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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 223 / 282
Prilocaine Approved DB00750
small molecule | CAS: 721-50-6

A local anesthetic that is similar pharmacologically to lidocaine. Currently, it is used most often for infiltration anesthesia in dentistry. (From AMA Drug Evaluations Annual, 1992, p165)

Kategori:
AmidesAminesAnesthetics +11
Target Protein:
Sodium channel protein type 5 subunit alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Primidone Approved DB00794
small molecule | CAS: 125-33-7

Primidone is an anticonvulsant used to treat essential tremor as well as grand mal, psychomotor, and focal epileptic seizures.[L11112] Primidone was developed by J Yule Bogue and H C Carrington in 1949.[A189522] Primidone was granted FDA Approval on 8 Marc…

Kategori:
Anti-epileptic AgentAnticholinergic AgentsAnticonvulsants +36
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-2Gamma-aminobutyric acid receptor subunit alpha-3Gamma-aminobutyric acid receptor subunit alpha-4 +8
Waktu ParuhThe half life of pr…
Vol. DistribusiThe volume of distr…
KlirensPrimidone is cleare…
Genetik -
Prinaberel DB06832
small molecule | CAS: 524684-52-4

Prinaberel is an estrogen receptor beta agonist.

Kategori:
Receptors, Estrogen, agonists
Target Protein:
Estrogen receptor betaNuclear receptor coactivator 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prinomastat DB05100
small molecule | CAS: 192329-42-3

Prinomastat is a synthetic hydroxamic acid derivative with potential antineoplastic activity. Prinomastat inhibits matrix metalloproteinases (MMPs) (specifically, MMP-2, 9, 13, and 14), thereby inducing extracellular matrix degradation, and inhibiting angioge…

Kategori:
Enzyme InhibitorsMatrix Metalloproteinase InhibitorsProtease Inhibitors
Target Protein:
72 kDa type IV collagenaseInterstitial collagenaseMatrilysin
Waktu Paruh2-5 hours
Vol. Distribusi-
Klirens-
Genetik -
Pristimerin DB17049
small molecule | CAS: 1258-84-0

Pristimerin is a quinone methide triterpenoid researched for its anti-cancer potential.[A253107]

Kategori:
TerpenesTriterpenes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pristinamycin DB13704
small molecule | CAS: 270076-60-3

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pritelivir DB11844
small molecule | CAS: 348086-71-5

Pritelivir has been used in trials studying the prevention of HSV-2 and Genital Herpes.

Kategori:
AmidesAnti-Infective AgentsAntiviral Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pritumumab DB17221
biotech | CAS: 499212-74-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

C-CAR039 is an autologous Chimeric Antigen Receptors (CAR) T-cell therapy expressing CD19/CD20 bi-specific CAR.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PRO 2000 DB05385
small molecule | CAS: 29321-75-3

PRO 2000 is an investigational medicine that is not yet approved by the FDA for use outside of clinical trials. It is being studied for the prevention of HIV infection and other sexually transmitted diseases. This medicine does not cure HIV infection or AIDS …

Kategori:
ArylsulfonatesArylsulfonic AcidsCompounds used in a research, industrial, or household setting +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PRO-542 DB05793
biotech

PRO 542 belongs to a new class of drugs, viral-entry inhibitor, which is intended to prevent HIV from entering and infecting cells. PRO 542 (CD4-immunoglobulin G2) is a tetravalent CD4-immunoglobulin fusion protein that broadly neutralizes primary HIV-1 isola…

Kategori:
Amino Acids, Peptides, and ProteinsAntigensAntigens, Surface +21
Target Protein:
Free fatty acid receptor 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1616927-79-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Probenecid Approved DB01032
small molecule | CAS: 57-66-9

The prototypical uricosuric agent. It inhibits the renal excretion of organic anions and reduces tubular reabsorption of urate. Probenecid has also been used to treat patients with renal impairment, and, because it reduces the renal tubular excretion of other…

Kategori:
Adjuvants, PharmaceuticAmidesAntigout Preparations +29
Target Protein:
Solute carrier family 22 member 6Solute carrier family 22 member 11Organic anion transporter 3 +2
Waktu Paruh6-12 hours
Vol. Distribusi-
Klirens-
Genetik -
Probiorinse DB15870
biotech

Probiorinse is an intranasal probiotic treatment composed of a pre-mixed and buffered sinus irrigation solution that contains the probiotic bacteria Lactococcus lactis W136.[L16368] This strain of bacteria is said to have salubrious effects on the microbiome …

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Probucol Approved DB01599
small molecule | CAS: 23288-49-5

A drug used to lower LDL and HDL cholesterol yet has little effect on serum-triglyceride or VLDL cholesterol. (From Martindale, The Extra Pharmacopoeia, 30th ed, p993).

Kategori:
Anticholesteremic AgentsAntioxidantsBenzene Derivatives +10
Target Protein:
Phospholipid-transporting ATPase ABCA1Liver carboxylesterase 1
Waktu ParuhRanges from 12 hour…
Vol. Distribusi-
Klirens-
Genetik -
Procainamide Approved DB01035
small molecule | CAS: 51-06-9

A derivative of procaine with less CNS action.

Kategori:
Acids, CarbocyclicAgents Causing Muscle ToxicityAgents that produce neuromuscular block (indirect) +32
Target Protein:
Voltage-gated inwardly rectifying potassium channel KCNH2Sodium channel protein type 5 subunit alphaDNA (cytosine-5)-methyltransferase 1
Waktu Paruh~2.5-4.5 hours
Vol. Distribusi* 2 L/kg
Klirens-
Genetik -
Procaine Approved DB00721
small molecule | CAS: 59-46-1

A local anesthetic of the ester type that has a slow onset and a short duration of action. It is mainly used for infiltration anesthesia, peripheral nerve block, and spinal block. (From Martindale, The Extra Pharmacopoeia, 30th ed, p1016). Procaine has also b…

Kategori:
Acids, CarbocyclicAgents for Treatment of Hemorrhoids and Anal Fissures for Topical UseAgents that reduce seizure threshold +25
Target Protein:
Sodium channel protein type 10 subunit alphaGlutamate receptor ionotropic, NMDA 3A5-hydroxytryptamine receptor 3A +8
Waktu Paruh7.7 minutes
Vol. Distribusi-
Klirens-
Genetik -
Procaine benzylpenicillin Approved DB09320
small molecule | CAS: 54-35-3

Procaine benzylpenicillin (INN), also known as procaine G penicillin, is an injectable antiobiotic. It is a poorly soluble salt form of penicillin which is a combination of naturally occuring benzylpenicillin (penicillin G) and the local anaesthetic agent pro…

Kategori:
Acids, CarbocyclicAmidesAminobenzoates +16
Target Protein:
Penicillin-binding protein
Waktu ParuhIntramuscular injec…
Vol. DistribusiThe drug is distrib…
Klirens-
Genetik -
Procaine merethoxylline Approved DB09364
small molecule | CAS: 60064-28-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Procalcitonin DB14812
biotech | CAS: 56645-65-9

Procalcitonin is under investigation in clinical trial NCT03440060 (Procalcitonin-guided Antibiotic Therapy During Severe Exacerbation of COPD).

Kategori:
Amino Acids, Peptides, and ProteinsBone Density Conservation AgentsCalcitonin Preparations +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Procarbazine Approved DB01168
small molecule | CAS: 671-16-9

An antineoplastic agent used primarily in combination with mechlorethamine, vincristine, and prednisone (the MOPP protocol) in the treatment of Hodgkin's disease.

Kategori:
Acids, CarbocyclicAgents Causing Muscle ToxicityAlkylating Activity +17
Target Protein:
Monoamine oxidaseDNA
Waktu Paruh10 minutes
Vol. Distribusi-
Klirens-
Genetik -
Procaterol Approved DB01366
small molecule | CAS: 72332-33-3

A long-acting beta-2-adrenergic receptor agonist. It is a potent bronchodilator that may be administered orally or by aerosol inhalation.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic beta-2 Receptor Agonists +21
Target Protein:
Beta-2 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prochlorperazine Approved DB00433
small molecule | CAS: 58-38-8

Prochlorperazine, also known as compazine, is a piperazine phenothiazine and first-generation antipsychotic drug that is used for the treatment of severe nausea and vomiting, as well as short-term management of psychotic disorders such as generalized non-psyc…

Kategori:
AntiemeticsAntipsychotic AgentsAntipsychotic Agents (First Generation [Typical]) +28
Target Protein:
D(2) dopamine receptorHistamine H1 receptorAlpha-1 adrenergic receptors +1
Waktu ParuhFollowing intraveno…
Vol. DistribusiIn a preliminary ph…
KlirensThe mean plasma cle…
Genetik -
Procinonide Approved DB18737
small molecule | CAS: 58497-00-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Procyclidine Approved DB00387
small molecule | CAS: 77-37-2

A muscarinic antagonist that crosses the blood-brain barrier and is used in the treatment of drug-induced extrapyramidal disorders and in parkinsonism.

Kategori:
Agents producing tachycardiaAnti-Dyskinesia AgentsAnti-Parkinson Drugs +8
Target Protein:
Muscarinic acetylcholine receptor M3Muscarinic acetylcholine receptor M5Muscarinic acetylcholine receptor M1 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Profadol DB17993
small molecule | CAS: 428-37-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Profenamine Approved DB00392
small molecule | CAS: 522-00-9

Profenamine (also known as ethopropazine) is a medication derived from phenothiazine. It is primarily used as an antidyskinetic to treat Parkinsonism. It is sold under the trade name Parsitan in Canada.[L46812] In the US, the marketing of profenamine has been…

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAgents producing tachycardia +12
Target Protein:
Histamine H1 receptorMuscarinic acetylcholine receptor M1Glutamate receptor ionotropic, NMDA 3A +1
Waktu Paruh1 to 2 hours
Vol. Distribusi-
Klirens-
Genetik -
Proflavine Approved DB01123
small molecule | CAS: 92-62-6

3,6-Diaminoacridine. Topical antiseptic used mainly in wound dressings.

Kategori:
AcridinesAminoacridinesAnti-Infective Agents +2
Target Protein:
DNAProthrombinHTH-type transcriptional regulator QacR +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Profoxydim DB14820
small molecule | CAS: 139001-49-3

Profoxydim is under investigation in clinical trial NCT02728011 (Pilot Trial Comparing Computerised Cognitive Exercises to Tetris in Adolescents With ADHD).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Progabide DB00837
small molecule | CAS: 62666-20-0

Progabide is an analog and prodrug of gamma-aminobutyric acid. It is commonly used in the treatment of epilepsy. It has agonistic activity for both the GABAA and GABAB receptors. In clinical trials, progabide has been investigated for Parkinson's disease, sch…

Kategori:
Acids, AcyclicAmino AcidsAmino Acids, Peptides, and Proteins +14
Target Protein:
Gamma-aminobutyric acid type B receptor subunit 2Gamma-aminobutyric acid receptor subunit alpha-1Gamma-aminobutyric acid type B receptor subunit 1
Waktu Paruh4 hours
Vol. Distribusi-
Klirens-
Genetik -
Progesterone Approved DB00396
small molecule | CAS: 57-83-0

Progesterone is a hormone that occurs naturally in females, and is essential for endometrial receptivity, embryo implantation, and the successful establishment of pregnancy. A low progesterone concentration or an insufficient response to progesterone can caus…

Kategori:
Adrenal Cortex HormonesBCRP/ABCG2 InducersBCRP/ABCG2 Inhibitors +47
Target Protein:
Progesterone receptorMineralocorticoid receptorEstrogen receptor +7
Waktu ParuhAbsorption half-lif…
Vol. DistribusiWhen administered v…
Klirens**Apparent clearanc…
Genetik -
Proglumetacin DB13527
small molecule | CAS: 57132-53-3

Deskripsi belum tersedia.

Kategori:
Acetic Acid Derivatives and Related SubstancesAgents causing hyperkalemiaAgents that produce hypertension +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Proglumide DB13431
small molecule | CAS: 6620-60-6

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismAmino AcidsAmino Acids, Basic +7
Target Protein:
Cholecystokinin receptor type A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Proguanil Approved DB01131
small molecule | CAS: 500-92-5

Proguanil is a prophylactic antimalarial drug, which works by stopping the malaria parasite, _Plasmodium falciparum_ and _Plasmodium vivax_, from reproducing once it is in the red blood cells. It does this by inhibiting the enzyme, dihydrofolate reductase, wh…

Kategori:
AmidinesAnti-Infective AgentsAntimalarials +15
Target Protein:
Dihydrofolate reductasePeptide deformylase, mitochondrialBifunctional dihydrofolate reductase-thymidylate synthase
Gen Terkait:
CYP2C19 CYP2C19
Waktu ParuhApproximately 20 ho…
Vol. Distribusi-
Klirens-
Genetik 2 Varian
biotech | CAS: 67422-14-4

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsBlood Glucose Lowering AgentsHormones +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prolactin G129R DB18431
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prolease-r-hFSH DB05826
biotech

Prolease-r-hFSH is a recombinant human follicle stimulating hormone (r-hFSH) with Alkermes' ProLease injectable sustained release drug delivery technology. It provides patients with long term therapeutic benefit from a single administration rather than multip…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prolectin-M DB16521
small molecule

Prolectin-M is a (1-6)-alpha-D-mannopyranose[L31338] and acts as an antagonist of galectin.[L31343] It is being investigated in the clinical trial NCT04512027 (Prolectin-M in COVID-19 Patients Having Mild to Moderate Symptoms Not Requiring Oxygen Support. (Pr…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prolgolimab DB16740
biotech | CAS: 2093956-19-3

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsMonoclonal antibodies and antibody drug conjugates +2
Target Protein:
Programmed cell death protein 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Proline DB00172
small molecule | CAS: 147-85-3

Proline is one of the twenty amino acids used in living organisms as the building blocks of proteins. Proline is sometimes called an imino acid, although the IUPAC definition of an imine requires a carbon-nitrogen double bond. Proline is a non-essential amino…

Kategori:
Amino AcidsAmino Acids, CyclicAmino Acids, Peptides, and Proteins +4
Target Protein:
Peptidyl-prolyl cis-trans isomerase BPeptidyl-prolyl cis-trans isomerase APyrroline-5-carboxylate reductase 1, mitochondrial +19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prolintane DB13438
small molecule | CAS: 493-92-5

Deskripsi belum tersedia.

Kategori:
Central Nervous System AgentsCentral Nervous System StimulantsNervous System +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Promazine Approved DB00420
small molecule | CAS: 58-40-2

A phenothiazine with actions similar to chlorpromazine but with less antipsychotic activity. It is primarily used in short-term treatment of disturbed behavior and as an antiemetic. It is currently not approved for use in the United States.

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +49
Target Protein:
D(2) dopamine receptorMuscarinic acetylcholine receptor M55-hydroxytryptamine receptor 2A +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Promegestone DB13602
small molecule | CAS: 34184-77-5

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Substrates +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Promestriene DB12487
small molecule | CAS: 39219-28-8

Promestriene (3-propyl ethyl, 17B-methyl estradiol) has been used in trials studying the prevention of Hypospadias. It is a synthetic estrogen analog, which is used in topical estrogen therapy. Promestriene’s potential for treating vaginal atrophy symptoms as…

Kategori:
Estradiol CongenersEstranesEstrenes +10
Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Promethazine Approved DB01069
small molecule | CAS: 60-87-7

Promethazine, originally known as 3,277 R.P., is an N-dimethylaminopropyl derivative of [phenothiazine] that was developed in France in 1946.[A189901] Promethazine antagonizes a variety of receptors, allowing it to be used for a number of indications includin…

Kategori:
Acid ReducersAgents producing tachycardiaAgents that reduce seizure threshold +44
Target Protein:
Histamine H1 receptorD(2) dopamine receptorMuscarinic acetylcholine receptor M1 +10
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe intravenous cle…
Genetik -
Propacetamol DB09288
small molecule | CAS: 66532-85-2

Propacetamol is a non-opioid analgesic devoid of the major contraindications.[A32051] It is a derivative of [acetaminophen], or paracetamol, with the molecular formula glycine, N, N-diethyl-,4-(acetylamino)phenyl ester. Propacetamol is a parenteral formulatio…

Kategori:
Acetaminophen and ProdrugsAcetanilidesAgents causing hyperkalemia +37
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2Transient receptor potential cation channel subfamily V member 1 +1
Waktu ParuhThe half-life of pr…
Vol. DistribusiThe volume of distr…
KlirensThe clearance rate …
Genetik -
Propafenone Approved DB01182
small molecule | CAS: 54063-53-5

An antiarrhythmia agent that is particularly effective in ventricular arrhythmias. It also has weak beta-blocking activity. The drug is generally well tolerated.

Kategori:
Adrenergic AntagonistsAdrenergic beta-AntagonistsAgents causing hyperkalemia +25
Target Protein:
Sodium channel protein type 5 subunit alphaVoltage-gated inwardly rectifying potassium channel KCNH2Beta-1 adrenergic receptor +1
Waktu Paruh2-10 hours
Vol. Distribusi* 252 L
Klirens-
Genetik -
Propagermanium DB17608
small molecule | CAS: 12758-40-6

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAntineoplastic AgentsElements +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propamidine DB13296
small molecule | CAS: 104-32-5

Deskripsi belum tersedia.

Kategori:
AmidinesAnti-Infective AgentsAntiparasitic Agents +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propanidid DB13234
small molecule | CAS: 1421-14-3

An intravenous anesthetic that has been used for rapid induction of anesthesia and for maintenance of anesthesia of short duration. (From Martindale, The Extra Pharmacopoeia, 30th ed, p918)

Kategori:
Acids, CarbocyclicAminesAnesthetics +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 11101–11150 dari 14063
Sebelumnya Halaman 223 / 282 Berikutnya