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15718

Total database: 17430
Struktur (SMILES)
10762 (68.5%)
Target
7957 (50.6%)
Genomik
112 (0.7%)
Referensi
15718 (100.0%)

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Hasil Pencarian (15718)

Halaman 222 / 315
Odetiglucan DB17468
biotech | CAS: 53238-80-5

Deskripsi belum tersedia.

Waktu Paruh-
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Odevixibat Approved DB16261
small molecule | CAS: 501692-44-0

Odevixibat, or A4250, is an ileal sodium/bile acid cotransporter inhibitor indicated for the treatment of pruritus in patients older than 3 months, with progressive familial intrahepatic cholestasis (PFIC).[A236808,L34793] Odevixibat is the first approved non…

Kategori:
Acids, AcyclicAlimentary Tract and MetabolismBenzazepines +9
Target Protein:
Ileal sodium/bile acid cotransporter
Waktu ParuhA 7.2 mg oral dose …
Vol. DistribusiThe majority of adu…
KlirensThe majority of adu…
Genetik -
Odiparcil DB06609
small molecule | CAS: 137215-12-4

Deskripsi belum tersedia.

Kategori:
Carbohydrates
Target Protein:
Prothrombin
Waktu Paruh-
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Genetik -
ODM-203 DB16843
small molecule | CAS: 1430723-35-5

Deskripsi belum tersedia.

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ODM-207 DB18820
small molecule | CAS: 1801503-93-4

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
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Genetik -
ODN M362 DB16485
biotech

Deskripsi belum tersedia.

Kategori:
Experimental Unapproved Treatments for COVID-19Nucleic Acids, Nucleotides, and NucleosidesNucleotides +2
Target Protein:
Toll-like receptor 9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Odocoileus virginianus hair Approved DB10868
biotech

White-tailed deer hair is used in allergenic testing.

Waktu Paruh-
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Odronextamab DB16684
biotech | CAS: 1801338-64-6

Odronextamab is a hinge-stabilized, fully human immunoglobulin G4 (IgG4)-based CD20×CD3 bispecific antibody currently evaluated for the treatment of relapsed/refractory (R/R) B-Cell non-Hodgkin lymphoma (NHL).[A254187,A254197] Preliminary studies have shown t…

Target Protein:
B-lymphocyte antigen CD20T-cell surface glycoprotein CD3
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Ofatumumab Approved DB06650
biotech | CAS: 679818-59-8

Ofatumumab is a novel anti-CD20 monoclonal antibody that targets B-cells. It is an IgG1? human monoclonal antibody produced from a recombinant murine cell line (NS0) via transgenic mouse and hybridoma technology.[L12612] Ofatumumab works by recognizing antige…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +17
Target Protein:
B-lymphocyte antigen CD20
Waktu ParuhIn patients with CL…
Vol. DistribusiIn patients with CL…
KlirensIn patients with CL…
Genetik -
Ofloxacin Approved DB01165
small molecule | CAS: 82419-36-1

A synthetic fluoroquinolone (fluoroquinolones) antibacterial agent that inhibits the supercoiling activity of bacterial DNA gyrase, halting DNA replication.

Kategori:
4-QuinolonesAgents Causing Muscle ToxicityAnti-Bacterial Agents +22
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA gyrase subunit A +2
Waktu Paruh9 hours
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1476737-24-2

Ofranergene obadenovec is under investigation in clinical trial NCT01229865 (Safety and Efficacy of VB-111 in Subjects With Advanced Differentiated Thyroid Cancer).

Waktu Paruh-
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Oftasceine Approved DB11184
small molecule | CAS: 1461-15-0

Oftasceine is also referred to as Fluorexon. It is used in ophthalmic solutions as a staining agent when fitting soft and hard lenses. It is a fluorescent dye or luminescent agent.

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Oglemilast DB12375
small molecule | CAS: 778576-62-8

Oglemilast has been investigated for the treatment of Pulmonary Disease, Chronic Obstructive.

Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4A3',5'-cyclic-AMP phosphodiesterase 4B3',5'-cyclic-AMP phosphodiesterase 4D
Waktu Paruh-
Vol. Distribusi-
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Oglufanide DB05779
small molecule | CAS: 38101-59-6

Oglufanide is a synthetic dipeptide immunomodulator in development for the treatment of chronic hepatitis C viral infection. Oglufanide was originally developed to treat severe infectious disease in Russia (where it is a registered pharmaceutical), and was ex…

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAngiogenesis Modulating Agents +10
Waktu Paruh-
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Ohmefentanyl DB01570
small molecule | CAS: 78995-14-9

Ohmefentanyl is an extremely potent opioid analgesic drug which selectively binds to the µ-opioid receptor. The Chinese have recorded ohmefentanyl as having a potency that is 6,300 times morphine. Ohmefentanyl is one of the most potent ? -receptor agonists kn…

Kategori:
AnalgesicsCentral Nervous System AgentsPeripheral Nervous System Agents +2
Waktu Paruh-
Vol. Distribusi-
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Genetik -
OKI-179 DB17583
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
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Okra Approved DB10660
biotech

Okra allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract +1
Waktu Paruh-
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Olacaftor DB16262
small molecule | CAS: 1897384-89-2

Olacaftor is under investigation in clinical trial NCT02951182 (A Study Evaluating the Safety and Efficacy of VX-440 Combination Therapy in Subjects With Cystic Fibrosis).

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Olafertinib DB17179
small molecule

Deskripsi belum tersedia.

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Olaflur DB13290
small molecule | CAS: 6818-37-7

Olaflur which is also referred to as elmex gel is an ingredient used in toothpaste which helps in the prevention of dental caries.

Kategori:
Alimentary Tract and MetabolismAminesAnions +9
Waktu Paruh-
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Olanexidine DB16889
small molecule | CAS: 146510-36-3

Deskripsi belum tersedia.

Kategori:
AmidinesGuanidines
Waktu Paruh-
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Olanzapine Approved DB00334
small molecule | CAS: 132539-06-1

Olanzapine is a thienobenzodiazepine classified as an atypical or second-generation antipsychotic agent.[A176996] The second-generation antipsychotics were introduced in the 90s and quickly gained traction due to their impressive efficacy, reduced risk for ex…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +50
Target Protein:
5-hydroxytryptamine receptor 2AD(2) dopamine receptorD(1A) dopamine receptor +17
Gen Terkait:
HTR1A
Waktu ParuhOlanzapine presents…
Vol. DistribusiThe volume of distr…
KlirensThe mean clearance …
Genetik 1 Varian
Olaparib Approved DB09074
small molecule | CAS: 763113-22-0

Olaparib is a selective and potent inhibitor of poly (ADP-ribose) polymerase (PARP) enzymes, PARP1 and PARP2.[L41100, L40908, L43792] PARP inhibitors represent a novel class of anti-cancer therapy and they work by taking advantage of a defect in DNA repair in…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Inhibitors +38
Target Protein:
Poly [ADP-ribose] polymerase 1Poly [ADP-ribose] polymerase 2Protein mono-ADP-ribosyltransferase PARP3 +1
Waktu ParuhFollowing a single …
Vol. DistribusiThe mean (± standar…
KlirensFollowing a single …
Genetik -
small molecule | CAS: 1380359-84-1

Olaparib-bodipy FL is under investigation in clinical trial NCT03085147 (A Dye for the Detection of Cancer of the Tongue and Mouth).

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Olaptesed Pegol DB11707
small molecule | CAS: 1390628-22-4

Olaptesed Pegol has been investigated for the treatment of Hematopoietic Stem Cell Transplantation.

Kategori:
Pegylated agents
Waktu Paruh-
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Olaratumab Approved DB06043
biotech | CAS: 1024603-93-7

Olaratumab (IMC-3G3) is a fully human IgG1 monoclonal antibody with antitumor activity that selectively binds the external domain of human platelet-derived growth factor receptor (PDGFR)-? with high affinity and blocks ligand binding. It is composed of two he…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +12
Target Protein:
Platelet-derived growth factor receptor alpha
Waktu ParuhEstimated value of …
Vol. Distribusi7.7 L at steady sta…
KlirensMean value of 0.56L…
Genetik -
biotech

Deskripsi belum tersedia.

Kategori:
AngiospermsBiological ProductsComplex Mixtures +9
Waktu Paruh-
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Olea europaea pollen Approved DB10378
biotech

Olea europaea pollen is the pollen of the Olea europaea plant. Olea europaea pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
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Oleandomycin DB11442
small molecule | CAS: 3922-90-5

Oleandomycin is a macrolide antibiotic, though it is less effective than erythromycin. It is synthesized from strains of _Streptomyces antibioticus_.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibacterials for Systemic Use +8
Waktu Paruh-
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Oleandrin DB12843
small molecule | CAS: 465-16-7

Oleandrin has been used in trials studying the treatment of Lung Cancer and Chemotherapeutic Agent Toxicity.

Kategori:
CardanolidesCardiac GlycosidesFused-Ring Compounds +2
Target Protein:
Sodium/potassium-transporting ATPase subunit alpha-1Sodium/potassium-transporting ATPase subunit alpha-2Sodium/potassium-transporting ATPase subunit alpha-3 +14
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Oleclumab DB15088
biotech | CAS: 1803176-05-7

Oleclumab is under investigation in clinical trial NCT03819465 (A Study of Novel Anti-cancer Agents in Patients With Previously Untreated NSCLC).

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Oleic Acid Approved DB04224
small molecule | CAS: 112-80-1

An unsaturated fatty acid that is the most widely distributed and abundant fatty acid in nature. It is used commercially in the preparation of oleates and lotions, and as a pharmaceutical solvent. (Stedman, 26th ed)

Kategori:
Fatty AcidsFatty Acids, MonounsaturatedFatty Acids, Unsaturated +2
Target Protein:
Fatty acid-binding protein, adipocyteFatty acid-binding protein, liverPeroxisome proliferator-activated receptor alpha +4
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiRadio-labelled olei…
KlirensNo pharmacokinetic …
Genetik -
small molecule | CAS: 111-58-0

Deskripsi belum tersedia.

Kategori:
AlcoholsAminesAmino Alcohols +10
Target Protein:
Peroxisome proliferator-activated receptor alphaG-protein coupled receptor 55Glucose-dependent insulinotropic receptor +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2096510-84-6

Olenasufligene relduparvovec is under investigation in clinical trial NCT03612869 (Study of aavrh10-h.sgsh Gene Therapy in Patients With Mucopolysaccharidosis Type IIIA (MPS IIIA)). It is an adeno-associated virus (AAV) vector that delivers a functional copy …

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
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Olendalizumab DB14834
biotech | CAS: 1337966-73-0

Olendalizumab is under investigation in clinical trial NCT01883544 (Study to Evaluate the Safety, Tolerability, Pharmacokinetics, and Pharmacodynamics of ALXN1007 in Healthy Male and Female Subjects).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oleoyl chloride DB14666
small molecule | CAS: 112-77-6

Deskripsi belum tersedia.

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Oleoyl-estrone DB04870
small molecule | CAS: 180003-17-2

Oleoyl-estrone (OE) is a fatty acid ester of estrone. This hormone occurs naturally and is found circulating in various animal species and humans. It has been shown in animal studies to promote the loss of body fat while maintaining body protein storage, main…

Kategori:
17-KetosteroidsAdrenal Cortex HormonesAnti-Obesity Agents +15
Target Protein:
Metabotropic glutamate receptor 3Metabotropic glutamate receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Olesoxime DB05185
small molecule | CAS: 22033-87-0

Olesoxime is a cholesterol-like small molecule that has demonstrated a remarkable neuroprotective profile in a battery of both in vitro and in vivo preclinical models. For example, it has demonstrated the ability to prevent neurodegeneration, enhance nerve fu…

Kategori:
CholestanesCholestenesFused-Ring Compounds +1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 76622-80-5

Deskripsi belum tersedia.

Kategori:
AminesOnium CompoundsQuaternary Ammonium Compounds +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Olezarsen DB18728
biotech | CAS: 2097587-83-0

Olezarsen is an antisense oligonucleotide targeting messenger RNA for apolipoprotein C-III (APOC3).

Waktu Paruh-
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Oliceridine Approved DB14881
small molecule | CAS: 1401028-24-7

Severe acute pain occurs through nociceptive signalling involving both ascending and descending spinal pathways, in which nerve conductance is mediated in part by the action of opioid receptors.[A218041, A218046] Opioid receptors are seven-transmembrane G-pro…

Kategori:
AnalgesicsAnestheticsCentral Nervous System Agents +18
Target Protein:
Mu-type opioid receptor
Waktu ParuhOliceridine has a h…
Vol. DistribusiOliceridine has a m…
KlirensHealthy volunteers …
Genetik -
Olinciguat DB15238
small molecule | CAS: 1628732-62-6

Olinciguat is under investigation in clinical trial NCT03892499 (A Trial to Evaluate the Effect of Itraconazole (ITZ), a CYP3A4 Inhibitor, on the Pharmacokinetics of the Soluble Guanylate Cyclase Stimulator, Olinciguat (IW-1701), in Healthy Volunteers).

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Olinvacimab DB16265
biotech | CAS: 2095504-49-5

Olinvacimab is under investigation in clinical trial NCT03033524 (Trial to Evaluate the Safety of Ttac-0001(tanibirumab) in Recurrent Glioblastoma).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Target Protein:
Vascular endothelial growth factor receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Olipudase alfa Approved DB12835
biotech | CAS: 927883-84-9

Olipudase alfa is recombinant human acid sphingomyelinase.[A251590] It is the first and only enzyme replacement therapy in the world for the treatment of Acid Sphingomyelinase Deficiency (ASMD), also known as Niemann–Pick disease.[L42740] ASMD is a rare lysos…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsEnzyme Replacement Therapy +7
Waktu ParuhAfter administratio…
Vol. DistribusiAfter administratio…
KlirensAfter administratio…
Genetik -
Olitigaltin DB12895
small molecule | CAS: 1450824-22-2

Olitigaltin has been investigated for the treatment of Idiopathic Pulmonary Fibrosis.

Kategori:
CarbohydratesGalactosidesGlycosides +2
Target Protein:
Galectin-3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Olive oil Approved DB09567
biotech | CAS: 8001-25-0

Oil extracted from olives [L857]. Consists primarily of the glycerides of the fatty acids linoleic, oleic and palmitic. Used as a source of fatty acids in total parenteral nutrition and as an additive in some cosmetic products [FDA Label].

Kategori:
Biological ProductsDiet, Food, and NutritionDietary Fats +10
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Olmesartan Approved DB00275
small molecule | CAS: 144689-24-7

Olmesartan belongs to the angiotensin II receptor blocker (ARB) family of drugs, which also includes [telmisartan], [candesartan], [losartan], [valsartan], and [irbesartan]. ARBs selectively bind to angiotensin receptor 1 (AT1) and prevent the protein angiote…

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing hyperkalemiaAngiotensin 2 Receptor Blocker +15
Target Protein:
Type-1 angiotensin II receptor
Waktu ParuhThe mean plasma olm…
Vol. Distribusi17 L[L5566]
KlirensTotal plasma cleara…
Genetik -
Olmutinib DB13164
small molecule | CAS: 1353550-13-6

Olmutinib is an orally active epidermal growth factor receptor inhibitor used in the treatment of T790M mutation positive non-small cell lung cancer. It is available under the brand name Olita made by Hanmi Pharmaceuticals [A19196]. Olmutinib was developed by…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsEpidermal growth factor receptor (EGFR) tyrosine kinase inhibitors +1
Target Protein:
Epidermal growth factor receptor
Waktu Paruh8-11h [L766].
Vol. DistribusiData not yet availa…
KlirensData not yet availa…
Genetik -
Olodanrigan DB16266
small molecule | CAS: 1316755-16-4

Olodanrigan is under investigation in clinical trial NCT03297294 (Safety and Efficacy of EMA401 in Patients With Painful Diabetic Neuropathy (PDN)).

Kategori:
Benzene DerivativesHeterocyclic Compounds, Fused-Ring
Target Protein:
Type-2 angiotensin II receptor
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Olodaterol Approved DB09080
small molecule | CAS: 868049-49-4

Olodaterol is a novel, long-acting beta2-adrenergic agonist (LABA) that exerts its pharmacological effect by binding and activating beta2-adrenergic receptors located primarily in the lungs. Beta2-adrenergic receptors are membrane-bound receptors that are nor…

Kategori:
Adrenergic AgonistsAdrenergic beta-1 Receptor AgonistsAdrenergic beta-2 Receptor Agonists +20
Target Protein:
Beta-2 adrenergic receptor
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe volume of distr…
KlirensTotal clearance of …
Genetik -
Menampilkan 11051–11100 dari 15718
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