Hasil Filter

17430

Total database: 17430
Struktur (SMILES)
12313 (70.6%)
Target
9368 (53.7%)
Genomik
112 (0.6%)
Referensi
17430 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (17430)

Halaman 224 / 349
MK-6325 DB15249
small molecule | CAS: 1263814-52-3

MK-6325 is under investigation in clinical trial NCT01329913 (Safety, Pharmacokinetics, and Pharmacodynamics of MK-6325 in Hepatitis C Virus (HCV) Infections (MK-6325-003)).

Target Protein:
Genome polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MK-7145 DB11968
small molecule | CAS: 1255204-84-2

MK-7145 has been used in trials studying the treatment of Hypertension and Renal Insufficiency.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MK-7288 DB17094
small molecule | CAS: 936626-07-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MK-7622 DB12897
small molecule | CAS: 1227923-29-6

MK-7622 has been used in trials studying the treatment of Alzheimer's Disease.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MK-8189 DB19153
small molecule | CAS: 1424371-93-6

MK-8189 is under investigation in clinical trial NCT04624243 (Efficacy and Safety of MK-8189 in Participants With an Acute Episode of Schizophrenia (MK-8189-008)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MK-8245 DB13024
small molecule | CAS: 1030612-90-8

MK-8245 has been used in trials studying the treatment of Type 2 Diabetes Mellitus.

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MK-8666 DB14937
small molecule | CAS: 1544739-75-4

MK-8666 is under investigation in clinical trial NCT01971554 (Safety, Tolerability, Pharmacodynamics, and Pharmacokinetics of MK-8666 in Participants With Type 2 Diabetes Mellitus (MK-8666-003)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MK-8719 DB16989
small molecule | CAS: 1382799-40-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MK-8776 DB11899
small molecule | CAS: 891494-63-6

Sch 900776 has been used in trials studying the treatment of Neoplasms, Hodgkin Disease, Adult Erythroleukemia, Lymphoma, Non-Hodgkin, and Myelogenous Leukemia, Acute, among others.

Target Protein:
Serine/threonine-protein kinase Chk1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MK-8777 DB18904
small molecule | CAS: 1026791-61-6

MK-8777 is under investigation in clinical trial NCT00610649 (Trial to Determine the Maximum Tolerated Dose (MTD) Based on Safety and Tolerability, of Org 26576 in Participants With Major Depressive Disorder (174001/P05704/MK-8777-001)).

Kategori:
Isoxazoles
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MK-886 DB16739
small molecule | CAS: 118414-82-7

MK-886 is an experimental inhibitor of leukotriene synthesis.

Kategori:
Benzene DerivativesEnzyme InhibitorsHeterocyclic Compounds, Fused-Ring +4
Target Protein:
Polyunsaturated fatty acid 5-lipoxygenaseArachidonate 5-lipoxygenase-activating protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MKC-1 DB05608
small molecule | CAS: 125313-92-0

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingProtein Kinase Inhibitors
Target Protein:
Cyclin-dependent kinase 4Cyclin-dependent kinase 2Cyclin-dependent kinase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MKC1106-PP DB06030
small molecule

MKC1106-PP is a 3-component investigational vaccine made up of a DNA plasmid (pPRA-PSM) and 2 peptides E-PRA and E-PSM. The plasmid portion is a recombinant plasmid expressing segments of the 2 target antigens, PRAME and PSMA. MKC1106-PP was under investigati…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MLN-977 DB05431
small molecule | CAS: 175212-04-1

MLN-977 is a small molecule compound that inhibits the production of leukotrienes, especially 5-lipoxygenase. It is developed by PharmaEngine to treat asthma and chronic obstructive pulmonary disease.

Target Protein:
Polyunsaturated fatty acid 5-lipoxygenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MLN0415 DB05183
small molecule

MLN0415 is a novel, small molecule IKK2 inhibitor, discovered by Millennium scientists. In preclinical studies, MLN0415 was shown to decrease NF-kB activation and down-regulate the expression of a number of inflammatory proteins. Because inflammatory proteins…

Target Protein:
Inhibitor of nuclear factor kappa-B kinase subunit beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MLN2222 DB06503
biotech

MLN2222 is a novel, proprietary recombinant protein that blocks both the C3 and C5 convertases, which are essential components of the complement activation pathway.

Target Protein:
Complement factor B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MLN2704 DB06513
biotech

A Phase 1/2 trial (NCT00070837) evaluated the safety, dosage, and pharmacokinetics of MLN2704 in patients with metastatic androgen-independent prostate cancer.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MLN3897 DB06505
small molecule | CAS: 849105-26-6

MLN3897, a novel CCR1 inhibitor, disrupts osteoclast formation and blocks the interaction between multiple myeloma cells and osteoclasts.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
C-C chemokine receptor type 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MLN576 DB06517
small molecule | CAS: 346689-77-8

XR11576 (MLN576) is a novel monophenazine with a mechanism of action that includes interaction with both topoisomerase (Topo) I and II.[A234609]

Kategori:
Antineoplastic AgentsEnzyme InhibitorsHeterocyclic Compounds, Fused-Ring +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MLN8054 DB13061
small molecule | CAS: 869363-13-3

MLN8054 has been used in trials studying the treatment of Colon Neoplasm, Breast Neoplasm, Bladder Neoplasm, Pancreatic Neoplasm, and Advanced Malignancies.

Kategori:
Heterocyclic Compounds, Fused-RingProtein Kinase Inhibitors
Target Protein:
Aurora kinase A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MM-093 DB05512
biotech

MM-093 is a recombinant version of human alpha-fetoprotein (hAFP), an immunomodulatory serum protein normally produced at very high levels by the fetus and present in low levels in the blood of adults and children. Research on AFP suggests that it may play a …

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MM-111 DB17983
biotech | CAS: 1361108-53-3

MM-111 is a novel bispecific antibody fusion protein that co-targets the the epidermal growth factor family receptor tyrosine kinases, ERBB2 and ERBB3.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MM3122 DB16737
small molecule

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsExperimental Unapproved Treatments for COVID-19Heterocyclic Compounds, Fused-Ring +2
Target Protein:
Transmembrane protease serine 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MMDA DB01442
small molecule | CAS: 13674-05-0

MMDA, or 3-methoxy-4,5-methylenedioxyamphetamine, is a member of the amphetamine drug class with stimulant and psychedelic properties. It also acts as an entheogen and an entactogen. MMDA bears resemblance to the psychopharmacologically active essential oils …

Kategori:
Agents producing tachycardiaAgents that produce hypertensionAmines +11
Target Protein:
5-hydroxytryptamine receptor 2ASodium-dependent dopamine transporterSodium-dependent serotonin transporter +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MMI-175 DB02378
small molecule

Deskripsi belum tersedia.

Target Protein:
Beta-secretase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MN-246 DB05981
small molecule

MN-246 is a novel ß3-adrenergic receptor agonist developed for the treatment of urinary incontinence by MediciNova Inc.

Target Protein:
Beta-3 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MN-305 DB05339
small molecule

MN-305 is a novel, potent and highly selective serotonin 5-HT1A receptor agonist under development by MediciNova for the treatment of anxiety disorders beginning with Generalized Anxiety Disorder (GAD).

Target Protein:
5-hydroxytryptamine receptor 1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mobocertinib Approved DB16390
small molecule | CAS: 1847461-43-1

Mobocertinib is a kinase inhibitor targeted against human epidermal growth factor receptor (EGFR). It is used specifically in the treatment of non-small cell lung cancer (NSCLC) caused by exon 20 insertion mutations in the _EGFR_ gene,[L38368] which are typic…

Kategori:
AminesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +15
Target Protein:
Epidermal growth factor receptor
Waktu ParuhAt steady-state, th…
Vol. DistribusiThe mean apparent v…
KlirensAt steady-state, th…
Genetik -
Mocemestrocel DB19154
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mocetinostat DB11830
small molecule | CAS: 726169-73-9

Mocetinostat has been used in trials studying the treatment of Lymphoma, Urothelial Carcinoma, Relapsed and Refractory, Myelodysplastic Syndrome, and Metastatic Leiomyosarcoma, among others.

Kategori:
Acids, CarbocyclicAmidesAntineoplastic Agents +6
Target Protein:
Histone deacetylase 1Histone deacetylase 3Histone deacetylase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Moclobemide Approved DB01171
small molecule | CAS: 71320-77-9

A reversible monoamine oxidase inhibitor (MAOI) selective for isoform A (RIMA) used to treat major depressive disorder. Most meta-analyses and most studies indicate that in the acute management of depression, moclobemide is more efficacious than placebo medic…

Kategori:
Acids, CarbocyclicAgents that produce hypertensionAgents that reduce seizure threshold +28
Target Protein:
Amine oxidase [flavin-containing] AMonoamine oxidaseAmine oxidase [flavin-containing] B
Waktu Paruh1-2 hours (4 hours …
Vol. Distribusi1-1.5 L/Kg [L1350]
KlirensClearance of 30-78 …
Genetik -
Mocravimod DB18151
small molecule | CAS: 509092-16-4

Deskripsi belum tersedia.

Kategori:
Sulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MOD-5014 DB17715
biotech

MOD-5014 is a long-acting carboxy-terminal peptide (CTP)-modified Factor IIa.[A259088] It is being investigated for the treatment of hemophilia.[L46173]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Modafinil Approved DB00745
small molecule | CAS: 68693-11-8

Modafinil is a stimulant drug marketed as a 'wakefulness promoting agent' and is one of the stimulants used in the treatment of narcolepsy. Narcolepsy is caused by dysfunction of a family of wakefulness-promoting and sleep-suppressing peptides, the orexins, w…

Kategori:
Benzene DerivativesBenzhydryl CompoundsCentral Nervous System Agents +35
Target Protein:
Sodium-dependent dopamine transporterAlpha-1B adrenergic receptor
Gen Terkait:
COMT COMT
Waktu Paruh23-215 hours
Vol. Distribusi* 0.9 L/kg
Klirens-
Genetik 2 Varian
Modakafusp alfa DB16399
biotech

Modakafusp alfa is under investigation in clinical trial NCT03215030 (A Study to Investigate the Safety, Tolerability, Efficacy, Pharmacokinetics, and Immunogenicity of TAK-573 in Participants With Refractory Multiple Myeloma (MM)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Moderna COVID-19 Vaccine Approved DB15654
biotech

The Moderna COVID-19 Vaccine (mRNA-1273) is a novel mRNA-based vaccine encapsulated in a lipid nanoparticle that encodes for a full-length pre-fusion stabilized spike (S) protein of severe acute respiratory syndrome coronavirus 2 (SARS-CoV-2). Coronavirus dis…

Kategori:
Biological ProductsCOVID-19 VaccinesExperimental Unapproved Treatments for COVID-19 +5
Waktu ParuhThere is limited ph…
Vol. DistribusiThere is limited ph…
KlirensThere is limited ph…
Genetik -
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
4-alpha-glucanotransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Nucleoside 2-deoxyribosyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Modified vaccinia ankara Approved DB15483
biotech

Modified Vaccinia Ankara (MVA) refers to an attenuated strain of the Vaccinia virus. Vaccines using MVA are live and non-replicating, and are produced using Modified Vaccinia Ankara-Bavarian Nordic (MVA-BN).[L42660,L42670]

Kategori:
Anti-Infective AgentsAntiviral AgentsBiological Products +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2171576-44-4

Modified vaccinia virus Ankara-85A antigen is under investigation in clinical trial NCT00953927 (A Study of MVA85A in Healthy Infants).

Kategori:
Amino Acids, Peptides, and ProteinsAntigensBacterial Vaccines +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Modimelanotide DB15314
small molecule | CAS: 926277-68-1

Modimelanotide is under investigation in clinical trial NCT01897519 (A Safety and Efficacy Trial of Multiple Dosing Regimens of ABT-719 for the Prevention of Acute Kidney Injury in Subjects Undergoing High Risk Surgery).

Kategori:
Pyridines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Modipafant DB16237
small molecule | CAS: 122957-06-6

Modipafant is under investigation in clinical trial NCT02569827 (Celgosivir or Modipafant as Treatment for Adult Participants With Uncomplicated Dengue Fever in Singapore).

Kategori:
Pyridines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Modithromycin DB16238
small molecule | CAS: 736992-12-4

Modithromycin is under investigation in clinical trial NCT00270517 (Comparative Study of EDP-420 Versus Another Antibiotic in the Treatment of Community Acquired Pneumonia).

Kategori:
LactonesPolyketides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Modotuximab DB14827
biotech | CAS: 1310460-86-6

Modotuximab is under investigation in clinical trial NCT03549338 (Sym004 Versus Futuximab or Modotuximab in Patients With mCRC).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Modufolin DB12676
small molecule | CAS: 31690-11-6

Modufolin is under investigation for the treatment of Osteosarcoma.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Moexipril Approved DB00691
small molecule | CAS: 103775-10-6

Moexipril is a non-sulfhydryl containing precursor of the active angiotensin-converting enzyme (ACE) inhibitor moexiprilat. It is used to treat high blood pressure (hypertension). It works by relaxing blood vessels, causing them to widen. Lowering high blood …

Kategori:
ACE Inhibitors and DiureticsAgents Acting on the Renin-Angiotensin SystemAgents causing angioedema +14
Target Protein:
Angiotensin-converting enzyme
Waktu ParuhMoexipril eliminati…
Vol. Distribusi* 183 L
Klirens* 441 mL/min
Genetik -
Moexiprilat DB14210
small molecule | CAS: 103775-14-0

The active metabolite of the prodrug [Moexipril].

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing angioedemaAngiotensin-Converting Enzyme Inhibitors +2
Target Protein:
Angiotensin-converting enzyme
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 11151–11200 dari 17430
Sebelumnya Halaman 224 / 349 Berikutnya