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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 222 / 282
Pralatrexate Approved DB06813
small molecule | CAS: 146464-95-1

Pralatrexate is an antifolate for the treatment of relapsed or refractory peripheral T-cell lymphoma [L37674]. Pralatrexate was developed in response due to the inferior responses of patients using the standard therapy for their B-cells counterparts.[A246693]…

Kategori:
AntimetabolitesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +10
Target Protein:
Dihydrofolate reductasePeptide deformylase, mitochondrialFolylpolyglutamate synthase, mitochondrial +1
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe steady-state vo…
KlirensThe total systemic …
Genetik -
Praliciguat DB16300
small molecule | CAS: 1628730-49-3

Praliciguat is under investigation in clinical trial NCT03254485 (A Study of the Effect of IW-1973 on the Exercise Capacity of Patients With Heart Failure With Preserved Ejection Fraction (Hfpef)).

Kategori:
Enzyme ActivatorsGastrointestinal AgentsGuanylyl Cyclase C Agonists
Target Protein:
Guanylate cyclase soluble subunit alpha-1Guanylate cyclase soluble subunit beta-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pralidoxime Approved DB00733
small molecule | CAS: 6735-59-7

Pralidoxime is an antidote to organophosphate pesticides and chemicals. Organophosphates bind to the esteratic site of acetylcholinesterase, which results initially in reversible inactivation of the enzyme. If given within 24 hours,after organophosphate expos…

Kategori:
AminesAntidotesCholinergic Agents +8
Target Protein:
AcetylcholinesteraseCholinesterase
Waktu Paruh74-77 minutes
Vol. Distribusi-
Klirens-
Genetik -
Pralmorelin DB18252
small molecule | CAS: 158861-67-7

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsGrowth Hormone-Releasing HormoneGrowth Substances +1
Target Protein:
Growth hormone secretagogue receptor type 16-phosphogluconate dehydrogenase, decarboxylating
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pralnacasan DB04875
small molecule | CAS: 192755-52-5

Pralnacasan is an orally bioavailable pro-drug of a potent, non-peptide inhibitor of interleukin-1beta converting enzyme (ICE).

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Caspase-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pralsetinib Approved DB15822
small molecule | CAS: 2097132-94-8

Pralsetinib, similar to the previously approved [selpercatinib], is a kinase inhibitor with enhanced specificity for RET tyrosine kinase receptors (RTKs) over other RTK classes.[A202055, A219751, L15986] Enhanced RET (Rearranged during transfection) oncogene …

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Inhibitors +38
Target Protein:
Proto-oncogene tyrosine-protein kinase receptor RetEpithelial discoidin domain-containing receptor 1NT-3 growth factor receptor +8
Waktu ParuhPralsetinib has a p…
Vol. DistribusiPralsetinib has a m…
KlirensPralsetinib has a m…
Genetik -
Pralurbactam DB19437
small molecule | CAS: 2163782-59-8

Pralurbactam is under investigation in clinical trial NCT06633718 (Study to Assess the Efficacy and Safety of Meropenem and Pralurbactam in CIAI).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pramiconazole DB06295
small molecule | CAS: 219923-85-0

Deskripsi belum tersedia.

Target Protein:
Lanosterol 14-alpha demethylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pramipexole Approved DB00413
small molecule | CAS: 104632-26-0

Pramipexole is a drug used to treat the symptoms of Parkinson's Disease (PD). It is a _non-ergot dopamine agonist_ drug that is efficacious in treating various Parkinson's symptoms such as tremor, rigidity, and bradykinesia (slow movement) [A176867]. It was …

Kategori:
Anti-Dyskinesia AgentsAnti-Parkinson Agents (Dopamine Agonist)Anti-Parkinson Drugs +17
Target Protein:
D(3) dopamine receptorD(2) dopamine receptorD(4) dopamine receptor +2
Waktu ParuhAbout 8.5-12 hours …
Vol. DistribusiThis drug is extens…
KlirensRenal clearance is …
Genetik -
Pramiracetam Approved DB13247
small molecule | CAS: 68497-62-1

Pramiracetam has been previously approved in some eastern European countries under the brand names Pramistar, Neupramir, and Remen. It was also previously approved in the United States with orphan drug designation [L1469]. Pramiracetam has been studied for th…

Kategori:
Nervous SystemPsychoanalepticsPsychostimulants, Agents Used for ADHD and Nootropics
Target Protein:
Muscarinic acetylcholine receptor M5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pramlintide Approved DB01278
small molecule | CAS: 151126-32-8

Pramlintide is a relatively new adjunct treatment for diabetes (both type 1 and 2), developed by Amylin Pharmaceuticals. It is derived from amylin, a hormone that is released into the bloodstream, in a similar pattern as insulin, after a meal. Like insulin, a…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsAmylin Agonists +12
Target Protein:
Glucagon-like peptide 1 receptorCalcitonin receptorReceptor activity-modifying protein 1 +2
Waktu ParuhApproximately 48 mi…
Vol. Distribusi-
Klirens-
Genetik -
Pranoprofen DB13514
small molecule | CAS: 52549-17-4

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAgents causing hyperkalemiaAgents that produce hypertension +17
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prasinezumab DB14788
biotech | CAS: 1960462-19-4

Prasinezumab is under investigation in clinical trial NCT03100149 (A Study to Evaluate the Efficacy of Prasinezumab (RO7046015/PRX002) in Participants With Early Parkinson's Disease).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prasterone Approved DB01708
small molecule | CAS: 53-43-0

Prasterone, also known as dehydroepiandrosterone (DHEA) is a major C19 steroid produced by the adrenal cortex. It is also produced in small quantities in the testis and the ovary. Dehydroepiandrosterone (DHEA) can be converted to testosterone; androstenedione…

Kategori:
17-KetosteroidsAdjuvants, ImmunologicAdrenal Cortex Hormones +32
Target Protein:
Glucose-6-phosphate 1-dehydrogenaseEstrogen receptorEstrogen receptor beta +7
Waktu Paruh12 hours
Vol. Distribusi-
Klirens-
Genetik -
Prasterone enantate Approved DB16625
small molecule | CAS: 23983-43-9

Deskripsi belum tersedia.

Kategori:
17-KetosteroidsAdrenal Cortex HormonesAndrostanes +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 651-48-9

DHEA sulfate is the major steroid of the fetal adrenal. DHEA-S is the principal adrenal androgen and is secreted together with cortisol under the control of ACTH and prolactin. DHEA-S is elevated with hyperprolactinemia.

Kategori:
17-KetosteroidsAdrenal Cortex HormonesAndrostanes +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prasugrel Approved DB06209
small molecule | CAS: 150322-43-3

Prasugrel, a thienopyridine derivative, is a platelet activation and aggregation inhibitor structurally and pharmacologically related to clopidogrel and ticlopidine. Similar to clopidogrel, prasugrel is a prodrug that requires enzymatic transformation in the …

Kategori:
AnticoagulantsAntiplatelet agentsBlood and Blood Forming Organs +15
Target Protein:
P2Y purinoceptor 12
Waktu ParuhThe active metaboli…
Vol. Distribusi44-68L
KlirensApparent clearance …
Genetik -
Pravastatin Approved DB00175
small molecule | CAS: 81093-37-0

Pravastatin is the 6-alpha-hydroxy acid form of [mevastatin].[T303] Pravastatin was firstly approved in 1991 becoming the second available statin in the United States. It was the first statin administered as the active form and not as a prodrug.[T274] This dr…

Kategori:
Agents Causing Muscle ToxicityAnticholesteremic AgentsBCRP/ABCG2 Inhibitors +20
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductaseHistone deacetylase 2
Gen Terkait:
KIF6 HMGCR
Waktu ParuhThe reported elimin…
Vol. DistribusiThe reported steady…
KlirensThe reported cleara…
Genetik 2 Varian
Pravibismane DB17784
small molecule | CAS: 175880-68-9

Deskripsi belum tersedia.

Kategori:
AlcoholsSulfhydryl CompoundsSulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prazepam Approved DB01588
small molecule | CAS: 2955-38-6

Prazepam is a benzodiazepine that is used in the treatment of anxiety disorders. It is a schedule IV drug in the U.S.

Kategori:
Anti-Anxiety AgentsBenzazepinesBenzodiazepines and benzodiazepine derivatives +14
Target Protein:
Translocator proteinGABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site
Waktu Paruh36-200 hours
Vol. Distribusi-
Klirens-
Genetik -
Praziquantel Approved DB01058
small molecule | CAS: 55268-74-1

Praziquantel is a pyrazino-isoquinolein derivative from the thioxantonic group used as a broad anthelmintic spectrum. Specifically, it is known as a treatment of trematodes and cestodes infections such as schistosomiasis, taeniasis, and cysticercosis.[A263201…

Kategori:
AnthelminticsAnti-Infective AgentsAntihelminthic +12
Target Protein:
Hematopoietic prostaglandin D synthaseSchistosome calcium ion (Ca2+) channels
Waktu ParuhFollowing oral admi…
Vol. DistribusiFollowing a single …
KlirensFollowing a single …
Genetik -
Prazosin Approved DB00457
small molecule | CAS: 19216-56-9

Prazosin is a drug used to treat hypertension. Prazosin is marketed by _Pfizer_ and was initially approved by the FDA in 1988.[L5828] It belongs to the class of drugs known as alpha-1 antagonists. Recently, many studies have evaluated the benefits of thi…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +16
Target Protein:
Alpha-1A adrenergic receptorAlpha-1B adrenergic receptorAlpha-1D adrenergic receptor +4
Waktu ParuhThe plasma half-lif…
Vol. DistribusiAbout 0.6 L/kg [A17…
KlirensIn patients with co…
Genetik -
Prednimustine DB12832
small molecule | CAS: 29069-24-7

Prednimustine has been used in trials studying the treatment of Lymphoma.

Kategori:
Alkylating DrugsAntineoplastic AgentsAntineoplastic Agents, Alkylating +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prednisolone Approved DB00860
small molecule | CAS: 50-24-8

Prednisolone is a glucocorticoid similar to [cortisol] used for its anti-inflammatory, immunosuppressive, anti-neoplastic, and vasoconstrictive effects.[A187463] Prednisolone was granted FDA approval on 21 June 1955.[L9431]

Kategori:
Adrenal Cortex HormonesAdrenalsAgents for Treatment of Hemorrhoids and Anal Fissures for Topical Use +45
Target Protein:
Glucocorticoid receptor
Waktu ParuhPrednisolone has a …
Vol. DistribusiA 0.15mg/kg dose of…
KlirensA 0.15mg/kg dose of…
Genetik -
Prednisolone acetate Approved DB15566
small molecule | CAS: 52-21-1

Prednisolone acetate is a [prednisolone] molecule bound to an acetate functional group by an ester bond.[L9449] Prednisolone acetate was granted FDA approval in 1955.[L9449]

Kategori:
Adrenal Cortex HormonesAnti-Inflammatory AgentsCorticosteroids +14
Target Protein:
Glucocorticoid receptor
Waktu ParuhOral prednisolone a…
Vol. DistribusiThe volume of distr…
KlirensData regarding the …
Genetik -
small molecule | CAS: 69164-69-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 2920-86-7

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesCorticosteroidsCytochrome P-450 CYP3A Inducers +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prednisolone phosphate Approved DB14631
small molecule | CAS: 302-25-0

Prednisolone phosphate is a glucocorticoid similar to [cortisol] used for its anti-inflammatory, immunosuppressive, anti-neoplastic, and vasoconstrictive effects.[A187463] Prednisolone phosphate was granted FDA Approval on 19 December 1973.[L14144]

Kategori:
Adrenal Cortex HormonesAdrenalsAnti-Inflammatory Agents +30
Target Protein:
Glucocorticoid receptorAnnexin A1
Waktu ParuhThe half life of pr…
Vol. DistribusiThe volume of distr…
Klirens-
Genetik -
Prednisolone tebutate Approved DB14632
small molecule | CAS: 7681-14-3

Deskripsi belum tersedia.

Kategori:
Fused-Ring CompoundsPregnadienesPregnadienetriols +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prednisone Approved DB00635
small molecule | CAS: 53-03-2

A synthetic anti-inflammatory glucocorticoid derived from [cortisone].[A187463] It is biologically inert and converted to [prednisolone] in the liver.[L10502] Prednisone was granted FDA approval on 21 February 1955.[L10496]

Kategori:
Adrenal Cortex HormonesAdrenalsAlimentary Tract and Metabolism +45
Target Protein:
Glucocorticoid receptor
Waktu ParuhPrednisone and its …
Vol. DistribusiData regarding the …
KlirensData regarding the …
Genetik -
Prednisone acetate Approved DB14646
small molecule | CAS: 125-10-0

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesAnti-Inflammatory AgentsAntineoplastic Agents +17
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prednylidene DB13208
small molecule | CAS: 599-33-7

Prednylidene is an experimental systemic glucocorticoid.

Kategori:
Adrenal Cortex HormonesCorticosteroidsCorticosteroids for Systemic Use +19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pregabalin Approved DB00230
small molecule | CAS: 148553-50-8

Pregabalin is structurally similar to gamma-aminobutyric acid (GABA) - an inhibitory neurotransmitter.[A173995] It may be used to manage neuropathic pain, postherpetic neuralgia, and fibromyalgia among other conditions.[A187190] Although as per the FDA Label …

Kategori:
Acids, AcyclicAgents causing angioedemaAmino Acids +24
Target Protein:
Voltage-dependent calcium channel subunit alpha-2/delta-1
Waktu ParuhThe elimination hal…
Vol. DistribusiAfter oral administ…
KlirensIn young healthy su…
Genetik -
Pregnenolone Approved DB02789
small molecule | CAS: 145-13-1

A 21-carbon steroid, derived from cholesterol and found in steroid hormone-producing tissues. Pregnenolone is the precursor to gonadal steroid hormones and the adrenal corticosteroids.

Kategori:
Adrenal Cortex HormonesCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Substrates +11
Target Protein:
Steroid hormone receptor ERR1Nuclear receptor subfamily 1 group I member 2Sulfotransferase 2B1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1778-02-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Preladenant DB11864
small molecule | CAS: 377727-87-2

Preladenant has been used in trials studying the treatment of Brain Diseases, Parkinson Disease, Movement Disorders, Antipsychotic Agents, and Parkinsonian Disorders, among others.

Target Protein:
Adenosine receptor A2a
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prenalterol DB13777
small molecule | CAS: 57526-81-5

Deskripsi belum tersedia.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic and Dopaminergic Agents +20
Target Protein:
Beta-3 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prenylamine Approved DB04825
small molecule | CAS: 390-64-7

Prenylamine was withdrawn from the Canadian, US, and UK markets in 1988 due to concerns regarding cardiac arrhythmias.

Kategori:
Adrenergic AgentsAgents causing hyperkalemiaAmines +19
Target Protein:
Myosin light chain kinase 2, skeletal/cardiac muscleCalmodulin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prephenic acid DB08427
small molecule | CAS: 126-49-8

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicCyclohexanesCycloparaffins
Target Protein:
Chorismate mutase AroH
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Presatovir DB12165
small molecule | CAS: 1353625-73-6

Presatovir has been used in trials studying the treatment of RSV Infection, Respiratory Syncytial Virus (RSV), Respiratory Syncytial Virus Infections, and Respiratory Syncytial Virus (RSV) Infections.

Kategori:
AmidesHeterocyclic Compounds, Fused-RingPyrazoles +2
Target Protein:
Fusion glycoprotein F0
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pretomanid Approved DB05154
small molecule | CAS: 187235-37-6

Persistent forms of tuberculosis (TB) have proven to be a major cause of global morbidity and mortality and a cause for significant concern. Research in recent years has been geared toward the development of novel therapies that target persistent forms of thi…

Kategori:
Antiinfectives for Systemic UseAntimycobacterialsCytochrome P-450 CYP3A Substrates +7
Target Protein:
Cyclopropane mycolic acid synthase 1Cyclopropane mycolic acid synthase 2Cyclopropane mycolic acid synthase 3 +5
Waktu ParuhThe elimination hal…
Vol. DistribusiA pharmacokinetic m…
KlirensThe clearance of pr…
Genetik -
Prexasertib DB12008
small molecule | CAS: 1234015-52-1

Prexasertib has been used in trials studying the treatment and basic science of mCRPC, Leukemia, Neoplasm, breast cancer, and Ovarian Cancer, among others.

Kategori:
Enzyme InhibitorsProtein Kinase Inhibitors
Target Protein:
Serine/threonine-protein kinase Chk1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prexigebersen DB17320
biotech | CAS: 202484-91-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prezatide DB11296
small molecule | CAS: 49557-75-7

Prezatide is a tripeptide consisting of glycine, histidine, and lysine which readily forms a complex with copper ions [A19503]. Prezatide is used in cosmetic products for the skin and hair. It is known to aid wound healing and its potential applications in ch…

Kategori:
Amino Acids, Peptides, and ProteinsGrowth SubstancesPeptides
Waktu ParuhPrezatide is rapidl…
Vol. Distribusi-
Klirens-
Genetik -
PRGN-2012 DB18342
biotech

PRGN-2012 is an adenoviral vector expressing human papillomavirus (HPV) 6 and HPV 11 antigens

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PRGN-3006 DB17229
biotech

PRGN-3006 are autologous CD3+ T cells genetically modified using a non-viral system to express a CD33 CAR, membrane-bound interleukin-15, and a truncated form of human HER1T (kill switch) on the cell surface.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PRI-724 DB15034
small molecule | CAS: 1198780-38-9

PRI-724 is under investigation in clinical trial NCT03620474 (Safety and Effectiveness of PRI-724 for Hepatitis C or B Virus Derived Liver Cirrhosis).

Kategori:
Pyrimidines
Target Protein:
CREB-binding protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pridinol DB13642
small molecule | CAS: 511-45-5

Deskripsi belum tersedia.

Kategori:
Central Nervous System DepressantsMuscle RelaxantsMuscle Relaxants, Centrally Acting Agents +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prifinium DB13254
small molecule | CAS: 10236-81-4

Prifinium is an antimuscarinic agent with antispasmodic and antiemetic properties. It may be useful for the treatment of irritable bowel syndrome [A175027].

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAnticholinergic Agents +3
Target Protein:
Muscarinic acetylcholine receptor M5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Priliximab DB16920
biotech | CAS: 147191-91-1

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 11051–11100 dari 14063
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