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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
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12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 225 / 252
Tagraxofusp Approved DB14731
biotech | CAS: 2055491-00-2

Tagraxofusp is a CD123-directed cytotoxin. It is a fusion protein composed of a human interleukin-3 (IL-3) that is genetically fused to the catalytic and translocation domains of truncated diphtheria toxin (DT) produced in _Escherichia coli_.[A253762, A253887…

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +7
Target Protein:
Interleukin-3 receptor subunit alpha
Waktu ParuhThe mean (SD) termi…
Vol. DistribusiFollowing administr…
KlirensMean clearance (SD)…
Genetik -
TAK-071 DB18954
small molecule | CAS: 1820812-16-5

TAK-071 is under investigation in clinical trial NCT04334317 (A Study of TAK-071 in People With Parkinson Disease).

Kategori:
Cholinergic AgentsCholinergic AgonistsHeterocyclic Compounds, Fused-Ring +2
Target Protein:
Muscarinic acetylcholine receptor M1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 667931-25-1

Deskripsi belum tersedia.

Kategori:
Receptors, Calcium-Sensing, antagonists & inhibitors
Target Protein:
Extracellular calcium-sensing receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TAK-243 DB15013
small molecule | CAS: 1450833-55-2

TAK-243 is under investigation in clinical trial NCT03816319 (TAK-243 in Treating Patients With Relapsed or Refractory Acute Myeloid Leukemia or Refractory Myelodysplastic Syndrome or Chronic Myelomonocytic Leukemia).

Kategori:
AmidesAnionsElectrolytes +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1818252-52-6

Deskripsi belum tersedia.

Kategori:
Sulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TAK-428 DB05499
small molecule

TAK-428 is a drug for treating diabetic neuropathy. It is based on the novel concept that peripheral nervous tissue that was damaged by diabetes can be repaired and regenerated by stimulating an increase in neurotrophic factors.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
TAK-448 DB11975
biotech | CAS: 1234319-68-6

TAK-448 has been used in trials studying the treatment of Prostate Cancer, Low Testosterone, Prostatic Neoplasms, and Hypogonadotropic Hypogonadism.

Kategori:
Amino Acids, Peptides, and ProteinsIntercellular Signaling Peptides and ProteinsNeoplasm Proteins +4
Target Protein:
Metastasis-suppressor KiSS-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TAK-475 DB05317
small molecule

TAK-475 is a "squalene synthase inhibitor", a type of cholesterol-lowering drug that has not yet been brought to market.

Kategori:
AzepinesFarnesyl-Diphosphate Farnesyltransferase, antagonists & inhibitors
Target Protein:
Squalene synthase3-hydroxy-3-methylglutaryl-coenzyme A reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TAK-593 DB13093
small molecule | CAS: 1005780-62-0

TAK-593 has been used in trials studying the treatment of Solid Tumors.

Kategori:
Aza CompoundsReceptors, Platelet-Derived Growth Factor, antagonists & inhibitors
Target Protein:
Vascular endothelial growth factor receptor 2Platelet-derived growth factor receptor beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TAK-603 DB17892
small molecule | CAS: 158146-85-1

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Interferon gamma
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TAK-653 DB16304
small molecule | CAS: 1358751-06-0

TAK-653 is under investigation in clinical trial NCT03312894 (Efficacy and Safety of TAK-653 in Treatment-resistant Depression).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TAK-715 DB16108
small molecule | CAS: 303162-79-0

TAK-715 is under investigation in clinical trial NCT00760864 (Safety and Efficacy of TAK-715 in Subjects With Rheumatoid Arthritis).

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TAK-733 DB12241
small molecule | CAS: 1035555-63-5

TAK-733 has been used in trials studying the treatment of Advanced Metastatic Melanoma, Advanced Nonhematologic Malignancies, and Advanced Non-hematologic Malignancies.

Kategori:
PyridinesPyrimidines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TAK-751S DB06432
small molecule

TAK-751S is a synthetic analog of Shiga toxin (Stx) receptor, Gb3, produced by enterohemorrhagic _Escherichia coli_.[A260296]

Kategori:
CarbohydratesOligosaccharidesPolysaccharides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TAK-754 DB17850
biotech

TAK-754 is an adeno-associated virus serotype 8 vector (AAV8) expressing B domain deleted codon optimized factor VIII. Developed by Takeda, it is being investigated for the treatment of hemophilia A.[A259831]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TAK-901 DB12756
small molecule | CAS: 934541-31-8

TAK-901 has been used in trials studying the treatment of Lymphoma, Myelofibrosis, Multiple Myeloma, Myeloid Metaplasia, and Advanced Solid Tumors, among others.

Kategori:
Heterocyclic Compounds, Fused-RingIndole AlkaloidsIndoles +3
Target Protein:
Aurora kinase BApoptosis regulator BAX
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Talacotuzumab DB14796
biotech | CAS: 1826831-79-1

Talacotuzumab is an IgG1 monoclonal antibody directed toward the IL3 receptor ?–subunit, also known as CD123. It is under investigation in clinical trial NCT01632852 (A Study of CSL362 in Patients With CD123+ Acute Myeloid Leukemia Currently in Remission).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 308240-58-6

Talactoferrin alfa is a novel immunomodulatory 80 kD protein with demonstrated oral anti-tumor properties. Lactoferrin, a protein found in breast milk is developed by Agennix. It increases body’s immune power and also works as a natural antioxidant, helping t…

Kategori:
Amino Acids, Peptides, and ProteinsAnimal Proteins, DietaryAntineoplastic Agents +21
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Taladegib DB12550
small molecule | CAS: 1258861-20-9

Taladegib has been used in trials studying the treatment of Solid Tumor, COLON CANCER, BREAST CANCER, Advanced Cancer, and Rhabdomyosarcoma, among others.

Kategori:
Pyridazines
Target Protein:
Protein smoothened
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Talampanel DB04982
small molecule | CAS: 161832-65-1

Talampanel is a substance that is being studied in the treatment of brain tumors and other brain disorders, such as epilepsy and Parkinson disease. It is a type of AMPA receptor antagonist.

Kategori:
BenzazepinesHeterocyclic Compounds, Fused-RingReceptors, AMPA, antagonists & inhibitors
Target Protein:
Glutamate receptor 1Glutamate receptor 2Glutamate receptor 3 +1
Waktu Paruh3-6 hours
Vol. Distribusi-
Klirens-
Genetik -
Talampicillin DB13814
small molecule | CAS: 47747-56-8

Deskripsi belum tersedia.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Talarozole DB13083
small molecule | CAS: 201410-53-9

Talarozole has been investigated for the treatment of Psoriasis and Cutaneous Inflammation.

Kategori:
Cytochrome P-450 Enzyme InhibitorsEnzyme InhibitorsHeterocyclic Compounds, Fused-Ring +1
Target Protein:
Substance-K receptorCytochrome P450 26A1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Talazoparib Approved DB11760
small molecule | CAS: 1207456-01-6

Talazoparib is an inhibitor of mammalian polyadenosine 5’-diphosphoribose polymerases (PARPs), enzymes responsible for regulating essential cellular functions, such as DNA transcription and DNA repair.[L47236] Developed by Pfizer, talazoparib was first app…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Substrates +7
Target Protein:
Poly [ADP-ribose] polymerase 1Poly [ADP-ribose] polymerase 2
Waktu ParuhThe mean terminal p…
Vol. DistribusiThe mean apparent v…
KlirensThe mean apparent o…
Genetik -
Talbutal Approved DB00306
small molecule | CAS: 115-44-6

Talbutal, also called 5-allyl-5-sec-butylbarbituric acid, is a barbiturate with a short to intermediate duration of action. Talbutal is a schedule III drug in the U.S.

Kategori:
Anticholinergic AgentsBarbiturates, PlainCentral Nervous System Depressants +6
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-2Gamma-aminobutyric acid receptor subunit gamma-3Gamma-aminobutyric acid receptor subunit alpha-3 +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Talc Approved DB09511
small molecule | CAS: 14807-96-6

Talc is a mineral composed primarily of magnesium, silicon and oxygen. It is a substance often found in cosmetic and personal hygiene products including baby powder, adult body powders and facial powders. Talc helps absorb moisture, freshen materials, and red…

Kategori:
AntiperspirantsCompounds used in a research, industrial, or household settingCosmetics +6
Waktu ParuhIntended for local …
Vol. DistribusiIntended for local …
KlirensIntended for local …
Genetik -
biotech | CAS: 1580555-26-5

Talditercept alfa is under investigation in clinical trial NCT03039686 (Clinical Trial to Evaluate the Efficacy, Safety, and Tolerability of RO7239361 in Ambulatory Boys With Duchenne Muscular Dystrophy).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
taletrectinib DB18711
small molecule | CAS: 1505515-69-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Talimogene laherparepvec Approved DB13896
biotech | CAS: 1187560-31-1

Talimogene laherparepvec is an oncolytic treatment used in local treatment of unresectable cutaneous, subcutaneous, and nodal lesions in patients with recurrent melanoma. It is a genetically administered herpes simplex virus 1 (HSV-1) that expresses human cyt…

Kategori:
AlphaherpesvirinaeAntineoplastic AgentsAntineoplastic Agents, Immunological +9
Target Protein:
Granulocyte-macrophage colony-stimulating factor
Waktu ParuhReadily accessible …
Vol. DistribusiTalimogene laherpar…
KlirensAlthough readily ac…
Genetik -
Talinolol DB11770
small molecule | CAS: 57460-41-0

Talinolol has been investigated for the basic science of Gastrointestinal Motility Disorder.

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-Antagonists +16
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tallimustine DB15466
small molecule | CAS: 115308-98-0

Tallimustine, a benzoyl mustard derivative of distamycin A, is an alkylating agent that binds to the minor groove of DNA.[A182036,A182039] It's association with severe myelotoxicity lead to the end of its development in favour of ?-halogenoacrylamide derivati…

Kategori:
Alkylating DrugsAmino Acids, Peptides, and ProteinsAntineoplastic Agents +6
Target Protein:
C-X-C chemokine receptor type 2DNA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Talmapimod DB05412
small molecule | CAS: 309913-83-5

Talmapimod is the first-generation oral p38 MAP kinase inhibitor developed by Scios. It has shown to be effective to cure inflammatory diseases such as Rheumatoid Arthritis.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Mitogen-activated protein kinase 14Tumor necrosis factorInterleukin-1 beta +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Talniflumate DB09295
small molecule | CAS: 66898-62-2

Talniflumate, is an anti-inflammatory molecule studied and used as a mucin regulator in the treatment of cystic fibrosis, chronic obstructive pulmonary disease (COPD) and asthma [L1400]. In addition, it is used in inflammatory conditions such as rheumatoid ar…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnti-Inflammatory Agents +5
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2Chloride channel protein ClC-Ka
Waktu ParuhApproximately 2h in…
Vol. DistribusiIn 12 subjects afte…
KlirensThis drug undergoes…
Genetik -
Talopram DB09190
small molecule | CAS: 7182-51-6

Talopram is a selective norepinephrine reuptake inhibitor (SNRI) that is structurally similar to citalopram and melitracen. It was researched in the 1960s and 1970s but never marketed.

Kategori:
Adrenergic Uptake InhibitorsAminesAntidepressive Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Talotrexin DB06178
small molecule | CAS: 113857-87-7

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +5
Target Protein:
Folate receptor alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Talquetamab Approved DB16678
biotech | CAS: 2226212-40-2

Talquetamab is a IgG4-PAA bispecific G protein-coupled receptor class C group 5 member D (GPRC5D)-directed CD3 T-cell engager. It consists of two arms - anti-GPRC5D and anti-CD3 arms - linked by two interchain disulfide bonds, each arm comprising a heavy and …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntineoplastic Agents +7
Target Protein:
T-cell surface glycoprotein CD3G-protein coupled receptor family C group 5 member D
Waktu ParuhThe mean (CV%) term…
Vol. DistribusiThe geometric mean …
KlirensTalquetamab clearan…
Genetik -
Talsaclidine DB12287
small molecule | CAS: 147025-53-4

Talsaclidine has been used in trials studying the treatment of Alzheimer Disease.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Talviraline DB07885
small molecule | CAS: 163451-80-7

Talviraline has been used in trials studying the treatment of HIV Infections.

Kategori:
Acquired Immunodeficiency SyndromeHeterocyclic Compounds, Fused-Ring
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tamarix gallica pollen Approved DB10725
biotech

Tamarix gallica pollen is the pollen of the Tamarix gallica plant. Tamarix gallica pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tamatinib DB07159
small molecule | CAS: 841290-80-0

Deskripsi belum tersedia.

Target Protein:
Tyrosine-protein kinase SYKProto-oncogene tyrosine-protein kinase receptor Ret
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tamibarotene DB04942
small molecule | CAS: 94497-51-5

Tamibarotene is a novel synthetic retinoid for acute promyelocytic leukaemia (APL). Tamibarotene is currently approved in Japan for treatment of recurrent APL, and is undergoing clinical trials in the United States.

Kategori:
Acids, CarbocyclicBenzene DerivativesNaphthalenes
Target Protein:
Retinoic acid receptor alphaRetinoic acid receptor beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Taminadenant DB18811
small molecule | CAS: 1337962-47-6

Deskripsi belum tersedia.

Target Protein:
Adenosine receptor A2a
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tamnorzatinib DB19201
small molecule | CAS: 1646839-59-9

Tamnorzatinib is under investigation in clinical trial NCT03176277 (A Study of ONO-7475 in Patients With Acute Leukemias).

Target Protein:
Tyrosine-protein kinase MerTyrosine-protein kinase receptor UFO
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tamoxifen Approved DB00675
small molecule | CAS: 10540-29-1

Tamoxifen is a non-steroidal antiestrogen used to treat estrogen receptor positive breast cancers as well as prevent the incidence of breast cancer in high risk populations.[A1025,L7799,L7802] Tamoxifen is used alone or as an adjuvant in these treatments.[L77…

Kategori:
Anti-EstrogensAntineoplastic AgentsAntineoplastic Agents, Hormonal +64
Target Protein:
Estrogen receptorEstrogen receptor betaProtein kinase C +7
Gen Terkait:
CYP2D6 F5
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of ta…
Genetik 2 Varian
Tamsulosin Approved DB00706
small molecule | CAS: 106133-20-4

Tamsulosin is a selective alpha-1A and alpha-1B adrenoceptor antagonist that exerts its greatest effect in the prostate and bladder, where these receptors are most common.[Label] It is indicated for the treatment of signs and symptoms of benign prostatic hype…

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +22
Target Protein:
Alpha-1A adrenergic receptorAlpha-1D adrenergic receptorAlpha-1B adrenergic receptor
Waktu ParuhThe half life in fa…
Vol. Distribusi16L after intraveno…
Klirens2.88L/h.[Label]
Genetik -
biotech

Tanacetum cinerariifolium flower allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tanaproget DB04787
small molecule | CAS: 304853-42-7

Tanaproget (NSP-989) is an investigational non-steroidal progestin. It is a high affinity, high efficacy agonist of the progesterone receptor (PR) with a much more selective binding profile relative to most conventional progestins. Because of this tanaproget …

Kategori:
Heterocyclic Compounds, Fused-RingOxazinesReceptors, Progesterone, agonists +1
Target Protein:
Progesterone receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tandospirone DB12833
small molecule | CAS: 87760-53-0

Tandospirone has been used in trials studying the treatment of Schizophrenia.

Kategori:
Anti-Anxiety AgentsAntidepressive AgentsCentral Nervous System Agents +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tandutinib DB05465
small molecule | CAS: 387867-13-2

MLN518 is a novel, oral, small molecule designed to inhibit type III receptor tyrosine kinases, including FLT3, (platelet-derived growth-factor receptor) PDGFR and c-KIT. Tyrosine kinases are enzymes involved in several cellular processes and are known to be …

Kategori:
Heterocyclic Compounds, Fused-RingPotential QTc-Prolonging AgentsQTc Prolonging Agents +1
Target Protein:
Receptor-type tyrosine-protein kinase FLT3Platelet-derived growth factor D
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tanespimycin DB05134
small molecule | CAS: 75747-14-7

Tanespimycin, manufactured by Conforma Therapeutics is under development as a small molecule inhibitor of heat shock protein 90 (HSP90). It is developed for the treatment of several types of cancer, solid tumors or chronic myelogenous leukemia.

Kategori:
AmidesHSP90 Heat-Shock Proteins, antagonists & inhibitorsLactams +2
Target Protein:
Heat shock protein HSP 90-alphaHeat shock protein HSP 90-beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tanezumab DB12335
biotech | CAS: 880266-57-9

Tanezumab has been investigated for the treatment of Osteoarthritis, Knee and Neuralgia, Postherpetic.

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsAntibodies +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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