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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

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Distribusi Wujud Zat

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Hasil Pencarian (14063)

Halaman 224 / 282
Propanoyl-CoA DB02912
small molecule | CAS: 317-66-8

Deskripsi belum tersedia.

Kategori:
Adenine NucleotidesCoenzymesEnzymes and Coenzymes +7
Target Protein:
Propionyl-CoA carboxylase complex B subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propantheline Approved DB00782
small molecule | CAS: 298-50-0

A muscarinic antagonist used as an antispasmodic, in rhinitis, in urinary incontinence, and in the treatment of ulcers. At high doses it has nicotinic effects resulting in neuromuscular blocking.

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAmines +13
Target Protein:
Muscarinic acetylcholine receptor M1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Proparacaine Approved DB00807
small molecule | CAS: 499-67-2

Proparacaine is a topical anesthetic drug of the amino ester group. It is found in ophthalmic solutions at a concentration of 0.5% as the hydrochloride salt.

Kategori:
Acids, CarbocyclicAminobenzoatesAnesthetics +18
Target Protein:
Sodium channel protein type 10 subunit alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 2921-92-8

Deskripsi belum tersedia.

Kategori:
AlcoholsAntianginal AgentsCardiac Therapy +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propenidazole DB13319
small molecule | CAS: 76448-31-2

Deskripsi belum tersedia.

Kategori:
Antiparasitic Products, Insecticides and RepellentsAntiprotozoalsGenito Urinary System and Sex Hormones +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propentofylline DB06479
small molecule | CAS: 55242-55-2

Deskripsi belum tersedia.

Kategori:
AlkaloidsAnti-Ulcer AgentsCentral Nervous System Agents +12
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propicillin DB13660
small molecule | CAS: 551-27-9

Deskripsi belum tersedia.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propidium DB02166
small molecule | CAS: 36015-30-2

Quaternary ammonium analog of ethidium; an intercalating dye with a specific affinity to certain forms of DNA and, used as diiodide, to separate them in density gradients; also forms fluorescent complexes with cholinesterase which it inhibits. [PubChem]

Kategori:
Coloring AgentsCompounds used in a research, industrial, or household settingHeterocyclic Compounds, Fused-Ring +4
Target Protein:
Acetylcholinesterase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propiolactone Approved DB09348
small molecule | CAS: 57-57-8

Propiolactone is a lactone compound with a four-membered ring. It is a colorless liquid with a pungent slightly sweet odor. Propiolactone is a disinfectant used for the sterilization of blood plasma, vaccines, tissue grafts, surgical instruments, and enzymes.…

Kategori:
Anti-Infective AgentsCompounds used in a research, industrial, or household settingDisinfectants +1
Target Protein:
DNA
Waktu ParuhThe half-life of pr…
Vol. Distribusi-
Klirens-
Genetik -
Propiomazine Approved DB00777
small molecule | CAS: 362-29-8

Propiomazine, an atypical antipsychotic agent, is used to treat both negative and positive symptoms of schizophrenia, acute mania with bipolar disorder, agitation, and psychotic symptoms in dementia. Future uses may include the treatment of obsessive-compulsi…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +20
Target Protein:
Histamine H1 receptorMuscarinic acetylcholine receptorAlpha-1A adrenergic receptor +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propionate ion DB19384
small molecule | CAS: 72-03-7

Propionate ion is under investigation in clinical trial NCT00846326 (Preventing Tolerance to Oxymetazoline in Allergic Rhinitis).

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propiopromazine DB11540
small molecule | CAS: 3568-24-9

Deskripsi belum tersedia.

Kategori:
Antipsychotic AgentsCentral Nervous System DepressantsHeterocyclic Compounds, Fused-Ring +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propiverine Approved DB12278
small molecule | CAS: 60569-19-9

Propiverine is a widely used antimuscarinic drug with a mixed mode of action in the treatment of symptoms associated with overactive bladder (OAB) [A32576]. Overactive bladder (OAB) is a chronic condition of the lower urinary tract characterized by urinary…

Kategori:
Acids, CarbocyclicAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +22
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M3 +4
Waktu ParuhIn three studies in…
Vol. DistribusiIn one study, the v…
KlirensMean total clearanc…
Genetik -
Propofol Approved DB00818
small molecule | CAS: 2078-54-8

Propofol is an intravenous anaesthetic agent used for induction and maintenance of general anaesthesia. IV administration of propfol is used to induce unconsciousness after which anaesthesia may be maintained using a combination of medications. Recovery from …

Kategori:
Agents Causing Muscle ToxicityAgents that produce hypertensionAgents that reduce seizure threshold +32
Target Protein:
Gamma-aminobutyric acid receptor subunit beta-2Gamma-aminobutyric acid receptor subunit beta-3GABA(A) Receptor +2
Waktu ParuhInitial distributio…
Vol. Distribusi* 60 L/kg [healthy …
Klirens* 23 - 50 mL/kg/min…
Genetik -
small molecule | CAS: 184869-48-5

Deskripsi belum tersedia.

Kategori:
AnestheticsAnesthetics, General
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propoxycaine Approved DB09342
small molecule | CAS: 86-43-1

Propoxycaine is a local anesthetic of the ester type that has a rapid onset of action and a longer duration of action than procaine hydrochloride [L1588]. This drug was removed from the US market in 1996. Although no longer available in the United States,…

Kategori:
Acids, CarbocyclicAminobenzoatesAnesthetics +11
Target Protein:
Voltage-gated sodium channel alpha subunit
Waktu Paruh-
Vol. Distribusi-
KlirensVia the kidneys, pr…
Genetik -
Propranolol Approved DB00571
small molecule | CAS: 525-66-6

Propranolol is a racemic mixture of 2 enantiomers where the S(-)-enantiomer has approximately 100 times the binding affinity for beta adrenergic receptors.[L6904] Propranolol is used to treat a number of conditions but most commonly is used for hypertension.[…

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-Antagonists +37
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptorBeta-3 adrenergic receptor +2
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of pr…
Genetik -
Propyl alcohol Approved DB03175
small molecule | CAS: 71-23-8

A colorless liquid made by oxidation of aliphatic hydrocarbons that is used as a solvent and chemical intermediate.

Kategori:
AlcoholsAntiseptics and DisinfectantsDermatologicals +1
Target Protein:
Lysozyme C
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propyl Gallate DB12450
small molecule | CAS: 121-79-9

Propyl Gallate is under investigation in clinical trial NCT01450098 (A Study of LY2484595 in Healthy Subjects).

Kategori:
Acids, CarbocyclicAntioxidantsBenzene Derivatives +7
Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propylene glycol Approved DB01839
small molecule | CAS: 57-55-6

A clear, colorless, viscous organic solvent and diluent used in pharmaceutical preparations.

Kategori:
AlcoholsCompounds used in a research, industrial, or household settingDrug Delivery Systems +7
Target Protein:
B12-independent glycerol dehydratase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propylthiouracil Approved DB00550
small molecule | CAS: 51-52-5

A thiourea antithyroid agent. Propythiouracil inhibits the synthesis of thyroxine and inhibits the peripheral conversion of throxine to tri-iodothyronine. It is used in the treatment of hyperthyroidism. (From Martindale, The Extra Pharmacopeoia, 30th ed, p534)

Kategori:
Agents Causing Muscle ToxicityAntimetabolitesAntithyroid agents +14
Target Protein:
Type I iodothyronine deiodinaseThyroid peroxidase
Waktu Paruh2 hours
Vol. Distribusi-
Klirens-
Genetik -
Propyphenazone DB13524
small molecule | CAS: 479-92-5

Deskripsi belum tersedia.

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Proquazone DB13649
small molecule | CAS: 22760-18-5

Deskripsi belum tersedia.

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Proscillaridin DB13307
small molecule | CAS: 466-06-8

Proscillaridin is a cardiac glycoside that is derived from plants of the genus Scilla and in Drimia maritima (Scilla maritima). Studies suggest the potential cytotoxic and anticancer property of proscillaridin, based on evidence of the drug potently disruptin…

Kategori:
BufanolidesCarbohydratesCardanolides +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 13367-85-6

Deskripsi belum tersedia.

Kategori:
AutacoidsBiological FactorsEicosanoids +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 41598-07-6

The principal cyclooxygenase metabolite of arachidonic acid. It is released upon activation of mast cells and is also synthesized by alveolar macrophages. Among its many biological actions, the most important are its bronchoconstrictor, platelet-activating-fa…

Kategori:
AutacoidsBiological FactorsEicosanoids +7
Target Protein:
Prostaglandin D2 receptorProstaglandin F2-alpha receptorProstaglandin E2 receptor EP1 subtype +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

A cyclic endoperoxide intermediate produced by the action of CYCLOOXYGENASE on ARACHIDONIC ACID. It is further converted by a series of specific enzymes to the series 2 prostaglandins. [PubChem]

Kategori:
AnionsAutacoidsBiological Factors +14
Target Protein:
Prostaglandin G/H synthase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prostalene DB11454
small molecule | CAS: 54120-61-5

Analog of prostaglandin F2 alpha.

Kategori:
AutacoidsBiological FactorsEicosanoids +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Protamine DB13700
small molecule | CAS: 9012-00-4

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntidotesCoagulants +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Protego-PD DB18279
biotech

Protego-PD is a post-delivery placental extract.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Protein C Approved DB11312
biotech

Protein C is an endogenously occurring plasma protein that plays a key role within the coagulation cascade. Protein C is a zymogen, or enzyme precursor, of a vitamin K-dependent anticoagulant glycoprotein (serine protease) that is synthesized in the liver. It…

Kategori:
Amino Acids, Peptides, and ProteinsAnticoagulantsBiological Factors +15
Target Protein:
Coagulation factor VCoagulation factor VIII
Waktu ParuhInitial half life =…
Vol. DistribusiVolume of distribut…
KlirensCL = 0.0533 dL/kg/h
Genetik -
Prothipendyl DB12958
small molecule | CAS: 303-69-5

Prothipendyl has been used in trials studying the treatment of Dementia, Depression, Schizophrenia, Anxiety Disorders, and Psychosomatic Disorders.

Kategori:
Antipsychotic AgentsCentral Nervous System DepressantsNervous System +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prothrombin Approved DB11311
biotech | CAS: 9001-26-7

Prothrombin Complex Concentrate (Human), is indicated for the urgent reversal of acquired coagulation factor deficiency induced by Vitamin K antagonist (VKA, e.g., warfarin) therapy in adult patients with acute major bleeding.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +7
Target Protein:
Fibrinogen alpha chainFibrinogen beta chainCoagulation factor XIII A chain +1
Waktu ParuhApproximately 60h […
Vol. Distribusi-
Klirens-
Genetik -
Protiofate DB13632
small molecule | CAS: 58416-00-5

Deskripsi belum tersedia.

Kategori:
Genito Urinary System and Sex HormonesGynecological Antiinfectives and Antiseptics
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Protionamide Approved DB12667
small molecule | CAS: 14222-60-7

Prothionamide has been used in trials studying the treatment of MDR-TB and HIV Infections.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntiinfectives for Systemic Use +5
Target Protein:
Enoyl-[acyl-carrier-protein] reductase [NADH]
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Protirelin Approved DB09421
small molecule | CAS: 24305-27-9

Protirelin is the pharmaceutically available synthetic analogue of the endogenous peptide thyrotropin-releasing hormone (TRH). It is a tri-peptide tropic hormone, released by the hypothalamus, that stimulates the release of Thyroid Stimulating Hormone (TSH) a…

Kategori:
Amino Acids, Peptides, and ProteinsDiagnostic AgentsHormones +12
Target Protein:
Thyrotropin-releasing hormone receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 139-85-5

Also known as protocatechuic aldehyde, protocatechualdehyde is a naturally-occuring phenolic aldehyde that is found in barley, green cavendish bananas, grapevine leaves and root of the herb S. miltiorrhiza [A27224]. Protocatechualdehyde possesses antiprolifer…

Kategori:
AldehydesAnticoagulantsBenzene Derivatives +2
Target Protein:
Amine oxidase [flavin-containing] B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Protoporphyrin DB02285
small molecule | CAS: 553-12-8

Deskripsi belum tersedia.

Kategori:
Biological FactorsDermatologicalsHeterocyclic Compounds, Fused-Ring +4
Target Protein:
Hematopoietic prostaglandin D synthaseFerritin light chain
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Prostaglandin G/H synthase 1Cytochrome c
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Protriptyline Approved DB00344
small molecule | CAS: 438-60-8

Protriptyline hydrochloride is a dibenzocycloheptene-derivative tricyclic antidepressant (TCA). TCAs are structurally similar to phenothiazines. They contain a tricyclic ring system with an alkyl amine substituent on the central ring. In non-depressed individ…

Kategori:
Adrenergic AgentsAdrenergic Uptake InhibitorsAgents that produce hypertension +24
Target Protein:
Sodium-dependent noradrenaline transporterSodium-dependent serotonin transporter
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Proxalutamide DB16065
small molecule | CAS: 1398046-21-3

Proxalutamide is under investigation in clinical trial NCT03899467 (The Safety and Tolerability of Proxalutamide (GT0918) in Subjects With Metastatic Castrate Resistant Prostate Cancer).

Kategori:
HydantoinsImidazolesImidazolidines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Proxibarbal Approved DB13253
small molecule | CAS: 2537-29-3

Proxibarbal is a derivative of barbiturates, which has been used to treat migraines. Proxibarbal was approved in France but was withdrawn from the market due to the risk of inducing immunoallergic thrombocytopenia [L5476].

Kategori:
Barbiturates, PlainCentral Nervous System AgentsCentral Nervous System Depressants +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prucalopride Approved DB06480
small molecule | CAS: 179474-81-8

Prucalopride is a dihydrobenzofurancarboxamide derivative from the benzofurane family that selectively stimulates 5-HT4 receptors and thus, it presents enterokinetic properties.[A37348] The high selectivity of prucalopride allowed further development as it pr…

Kategori:
Alimentary Tract and MetabolismAntidepressive AgentsCentral Nervous System Depressants +17
Target Protein:
5-hydroxytryptamine receptor 4
Waktu ParuhThe reported half-l…
Vol. DistribusiThe mean volume of …
KlirensPrucalopride renal …
Genetik -
Prulifloxacin DB11892
small molecule | CAS: 123447-62-1

Prulifloxacin has been investigated for the treatment of Urinary Tract Infection.

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +15
Target Protein:
DNA topoisomerase 4 subunit ADNA gyrase subunit ADNA gyrase subunit B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pruvanserin DB13094
small molecule | CAS: 443144-26-1

Pruvanserin has been used in trials studying the treatment of Sleep Initiation and Maintenance Disorders.

Target Protein:
5-hydroxytryptamine receptor 2A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PRX-03140 DB05596
small molecule | CAS: 869493-21-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PRX-07034 DB05993
small molecule | CAS: 903580-39-2

Deskripsi belum tersedia.

Target Protein:
5-hydroxytryptamine receptor 6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PRX-08066 DB05607
small molecule

Deskripsi belum tersedia.

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsSerotonin 5-HT2 Receptor Antagonists +3
Target Protein:
5-hydroxytryptamine receptor 2B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PS386113 DB05211
small molecule

PS386113 is a small molecule drug candidate under investigation for the treatment of inflammatory disorders. It is being developed by Schering-Plough and Pharmacopeia. Little information has been released about PS386113.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pseudoephedrine Approved DB00852
small molecule | CAS: 90-82-4

Pseudoephedrine is structurally related to [ephedrine] but exerts a weaker effect on the sympathetic nervous system.[A188820,A188823] Both drugs naturally occur in in ephedra plant which have a history of use in traditional Eastern medicine and were first res…

Kategori:
Adrenergic AgonistsAdrenergic alpha-1 Receptor AgonistsAdrenergic alpha-2 Receptor Agonists +30
Target Protein:
Sodium-dependent noradrenaline transporterD(2) dopamine receptorSodium-dependent dopamine transporter +10
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe apparent volume…
KlirensA 60mg oral dose of…
Genetik -
Menampilkan 11151–11200 dari 14063
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