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13591

Total database: 17430
Struktur (SMILES)
10177 (74.9%)
Target
7625 (56.1%)
Genomik
104 (0.8%)
Referensi
13591 (100.0%)

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Hasil Pencarian (13591)

Halaman 226 / 272
Rocacetrapib DB15437
small molecule | CAS: 1402796-27-3

Rocacetrapib is under investigation in clinical trial NCT02156544 (Study to Investigate the Safety/Tolerability and Pharmacokinetics/Pharmacodynamics of CKD-519).

Kategori:
Hydrocarbons, Halogenated
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rocaglamide DB15495
small molecule | CAS: 84573-16-0

Rocaglamide, also referred to as rocaglamide-A, is the eponymous member of a class of anti-cancer phytochemicals known as rocaglamides.[A186760] Rocaglamides are secondary metabolites of the plant genus _Aglaia_, and extracts of the plant have traditionally b…

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Prohibitin 1Transcription factor RelBNuclear factor NF-kappa-B p100 subunit +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2253753-17-0

Rocakinogene sifuplasmid is under investigation in clinical trial NCT03491683 (INO-5401 and INO-9012 Delivered by Electroporation (EP) in Combination With Cemiplimab (REGN2810) in Newly-diagnosed Glioblastoma (GBM)).

Kategori:
Amino Acids, Peptides, and ProteinsAntigensBiological Factors +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rocapuldencel-T DB17588
biotech

Rocapuldencel-T is an autologous dendritic cell immunotherapy that was investigated in NCT02662634 (A Safety and Feasibility Study of AGS-003-LNG for the Treatment of Stage 3 Non Small Cell Lung Cancer).

Kategori:
Autologous Cellular Immunotherapy
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rocatinlimab DB18809
biotech | CAS: 2431972-52-8

Rocatinlimab is a subcutaneously administered anti-OX40 antibody developed for the treatment of moderate-to-severe atopic dermatitis. In clinical trials, it has shown significant efficacy and safety compared to a placebo. The drug works by targeting the OX40 …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Target Protein:
Tumor necrosis factor receptor superfamily member 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rocbrutinib DB19445
small molecule | CAS: 2485861-07-0

Rocbrutinib is under investigation in clinical trial NCT05716087 (A Study of Rocbrutinib in Participants With Relapse or Refractory Mantle Cell Lymphoma).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rociletinib DB11907
small molecule | CAS: 1374640-70-6

Rociletinib has been used in trials studying the treatment and prevention of Nonsmall Cell Lung Cancer, Non-small Cell Lung Cancer, and Locally Advanced or Metastatic Non-small Cell Lung Cancer.

Kategori:
Acids, AcyclicAcrylatesAmides +4
Target Protein:
Epidermal growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rociverine DB13581
small molecule | CAS: 53716-44-2

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAgents producing tachycardiaAlimentary Tract and Metabolism +9
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M3 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rocuronium Approved DB00728
small molecule | CAS: 143558-00-3

Rocuronium (rapid onset-curonium) is a desacetoxy analogue of vecuronium with a more rapid onset of action. It is an aminosteroid non-depolarizing neuromuscular blocker or muscle relaxant used in modern anaesthesia, to facilitate endotracheal intubation and t…

Kategori:
Agents producing tachycardiaAndrostanesAndrostanols +16
Target Protein:
Neuronal acetylcholine receptor subunit alpha-2Muscarinic acetylcholine receptor M25-hydroxytryptamine receptor 3A
Waktu ParuhThe rapid distribut…
Vol. Distribusi* 0.3 L/kg [3 to <1…
Klirens* 0.25 L/kg/hr [Adu…
Genetik -
Rodatristat DB18478
small molecule | CAS: 1673568-73-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1673571-51-1

Deskripsi belum tersedia.

Target Protein:
Tryptophan 5-hydroxylase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rofecoxib Approved DB00533
small molecule | CAS: 162011-90-7

Rofecoxib is used for the treatment of osteoarthritis, rheumatoid arthritis, acute pain in adults, and primary dysmenorrhea, as well as acute treatment of migraine attacks with or without auras. Rofecoxib is a solid. This compound belongs to the stilbenes. Th…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +29
Target Protein:
Prostaglandin G/H synthase 2Elastin
Waktu Paruh17 hours
Vol. Distribusi-
Klirens-
Genetik -
Roflumilast Approved DB01656
small molecule | CAS: 162401-32-3

Roflumilast is a highly selective phosphodiesterase-4 (PDE4) inhibitor.[A251385] PDE4 is a major cyclic-3',5?-adenosinemonophosphate (cyclic AMP, cAMP)-metabolizing enzyme [L37564] expressed on nearly all immune and pro-inflammatory cells, in addition to stru…

Kategori:
Acids, CarbocyclicAgents to Treat Airway DiseaseAmides +17
Target Protein:
cAMP-specific 3',5'-cyclic phosphodiesterase 4 (PDE4)
Waktu ParuhFollowing oral admi…
Vol. DistribusiFollowing a single …
KlirensPlasma clearance of…
Genetik -
Rogaratinib DB15078
small molecule | CAS: 1443530-05-9

Rogaratinib is under investigation in clinical trial NCT03762122 (Rogaratinib in Patients With Advanced Pretreated Squamous-cell Non-small Cell Lung Cancer (SQCLC)).

Kategori:
Sulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Roginolisib DB18088
small molecule | CAS: 1305267-37-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rokitamycin DB13409
small molecule | CAS: 74014-51-0

Deskripsi belum tersedia.

Kategori:
Anti-Bacterial AgentsAntibacterials for Systemic UseAntiinfectives for Systemic Use +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rolapitant Approved DB09291
small molecule | CAS: 552292-08-7

Rolapitant is a potent, highly selective, long-acting Neurokinin-1 (NK-1) receptor antagonist approved for the prevention of delayed chemotherapy-induced nausea and vomiting (CINV) in adults. Delayed-phase CINV typically occurs >24 hours after chemotherapy tr…

Kategori:
Alimentary Tract and MetabolismAntiemetics and AntinauseantsBCRP/ABCG2 Inhibitors +11
Target Protein:
Substance-P receptor
Waktu ParuhMean terminal half …
Vol. Distribusi460 L
Klirens0.96 L/hour
Genetik -
Roledumab DB16317
biotech | CAS: 1174008-79-7

Roledumab is under investigation in clinical trial NCT02287896 (Pharmacokinetics and Safety of Roledumab in Rhd-negative Pregnant Women Carrying an Rhd-positive Foetus).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rolicyclidine DB01549
small molecule | CAS: 2201-39-0

Rolicyclidine (PCPy) is classified as a dissociative anesthetic agent. It also has hallucinogenic and sedative properties. Because of its pharmacodynamic similarity to the drug phencyclidine (PCP), rolicyclidine was added to the Schedule I list of illegal dr…

Kategori:
Piperidines
Target Protein:
Glutamate receptor ionotropic, NMDA 3AD(2) dopamine receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rolipram DB01954
small molecule | CAS: 61413-54-5

A phosphodiesterase inhibitor with antidepressant properties.

Kategori:
Antidepressive AgentsCentral Nervous System AgentsCentral Nervous System Depressants +6
Target Protein:
cGMP-specific 3',5'-cyclic phosphodiesterase3',5'-cyclic-AMP phosphodiesterase 4AcAMP-specific 3',5'-cyclic phosphodiesterase 4 (PDE4) +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rolitetracycline Approved DB01301
small molecule | CAS: 751-97-3

A pyrrolidinylmethyl tetracycline.

Kategori:
Agents that produce neuromuscular block (indirect)Anti-Bacterial AgentsAnti-Infective Agents +4
Target Protein:
30S ribosomal protein S916S ribosomal RNA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rolofylline DB12670
small molecule | CAS: 136199-02-5

Rolofylline is under clinical development by pharmaceutical company NovaCardia for the treatment of congestive heart failure.

Kategori:
AlkaloidsDiureticsHeterocyclic Compounds, Fused-Ring +3
Target Protein:
Adenosine receptor A1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Roluperidone DB13080
small molecule | CAS: 359625-79-9

Roluperidone has been used in trials studying the treatment of Schizophrenia.

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsHeterocyclic Compounds, Fused-Ring +4
Target Protein:
Sigma intracellular receptor 25-hydroxytryptamine receptor 2A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Romifidine DB11543
small molecule | CAS: 65896-16-4

Romifidine is a veterinary drug utilized as a sedative primarily in large animals, most frequently horses. It is also used less commonly in a wide variety of other animal species. This drug's chemical structure closely resembles that of clonidine, however, ro…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-2 Receptor Agonists +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Romilkimab DB16318
biotech | CAS: 1399584-78-1

Romilkimab is under investigation in clinical trial NCT02345070 (Efficacy and Safety of SAR156597 in the Treatment of Idiopathic Pulmonary Fibrosis).

Target Protein:
Interleukin-13Interleukin-4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Romiplostim Approved DB05332
biotech | CAS: 267639-76-9

Romiplostim is a thrombopoiesis stimulating dimer Fc-peptide fusion protein (peptibody) to increase platelet production through activation of the thrombopoietin receptor. The peptibody molecule has two identical single-chain subunits, each one is made up of 2…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood and Blood Forming Organs +17
Target Protein:
Thrombopoietin receptor
Waktu ParuhImmune thrombocytop…
Vol. DistribusiIn healthy voluntee…
Klirens-
Genetik -
Romosozumab Approved DB11866
biotech | CAS: 909395-70-6

Romosozumab is a humanized monoclonal antibody indicated for the treatment of osteoperosis in postmenopausal women at high risk of fracture and patients who have failed in other treatments or are intolerant to other osteoperosis therapies[L9554]. Romosozumab …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +12
Target Protein:
Sclerostin
Waktu Paruh12.8 days[L9554].
Vol. Distribusi3.92L[L9554].
Klirens0.38mL/hr/kg[L9554].
Genetik -
Ronacaleret DB05255
small molecule | CAS: 753449-67-1

Ronacaleret is a calcium-sensing receptor antagonist.

Kategori:
Acids, CarbocyclicIndenes
Target Protein:
Extracellular calcium-sensing receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Roneparstat DB17153
biotech | CAS: 1407492-04-9

Deskripsi belum tersedia.

Kategori:
CarbohydratesGlycosaminoglycansPolysaccharides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Roniciclib DB12974
small molecule | CAS: 1223498-69-8

Roniciclib has been investigated for the treatment of Small Cell Lung Carcinoma.

Kategori:
Sulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ronifibrate DB13460
small molecule | CAS: 42597-57-9

Deskripsi belum tersedia.

Kategori:
Agents Causing Muscle ToxicityFibric AcidsLipid Modifying Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ronnel DB11456
small molecule | CAS: 299-84-3

Deskripsi belum tersedia.

Kategori:
Organophosphorus CompoundsSulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ronopterin DB12575
small molecule | CAS: 185243-78-1

Ronopterin has been used in trials studying the treatment of Traumatic Brain Injury.

Kategori:
CoenzymesEnzymes and CoenzymesHeterocyclic Compounds, Fused-Ring +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rontalizumab DB12844
biotech | CAS: 948570-30-7

Rontalizumab has been used in trials studying the treatment of Systemic Lupus Erythematosus.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ropanicant DB19134
small molecule | CAS: 2414674-70-5

Ropanicant is under investigation in clinical trial NCT06126497 (Study Evaluating Safety and Efficacy of Ropanicant in MDD Patients).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ropeginterferon alfa-2b Approved DB15119
biotech | CAS: 1335098-50-4

Polycythemia vera (PV) is the most common Philadelphia chromosome-negative myeloproliferative neoplasm (MPN), characterized by increased hematocrit and platelet/leukocyte counts, an increased risk for hemorrhage and thromboembolic events, and a long-term prop…

Kategori:
Adjuvants, ImmunologicAlfa InterferonsAntineoplastic and Immunomodulating Agents +12
Target Protein:
Interferon alpha/beta receptor (IFNAR)
Waktu ParuhRopeginterferon alf…
Vol. DistribusiRopeginterferon alf…
KlirensRopeginterferon alf…
Genetik -
Ropidoxuridine DB06485
small molecule | CAS: 93265-81-7

Ropidoxuridine is a novel, orally available, thymidine analogue and prodrug for IUdR, which demonstrated a survival advantage in Phase II studies in anaplastic astrocytoma, a type of brain tumor.

Kategori:
Antineoplastic AgentsNucleic Acids, Nucleotides, and NucleosidesNucleosides +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ropinirole Approved DB00268
small molecule | CAS: 91374-21-9

Ropinirole, also known as _ReQuip_, is a non-ergoline dopamine agonist used in Parkinson's disease and restless legs syndrome [FDA label], [A174547]. It is manufactured by GlaxoSmithKline Pharmaceuticals. Ropinirole was initially approved in 1997 by the FDA…

Kategori:
Anti-Dyskinesia AgentsAnti-Parkinson Agents (Dopamine Agonist)Anti-Parkinson Drugs +10
Target Protein:
D(3) dopamine receptorD(2) dopamine receptorD(4) dopamine receptor +1
Waktu ParuhApproximately 6 hou…
Vol. DistribusiRopinirole is found…
KlirensThe clearance of ro…
Genetik -
Ropsacitinib DB18709
small molecule | CAS: 2127109-84-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Roquinimex DB11366
small molecule | CAS: 84088-42-6

Roquinimex is a derivative of quinoline that presents immunostimulant properties. Its effects are suggested to increase the activity of NK cells and macrophage cytotoxicity. Additionally, roquinimex is known to inhibit angiogenesis and to decrease the synthes…

Kategori:
Adjuvants, ImmunologicAngiogenesis InhibitorsAngiogenesis Modulating Agents +7
Target Protein:
Interleukin-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Rosa centifolia flower oil is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rose bengal Approved DB11182
small molecule

Rose bengal is a pink stain derived as an analogue of fluorescein. Its disodium salt in ophthalmic solutions has been used as a diagnostic agent in suspected damage to conjunctival and corneal cells. It is also used in laboratory settings, including the prepa…

Kategori:
Coloring AgentsColouring AgentsCompounds used in a research, industrial, or household setting +12
Waktu ParuhDoses between 0.01 …
Vol. DistribusiNo information avai…
KlirensNo information avai…
Genetik -
Rose bengal I-131 Approved DB09388
small molecule | CAS: 99689-97-1

Deskripsi belum tersedia.

Kategori:
Radiopharmaceuticals
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rosiglitazone Approved DB00412
small molecule | CAS: 122320-73-4

Rosiglitazone is an anti-diabetic drug in the thiazolidinedione class of drugs. It is marketed by the pharmaceutical company GlaxoSmithKline as a stand-alone drug (Avandia) and in combination with metformin (Avandamet) or with glimepiride (Avandaryl). Like ot…

Kategori:
Alimentary Tract and MetabolismBlood Glucose Lowering AgentsBSEP/ABCB11 Substrates +33
Target Protein:
Peroxisome proliferator-activated receptor gammaLong-chain-fatty-acid--CoA ligase 4Peroxisome proliferator-activated receptor alpha +4
Waktu Paruh3-4 hours (single o…
Vol. Distribusi* 17.6 L [oral volu…
Klirens* Oral clearance (C…
Genetik -
Rosmarinic acid DB16865
small molecule | CAS: 20283-92-5

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAldehyde Reductase, antagonists & inhibitorsAnalgesics +22
Target Protein:
TyrosinaseInduced myeloid leukemia cell differentiation protein Mcl-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rosnilimab DB18851
biotech | CAS: 2412764-40-8

Rosnilimab is under investigation in clinical trial NCT06041269 (A Study of Efficacy and Safety of Rosnilimab in Subjects With Moderate to Severe Rheumatoid Arthritis (RENOIR)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rosomidnar DB17154
biotech | CAS: 871597-03-4

Deskripsi belum tersedia.

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesOligonucleotides +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rosoxacin Approved DB00817
small molecule | CAS: 40034-42-2

Rosoxacin is a quinolone derivative antibiotic for the treatment of bacterial infection of respiratory tract, urinary tract, GI, CNS and immuno compromised patients. Rosoxacin is known to be effective against penicillin resistant strains and is a single dose …

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibacterials for Systemic Use +9
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-betaDNA gyrase subunit B +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rostafuroxin DB12350
small molecule | CAS: 156722-18-8

Rostafuroxin has been used in trials studying the treatment of Essential Hypertension.

Kategori:
AndrostanesFused-Ring CompoundsSteroids
Target Protein:
Sodium/potassium-transporting ATPase subunit beta-1Sodium/potassium-transporting ATPase subunit beta-2Sodium/potassium-transporting ATPase subunit beta-3 +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rosuvastatin Approved DB01098
small molecule | CAS: 287714-41-4

Rosuvastatin, also known as the brand name product Crestor, is a lipid-lowering drug that belongs to the statin class of medications, which are used to lower the risk of cardiovascular disease and manage elevated lipid levels by inhibiting the endogenous prod…

Kategori:
Agents Causing Muscle ToxicityAlimentary Tract and MetabolismAmides +32
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductaseIntegrin alpha-L
Gen Terkait:
KIF6 HMGCR ABCG2
Waktu ParuhThe elimination hal…
Vol. DistribusiRosuvastatin underg…
Klirens-
Genetik 3 Varian
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