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2279

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866 (38.0%)
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1100 (48.3%)
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Halaman 22 / 46
Hydroxyzine Approved DB00557
small molecule | CAS: 68-88-2

Hydroxyzine is a first-generation histamine H<sub>1</sub>-receptor antagonist of the dephenylmethane and piperazine classes that exhibits sedative, anxiolytic, and antiemetic properties.[A1257,A187589] It was first developed in 1955,[A189726] and has since re…

Kategori:
Anti-Anxiety AgentsAntipruriticsCentral Nervous System Depressants +21
Target Protein:
Histamine H1 receptorVoltage-gated inwardly rectifying potassium channel KCNH2
Waktu ParuhThe half-life of hy…
Vol. DistribusiThe mean volume of …
KlirensClearance of hydrox…
Genetik -
Ibalizumab Approved DB12698
biotech | CAS: 680188-33-4

Ibalizumab (also known as _ibalizumab-uiyk_ and formerly known as TNX-355) is a monoclonal antibody that binds to CD4 receptors on the surface of CD4-positive cells, preventing HIV particle entry into the lymphocytes. It is an advanced and current antibody in…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-HIV AgentsAnti-Infective Agents +19
Target Protein:
C-C chemokine receptor type 5C-X-C chemokine receptor type 4T-cell surface glycoprotein CD4
Waktu ParuhThe half-life of ib…
Vol. Distribusi4.8 L [FDA label]
KlirensFollowing single-do…
Genetik -
Iboctadekin DB14920
biotech | CAS: 479198-61-3

Iboctadekin is under investigation in clinical trial NCT00500058 (A Phase I, Dose-Escalation Study to Assess the Safety and Biological Activity of Recombinant Human Interleukin-18).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ibrexafungerp Approved DB12471
small molecule | CAS: 1207753-03-4

Ibrexafungerp, also known as SCY-078 or MK-3118, is a novel enfumafungin derivative oral triterpene antifungal approved for the treatment of vulvovaginal candidiasis (VVC), also known as a vaginal yeast infection.[A235384,L34349] It was developed out of a nee…

Kategori:
Anti-Infective AgentsAntifungal AgentsAntiinfectives for Systemic Use +17
Target Protein:
1,3-beta-glucan synthase component GSC2GTP-binding protein RHO1
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensClearance values of…
Genetik -
Ibrutinib Approved DB09053
small molecule | CAS: 936563-96-1

Ibrutinib is a small molecule that acts as an irreversible potent inhibitor of Burton's tyrosine kinase. It is designated as a targeted covalent drug and presented as a promising activity in B-cell malignancies in clinical trials.[A32299] Ibrutinib was develo…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBruton's tyrosine kinase (BTK) inhibitors +15
Target Protein:
Tyrosine-protein kinase BTK
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensIn patients with no…
Genetik -
Icariin DB12052
small molecule | CAS: 489-32-7

Icariin has been investigated for the basic science of the Pharmacokinetic Profile of Icariin in Humans.

Kategori:
BenzopyransChromonesDrugs, Chinese Herbal +3
Target Protein:
cGMP-specific 3',5'-cyclic phosphodiesterase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Idarucizumab Approved DB09264
biotech | CAS: 1362509-93-0

Idarucizumab is a humanized monoclonal antibody fragment (Fab) derived from an immunoglobulin G1 isotype molecule that binds to and inactivates the oral anticoagulant dabigatran, thereby reversing its anticoagulant effect. As a direct acting oral anticoagulan…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Waktu Paruhinitial half-life: …
Vol. Distribusi8.9 L
Klirens47.0 mL/min
Genetik -
Idecabtagene vicleucel Approved DB16665
biotech

Multiple myeloma is a cancer where plasma cells rapidly divide out of control.[A232563] These cancerous cells generally express the B-cell maturation antigen, while it is rarely expressed on non-cancerous cells.[A232563] Multiple myeloma is typically treated …

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic AgentsAntineoplastic Agents, Immunological +11
Target Protein:
Tumor necrosis factor receptor superfamily member 17
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
IDM-4 DB05438
biotech

IDM-4 is an immuno-designed molecule that completed phase I/II of investigation for the treatment of Leukemia. It is a monoclonal antibody-specific antigen that can selectively target cancer-affected cells by coupling with tumor cell-killing MAK cells, which …

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Idursulfase Approved DB01271
biotech | CAS: 50936-59-9

Idursulfase is a purified form of human iduronate-2-sulfatase, a lysosomal enzyme. Idursulfase is produced by recombinant DNA technology in a human cell line. Idursulfase is an enzyme that hydrolyzes the 2-sulfate esters of terminal iduronate sulfate residues…

Kategori:
Alimentary Tract and MetabolismEnzymesEnzymes and Coenzymes +4
Target Protein:
Dermatan sulfateHeparan sulfatePerilipin-3
Waktu Paruh44 &plusmn; 19 minu…
Vol. Distribusi-
Klirens* 3 mL/min/kg [Pati…
Genetik -
biotech | CAS: 1271734-34-9

Idursulfase beta is under investigation in clinical trial NCT01645189 (Safety and Efficacy of Hunterase).

Kategori:
Alimentary Tract and MetabolismEnzymesEnzymes and Coenzymes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2484870-92-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
IGN311 DB04988
biotech

IGN311 is a humanized monoclonal antibody (mab) against the Lewis Y carbohydrate antigen, a blood-group-related oligosaccharide.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Target Protein:
Epidermal growth factor receptorReceptor tyrosine-protein kinase erbB-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
IL-2 pDNA DB05935
small molecule

Vical incorporated has initiated a human Phase 1 study of an investigational method of delivering interleukin-2 (IL-2), a potent immune system stimulant, for patients with recurrent metastatic melanoma.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Iloperidone Approved DB04946
small molecule | CAS: 133454-47-4

Iloperidone is a benzisoxazole [A263557] and an atypical antipsychotic agent that was first approved by the FDA on May 6, 2009.[A3024] It is considered to be a second-generation antipsychotic drug [A263552] with multiple receptor binding profile, although it …

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +31
Target Protein:
5-hydroxytryptamine receptor 2AD(2) dopamine receptor5-hydroxytryptamine receptor 1A +14
Waktu ParuhThe observed mean e…
Vol. DistribusiThe apparent volume…
KlirensIloperidone has an …
Genetik -
Iltamiocel DB19059
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Iluzanebart DB18275
biotech | CAS: 2733621-19-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 138660-99-8

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Imdevimab Approved DB15940
biotech | CAS: 2415933-40-1

Imdevimab is a monoclonal antibody combined with [casirivimab] in Regeneron's antibody cocktail known as REGEN-COV2 for the treatment of COVID-19.[L23539] This drug is a combination of antibodies derived from humanized VelocImmune® mice in addition to blood …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Target Protein:
Spike glycoprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Imetelstat Approved DB14909
small molecule | CAS: 868169-64-6

Imetelstat is a first-in-class 18-amino acid oligonucleotide that directly and competitively inhibits human telomerase.[A263973] It is used to treat anemia in patients with myelodysplastic syndromes (MDS), a group of hematologic disorders characterized by ine…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsEnzyme Inhibitors +6
Target Protein:
Telomerase reverse transcriptaseHuman telomerase RNA component
Waktu ParuhThe geometric mean …
Vol. DistribusiThe geometric mean …
Klirens-
Genetik -
IMGN632 DB17337
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Imidacloprid DB11421
small molecule | CAS: 105827-78-9

Imidacloprid is a neonicotinoid, which is a class of neuro-active insecticides modeled after nicotine. Imidacloprid is a patented chemical, Imidacloprid is manufactured by Bayer Cropscience (part of Bayer AG) and sold under trade names Kohinor, Admire, Advant…

Kategori:
AgrochemicalsCholinergic AgentsCompounds used in a research, industrial, or household setting +4
Target Protein:
CHRNA7-FAM7A fusion protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Imiglucerase Approved DB00053
biotech | CAS: 154248-97-2

Human Beta-glucocerebrosidase or Beta-D-glucosyl-N-acylsphingosine glucohydrolase E.C. 3.2.1.45. 497 residue protein with N-linked carbohydrates, MW=59.3 kD. Alglucerase is prepared by modification of the oligosaccharide chains of human Beta-glucocerebrosidas…

Kategori:
Alimentary Tract and MetabolismEnzyme Replacement TherapyEnzymes +6
Target Protein:
Glucocerebroside
Waktu Paruh3.6-10.4 min
Vol. Distribusi* 0.09 to 0.15 L/kg
Klirens* 14.5 +/- 4.0 mL/m…
Genetik -
Imipenem Approved DB01598
small molecule | CAS: 64221-86-9

Imipenem is a semisynthetic thienamycin that has a wide spectrum of antibacterial activity against gram-negative and gram-positive aerobic and anaerobic bacteria, including many multiresistant strains.[label] It is stable to many beta-lactamases. Similar comp…

Kategori:
Agents that reduce seizure thresholdAmidesAnti-Bacterial Agents +12
Target Protein:
Penicillin-binding protein 2Penicillin-binding protein 1BPenicillin-binding protein 1A +3
Waktu ParuhWhen given via IV i…
Vol. DistribusiThe reported volume…
KlirensThe total clearance…
Genetik -
Imlifidase Approved DB15258
biotech | CAS: 1947415-68-0

Chronic kidney disease (CKD) is a progressive and irreversible disease that represents a significant burden for both the individual and healthcare system at large.[A225916] Currently available treatments for end-stage renal disease are limited to dialysis and…

Kategori:
Antineoplastic and Immunomodulating AgentsEndopeptidasesImmunosuppressive Agents +2
Target Protein:
IgG heavy chain
Waktu ParuhThe mean distributi…
Vol. DistribusiThe volume of distr…
KlirensThe mean clearance …
Genetik -
IMMU-114 DB18458
biotech

IMMU-114 is antibody-drug conjugate consisting of humanized anti-HLA-DR IgG4 monoclonal antibody specific for alpha-chain linked to SN-38 via a CL2A linker.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Immucin DB17403
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Inavolisib Approved DB15275
small molecule | CAS: 2060571-02-8

_PIK3CA_ is one of the most frequently mutated oncogenes, with the resulting mutated p110? protein it encodes playing a central role in tumor cell proliferation.[A264563] Chemotherapeutic agents targeting the PI3K p110? catalytic subunit have shown antitumor …

Kategori:
BCRP/ABCG2 SubstratesCytochrome P-450 CYP2B6 InducersCytochrome P-450 CYP2B6 Inducers (strength unknown) +4
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoformPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
Waktu ParuhThe elimination hal…
Vol. DistribusiThe apparent volume…
KlirensThe total clearance…
Genetik -
Inbakicept DB16479
biotech | CAS: 2135939-52-3

Inbakicept is a dimeric human IL-15 receptor ? (IL-15R?) sushi domain/human IgG1 Fc fusion protein. It is one of the active ingredients in Anktiva, a combination product also containing [nogapendekin alfa], where a single inbakicept is complexed with two noga…

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic AgentsExperimental Unapproved Treatments for COVID-19 +4
Target Protein:
Interleukin-2 receptor subunit betaCytokine receptor common subunit gamma
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
INBRX-101 DB18384
biotech

INBRX-101 is a recombinant human alpha-1 antitrypsin (AAT)-Fc fusion protein.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Indacaterol Approved DB05039
small molecule | CAS: 312753-06-3

Indacaterol is a novel, ultra-long-acting, rapid onset ?(2)-adrenoceptor agonist developed for Novartis for the once-daily management of asthma and chronic obstructive pulmonary disease. It was approved by the European Medicines Agency (EMA) on 30 November 20…

Kategori:
Adrenergic AgonistsAdrenergic beta-2 Receptor AgonistsAdrenergic beta-Agonists +17
Target Protein:
Beta-2 adrenergic receptor
Waktu ParuhIndacaterol serum c…
Vol. DistribusiAfter intravenous i…
KlirensRenal clearance of …
Genetik -
Inebilizumab Approved DB12530
biotech | CAS: 1299440-37-1

Inappropriate growth of or self-directed antibody production by B-cells is the etiological underpinning of a variety of conditions, including the multiple sclerosis-like neurological condition neuromyelitis optica spectrum disorder (NMOSD).[A214283, A214286] …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +12
Target Protein:
B-lymphocyte antigen CD19
Waktu ParuhInebilizumab exhibi…
Vol. DistribusiInebilizumab has an…
KlirensInebilizumab has an…
Genetik -
Infliximab Approved DB00065
biotech | CAS: 170277-31-3

Infliximab is a tumor necrosis factor (TNF-alpha or TNF-?) blocker and a chimeric monoclonal IgG1 antibody composed of human constant (75%) and murine variable (25%) regions [A31469]. Infliximab is produced by a recombinant cell line cultured by continuous pe…

Kategori:
Agents Causing Muscle ToxicityAgents reducing cytokine levelsAmino Acids, Peptides, and Proteins +21
Target Protein:
Tumor necrosis factor
Gen Terkait:
FCGR3A
Waktu ParuhThe median terminal…
Vol. DistribusiBased on a pharmaco…
KlirensIn patients with Cr…
Genetik 1 Varian
biotech

A seasonally-specific component of the influenza vaccine. The influenza vaccine, also known as the "flu shot", is a vaccine that helps to protect against infection from influenza viruses. These vaccines provide protection from influenza by exposing the immune…

Kategori:
Inactivated Influenza A Virus VaccineInfluenza VaccinesVaccines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

A seasonally-specific component of the influenza vaccine. The influenza vaccine, also known as the "flu shot", is a vaccine that helps to protect against infection from influenza viruses. These vaccines provide protection from influenza by exposing the immune…

Kategori:
Influenza VaccinesRecombinant influenza vaccinesVaccines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

A seasonally-specific component of the influenza vaccine. The influenza vaccine, also known as the "flu shot", is a vaccine that helps to protect against infection from influenza viruses. These vaccines provide protection from influenza by exposing the immune…

Kategori:
Inactivated Influenza A Virus VaccineInfluenza VaccinesVaccines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

A seasonally-specific component of the influenza vaccine. The influenza vaccine, also known as the "flu shot", is a vaccine that helps to protect against infection from influenza viruses. These vaccines provide protection from influenza by exposing the immune…

Kategori:
Inactivated Influenza A Virus VaccineInfluenza VaccinesVaccines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

A seasonally-specific component of the influenza vaccine. The influenza vaccine, also known as the "flu shot", is a vaccine that helps to protect against infection from influenza viruses. These vaccines provide protection from influenza by exposing the immune…

Kategori:
Influenza VaccinesRecombinant influenza vaccinesVaccines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

A seasonally-specific component of the influenza vaccine. The influenza vaccine, also known as the "flu shot", is a vaccine that helps to protect against infection from influenza viruses. These vaccines provide protection from influenza by exposing the immune…

Kategori:
Influenza VaccinesLive Attenuated Influenza A Virus VaccineVaccines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

A seasonally-specific component of the influenza vaccine. The influenza vaccine, also known as the "flu shot", is a vaccine that helps to protect against infection from influenza viruses. These vaccines provide protection from influenza by exposing the immune…

Kategori:
Inactivated Influenza A Virus VaccineInfluenza VaccinesVaccines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

A seasonally-specific component of the influenza vaccine. The influenza vaccine, also known as the "flu shot", is a vaccine that helps to protect against infection from influenza viruses. These vaccines provide protection from influenza by exposing the immune…

Kategori:
Inactivated Influenza A Virus VaccineInfluenza VaccinesVaccines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

A seasonally-specific component of the influenza vaccine. The influenza vaccine, also known as the "flu shot", is a vaccine that protects against infection from the influenza viruses. Vaccines provide protection from influenza by exposing the immune system to…

Kategori:
Inactivated Influenza A Virus VaccineInfluenza VaccinesVaccines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

A seasonally-specific component of the influenza vaccine. The influenza vaccine, also known as the "flu shot", is a vaccine that protects against infection from the influenza viruses. Vaccines provide protection from influenza by exposing the immune system to…

Kategori:
Influenza VaccinesLive Attenuated Influenza A Virus VaccineVaccines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Kategori:
Influenza VaccinesRecombinant influenza vaccinesVaccines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

A seasonally-specific component of the influenza vaccine. The influenza vaccine, also known as the "flu shot", is a vaccine that protects against infection from the influenza viruses. Vaccines provide protection from influenza by exposing the immune system to…

Kategori:
Inactivated Influenza A Virus VaccineInfluenza VaccinesVaccines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

A seasonally-specific component of the influenza vaccine. The influenza vaccine, also known as the "flu shot", is a vaccine that protects against infection from the influenza viruses. Vaccines provide protection from influenza by exposing the immune system to…

Kategori:
Inactivated Influenza A Virus VaccineInfluenza VaccinesVaccines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

A seasonally-specific component of the influenza vaccine. The influenza vaccine, also known as the "flu shot", is a vaccine that helps to protect against infection from influenza viruses. These vaccines provide protection from influenza by exposing the immune…

Kategori:
Inactivated Influenza A Virus VaccineInfluenza VaccinesVaccines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

A seasonally-specific component of the influenza vaccine. The influenza vaccine, also known as the "flu shot", is a vaccine that helps to protect against infection from influenza viruses. These vaccines provide protection from influenza by exposing the immune…

Kategori:
Inactivated Influenza A Virus VaccineInfluenza VaccinesVaccines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

A seasonally-specific component of the influenza vaccine. The influenza vaccine, also known as the "flu shot", is a vaccine that helps to protect against infection from influenza viruses. These vaccines provide protection from influenza by exposing the immune…

Kategori:
Influenza VaccinesLive Attenuated Influenza A Virus VaccineVaccines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

A seasonally-specific component of the influenza vaccine. The influenza vaccine, also known as the "flu shot", is a vaccine that helps to protect against infection from influenza viruses. These vaccines provide protection from influenza by exposing the immune…

Kategori:
Inactivated Influenza A Virus VaccineInfluenza VaccinesVaccines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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