Hasil Filter

11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (11778)

Halaman 224 / 236
Tubimod DB17745
biotech

Deskripsi belum tersedia.

Kategori:
Biological ProductsComplex MixturesVaccines +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tubocurarine Approved DB01199
small molecule | CAS: 57-95-4

Tubocurarine is a non-depolarizing neuromuscular blocking agent and the first identified curare alkaloid.[A216008] Curare is one of the names used to describe plant-derived poisons used by indigenous South Americans to coat the tips of hunting arrows and dart…

Kategori:
AlkaloidsAminesAnticholinergic Agents +23
Target Protein:
Neuronal acetylcholine receptor subunit alpha-25-hydroxytryptamine receptor 3AAcetylcholinesterase +1
Waktu Paruh1-2 hours
Vol. Distribusi-
Klirens-
Genetik -
Tucaresol DB13027
small molecule | CAS: 84290-27-7

Tucaresol has been used in trials studying the treatment of HIV Infections.

Kategori:
Acids, CarbocyclicAldehydesBenzene Derivatives
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tucatinib Approved DB11652
small molecule | CAS: 937263-43-9

Tucatinib is a kinase inhibitor drug used with [trastuzumab] and [capecitabine] in the treatment of unresectable or metastatic HER-2 positive breast cancer. It was developed by Seattle Genetics and approved by the FDA on April 17, 2020.[L12951] Tucatinib is a…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Substrates +18
Target Protein:
Receptor tyrosine-protein kinase erbB-2Receptor tyrosine-protein kinase erbB-3
Waktu ParuhA pharmacokinetic s…
Vol. DistribusiThe volume of distr…
KlirensThe apparent cleara…
Genetik -
Tucidinostat DB06334
small molecule | CAS: 1616493-44-7

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesAmines +7
Target Protein:
Histone deacetylase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 339986-90-2

Tucotuzumab celmoleukin is under investigation in clinical trial NCT00016237 (Interleukin-2 Combined With Monoclonal Antibody Therapy in Treating Patients With Kidney, Bladder, or Lung Cancer That Has Not Responded to Previous Treatment).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tulathromycin A DB11474
small molecule | CAS: 217500-96-4

Tulathromycin is a macrolide antibiotic used to treat bovine respiratory disease in cattle and swine respiratory disease in pigs. It is marketed by Pfizer Inc. under the tradename Draxxin.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsCarbohydrates +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tulisokibart DB18719
biotech | CAS: 2648504-55-4

PRA023 is a humanized monoclonal antibody directed to vascular endothelial growth inhibitor, also known as tumour necrosis factor (TNF)-like ligand 1A (TL1A) and TNF superfamily member 15. It is being investigated for ulcerative colitis.

Target Protein:
Tumor necrosis factor ligand superfamily member 15
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tulmimetostat DB19446
small molecule | CAS: 2567686-02-4

Tulmimetostat is under investigation in clinical trial NCT05467748 (EZH2 Inhibitor, Tulmimetostat, and PD-1 Blockade for Treatment of Advanced Non-small Cell Lung Cancer).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tulobuterol DB12248
small molecule | CAS: 41570-61-0

Tulobuterol has been used in trials studying the treatment of Chronic Obstructive Pulmonary Disease.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic beta-Agonists +17
Target Protein:
Beta-2 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tulrampator DB16344
small molecule | CAS: 1038984-31-4

Tulrampator is under investigation in clinical trial NCT02626572 (Efficacy and Safety of 3 Doses of S47445 Versus Placebo in Patients With Alzheimer's Disease at Mild to Moderate Stages With Depressive Symptoms).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tuna Approved DB10574
biotech

Tuna allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tunicamycin DB13172
small molecule | CAS: 11089-65-9

Tunicamycin is a mixture of homologous nucleoside antibiotics that inhibits the UDP-HexNAc: polyprenol-P HexNAc-1-P family of enzymes. One member of this family is the enzyme GlcNAc phosphotransferase (GPT), which catalyzes the transfer of N-acetylglucosamine…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsNucleic Acids, Nucleotides, and Nucleosides +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tunlametinib DB18791
small molecule | CAS: 1801756-06-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tuparstobart DB19118
biotech | CAS: 2649466-03-3

Tuparstobart is under investigation in clinical trial NCT05287113 (Study of Retinfanlimab in Combination With INCAGN02385 and INCAGN02390 as First-line Treatment in Participants With Pd-l1-positive (CPS ? 1) Recurrent/metastatic Squamous Cell Carcinoma of the…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Turkey Approved DB10575
biotech

Turkey allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Turmeric Approved DB14276
biotech

Turmeric is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
AngiospermsAntioxidantsBiological Factors +16
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Turoctocog alfa Approved DB09109
biotech | CAS: 1192451-26-5

Turoctocog alfa is a recombinant factor VIII (rFVIII) with a truncated B-domain made from the sequence coding for 10 amino acids from the N-terminus and 11 amino acids from the C-terminus of the naturally occurring B-domain. Turoctocog alfa is produced in Chi…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +5
Target Protein:
Coagulation factor IXCoagulation factor XProthrombin
Waktu ParuhIn pre-clinical stu…
Vol. DistribusiIn pre-clinical stu…
KlirensIn pre-clinical stu…
Genetik -
Turoctocog alfa pegol Approved DB14738
biotech | CAS: 1309086-46-1

Turoctocog alfa pegol is a pegylated version of [turoctocog alfa]. Novo Nordisk's brand name Esperoct (turoctocog alfa pegol, N8-GP) was approved by the US FDA on February 19, 2019. Fundamentally, the N8-GP moiety is identical to [turoctocog alfa], a recom…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +5
Target Protein:
Coagulation factor IXCoagulation factor XProthrombin +1
Waktu ParuhThe mean plasma hal…
Vol. DistribusiThe mean volume of …
KlirensThe mean clearance …
Genetik -
small molecule | CAS: 629664-81-9

Fxr 450 is under investigation in clinical trial NCT00509756 (Study Evaluating Turofexorate isopropyl in Healthy Japanese Men).

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Bile acid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Turpentine Approved DB11120
small molecule | CAS: 9005-90-7

Turpentine, also known as spirit of turpentine, oil of turpentine, and wood turpentine, is a liquid extracted from live trees, mainly pine, through distillation of resin. It is used as a solvent and base material in organic synthesis reactions. Turpentine is …

Kategori:
Biological ProductsComplex MixturesCompounds used in a research, industrial, or household setting +9
Target Protein:
Mitogen-activated protein kinase 1
Waktu ParuhEight male voluntee…
Vol. DistribusiTurpentine, as a li…
Klirens-
Genetik -
biotech | CAS: 2254086-60-5

Tusamitamab ravtansine is an antibody-drug conjugate that targets carcinoembryonic antigen-related cell adhesion molecule-5 (CEACAM5).

Kategori:
Amino Acids, Peptides, and ProteinsBlood ProteinsGlobulins +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tuspetinib DB15343
small molecule

Tuspetinib (HM-43239) is under investigation in clinical trial NCT03850574 (Clinical Trial to Evaluate the Safety, Tolerability, Pharmacokinetics and Pharmacodynamics of HM43239 in Patients With Relapsed or Refractory Acute Myeloid Leukemia).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tuvirumab DB17752
biotech | CAS: 138660-97-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tuvusertib DB18790
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TVI-Brain-1 DB17227
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TW-37 DB17059
small molecule | CAS: 877877-35-5

TW-37 is a small-molecule inhibitor of Bcl-2 investigated for its anti-cancer properties.[A253157]

Target Protein:
Apoptosis regulator Bcl-2Induced myeloid leukemia cell differentiation protein Mcl-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TY027 DB16500
biotech

Deskripsi belum tersedia.

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tylosin DB11475
small molecule | CAS: 1401-69-0

Tylosin is a bacteriostatic macrolide antibiotic and feed additive used in veterinary medicine. It has a broad spectrum of activity against Gram-positive organisms and a limited range of Gram-negative organisms. Tylosin is produced as a fermentation product o…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsLactones +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tymazoline DB08803
small molecule | CAS: 24243-97-8

Tymazoline is a nasal preparation.

Kategori:
Nasal PreparationsSympathomimetics, Plain
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tyramine DB08841
small molecule | CAS: 51-67-2

Tyramine (4-hydroxyphenethylamine; para-tyramine, mydrial or uteramin) is a naturally occurring monoamine compound and trace amine derived from the amino acid tyrosine. Tyramine acts by inducing the release of catecholamine. An important characteristic of thi…

Kategori:
Adrenergic AgentsAgents producing tachycardiaAgents that produce hypertension +9
Target Protein:
Trace amine-associated receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tyropanoic acid Approved DB09340
small molecule | CAS: 27293-82-9

Tyropanoic acid is a radiocontrast agent used in cholecystography, the X-ray diagnosis of gallstones under the trade names include Bilopaque, Lumopaque, Tyropaque, and Bilopac. The molecule contains three heavy iodine atoms which obstruct X-rays in the same w…

Kategori:
Benzene DerivativesCompounds used in a research, industrial, or household settingContrast Media +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tyroserleutide DB17300
small molecule | CAS: 138168-48-6

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tyrosinal DB03978
small molecule

Deskripsi belum tersedia.

Target Protein:
Tyrosine--tRNA ligaseTyrosine--tRNA ligase, cytoplasmicTyrosine--tRNA ligase +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 133550-34-2

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesBenzylidene CompoundsHeterocyclic Compounds, Fused-Ring +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 133550-37-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 148741-30-4

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesBenzylidene CompoundsHeterocyclic Compounds, Fused-Ring +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tyrphostin B44 DB16762
small molecule | CAS: 133550-32-0

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesBenzylidene CompoundsHeterocyclic Compounds, Fused-Ring +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tyrphostin B48 DB16774
small molecule | CAS: 133550-35-3

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesBenzylidene CompoundsHeterocyclic Compounds, Fused-Ring +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tyrphostin B56 DB16775
small molecule | CAS: 149092-35-3

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesBenzylidene CompoundsHeterocyclic Compounds, Fused-Ring +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
U-0126 DB17060
small molecule | CAS: 218601-62-8

U-0126 is a direct inhibitor of the mitogen-activated protein-kinase kinase family members, MEK-1 and MEK-2.[A253162]

Kategori:
AlkadienesAlkenesEnzyme Inhibitors +2
Target Protein:
Mitogen-activated protein kinase kinase kinase 2Mitogen-activated protein kinase kinase kinase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
UB-612 DB16444
biotech

The UB-612 COVID-19 vaccine was developed by United Biomedical Inc Asia in Taipei as the first COVID-19 “multi-tope” protein-peptide vaccine made up of eight rationally designed components[L30653]. The vaccine incorporates a strong S1-RBD component linked to …

Kategori:
Biological ProductsComplex MixturesVaccines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ubamatamab DB18875
biotech | CAS: 2305629-50-7

Ubamatamab is under investigation in clinical trial NCT03564340 (Study of REGN4018 Administered Alone or in Combination With Cemiplimab in Adult Patients With Recurrent Ovarian Cancer or Other Recurrent Mucin-16 Expressing (MUC16+) Cancers).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ubenimex DB03424
small molecule | CAS: 58970-76-6

Ubenimex (also known as bestatin) is a competitive protease inhibitor. It is an inhibitor of aminopeptidase B, leukotriene A4 hydrolase, aminopeptidase N. It is being studied for use in the treatment of acute myelocytic leukemia.

Kategori:
Adjuvants, ImmunologicAmino AcidsAmino Acids, Branched-Chain +9
Target Protein:
Leukotriene A-4 hydrolaseBacterial leucyl aminopeptidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ubidecarenone Approved DB09270
small molecule | CAS: 303-98-0

Ubidecarenone, also called coenzyme Q10, is a 1,4-benzoquinone. From its name (Q10), the Q refers to the constitutive quinone group, and 10 is related to the number of isoprenyl subunits in its tail.[A7874] It is a powerful antioxidant, a lipid-soluble and es…

Kategori:
Agents Causing Muscle ToxicityBenzoquinonesCardiac Therapy +13
Target Protein:
NADH dehydrogenase [ubiquinone] flavoprotein 3, mitochondrialSuccinate dehydrogenase [ubiquinone] flavoprotein subunit, mitochondrial
Waktu ParuhThe pharmacokinetic…
Vol. DistribusiUbidecarenone is di…
KlirensIn preclinical stud…
Genetik -
Ubiquinol Approved DB11340
small molecule | CAS: 992-78-9

Ubiquinol (CoQH2) is a reduced form of coenzyme Q10 (CoQ10) that acts as an active antioxidant that prevents the initiation and propagation of lipid peroxidation in biological membranes and human low-density lipoprotein (LDL). It plays an essential role in ma…

Kategori:
BenzoquinonesCoenzymesEnzymes and Coenzymes +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ubiquinone Q1 DB08689
small molecule | CAS: 727-81-1

Deskripsi belum tersedia.

Kategori:
BenzoquinonesCoenzymesEnzymes and Coenzymes +1
Target Protein:
Photosynthetic reaction center cytochrome c subunitReaction center protein H chainReaction center protein L chain +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ublituximab Approved DB11850
biotech | CAS: 1174014-05-1

CD20, an antigen expressed by various B and T cells, is an attractive therapeutic target in various cancers and autoimmune conditions.[A244195, A244200, A244205] Monoclonal antibodies for B cell depletion rely on their binding affinity and ability to clear bo…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +11
Target Protein:
B-lymphocyte antigen CD20
Waktu ParuhThe estimated mean …
Vol. DistribusiThe estimated centr…
Klirens-
Genetik -
Ubrogepant Approved DB15328
small molecule | CAS: 1374248-77-7

Ubrogepant is indicated for the acute treatment of migraine headaches with or without aura in adults.[L10926] It was approved by the FDA on December 23, 2019, and is the first oral calcitonin gene-related peptide (CGRP) receptor antagonist approved for the ac…

Kategori:
AnalgesicsAntimigraine PreparationsBCRP/ABCG2 Substrates +23
Target Protein:
Calcitonin gene-related peptide type 1 receptor
Waktu ParuhUbrogepant has an e…
Vol. DistribusiThe apparent centra…
KlirensThe apparent oral c…
Genetik -
UC-781 DB05871
small molecule | CAS: 178870-32-1

UC-781 is a thiocarboxanilide non-nucleoside reverse transcriptase inhibitor (NNRTI). It is a topical microbicide targeted against the AIDS virus.

Kategori:
AmidesAnti-Infective AgentsAnti-Retroviral Agents +2
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 11151–11200 dari 11778
Sebelumnya Halaman 224 / 236 Berikutnya