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13591

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10177 (74.9%)
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7625 (56.1%)
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104 (0.8%)
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13591 (100.0%)

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Hasil Pencarian (13591)

Halaman 221 / 272
biotech | CAS: 2610074-57-0

Raludotatug deruxtecan is under investigation in clinical trial NCT06660654 (A Study of Raludotatug Deruxtecan in Participants With Advanced/metastatic Solid Tumors (Rejoice-pantumor01)).

Waktu Paruh-
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Raluridine DB12894
small molecule | CAS: 119644-22-3

Raluridine has been used in trials studying the treatment of HIV Infections.

Kategori:
DeoxyribonucleosidesNucleic Acids, Nucleotides, and NucleosidesNucleosides
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ramatercept DB15116
biotech | CAS: 1169766-01-1

Ramatercept is under investigation in clinical trial NCT00952887 (A Safety, Tolerability, Pharmacokinetic and Pharmacodynamic Study of ACE-031 in Healthy Postmenopausal Women).

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Ramatroban DB13036
small molecule | CAS: 116649-85-5

Ramatroban has been used in trials studying the treatment of Asthma.

Kategori:
AmidesAntiplatelet agentsHematologic Agents +5
Target Protein:
Thromboxane A2 receptorProstaglandin D2 receptor 2
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Ramipril Approved DB00178
small molecule | CAS: 87333-19-5

Ramipril is a prodrug belonging to the angiotensin-converting enzyme (ACE) inhibitor class of medications. It is metabolized to ramiprilat in the liver and, to a lesser extent, kidneys. Ramiprilat is a potent, competitive inhibitor of ACE, the enzyme responsi…

Kategori:
ACE Inhibitors and Calcium Channel BlockersACE Inhibitors and DiureticsAgents Acting on the Renin-Angiotensin System +14
Target Protein:
Angiotensin-converting enzymeB1 bradykinin receptor
Gen Terkait:
ACE
Waktu ParuhPlasma concentratio…
Vol. Distribusi-
KlirensThe renal clearance…
Genetik 1 Varian
Ramosetron DB09290
small molecule | CAS: 132036-88-5

Ramosetron is a _serotonin 5-HT3 receptor antagonist_ commonly employed to treat nausea and vomiting, in addition to certain diarrheal conditions. It is believed to have higher potency and longer antiemetic action than other 1st generation 5-HT3 antagonists s…

Kategori:
Antidepressive AgentsAntiemeticsAutonomic Agents +10
Target Protein:
5-hydroxytryptamine receptor 3A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ramucirumab Approved DB05578
biotech | CAS: 947687-13-0

Ramucirumab is a human monoclonal antibody (IgG1) against vascular endothelial growth factor receptor 2 (VEGFR2), a type II trans-membrane tyrosine kinase receptor expressed on endothelial cells. By binding to VEGFR2, ramucirumab prevents binding of its ligan…

Kategori:
Amino Acids, Peptides, and ProteinsAngiogenesis InhibitorsAngiogenesis Modulating Agents +20
Target Protein:
Vascular endothelial growth factor receptor 2
Waktu Paruh15 days
Vol. Distribusi5.5 L
Klirens0.014 L/hour
Genetik -
Ranibizumab Approved DB01270
biotech | CAS: 347396-82-1

Ranibizumab is a recombinant humanized IgG1 kappa isotype monoclonal antibody fragment directed against human vascular endothelial growth factor A (VEGF-A), which is a glycoprotein implicated in the pathophysiology of age-related macular degeneration.[A2301, …

Kategori:
Amino Acids, Peptides, and ProteinsAngiogenesis InhibitorsAngiogenesis Modulating Agents +19
Target Protein:
Vascular endothelial growth factor A, long form
Waktu ParuhThe estimated avera…
Vol. DistribusiThe apparent volume…
KlirensIn patients with re…
Genetik -
Ranimustine DB13832
small molecule | CAS: 58994-96-0

Deskripsi belum tersedia.

Kategori:
Alkylating DrugsAmidesAntineoplastic Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ranirestat DB05327
small molecule | CAS: 147254-64-6

Ranirestat is a structurally novel and stereospecifically potent aldose reductase (AKR1B; EC 1.1.1.21) inhibitor, which contains a succinimide ring that undergoes ring-opening at physiological pH levels. It has been used in trials studying the treatment of M…

Kategori:
Aldehyde Reductase, antagonists & inhibitorsEnzyme Inhibitors
Target Protein:
Aldo-keto reductase family 1 member B1
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Ranitidine Approved DB00863
small molecule | CAS: 66357-35-5

Ranitidine is a commonly used drug, classified as a histamine H2-receptor antagonist, and belongs to the same drug class as [cimetidine] and [famotidine]. This drug helps to prevent and treat gastric-acid associated conditions, including ulcers, because of it…

Kategori:
Acid ReducersAgents Causing Muscle ToxicityAlimentary Tract and Metabolism +29
Target Protein:
Histamine H2 receptorAcetylcholinesterase
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensRenal clearance is …
Genetik -
Ranolazine Approved DB00243
small molecule | CAS: 95635-55-5

Chronic angina is a common cardiovascular condition affecting millions worldwide and causes significant disability while interfering with daily activities.[A189234] Ranolazine is a well-tolerated piperazine derivative used for the management of this condition…

Kategori:
AcetamidesAntianginal AgentsBSEP/ABCB11 Substrates +26
Target Protein:
PlasminogenSodium channel proteinInward rectifier potassium channel +4
Waktu ParuhThe apparent termin…
Vol. DistribusiThe mean apparent v…
KlirensThe reported cleara…
Genetik -
biotech | CAS: 2143578-32-7

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RAPA-501-Allo DB15890
biotech

RAPA-501-ALLO is composed of T-cells extracted from healthy volunteers; these cells are then reprogrammed _ex vivo_ in a process that involves de-differentiation and re-differentiation.[L16483]

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Rapacuronium Approved DB04834
small molecule | CAS: 465499-11-0

Rapacuronium was withdrawn in 2001 in many countries due to risk of fatal bronchospasm.

Kategori:
Agents producing tachycardiaAndrostanesAndrostanols +9
Target Protein:
Muscarinic acetylcholine receptor M2
Waktu Paruh141 minutes (mean)
Vol. Distribusi-
Klirens-
Genetik -
Rasagiline Approved DB01367
small molecule | CAS: 136236-51-6

Rasagiline is an irreversible inhibitor of monoamine oxidase and is used as a monotherapy in early Parkinson's disease or as an adjunct therapy in more advanced cases.

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAnti-Parkinson Drugs +19
Target Protein:
Amine oxidase [flavin-containing] BApoptosis regulator Bcl-2
Waktu ParuhRasagiline has a me…
Vol. Distribusi* 87 L
Klirens-
Genetik -
Rasburicase Approved DB00049
biotech | CAS: 134774-45-1

Rasburicase is a recombinant urate-oxidase enzyme produced by a genetically modified <i>Saccharomyces cerevisiae</i> strain. The cDNA coding for rasburicase was cloned from a strain of _Aspergillus flavus_.

Kategori:
Antigout PreparationsDetoxifying Agents for Antineoplastic TreatmentEnzymes +7
Target Protein:
Uric acid
Waktu Paruh18 hours
Vol. Distribusi* 110 to 127 mL/kg …
Klirens-
Genetik -
biotech | CAS: 1587257-96-2

Rasdegafusp alfa is under investigation in clinical trial NCT03206047 (Atezolizumab, Guadecitabine, and CDX-1401 Vaccine in Treating Patients With Recurrent Ovarian, Fallopian Tube, or Primary Peritoneal Cancer).

Waktu Paruh-
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Raspberry Approved DB10636
biotech

Raspberry allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Raubasine DB15949
small molecule | CAS: 483-04-5

Deskripsi belum tersedia.

Kategori:
AlkaloidsCardiovascular AgentsHeterocyclic Compounds, Fused-Ring +5
Target Protein:
Beta-1 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 8063-17-0

Rauwolfia (Rauwolfia serpentina), also spelled _ravolphia_, is a medicinal plant in the milkweed family. The root of the plant is ground into a powder or sold in tablets or capsules. It is a compound commonly used in Asian medicine, which includes traditional…

Kategori:
AlkaloidsAntiadrenergic Agents, Centrally ActingAntihypertensive Agents +6
Target Protein:
Synaptic vesicular amine transporter
Waktu ParuhAfter oral ingestio…
Vol. Distribusi-
KlirensHepatically and ren…
Genetik -
Ravagalimab DB16676
biotech | CAS: 2050816-56-1

Ravagalimab is under investigation in clinical trial NCT03695185 (A Study to Investigate How Well Ravagalimab (ABBV-323) Works and How Safe It Is in Participants With Moderate to Severe Ulcerative Colitis Who Failed Prior Therapy).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Ravidasvir DB15652
small molecule | CAS: 1242087-93-9

Ravidasvir is under investigation in clinical trial NCT02961426 (Sofosbuvir Plus Ravidasvir for the Treatment of HCV Chronic Infection).

Kategori:
Amino AcidsAmino Acids, Branched-ChainAmino Acids, Peptides, and Proteins +6
Target Protein:
Genome polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Ravoxertinib DB15281
small molecule | CAS: 1453848-26-4

Ravoxertinib is under investigation in clinical trial NCT01875705 (A Dose-Escalation Study of GDC-0994 in Patients With Locally Advanced or Metastatic Solid Tumors).

Kategori:
Antineoplastic AgentsEnzyme InhibitorsProtein Kinase Inhibitors +1
Target Protein:
Mitogen-activated protein kinase 3Mitogen-activated protein kinase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ravulizumab Approved DB11580
biotech | CAS: 1803171-55-2

Ravulizumab is a potent and selective complement 5 (C5) inhibitor. It is a humanized monoclonal IgG2/4 kappa antibody produced in Chinese hamster ovary (CHO) cells.[L39690] Ravulizumab was engineered from [eculizumab], another complement inhibitor, to increas…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +15
Target Protein:
Complement C5
Waktu ParuhThe mean (%CV) term…
Vol. DistribusiThe mean (%CV) volu…
KlirensThe mean (%CV) clea…
Genetik -
Raxibacumab Approved DB08902
biotech | CAS: 565451-13-0

Raxibacumab is a human IgG1? monoclonal antibody that binds the protective antigen (PA) component of B. anthracis toxin. Raxibacumab has a molecular weight of approximately 146 kilodaltons. Raxibacumab is produced by recombinant DNA technology in a murine cel…

Kategori:
Amino Acids, Peptides, and ProteinsAnthrax Protective Antigen-directed AntibodyAnthrax Protective Antigen-directed Antibody Interactions +12
Target Protein:
Protective antigen
Waktu ParuhMean terminal elimi…
Vol. DistribusiSteady state volume…
KlirensClearance values we…
Genetik -
Razupenem DB12587
small molecule | CAS: 426253-04-5

Razupenem has been used in trials studying the treatment of Skin Infections.

Kategori:
Amidesbeta-LactamsHeterocyclic Compounds, Fused-Ring +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Razuprotafib DB16353
small molecule | CAS: 1008510-37-9

Razuprotafib, also known as AKB-9778, is a small-molecule inhibitor restoring Tie2 activation by inhibiting VE-PTP.[L27171,L27176] In investigations against diabetes and COVID-19, razuprotafib is self-administered by patients through subcutaneous injection.

Kategori:
AcidsAcids, NoncarboxylicAmines +2
Target Protein:
Receptor-type tyrosine-protein phosphatase betaAngiopoietin-1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RCT1100 DB18830
biotech

RCT1100 is an investigational mRNA-based therapeutic that aims to treat primary ciliary dyskinesia caused by pathogenic mutations in DNAI1.[L50788]

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Genetik -
small molecule

Deskripsi belum tersedia.

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Genetik -
small molecule

Deskripsi belum tersedia.

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Rebastinib DB13005
small molecule | CAS: 1020172-07-9

Rebastinib has been used in trials studying the treatment of Chronic Myeloid Leukemia. It is an inhibitor of Tie2 tyrosine kinase receptor and an antineoplastic agent.

Kategori:
Antineoplastic AgentsEnzyme InhibitorsHeterocyclic Compounds, Fused-Ring +2
Target Protein:
Tyrosine-protein kinase ABL1Angiopoietin-1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rebaudioside A DB15136
small molecule | CAS: 58543-16-1

Rebaudioside A is under investigation in clinical trial NCT03510624 (Acute Effect of Rebaudioside A on Glucose Excursion During an Oral Glucose Tolerance Test in Type 2 Diabetes Mellitus).

Kategori:
AlkaloidsDiterpene AlkaloidsDiterpenes +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rebeccamycin DB14729
small molecule | CAS: 93908-02-2

Rebeccamycin is a weak topoisomerase I inhibitor isolated from _Nocardia sp_.

Kategori:
Heterocyclic Compounds, Fused-RingIndoles
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rebimastat DB06573
small molecule | CAS: 259188-38-0

Deskripsi belum tersedia.

Kategori:
Matrix Metalloproteinases
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Reboxetine Approved DB00234
small molecule | CAS: 71620-89-8

Reboxetine is an antidepressant drug used in the treatment of clinical depression, panic disorder and ADD/ADHD. Its mesylate (i.e. methanesulfonate) salt is sold under tradenames including Edronax, Norebox, Prolift, Solvex, Davedax or Vestra. Reboxetine has t…

Kategori:
Adrenergic AgentsAdrenergic Uptake InhibitorsAntidepressive Agents +20
Target Protein:
Sodium-dependent noradrenaline transporter
Waktu Paruh12.5 hours
Vol. Distribusi-
Klirens-
Genetik -
Recaticimab DB19302
biotech | CAS: 2361290-85-7

Recaticimab is under investigation in clinical trial NCT06467617 (Adebrelimab Plus Chemo and Recaticimab Perioperative Treatment for Resectable NSCLC).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech

Receptor binding domain SARS-CoV-2 Hepatitis B surface antigen virus-like particle vaccine (RBD SARS-CoV-2 HBsAg VLP vaccine), is a virus-like particle vaccine candidate where the RBD antigen is conjugated to the hepatitis B surface antigen[A226593]. Virus-li…

Waktu Paruh-
Vol. Distribusi-
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Recifercept DB17899
biotech | CAS: 2226238-09-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Recilisib DB18310
small molecule | CAS: 334969-03-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Recoflavone DB12058
small molecule | CAS: 203191-10-0

Recoflavone has been used in trials studying the treatment of Acute Gastritis, Dry Eye Syndrome, and Chronic Gastritis.

Kategori:
BenzopyransChromonesHeterocyclic Compounds, Fused-Ring +1
Target Protein:
Nuclear factor NF-kappa-B p105 subunitTranscription factor RelBNuclear factor NF-kappa-B p100 subunit +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 122320-05-2

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsEnzyme InhibitorsPeptides +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

B38-CAP is structured as a carboxypeptidase and derived from _Paenibacillus sp._ The molecule, an Angiotensin Converting Enzyme 2 (ACE2)-like enzyme, shares structural similarities to the mammalian ACE2. B38-CAP is an ACE2-like enzyme which decreases angioten…

Waktu Paruh-
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Genetik -
biotech

Deskripsi belum tersedia.

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biotech

Recombinant CD40-ligand is under investigation in clinical trial NCT00053391 (Vaccine Therapy in Treating Patients With Stage III or Stage IV Melanoma).

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCarbohydrates +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Recombinant Cholera Toxin B Subunit is an ingredient in the EMA-authorised product Dukoral.

Kategori:
Adjuvants, ImmunologicADP Ribose TransferasesBacterial Toxins +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech | CAS: 389069-73-2

Recombinant human kallikrein-1 is under investigation in clinical trial NCT01845064 (A Study to Evaluate the Safety and Effectiveness of DM199 in Healthy Subjects and Type 2 Diabetes Patients).

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

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biotech

Recombinant human thrombopoietin is a full-length glycosylated cytokine produced by Chinese hamster ovary cells and is used to promote the generation of megakaryocytes and platelets.[A225691, A225696] This drug is used in the treatment of thrombocytopenia.

Waktu Paruh-
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Menampilkan 11001–11050 dari 13591
Sebelumnya Halaman 221 / 272 Berikutnya