-25-5

Tanzisertib has been used in trials studying the treatment of Fibrosis, Discoid Lupus, Pulmonary Fibrosis, Interstitial Lung Disease, and Lung Diseases, Interstitial, among others.

Kategori:
AlcoholsCarbon RadioisotopesCyclohexanes +6
Target Protein:
Mitogen-activated protein kinase 8Mitogen-activated protein kinase 9Mitogen-activated protein kinase 10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tapencarium DB17821
small molecule

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingIndoles
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tapentadol Approved DB06204
small molecule | CAS: 175591-23-8

Tapentadol is a centrally-acting synthetic analgesic with a dual mechanism of action. It is a mu-opioid receptor agonist that also inhibits norepinephrine reuptake.[A260721, A36596] Tapentadol was first approved by the FDA on November 20, 2008. The extende…

Kategori:
Adrenergic AgentsAdrenergic Uptake InhibitorsAnalgesics +25
Target Protein:
Mu-type opioid receptorSodium-dependent noradrenaline transporterKappa-type opioid receptor +2
Waktu ParuhThe terminal half-l…
Vol. DistribusiTapentadol is widel…
KlirensThe total clearance…
Genetik -
Tapinarof Approved DB06083
small molecule | CAS: 79338-84-4

Tapinarof is a novel, first-in-class, small-molecule AhR agonist that is indicated for the treatment of adult psoriasis. It is available as a topical cream to be applied to the affected area once daily.[L41845, A248790] Tapiranof was first discovered as a met…

Kategori:
AntipsoriaticsAntipsoriatics for Topical UseAryl Hydrocarbon Receptor Agonist +11
Target Protein:
Aryl hydrocarbon receptor
Waktu ParuhDue to the insuffic…
Vol. DistribusiThe Vss of tapinaro…
Klirens-
Genetik -
Taprenepag DB12623
small molecule | CAS: 752187-80-7

Taprenepag has been used in trials studying the treatment of Ocular Hypertension and Glaucoma, Open-Angle.

Kategori:
Acids, AcyclicAmidesFatty Acids +5
Target Protein:
Prostaglandin E2 receptor EP2 subtype
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tarafenacin DB18810
small molecule | CAS: 385367-47-5

Deskripsi belum tersedia.

Target Protein:
Muscarinic acetylcholine receptor M3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Taranabant DB06624
small molecule | CAS: 701977-09-5

Deskripsi belum tersedia.

Kategori:
Cannabinoid Receptor AgonistsCannabinoids and similarsHormones +2
Target Protein:
Cannabinoid receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Taraxacum officinale pollen Approved DB10755
biotech

Taraxacum officinale pollen is the pollen of the Taraxacum officinale plant. Taraxacum officinale pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tarazepide DB06435
small molecule | CAS: 141374-81-4

Deskripsi belum tersedia.

Kategori:
BenzazepinesHeterocyclic Compounds, Fused-Ring
Target Protein:
Cholecystokinin receptor type A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2411896-53-0

Tarcocimab tedromer is under investigation in clinical trial NCT06270836 (A Study to Evaluate the Efficacy and Safety of Tarcocimab Tedromer Compared With Sham Treatment in Participants With Moderately Severe to Severe Non-proliferative Diabetic Retinopathy (…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tarenflurbil DB05289
small molecule | CAS: 51543-40-9

Tarenflurbil is an investigational drug that was studied in patients with mild Alzheimer's disease. It is a selective amyloid lowering agent (SALA) that reduces levels of the toxic peptide amyloid beta 42 (A?42) in cultured human cells and in animal models. A…

Kategori:
Acids, AcyclicAnalgesicsAnalgesics, Non-Narcotic +11
Target Protein:
Gamma-secretase subunit APH-1BNicastrinGamma-secretase subunit APH-1A +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tarextumab DB12104
biotech | CAS: 1359940-55-8

Tarextumab has been used in trials studying the treatment of Solid Tumors, Stage IV Pancreatic Cancer, and Stage IV Small Cell Lung Cancer.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Taribavirin DB06408
small molecule | CAS: 119567-79-2

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAntiviral AgentsNucleic Acids, Nucleotides, and Nucleosides +3
Target Protein:
Inosine-5'-monophosphate dehydrogenase 1DNARNA-directed RNA polymerase L +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tarlatamab Approved DB17256
biotech | CAS: 2307488-83-9

Tarlatamab is a first-in-class T-cell engager used to treat extensive-stage small cell lung cancer.[L50748] It is a bispecific monoclonal antibody that targets CD3 expressed on the surface of T-cells and delta-like ligand 3 (DLL3), an inhibitory ligand that s…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalBispecific Monoclonal Antibodies +5
Target Protein:
Delta-like protein 3T-cell surface glycoprotein CD3
Waktu ParuhThe median terminal…
Vol. DistribusiAt steady-state, th…
KlirensThe systemic cleara…
Genetik -
Tarloxotinib DB14944
small molecule | CAS: 1636938-13-0

Tarloxotinib is under investigation in clinical trial NCT03743350 (NSCLC Exon 20 or HER2-activating Mutations).

Target Protein:
Receptor tyrosine-protein kinase erbB-2Epidermal growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TAS-106 DB06656
small molecule | CAS: 180300-43-0

TAS-106 is a new nucleoside antimetabolite. TAS-106 has demonstrated strong antitumor activity without serious toxicity in nude rat models bearing human tumours [A31693].

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleosidesPyrimidine Nucleosides +2
Target Protein:
DNA-directed RNA polymerase subunit betaDNA-directed RNA polymerase subunit beta'
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TAS-108 DB05966
small molecule | CAS: 229634-97-3

Deskripsi belum tersedia.

Target Protein:
Estrogen receptorEstrogen receptor beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TAS-116 DB14876
small molecule | CAS: 1260533-36-5

TAS-116 is under investigation in clinical trial NCT02965885 (A Study of TAS-116 in Patients With Solid Tumors).

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +1
Target Protein:
Heat shock protein HSP 90-beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TAS-117 DB15054
small molecule | CAS: 1402602-94-1

TAS-117 is under investigation in clinical trial NCT03017521 (K-BASKET, TAS-117, PI3K/AKT Gene Aberration).

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tasadenoturev DB17178
biotech | CAS: 1448774-00-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Taselisib DB12108
small molecule | CAS: 1282512-48-4

Taselisib has been used in trials studying the treatment and basic science of LYMPHOMA, Breast Cancer, Ovarian Cancer, Solid Neoplasm, and HER2/Neu Negative, among others.

Kategori:
Antineoplastic AgentsAzepinesPhosphatidylinositol 3-Kinases, antagonists & inhibitors
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoformPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tasisulam DB11941
small molecule | CAS: 519055-62-0

Tasisulam has been used in trials studying the treatment and basic science of Melanoma, Lymphoma, Solid Tumors, Breast Cancer, and Ovarian Cancer, among others.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tasonermin Approved DB11626
biotech | CAS: 94948-59-1

Tasonermin is recombinant soluble form tumor necrosis factor α produced via _Escherichia coli_ cell culture. It was approved for use by the European Medicines Agency in April of 1999 for use as an adjunt to surgery for the subsequent removal of the tum…

Kategori:
Adjuvants, ImmunologicAntineoplastic and Immunomodulating Agents
Target Protein:
Tumor necrosis factor receptor superfamily member 1ATumor necrosis factor receptor superfamily member 1B
Waktu ParuhTasonermin has a te…
Vol. DistribusiThe estimated volum…
KlirensClearance was estim…
Genetik -
Tasosartan DB01349
small molecule | CAS: 145733-36-4

Tasosartan is a long-acting angiotensin II (AngII) receptor blocker. Its long duration of action has been attributed to its active metabolite enoltasosartan. It is used to treat patients with essential hypertension.

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing hyperkalemiaAngiotensin II receptor blockers (ARBs), plain +4
Target Protein:
Type-1 angiotensin II receptorType-2 angiotensin II receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Taspoglutide DB14027
small molecule | CAS: 275371-94-3

Taspoglutide is a pharmaceutical drug, a glucagon-like peptide-1 agonist (GLP-1 agonist), under investigation for treatment of type 2 diabetes being codeveloped by Ipsen and Roche. In September 2010 Roche halted Phase III clinical trials due to incidences of …

Kategori:
Amino Acids, Peptides, and ProteinsBlood Glucose Lowering AgentsGastrointestinal Hormones +5
Target Protein:
Glucagon-like peptide 1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tasquinimod DB05861
small molecule | CAS: 254964-60-8

The quinoline-3-carboxamide anti-angiogenic agent, tasquinimod, enhances the anti-prostate cancer efficacy of androgen ablation and taxotere without effecting serum PSA directly in human xenografts

Kategori:
Heterocyclic Compounds, Fused-RingQuinolines
Target Protein:
Protein S100-A9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Taurine Approved DB01956
small molecule | CAS: 107-35-7

Taurine, whose chemical name is 2-aminoethanesulfonic acid, is one of the most abundant amino acids in several organs. It plays important role in essential biological processes.[A31396] This conditional amino acid can be either be manufactured by the body or …

Kategori:
AlkanesAlkanesulfonic AcidsAmino Acids +5
Target Protein:
Glutamate receptor ionotropic, NMDA 2BGlycine receptor subunit betaGlycine receptor subunit alpha-2 +6
Waktu ParuhOral administration…
Vol. DistribusiThe distribution of…
KlirensThe clearance rate …
Genetik -
small molecule | CAS: 516-35-8

Taurochenodeoxycholic acid is an experimental drug that is normally produced in the liver. Its physiologic function is to emulsify lipids such as cholesterol in the bile. As a medication, taurochenodeoxycholic acid reduces cholesterol formation in the liver, …

Kategori:
AlkanesAlkanesulfonic AcidsBile Acids and Salts +18
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Taurolidine Approved DB12473
small molecule | CAS: 19388-87-5

Taurolidine is an antimicrobial used for the prevention of catheter-related infections. It is a derivative of the amino acid [taurine]. It was first synthesized in the 1970s and was originally used as a prophylactic against intraperitoneal bacterial infect…

Kategori:
AlkanesAlkanesulfonic AcidsAnti-Infective Agents +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 75018-71-2

Deskripsi belum tersedia.

Kategori:
Acids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tauroursodeoxycholic acid Approved DB08834
small molecule | CAS: 14605-22-2

Tauroursodeoxycholic acid, also known as ursodoxicoltaurine, is a highly hydrophilic tertiary bile acid [A249070] that is produced in humans at a low concentration.[A249070] It is a taurine conjugate of [ursodeoxycholic acid] [A249065] with comparable therape…

Kategori:
Alimentary Tract and MetabolismBile acids and derivativesBile Acids and Salts +10
Target Protein:
Integrin alpha-5
Waktu Paruh-
Vol. DistribusiThere is evidence t…
Klirens-
Genetik -
Tavaborole Approved DB09041
small molecule | CAS: 174671-46-6

Tavaborale is a novel, boron-based topical antifungal medication for the treatment of onychomycosis, a fungal infection of the nail and nail bed due to *Trichophyton rubrum* or *Trichophyton mentagrophytes* infection. Tavaborole functions by inhibiting Leucyl…

Kategori:
Anti-Infective AgentsAntifungal AgentsAntifungals for Dermatological Use +4
Target Protein:
leucine--tRNA ligase
Waktu Paruh28.5 hr
Vol. Distribusi-
Klirens-
Genetik -
Tavapadon DB14899
small molecule | CAS: 1643489-24-0

Tavapadon is under investigation in clinical trial NCT02262767 (A Study to Investigate the Safety, Tolerability, and Pharmacokinetics of PF-06649751 Co-administered With Trimethobenzamide Hydrochloride in Healthy Subjects).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tavilermide DB12441
small molecule | CAS: 263251-78-1

Tavilermide has been investigated for the treatment of Dry Eye Syndromes.

Target Protein:
High affinity nerve growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1971880-37-1

Tavokinogene telseplasmid consists of a DNA Plasmid Vector Encoding IL-12.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tavolixizumab DB15042
biotech | CAS: 1635395-25-3

Tavolixizumab is under investigation in clinical trial NCT02318394 (A Phase 1 Study of MEDI0562 in Adult Subjects With Selected Advanced Solid Tumors).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Taxifolin DB02224
small molecule | CAS: 480-18-2

Deskripsi belum tersedia.

Kategori:
Agents that produce hypertensionAnalgesicsAnalgesics, Non-Narcotic +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tazemetostat Approved DB12887
small molecule | CAS: 1403254-99-8

Tazemetostat is a methyltransferase inhibitor used to treat metastatic or locally advanced epithelioid sarcoma not eligible for complete resection.[L11476] Tazemetostat was first named in literature as EPZ-6438.[A190363] Tazemetaostat was granted FDA appro…

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +16
Target Protein:
Histone-lysine N-methyltransferase EZH2Histone-lysine N-methyltransferase EZH1
Waktu ParuhTazemetostat has a …
Vol. DistribusiTazemetostat has a …
KlirensTazemetostat has an…
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Beta-lactamase SHV-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TB-402 DB06050
biotech

TB-402 is a human antibody binding to Factor VIII, which plays a crucial role in the coagulation of the blood. It is expected to be developed as a potential treatment to prevent blood clot formation in connection with certain types of heart arrhythmia, such a…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Target Protein:
Coagulation factor VIII
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TBA-7371 DB16243
small molecule | CAS: 1494675-86-3

TBA-7371 is under investigation in clinical trial NCT04176250 (Early Bactericidal Activity of TBA-7371 in Pulmonary Tuberculosis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TBC-3711 DB05407
small molecule | CAS: 349453-49-2

TBC3711 is a next-generation endothelin antagonist that is being studied through oral and intravenous formulations by Encysive Pharmaceuticals.

Kategori:
Endothelin A Receptor AntagonistsEndothelin Receptor AntagonistsSulfur Compounds
Target Protein:
Endothelin-1 receptorEndothelin-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TBI-223 DB18911
small molecule | CAS: 2071265-08-0

TBI-223 is under investigation in clinical trial NCT06192160 (Trial of Novel Regimens for the Treatment of Pulmonary Tuberculosis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 11251–11300 dari 12560
Sebelumnya Halaman 226 / 252 Berikutnya