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2677

Total database: 17430
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1588 (59.3%)
Target
1494 (55.8%)
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51 (1.9%)
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2677 (100.0%)

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Hasil Pencarian (2677)

Halaman 22 / 54
Halofuginone DB04866
small molecule | CAS: 55837-20-2

Halofuginone is a low molecular weight quinazolinone alkaloid, and a potent inhibitor of collagen alpha1(I) and matrix metalloproteinase 2 (MMP-2) gene expression. Halofuginone also effectively suppresses tumor progression and metastasis in mice. Collgard Bio…

Kategori:
Angiogenesis InhibitorsAngiogenesis Modulating AgentsAnti-Infective Agents +10
Target Protein:
Collagen alpha-1(I) chain72 kDa type IV collagenase
Waktu Paruh23.8 to 72.1 hours
Vol. Distribusi-
Klirens-
Genetik -
Haloperidol Approved DB00502
small molecule | CAS: 52-86-8

Haloperidol is a high potency first-generation (typical) antipsychotic and one of the most frequently used antipsychotic medications used worldwide.[A180616] While haloperidol has demonstrated pharmacologic activity at a number of receptors in the brain,[A274…

Kategori:
Agents that reduce seizure thresholdAnti-Dyskinesia AgentsAntidepressive Agents +50
Target Protein:
5-hydroxytryptamine receptor 2CD(2) dopamine receptor5-hydroxytryptamine receptor 2A +15
Waktu ParuhFollowing oral admi…
Vol. DistribusiThe apparent volume…
KlirensFollowing intraveno…
Genetik -
biotech

Deskripsi belum tersedia.

Kategori:
AngiospermsBiological ProductsComplex Mixtures +10
Waktu Paruh-
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Genetik -
Helium Approved DB09155
small molecule | CAS: 7440-59-7

Helium is a second most abundant chemical element in the universe with symbol He and atomic number 2. It is a colorless, odorless, tasteless, non-toxic, inert, monatomic gas located at the top of the noble gases on the periodic table. Its boiling and melting …

Kategori:
ElementsGasesMedical Gases +3
Waktu Paruh0.8 seconds
Vol. Distribusi-
Klirens-
Genetik -
Hemoglobin Approved DB04945
biotech | CAS: 9008-02-0

The respiratory protein of the red blood cells. It consists primarily of globin and heme.

Kategori:
Amino Acids, Peptides, and ProteinsBlood ProteinsGlobins +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Heparin Approved DB01109
small molecule | CAS: 9005-49-6

Unfractionated heparin (UH) is a heterogenous preparation of anionic, sulfated glycosaminoglycan polymers with weights ranging from 3000 to 30,000 Da. It is a naturally occurring anticoagulant released from mast cells. It binds reversibly to antithrombin III …

Kategori:
Agents causing hyperkalemiaAnticoagulantsAntivaricose Therapy +16
Target Protein:
Antithrombin-IIICoagulation factor XP-selectin +9
Waktu ParuhThe plasma half-lif…
Vol. DistribusiThe volume of distr…
KlirensThe clearance in ad…
Genetik -
Hepatitis B immune globulin Approved DB05276
biotech

Long-term hepatitis B immune globulin (HBIG) has been shown to reduce hepatitis B virus (HBV) reinfection in patients transplanted for hepatitis B. Infection with hepatitis B may lead to hepatocellular carcinoma, a type of liver cancer. Therefore, the hepatit…

Kategori:
Amino Acids, Peptides, and ProteinsAntiinfectives for Systemic UseBlood Proteins +12
Target Protein:
HBsAg
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Hepatitis B Vaccine is an ingredient in the EMA-withdrawn product Quintanrix. It is marketed in Canada as Engerix B. It is also a part of Twinrix (Hep A/Hep B vaccine) available also in Canada. The hepatitis B virus induces a severe form of viral hepatitis. …

Kategori:
Actively Acquired ImmunityAmino Acids, Peptides, and ProteinsAntigens +19
Waktu ParuhEvaluation of pharm…
Vol. DistribusiEvaluation of pharm…
KlirensEvaluation of pharm…
Genetik -
Heptabarbital DB01354
small molecule | CAS: 509-86-4

Heptabarbital is an intermediate or short term barbiturate used mainly for sedation and hypnosis.

Kategori:
Anticholinergic AgentsBarbiturates, PlainCentral Nervous System Depressants +6
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1Gamma-aminobutyric acid receptor subunit alpha-2Gamma-aminobutyric acid receptor subunit alpha-3 +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Hesperidin Approved DB04703
small molecule | CAS: 520-26-3

Hesperidin is a flavan-on glycoside found in citrus fruits.

Kategori:
BenzopyransCarbohydratesChromones +5
Target Protein:
Voltage-dependent N-type calcium channel subunit alpha-1BAurora kinase B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Hexachlorophene Approved DB00756
small molecule | CAS: 70-30-4

A chlorinated bisphenol antiseptic with a bacteriostatic action against Gram-positive organisms, but much less effective against Gram-negative organisms. It is mainly used in soaps and creams and is an ingredient of various preparations used for skin disorder…

Kategori:
Anti-Infective AgentsAnti-Infective Agents, LocalAntiseptics and Disinfectants +8
Target Protein:
D-lactate dehydrogenaseSuccinate dehydrogenase [ubiquinone] cytochrome b small subunit, mitochondrialGlutamate dehydrogenase 1, mitochondrial +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Hydrocarbons, FluorinatedHydrocarbons, HalogenatedKetones
Waktu Paruh-
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Genetik -
Hexaminolevulinate Approved DB06261
small molecule | CAS: 140898-97-1

Hexaminolevulinate is an optical imaging drug. In solution form it is instilled intravesically for use with photodynamic blue light cystoscopy as an adjunct to white light cystoscopy. On May 28, 2010, the U.S. Food and Drug Administration (FDA) granted approv…

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsCarbon Radioisotopes +5
Waktu ParuhBiphasic eliminatio…
Vol. Distribusi-
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Genetik -
Hexobarbital DB01355
small molecule | CAS: 56-29-1

A barbiturate that is effective as a hypnotic and sedative.

Kategori:
AdjuvantsAnestheticsAnesthetics, General +18
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-2Gamma-aminobutyric acid receptor subunit alpha-3Gamma-aminobutyric acid receptor subunit alpha-4 +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Histrelin Approved DB06788
small molecule | CAS: 76712-82-8

Histrelin is a gonadotropin-releasing hormone (GnRH) agonist that acts as a potent inhibitor of gonadotropin when administered as an implant delivering continuous therapeutic doses. This drug is a synthetic analog of naturally occurring GnRH with a higher pot…

Kategori:
Adrenal Cortex HormonesAmino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating Agents +17
Target Protein:
Gonadotropin-releasing hormone receptor
Waktu ParuhIn healthy voluntee…
Vol. DistribusiThe apparent volume…
KlirensIn prostate cancer …
Genetik -
Homatropine Approved DB11181
small molecule | CAS: 87-00-3

Homatropine is an anticholinergic drug that acts as an antagonist at muscarinic acetylcholine receptors. It is present in antitussives, under the trade name Hycodan, in combination with hydrocodone (dihydrocodeinone) bitartrate indicated for the symptomatic r…

Kategori:
AlkaloidsAnticholinergic AgentsAutonomic Agents +8
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M3 +2
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Honey Approved DB14242
biotech | CAS: 8028-66-8

Honey is an animal extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
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HQP1351 DB16185
small molecule | CAS: 1257628-77-5

HQP1351 is under investigation in clinical trial NCT03883100 (A Pivotal Study of HQP1351 in Patients of Chronic Myeloid Leukemia in Accelerated Phase With T315I Mutation).

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +2
Waktu Paruh-
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HSK-3486 DB16295
small molecule | CAS: 1637741-58-2

HSK-3486 is under investigation in clinical trial NCT04620031 (A Study Evaluating Sedation of Intravenous Administration of HSK3486 Injectable Emulsion in ICU Patients Undergoing Mechanical Ventilation).

Kategori:
Benzene Derivatives
Waktu Paruh-
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Genetik -
biotech

Human amniotic fluid is the liquid surrounding the human embryo and fetus.[L16373] Physically, the fluid provides protection through cushioning. Chemically, the fluid provides protection through its inherent antibacterial properties. The fluid contains carboh…

Waktu Paruh-
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Genetik -
biotech

Infant botulism is a rare infectious disease occurring in infants in which _Clostridium botulinum_ colonize the large intestine and being to produce botulinum neurotoxin directly in the gut. As these neurotoxins interfere with cholinergic nervous transmission…

Kategori:
Bacterial Neurotoxin NeutralizationHuman Immunoglobulin GPassively Acquired Immunity
Waktu ParuhThe half-life of hu…
Vol. Distribusi-
Klirens-
Genetik -
Human calcitonin Approved DB06773
biotech | CAS: 21215-62-3

Calcitonin was first discovered in isolated parathyroid tissue as a substance with a serum-calcium-lowering effect.[A32099] It is constituted as a 32-amino acid single chain polypeptide structure that gets secreted as a regulatory agent in calcium-phosphorus …

Kategori:
Bone Density Conservation AgentsCalcitonin PreparationsCalcium Homeostasis +1
Target Protein:
Alpha-actinin-1
Waktu ParuhIntravenous adminis…
Vol. Distribusi-
KlirensThe metabolic clear…
Genetik -
biotech

Human cord blood hematopoietic progenitor cells consist of hematopoietic progenitor cells, monocytes, lymphocytes, and granulocytes from human cord blood. They are used during allogeneic unrelated and related hematopoietic stem cell transplantation procedures…

Kategori:
Allogeneic Cord Blood Hematopoietic Progenitor Cell Therapy
Waktu ParuhPharmacokinetic par…
Vol. DistribusiPharmacokinetic par…
KlirensPharmacokinetic par…
Genetik -
biotech | CAS: 339086-15-6

Cytomegalovirus immunoglobulin is obtained from pooled adult human plasma selected for high titers of antibody for cytomegalovirus (CMV). It contains purified immunoglobulin G (IgG) antibodies targeting cytomegalovirus (CMV)[FDA label]. Cytomegalovirus, a …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntiinfectives for Systemic Use +15
Waktu ParuhIgG1 has a half-lif…
Vol. DistribusiIgG is distributed …
Klirens-
Genetik -
Human interferon beta Approved DB14999
biotech | CAS: 74899-71-1

Human interferon beta is a polypeptide used in the management of relapsing forms of Multiple Sclerosis (MS), and was initially approved by the FDA in 1992.[L12081] Multiple Sclerosis is a devastating neurodegenerative disease that is usually progressive and s…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsBiological Factors +7
Target Protein:
Interferon alpha/beta receptor 1
Waktu ParuhThe mean terminal e…
Vol. DistribusiThe average state v…
KlirensAverage serum clear…
Genetik -
biotech

Human interferon omega 1 (IFN-omega 1 = IFN-alpha II1) is a recently discovered protein structurally related to IFN-alpha and -beta. It occurs naturally in the human body and is currently being manufactured by Intarcia through genetic engineering. There are m…

Kategori:
Immunosuppressive AgentsMyelosuppressive Agents
Target Protein:
Interferon alpha/beta receptor 1Interferon alpha/beta receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Stem cells are self-renewing and proliferate without differentiation, with the two major groups being embryonic stem cells (ESCs) and adult stem cells (ASC). Differentiation occurs under different conditions into different cell types. ESCs are from the inner …

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Human papillomavirus type 11 L1 capsid protein antigen is contained in Gardasil, or a recombinant Human Papillomavirus Quadrivalent (Types 6, 11, 16, and 18) vaccine for intramuscular injection. It is an immunization for young men and women 9-26 years of age …

Kategori:
Actively Acquired ImmunityCancer immunotherapyImmunotherapy +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Human papillomavirus type 16 L1 capsid protein antigen is contained in Gardasil, or a recombinant Human Papillomavirus Quadrivalent (Types 6, 11, 16, and 18) vaccine for intramuscular injection. It is an immunization for young men and women 9-26 years of age …

Kategori:
Actively Acquired ImmunityAmino Acids, Peptides, and ProteinsCancer immunotherapy +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Human papillomavirus type 18 L1 capsid protein antigen is contained in Gardasil, or a recombinant Human Papillomavirus Quadrivalent (Types 6, 11, 16, and 18) vaccine for intramuscular injection. It is an immunization for young men and women 9-26 years of age …

Kategori:
Actively Acquired ImmunityCancer immunotherapyImmunotherapy +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Human papillomavirus type 31 L1 capsid protein antigen is contained in Gardasil is a vaccine for intramuscular injection. It is an immunization for young men and women 9-26 years of age for the prevention of diseases caused by Human Papillomavirus (HPV) type …

Kategori:
Cancer immunotherapyImmunotherapy
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Human papillomavirus type 33 L1 capsid protein antigen is contained in Gardasil is a vaccine for intramuscular injection. It is an immunization for young men and women 9-26 years of age for the prevention of diseases caused by Human Papillomavirus (HPV) type …

Kategori:
Cancer immunotherapyImmunotherapy
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Human papillomavirus type 45 L1 capsid protein antigen is contained in Gardasil is a vaccine for intramuscular injection. It is an immunization for young men and women 9-26 years of age for the prevention of diseases caused by Human Papillomavirus (HPV) type …

Kategori:
Cancer immunotherapyImmunotherapy
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Human papillomavirus type 52L1 capsid protein antigen is contained in Gardasil is a vaccine for intramuscular injection. It is an immunization for young men and women 9-26 years of age for the prevention of diseases caused by Human Papillomavirus (HPV) type 5…

Kategori:
Cancer immunotherapyImmunotherapy
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Human papillomavirus type 58 L1 capsid protein antigen is contained in Gardasil is a vaccine for intramuscular injection. It is an immunization for young men and women 9-26 years of age for the prevention of diseases caused by Human Papillomavirus (HPV) type …

Kategori:
Cancer immunotherapyImmunotherapy
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Human papillomavirus type 6 L1 capsid protein antigen is contained in Gardasil, or a recombinant Human Papillomavirus Quadrivalent (Types 6, 11, 16, and 18) vaccine for intramuscular injection. It is an immunization for young men and women 9-26 years of age f…

Kategori:
Actively Acquired ImmunityCancer immunotherapyImmunotherapy +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Transplantation with human umbilical cord blood mononuclear cells (HUCBC) has demonstrated promising results in various disease states. While some of the positive results are credited to HUCBCs’ differentiation potential, the growth factors and cytokines thes…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech

Stem cells obtained from amniotic fluid, the umbilical cord (UC), and placenta are gaining in popularity. Stem cells from the umbilical cord offer several advantages, including: non-invasive collection procedures, more hearty and steady growth than bone-marro…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech

Human vaccinia immune globulin (VIG) is a sterile solution containing the purified gamma globulin (IgG) fraction of plasma taken from healthy donors previously vaccinated with live vaccinia virus vaccine who possess high titers of anti-vaccinia virus antibody…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +10
Waktu ParuhThe mean half-life …
Vol. DistribusiThe volume of distr…
KlirensReadily accessible …
Genetik -
biotech

Human varicella-zoster immune globulin is a solvent/detergent-treated sterile liquid preparation of purified human immune globulin G (IgG) containing antibodies to varicella zoster virus (anti-VZV). It is prepared from pools of healthy human donors' plasma vi…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBiological Products +13
Waktu ParuhHuman Varicella-Zos…
Vol. DistribusiFollowing intraveno…
Klirens-
Genetik -
Huperzine A Approved DB04864
small molecule | CAS: 102518-79-6

Huperzine A, is a naturally occurring sesquiterpene alkaloid found in the extracts of the firmoss _Huperzia serrata_. The botanical has been used in China for centuries for the treatment of swelling, fever and blood disorders. Recently in clinical trials in C…

Kategori:
Central Nervous System AgentsCholinergic AgentsCholinesterase Inhibitors +6
Target Protein:
Acetylcholinesterase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
HY10275 DB05079
small molecule

HY10275 is a novel compound specifically designed to modulate two key neurobiological mechanisms that interfere with the sleeping process. HY10275 is highly selective for histamine H1 and serotonin 5HT2a, two chemical receptors that are known to impact the ab…

Target Protein:
Histamine H1 receptor5-hydroxytryptamine receptor 2A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Hyaluronic acid Approved DB08818
small molecule | CAS: 9004-61-9

Hyaluronic acid (HA) is an anionic, nonsulfated glycosaminoglycan found in connective, epithelial, and neural tissues; it was first isolated in 1934. Karl Meyer and John Palmer obtained glycosaminoglycan (GAG) from the bovine eye, giving it the name “hyaluron…

Kategori:
Adjuvants, ImmunologicBiocompatible MaterialsCarbohydrates +16
Target Protein:
CD44 antigenIntercellular adhesion molecule 1Hyaluronan mediated motility receptor +12
Waktu ParuhWhen injected by th…
Vol. DistribusiThere is limited in…
KlirensThere is limited in…
Genetik -
biotech | CAS: 757971-58-7

A purified preparation of the enzyme recombinant human hyaluronidase. Hyaluronidase (human recombinant) (INN Vorhyaluronidase alfa) is produced by genetically engineered Chinese Hamster Ovary (CHO) cells containing a DNA plasmid encoding for a soluble fragmen…

Kategori:
Blood and Blood Forming OrgansCarbon-Oxygen LyasesEnzymes +6
Target Protein:
Hyaluronic acidTransforming growth factor beta-1 proprotein
Waktu ParuhHyaluronidase has a…
Vol. DistribusiData regarding the …
KlirensData regarding the …
Genetik -
Hyaluronidase (ovine) Approved DB00070
biotech | CAS: 488712-31-8

Highly purified sheep hyaluronidase for administration by injection into the vitreous of the eye.

Kategori:
EnzymesEnzymes and CoenzymesGlycoside Hydrolases
Target Protein:
Transforming growth factor beta-1 proprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Hydrocodone Approved DB00956
small molecule | CAS: 125-29-1

Hydrocodone is a synthetic opioid derivative of codeine.[T116] It is commonly used in combination with [acetaminophen] to control moderate to severe pain. Historically, hydrocodone has been used as a cough suppressant although this has largely been replaced b…

Kategori:
AlkaloidsAnalgesicsAntitussive Agents +23
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorSigma non-opioid intracellular receptor 1
Waktu ParuhThe half-life of el…
Vol. DistribusiThe apparent volume…
KlirensOfficial FDA labeli…
Genetik -
Hydrocortisone butyrate Approved DB14540
small molecule | CAS: 13609-67-1

Deskripsi belum tersedia.

Kategori:
11-Hydroxycorticosteroids17-HydroxycorticosteroidsAdministration, Topical +26
Target Protein:
Annexin A1Glucocorticoid receptor11-beta-hydroxysteroid dehydrogenase type 2 +1
Waktu Paruh6-8 hours
Vol. Distribusi-
Klirens-
Genetik -
Hydrocortisone probutate Approved DB14543
small molecule | CAS: 72590-77-3

Deskripsi belum tersedia.

Kategori:
11-Hydroxycorticosteroids17-HydroxycorticosteroidsAdrenal Cortex Hormones +26
Target Protein:
Annexin A1Glucocorticoid receptor11-beta-hydroxysteroid dehydrogenase type 2 +1
Waktu Paruh6-8 hours
Vol. Distribusi-
Klirens-
Genetik -
Hydrocortisone valerate Approved DB14544
small molecule | CAS: 57524-89-7

Deskripsi belum tersedia.

Kategori:
11-Hydroxycorticosteroids17-HydroxycorticosteroidsAdrenal Cortex Hormones +23
Target Protein:
Annexin A1Glucocorticoid receptor11-beta-hydroxysteroid dehydrogenase type 2 +1
Waktu Paruh6-8 hours
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 8016-70-4

Extracted from the seeds of the soybean (Glycine soja), hydrogenated soybean oil is a major food fat used in the production of margarine, shortening, and salad and cooking oils. According to the FDA, hydrogenated soybean oil is generally recognized as safe (G…

Waktu Paruh-
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