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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 222 / 236
Trichophyton tonsurans Approved DB10970
biotech

Trichophyton tonsurans is a fungus which can provoke allergic reactions. Trichophyton tonsurans extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trichosporon cutaneum Approved DB10974
biotech

Trichosporon cutaneum allergenic extract is used in allergenic testing.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trichostatin A DB04297
small molecule | CAS: 58880-19-6

Deskripsi belum tersedia.

Kategori:
AminesAnti-Infective AgentsAntifungal Agents +9
Target Protein:
Histone deacetylase 7Histone deacetylase 8Acetoin utilization protein +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Triclabendazole Approved DB12245
small molecule | CAS: 68786-66-3

Triclabendazole, manufactured by Novartis pharmaceuticals, is an antihelminthic drug that was approved by the FDA in February 2019 for the treatment of fascioliasis in humans.[FDA label, L5452] Fascioliasis is a parasitic infection often caused by the helmi…

Kategori:
AnthelminticsAnti-Infective AgentsAntihelminthic +34
Target Protein:
CruzipainExcretory Secretory (ES) proteins
Waktu ParuhThe plasma eliminat…
Vol. DistribusiThe apparent volume…
Klirens-
Genetik -
Triclocarban Approved DB11155
small molecule | CAS: 101-20-2

Triclocarban, with the chemical formula C13H9Cl3N2O [L2675] is an antibacterial agent that is particularly effective against Gram-positive bacteria such as *Staphylococcus aureus*. It is a bacteriostatic compound that has been found in antibacterial soaps and…

Kategori:
AmidesAminesAnilides +10
Target Protein:
Enoyl-[acyl-carrier-protein] reductase [NADPH] FabI
Waktu Paruh10 hours [L2680]
Vol. Distribusi-
KlirensAfter a pharmacokin…
Genetik -
Triclofos Approved DB06753
small molecule | CAS: 306-52-5

Deskripsi belum tersedia.

Kategori:
Central Nervous System DepressantsHypnotics and SedativesNervous System +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 2433-96-7

Deskripsi belum tersedia.

Kategori:
Fatty AcidsLipids
Target Protein:
Lipase 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tricyclazole DB02891
small molecule | CAS: 41814-78-2

Deskripsi belum tersedia.

Kategori:
Sulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tridecactide DB15687
small molecule | CAS: 22006-64-0

Tridecactide, also known as alpha-corticotropin 1-13, is a deacetylated and deaminated alpha-melanocyte stimulating hormone, which may have antipyretic, anti-inflammatory, and antimicrobial effects.[A203210] Tridecactide, along with [metenkefalin], are under …

Kategori:
Experimental Unapproved Treatments for COVID-19Melanocyte-Stimulating Hormones
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tridolgosir DB02034
small molecule | CAS: 72741-87-8

An indolizidine alkaloid from the plant Swainsona canescens that is a potent alpha-mannosidase inhibitor. Swainsonine also exhibits antimetastatic, antiproliferative, and immunomodulatory activity.

Target Protein:
Alpha-mannosidase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 2943-75-1

Deskripsi belum tersedia.

Kategori:
NaphthalenesQuinonesSilicon Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 77-93-0

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicTricarboxylic Acids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 78-40-0

Deskripsi belum tersedia.

Kategori:
Organophosphorus Compounds
Target Protein:
Parathion hydrolaseCellular tumor antigen p53Parathion hydrolase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 112-27-6

Deskripsi belum tersedia.

Kategori:
AlcoholsCompounds used in a research, industrial, or household settingEthylene Glycols +3
Target Protein:
Acetolactate synthase, catabolicArabinogalactan endo-beta-1,4-galactanasePhosphoserine aminotransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Triethylenetetramine Approved DB06824
small molecule | CAS: 112-24-3

Triethylenetatramine (TETA), also known as trientine, is a potent and selective copper (II)-selective chelator. It is a structural analog of linear polyamine compounds, [spermidine] and [spermine]. TETA was first developed in Germany in 1861 and its chelating…

Kategori:
Alimentary Tract and MetabolismAminesChelating Agents +11
Target Protein:
Carbonic anhydrase 14
Waktu ParuhThe mean terminal h…
Vol. DistribusiTETA is widely dist…
KlirensIn healthy adult vo…
Genetik -
small molecule | CAS: 7360-38-5

Triethylhexanoin is an ingredient of cosmetic products as a fragrant solvent.

Kategori:
Acids, AcyclicCompounds used in a research, industrial, or household settingExcipients +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trifarotene Approved DB12808
small molecule | CAS: 895542-09-3

Trifarotene is a topical retinoid cream used in the treatment of acne vulgaris that was first approved for use in the United States in October 2019.[L9013] Retinoids are a class of medications structurally and functionally analogous to [vitamin A], though lat…

Kategori:
AlkenesAnti-Acne PreparationsAnti-Acne Preparations for Topical Use +11
Target Protein:
Retinoic acid receptor gammaRetinoic acid receptor betaRetinoic acid receptor alpha
Waktu ParuhThe terminal half-l…
Vol. Distribusi-
Klirens-
Genetik -
Trifluoperazine Approved DB00831
small molecule | CAS: 117-89-5

A phenothiazine with actions similar to chlorpromazine. It is used as an antipsychotic and an antiemetic.

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +29
Target Protein:
D(2) dopamine receptorCalmodulin-1Calmodulin-3 +6
Waktu Paruh10-20 hours
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Myosin-14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 75-89-8

A non-aqueous co-solvent that serves as tool to study protein folding. It is also used in various pharmaceutical, chemical and engineering applications.

Kategori:
Alcohols
Target Protein:
Alcohol dehydrogenase 1CGTPase HRasAlcohol dehydrogenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, NeutralAmino Acids, Peptides, and Proteins +2
Target Protein:
Methionine--tRNA ligaseMethionine aminopeptidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trifluperidol DB13552
small molecule | CAS: 749-13-3

Deskripsi belum tersedia.

Kategori:
Antipsychotic AgentsButyrophenone DerivativesButyrophenones +11
Target Protein:
Chymase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trifluridine Approved DB00432
small molecule | CAS: 70-00-8

Trifluridine is a fluorinated pyrimidine nucleoside that is structurally related to [idoxuridine] [A35271]. It is an active antiviral agent in ophthalmic solutions used mainly in the treatment of primary keratoconjunctivitis and recurrent epithelial keratitis…

Kategori:
Anti-Infective AgentsAntimetabolitesAntineoplastic Agents +20
Target Protein:
Thymidylate synthaseDNAThymidylate synthase
Waktu ParuhAfter administratio…
Vol. DistribusiFollowing a single …
KlirensFollowing a single …
Genetik -
Triflusal Approved DB08814
small molecule | CAS: 322-79-2

Triflusal is a 2-acetoxy-4-trifluoromethylbenzoic acid and it is an aspirin chemically-related molecule but not a derivative. The benefits of this agent are the lack of action over the arachidonic acid pathway, the driven production of nitric oxide and the in…

Kategori:
Acids, CarbocyclicAnticoagulantsAntiplatelet agents +8
Target Protein:
Prostaglandin G/H synthase 1Nuclear factor NF-kappa-B p105 subunitNitric oxide synthase, inducible +1
Waktu ParuhIn the healthy huma…
Vol. DistribusiThe reported volume…
KlirensRenal clearance is …
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Folic Acid and DerivativesVitamin B ComplexVitamins
Target Protein:
Serine hydroxymethyltransferase, cytosolic
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Triglyme DB02078
small molecule | CAS: 112-49-2

Triethylene glycol dimethyl ether (also called triglyme) is a glycol ether used as a solvent.

Kategori:
AlcoholsCompounds used in a research, industrial, or household settingEthylene Glycols +3
Target Protein:
Tyrosine-protein kinase FynProfilin-2Outer-membrane lipoprotein LolB +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trigonellamide DB11710
small molecule | CAS: 3106-60-3

Trigonellamide is under investigation in clinical trial NCT01930240 (The Safety of a Hypolipidemic Agent in Healthy Normal Volunteers).

Kategori:
Nicotinic AcidsPyridines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Triheptanoin Approved DB11677
small molecule | CAS: 620-67-7

Triheptanoin is a source of heptanoate fatty acids, which can be metabolized without the enzymes of long chain fatty acid oxidation.[L14612] In clinical trials, patients with long chain fatty acid oxidation disorders (lc-FAODs) treated with triheptanoin are l…

Kategori:
Alimentary Tract and MetabolismCaloric AgentsGlycerides +5
Waktu ParuhDue to multiple pea…
Vol. Distribusi-
KlirensA single dose of 0.…
Genetik -
Trihexyphenidyl Approved DB00376
small molecule | CAS: 144-11-6

Trihexyphenidyl is a centrally acting muscarinic antagonist used for treatment of parkinsonism and drug-induced extrapyramidal disorders.[L31773,L31778] Its discovery was published in 1949 in a study looking for drugs with antispasmodic activity.[A229103] Tri…

Kategori:
Agents producing tachycardiaAnti-Dyskinesia AgentsAnti-Parkinson Drugs +8
Target Protein:
Muscarinic acetylcholine receptor M1Beta-3 adrenergic receptorMuscarinic acetylcholine receptor M2 +3
Waktu ParuhThe mean eliminatio…
Vol. Distribusi-
Klirens-
Genetik -
Trilaciclib Approved DB15442
small molecule | CAS: 1374743-00-6

Trilaciclib, or G1T28, is a CDK4 and CDK6 inhibitor, indicated to reduce the incidence of chemotherapy induced myelosuppression in patients before topotecan-containing or platinum and etoposide-containing chemotherapy for extensive stage small cell lung cance…

Kategori:
BCRP/ABCG2 SubstratesCyclin-dependent Kinase 4 InhibitorsCyclin-dependent Kinase 6 Inhibitors +16
Target Protein:
Cyclin-dependent kinase 4Cyclin-dependent kinase 6Cyclin-dependent kinase 9 +3
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of tr…
Genetik -
Trilostane Approved DB01108
small molecule | CAS: 13647-35-3

Trilostane is an inhibitor of 3 beta-hydroxysteroid dehydrogenase used in the treatment of Cushing's syndrome. It was withdrawn from the United States market in April 1994.

Kategori:
Abortifacient AgentsAbortifacient Agents, SteroidalAdrenal Cortex Hormones +20
Target Protein:
3 beta-hydroxysteroid dehydrogenase/Delta 5-->4-isomerase type 13 beta-hydroxysteroid dehydrogenase/Delta 5-->4-isomerase type 2Estrogen receptor +1
Waktu Paruh8 hours.
Vol. Distribusi-
Klirens-
Genetik -
Trimazosin DB09206
small molecule | CAS: 35795-16-5

Trimazosin is a sympatholytic alpha blocker.

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +7
Target Protein:
Alpha-1D adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trimegestone DB13129
small molecule | CAS: 74513-62-5

Trimegestone has been used in trials studying the treatment of Postmenopause.

Kategori:
Fused-Ring CompoundsGenito Urinary System and Sex HormonesNorpregnadienes +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trimetazidine Approved DB09069
small molecule | CAS: 5011-34-7

Trimetazidine is a piperazine derivative indicated for the symptomatic treatment of stable angina pectoris in patients inadequately controlled or intolerant to first line therapies.[L33015] Trimetazidine has been studied as a treatment for angina pectoris sin…

Kategori:
Cardiac TherapyCardiovascular AgentsPiperazines +1
Target Protein:
3-ketoacyl-CoA thiolase, mitochondrial
Waktu ParuhIn young, healthy s…
Vol. DistribusiThe volume of distr…
KlirensTrimetazidine clear…
Genetik -
Trimethadione Approved DB00347
small molecule | CAS: 127-48-0

An anticonvulsant effective in absence seizures, but generally reserved for refractory cases because of its toxicity. (From AMA Drug Evaluations Annual, 1994, p378)

Kategori:
Agents causing hyperkalemiaAnti-epileptic AgentAntiarrhythmic agents +18
Target Protein:
Voltage-dependent T-type calcium channel subunit alpha-1G
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trimethaphan Approved DB01116
small molecule | CAS: 7187-66-8

A nicotinic antagonist that has been used as a ganglionic blocker in hypertension, as an adjunct to anesthesia, and to induce hypotension during surgery.

Kategori:
Adjuvants, AnesthesiaAntiadrenergic Agents, Ganglion-BlockingAnticholinergic Agents +13
Target Protein:
Neuronal acetylcholine receptor subunit alpha-4Neuronal acetylcholine receptor subunit alpha-10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trimethobenzamide Approved DB00662
small molecule | CAS: 138-56-7

Trimethobenzamide is a novel antiemetic which prevents nausea and vomiting in humans. Its actions are unclear but most likely involves the chemoreceptor trigger zone (CTZ). In dogs pretreated with trimethobenzamide HCl, the emetic response to apomorphine is i…

Kategori:
Acids, CarbocyclicAmidesAminoalkyl Ethers +10
Target Protein:
D(2) dopamine receptor
Waktu ParuhThe mean eliminatio…
Vol. Distribusi-
Klirens-
Genetik -
Trimethoprim Approved DB00440
small molecule | CAS: 738-70-5

Trimethoprim is an antifolate antibacterial agent that inhibits bacterial dihydrofolate reductase (DHFR), a critical enzyme that catalyzes the formation of tetrahydrofolic acid (THF) - in doing so, it prevents the synthesis of bacterial DNA and ultimately con…

Kategori:
Agents causing hyperkalemiaAgents Causing Muscle ToxicityAnti-Infective Agents +32
Target Protein:
Dihydrofolate reductaseDihydrofolate reductase
Waktu ParuhTrimethoprim half-l…
Vol. DistribusiTrimethoprim is ext…
KlirensFollowing oral admi…
Genetik -
small molecule | CAS: 13957-55-6

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismDrugs for Functional Gastrointestinal Disorders
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trimethyllysine DB03977
small molecule | CAS: 19253-88-4

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +3
Target Protein:
Calmodulin-2Calmodulin-1Calmodulin-3 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 10182-92-0

Deskripsi belum tersedia.

Kategori:
AminesCompounds used in a research, industrial, or household settingDetergents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trimetrexate Approved DB01157
small molecule | CAS: 52128-35-5

A nonclassical folic acid inhibitor through its inhibition of the enzyme dihydrofolate reductase. It is being tested for efficacy as an antineoplastic agent and as an antiparasitic agent against pneumocystis pneumonia in AIDS patients. Myelosuppression is its…

Kategori:
Acids, AcyclicAcids, AldehydicAnti-Infective Agents +18
Target Protein:
Peptide deformylase, mitochondrialDihydrofolate reductase
Waktu Paruh11 to 20 hours
Vol. Distribusi* 20 ± 8 L/m2 * 36…
Klirens* 38 +/- 15 mL/min/…
Genetik -
Trimipramine Approved DB00726
small molecule | CAS: 739-71-9

Tricyclic antidepressant similar to imipramine, but with more antihistaminic and sedative properties.

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +44
Target Protein:
Sodium-dependent serotonin transporterSodium-dependent noradrenaline transporterSodium-dependent dopamine transporter +15
Gen Terkait:
CYP2D6 CYP2D6 CYP2D6 +5
Waktu Paruh11-18 hrs
Vol. Distribusi-
Klirens-
Genetik 8 Varian
Trinitrotoluene DB01676
small molecule | CAS: 118-96-7

Trinitrotoluene is an explosive chemical that can cause skin irritation and other toxic consequences.

Kategori:
Benzene DerivativesCompounds used in a research, industrial, or household settingExplosive Agents
Target Protein:
Pentaerythritol tetranitrate reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trioxsalen Approved DB04571
small molecule | CAS: 3902-71-4

Trioxsalen (trimethylpsoralen, trioxysalen or trisoralen) is a furanocoumarin and a psoralen derivative obtained from several plants, mainly Psoralea corylifolia. Like other psoralens it causes photosensitization of the skin. It is administered either topical…

Kategori:
AntipsoriaticsAntipsoriatics for Systemic UseAntipsoriatics for Topical Use +11
Target Protein:
DNA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tripamide DB15959
small molecule | CAS: 73803-48-2

Deskripsi belum tersedia.

Kategori:
DiureticsHeterocyclic Compounds, Fused-RingMembrane Transport Modulators +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tripelennamine Approved DB00792
small molecule | CAS: 91-81-6

A histamine H1 antagonist with low sedative action but frequent gastrointestinal irritation. It is used to treat asthma; HAY fever; urticaria; and rhinitis; and also in veterinary applications. Tripelennamine is administered by various routes, including topic…

Kategori:
AminesAminopyridinesAnti-Allergic Agents +17
Target Protein:
Histamine H1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Triphendiol DB06588
small molecule | CAS: 1213777-80-0

Deskripsi belum tersedia.

Kategori:
BenzopyransChromonesFlavonoids +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Dehydrosqualene synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 11051–11100 dari 11778
Sebelumnya Halaman 222 / 236 Berikutnya