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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
Referensi
12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 224 / 252
SUVN-502 DB06140
small molecule | CAS: 701205-60-9

SUVN-502 is a novel, potent, safe, highly selective and orally active antagonist at a central nervous system serotonin receptor site 5-HT6 intended for treatment of cognitive disorders such as Alzheimer’s and Schizophrenia, an unmet medical need.

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsHeterocyclic Compounds, Fused-Ring +3
Target Protein:
5-hydroxytryptamine receptor 6
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SUVN-G3031 DB14835
small molecule | CAS: 1394808-82-2

SUVN-G3031 is under investigation in clinical trial NCT02342041 (A Study to Investigate the Safety, Tolerability and Pharmacokinetics of SUVN-G3031 in Healthy Subjects).

Kategori:
Oxazines
Target Protein:
Histamine H3 receptor
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Suvodirsen DB17940
biotech | CAS: 2095270-67-8

Suvodirsen is an antisense oligonucleotide that has been investigated for the treatment of Duchenne muscular dystrophy.

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Suvratoxumab DB15172
biotech | CAS: 1629620-18-3

Suvratoxumab is under investigation in clinical trial NCT02296320 (Study of the Efficacy and Safety of MEDI4893).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
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Suxibuzone DB13232
small molecule | CAS: 27470-51-5

Deskripsi belum tersedia.

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +13
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Suzetrigine DB18927
small molecule | CAS: 2649467-58-1

Suzetrigine is under investigation in clinical trial NCT05558410 (Evaluation of Efficacy and Safety of VX-548 for Acute Pain After an Abdominoplasty).

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Sweet cherry Approved DB10853
biotech

Sweet cherry allergenic extract is used in allergenic testing.

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Swordfish Approved DB10625
biotech

Swordfish allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
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SX-682 DB19210
small molecule | CAS: 1648843-04-2

SX-682 is under investigation in clinical trial NCT04574583 (Phase I/II Trial Investigating the Safety, Tolerability, Pharmacokinetics, Immune and Clinical Activity of SX-682 in Combination With Bintrafusp Alfa (M7824 or Tgf-beta "Trap"/pd-l1) With CV301 TRIC…

Target Protein:
C-X-C chemokine receptor type 2C-X-C chemokine receptor type 1
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SY-5609 DB17099
small molecule | CAS: 2417302-07-7

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
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SYD-003 DB17106
small molecule | CAS: 249937-52-8

Deskripsi belum tersedia.

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small molecule | CAS: 30344-00-4

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +1
Target Protein:
Haloalkane dehalogenase
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SYN-101 DB05958
biotech

SYN-101 is an investigational antibody-drug conjugate developed for the treatment of cancer. SYN101 is comprised of an immune cell specific antibody linked to an ALK5 inhibitor payload to selectively block TGF-b signalling in immune cells.

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SYNB1020 DB17667
biotech

SYNB1020 is an engineered strain of _Escherichia coli_ Nissle 1917 developed by Synlogic Inc. It was initially designed to convert ammonia to L-arginine [A258838] and granted orphan designation by the FDA for the treatment of urea cycle disorders in August 20…

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SYNB1353 DB17666
biotech

SYNB1353 is a strain of the probiotic bacteria _Escherichia coli_ (_E. coli_) type Nissle and an engineered probiotic drug.[A258833] Developed by Synlogic Operating Company, Inc., SYNB1353 is being investigated for the treatment of homocystinuria. It is desig…

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SYNB1891 DB17541
biotech

SYNB1891 is a live, modified strain of the probiotic _Escherichia coli_ Nissle engineered to produce cyclic di-AMP (CDA), a stimulator of the STING (STimulator of INterferon Genes) pathway.[A256733] SYNB1891 is under investigation in clinical trial NCT0416713…

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Synephrine DB09203
small molecule | CAS: 94-07-5

Synephrine, also referred to as, p-synephrine, is naturally occurring alkaloid. It is present in approved drug products as neo-synephrine, its m-substituted analog. p-synephrine and m-synephrine are known for their longer acting adrenergic effects compared to…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-Agonists +23
Target Protein:
Alpha-1 adrenergic receptors
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SynKIR-110 DB17365
biotech

SynKIR-110 are autologous T cells genetically engineered to express an anti-mesothelin killer immunoglobulin-like receptor-chimeric antigen receptor (KIR-CAR).

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SynOV1.1 DB17539
biotech

SynOV1.1 is an investigational cancer immunotherapy developed by SyngenTech. It is a recombinant oncolytic adenovirus, controlled by synthetic gene circuit, encoding the human immunostimulating factor cytokine granulocyte-macrophage colony-stimulating factor …

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Synthetic camphor Approved DB14156
small molecule | CAS: 76-22-2

Deskripsi belum tersedia.

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small molecule

Synthetic conjugated estrogens A are composed of a blend of the following nine synthetic estrogenic substances: estrone sulfate, sodium equilin sulfate, sodium 17?-dihydroequilin sulfate, sodium 17?-estradiol sulfate, sodium 17?­ dihydroequilin sulfate, sodiu…

Kategori:
Cytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 SubstratesCytochrome P-450 Substrates +7
Target Protein:
Estrogen receptor
Waktu ParuhThe half life of ba…
Vol. DistribusiThe distribution of…
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small molecule | CAS: 746658-13-9

Synthetic conjugated estrogens, B tablets contain a blend of ten synthetic estrogenic substances. The estrogenic substances are: sodium estrone sulfate, sodium equilin sulfate, sodium 17?-dihydroequilin sulfate, sodium 17?-estradiol sulfate, sodium 17?­ dihyd…

Kategori:
Cytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 SubstratesCytochrome P-450 Substrates +7
Target Protein:
Estrogen receptor
Waktu ParuhThe half life of ba…
Vol. DistribusiThe distribution of…
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SYRINGATE DB08589
small molecule

Deskripsi belum tersedia.

Target Protein:
Endo-1,4-beta-xylanase Y
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Syrosingopine Approved DB19379
small molecule | CAS: 84-36-6

Deskripsi belum tersedia.

Kategori:
AlkaloidsAntihypertensive AgentsHeterocyclic Compounds, Fused-Ring +5
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T-2000 DB11654
small molecule | CAS: 97846-21-4

T2000 has been used in trials studying the treatment of Myoclonus and Essential Tremor.

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T-5224 DB05998
small molecule | CAS: 530141-72-1

T-5224 is an investigational drug developed to treat Sepsis-induced Acute Kidney Injury. It's mechanism of action is to inhibit c-Fos/activator protein-1.

Kategori:
Benzene DerivativesKetones
Target Protein:
Transcription factor Jun
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T-900607 DB12068
small molecule | CAS: 261944-52-9

T900607 has been used in trials studying the treatment of Liver Cancer and Gastric Cancer.

Kategori:
AmidesSulfonesSulfur Compounds
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T-Guard DB18357
biotech

Deskripsi belum tersedia.

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T487 DB05474
small molecule

T487 is a small molecule chemokine receptor antagonist to correct or modify immune system responses. It binds selectively and potently to CXCR3. The formulation is administered orally and has anti-inflammatory effects in conditions such as rheumatoid arthriti…

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T611 DB06391
small molecule | CAS: 350595-61-8

T611 is an investigational oral anti-cytomegalovirus (CMV) drug candidate.

Target Protein:
Transmembrane anterior posterior transformation protein 1 homolog
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TA-CIN DB05809
biotech

TA-CIN is a subunit vaccine comprising L2/E6/E7 proteins from Human Papillomavirus (HPV16), designed to generate a strong cellular immune response against HPV-infected cells.

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TA-NIC DB05445
biotech

TA-NIC is a novel and proprietary vaccine in development as an aid to quitting smoking in motivated patients. It is designed to raise anti-nicotine antibodies which bind to nicotine molecules in the patient's blood stream, reducing the rate and quantity of ni…

Kategori:
Biological ProductsComplex Mixtures
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Tabalumab DB11657
biotech | CAS: 1143503-67-6

Tabalumab has been used in trials studying the treatment of Autoimmune Disease, Rheumatoid Arthritis, Kidney Failure, Chronic, Connective Tissue Disease, and Systemic Lupus Erythematosus, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
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Tabelecleucel Approved DB17072
biotech

Tabelecleucel is an innovative therapy that uses Epstein-Barr virus (EBV)-specific allogeneic cytotoxic T cells (CTLs). It is produced by mixing T-cells with B-cells that have been infected with the Epstein-Barr virus (EBV). Both T-cells and B-cells are obtai…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsAntineoplastic cell and gene therapy
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biotech | CAS: 943980-47-0

Taberminogene vadenovec (EG004) is a novel product consisting of a local delivery device and a gene-based medicine, being developed to prevent the blocking of veins and arteries that frequently occurs after vascular surgery. The initial target market is haemo…

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small molecule | CAS: 2412170-98-8

Tabirafusp tedromer is under investigation in clinical trial NCT06556368 (A Study to Evaluate the Efficacy and Safety of Tarcocimab Tedromer and Tabirafusp Tedromer Compared to Aflibercept in Participants With Neovascular (Wet) Age-related Macular Degeneratio…

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small molecule | CAS: 1612758-88-9

Deskripsi belum tersedia.

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Tacalcitol DB13689
small molecule | CAS: 57333-96-7

Deskripsi belum tersedia.

Kategori:
Anti-Inflammatory AgentsAntipsoriaticsAntipsoriatics for Topical Use +13
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Tacedinaline DB12291
small molecule | CAS: 112522-64-2

Tacedinaline has been used in trials studying the treatment of Lung Cancer, Multiple Myeloma, and Pancreatic Cancer.

Kategori:
Acids, CarbocyclicAmidesAmines +8
Target Protein:
Histone deacetylase 1
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Tacrine Approved DB00382
small molecule | CAS: 321-64-2

A centerally active cholinesterase inhibitor that has been used to counter the effects of muscle relaxants, as a respiratory stimulant, and in the treatment of Alzheimer's disease and other central nervous system disorders. Tacrine has been discontinued for t…

Kategori:
AcridinesAgents Causing Muscle ToxicityAminoacridines +16
Target Protein:
CholinesteraseAcetylcholinesteraseLiver carboxylesterase 1
Waktu Paruh2 to 4 hours
Vol. Distribusi* 349 ± 193 L
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Tacrolimus Approved DB00864
small molecule | CAS: 104987-11-3

Tacrolimus (also FK-506 or Fujimycin) is an immunosuppressive drug whose main use is after organ transplant to reduce the activity of the patient's immune system and so the risk of organ rejection. It is also used in a topical preparation in the treatment of …

Kategori:
Agents causing hyperkalemiaAgents Causing Muscle ToxicityAgents for Dermatitis, Excluding Corticosteroids +33
Target Protein:
Protein phosphatase 3 catalytic subunit alphaPeptidyl-prolyl cis-trans isomerase FKBP1A
Gen Terkait:
CYP3A5 ABCB1
Waktu ParuhThe elimination hal…
Vol. Distribusi* 2.6 ± 2.1 L/kg [p…
Klirens* 0.040 L/hr/kg [he…
Genetik 2 Varian
Tadalafil Approved DB00820
small molecule | CAS: 171596-29-5

Tadalafil is a selective phosphodiesterase-5 inhibitor that is used in the treatment of erectile dysfunction (ED), pulmonary arterial hypertension (PAH), and benign prostatic hypertrophy.[L39100, L39105] It was first approved in 2003 by the FDA for use in ED …

Kategori:
5-alpha Reductase InhibitorsAntihypertensive AgentsAntihypertensives for Pulmonary Arterial Hypertension +20
Target Protein:
cGMP-specific 3',5'-cyclic phosphodiesteraseDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11ARetinal rod rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit gamma
Waktu ParuhThe mean half-life …
Vol. DistribusiTadalafil has a mea…
KlirensThe mean apparent o…
Genetik -
Tadekinig alfa DB14858
biotech | CAS: 220712-29-8

Tadekinig alfa is under investigation in clinical trial NCT03113760 (Therapeutic Use of Tadekinig Alfa in NLRC4 Mutation and XIAP Deficiency).

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TAFA-93 DB05887
small molecule

TAFA93 is a novel prodrug of the mTOR inhibitor rapamycin which has successfully completed Phase 1 clinical development. mTOR inhibitors are currently used in the prevention of organ rejection in transplantation, the treatment of autoimmune and oncological di…

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Tafamidis Approved DB11644
small molecule | CAS: 594839-88-0

Tafamidis and tafamidis meglumine (FX-1006A) are benzoxazole derivatives[A27206] developed by FoldRX.[A189717] Tafamidis is structurally similar to diflusinal.[A189717] Tafamidis was granted an EMA market authorisation on 16 November 2011[L6247] and FDA ap…

Kategori:
Anti-Inflammatory AgentsBCRP/ABCG2 InhibitorsFused-Ring Compounds +8
Target Protein:
Transthyretin
Waktu ParuhThe half life of ta…
Vol. DistribusiThe apparent volume…
KlirensThe oral clearance …
Genetik -
Tafasitamab Approved DB15044
biotech | CAS: 1422527-84-1

Tafasitamab is a humanized, CD19-directed cytolytic monoclonal antibody intended for the treatment of B-cell malignancies.[L15302] It is produced using recombinant DNA technology in Chinese hamster ovary cells, and contains an IgG1/2 hybrid Fc-domain which ha…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +13
Target Protein:
B-lymphocyte antigen CD19
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe total volume of…
KlirensThe clearance of ta…
Genetik -
Tafenoquine Approved DB06608
small molecule | CAS: 106635-80-7

Tafenoquine is an 8-aminoquinoline analogue of primaquine which varies only on the presence of a 5-phenoxy group.[A35671, A35690] It was discovered by the scientists at the Walter Reed Army Institute of Research in 1978 as a substitute for primaquine that wou…

Kategori:
AminoquinolinesAnti-Infective AgentsAntimalarials +11
Waktu ParuhTafenoquine present…
Vol. DistribusiTafenoquine present…
KlirensTafenoquine present…
Genetik -
Tafolecimab DB16336
biotech | CAS: 2225109-03-3

Tafolecimab is under investigation in clinical trial NCT04031742 (A Study to Evaluate Safety and Efficacy of IBI306, a PCSK9 Monoclonal Antibody in Chinese Subjects With Homozygous Familial Hypercholesterolemia).

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Tagatose DB04936
small molecule | CAS: 87-81-0

Tagatose is a functional sweetener. It is a naturally occurring monosaccharide, specifically a hexose. It is commonly found in dairy with a similar texture and sweetened capacity to sucrose but with only a third of the calories. It is approved as a food addit…

Kategori:
CarbohydratesChelating AgentsCompounds used in a research, industrial, or household setting +3
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Tagetitoxin DB04788
small molecule | CAS: 87913-21-1

Tagetitoxin is a bacterial phytotoxin. It preferentially inhibits eukaryotic RNA polymerase.

Kategori:
Acids, AcyclicBacterial Toxins
Target Protein:
DNA-directed RNA polymerase subunit betaDNA-directed RNA polymerase subunit beta'
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