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6694

Total database: 17430
Struktur (SMILES)
4518 (67.5%)
Target
3751 (56.0%)
Genomik
81 (1.2%)
Referensi
6694 (100.0%)

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Halaman 22 / 134
Angelica archangelica root Approved DB14283
biotech

Angelica archangelica root is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Angiotensin II Approved DB11842
biotech | CAS: 4474-91-3

Angiotensin II is under investigation for the treatment of Sepsis, Septic Shock, Diabetes Mellitus, and Acute Renal Failure. Angiotensin II has been investigated for the treatment, basic science, and diagnostic of Hypertension, Renin Angiotensin System, and I…

Kategori:
Amino Acids, Peptides, and ProteinsAngiotensin II, antagonists & inhibitorsAngiotensins +16
Target Protein:
Type-2 angiotensin II receptorType-1 angiotensin II receptor
Waktu ParuhThe plasma half-lif…
Vol. DistribusiThe official prescr…
KlirensThe official prescr…
Genetik -
small molecule | CAS: 38390-45-3

Anhydrovinblastine has been used in trials studying the treatment of Unspecified Adult Solid Tumor, Protocol Specific.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anifrolumab Approved DB11976
biotech | CAS: 1326232-46-5

Anifrolumab, or MEDI-546, is a type 1 interferon receptor (IFNAR) inhibiting IgG1? monoclonal antibody indicated in the treatment of adults with moderate to severe systemic lupus erythematosus.[A237074,L34929] The standard therapy for systemic lupus erythemat…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Target Protein:
Interferon alpha/beta receptor 1
Waktu ParuhThe serum eliminati…
Vol. DistribusiBased on population…
KlirensFollowing the admin…
Genetik -
Anileridine Approved DB00913
small molecule | CAS: 144-14-9

Anileridine is a synthetic opioid and strong analgesic medication. It is a narcotic pain reliever used to treat moderate to severe pain. Narcotic analgesics act in the central nervous system (CNS) to relieve pain. Some of their side effects are also caused by…

Kategori:
AnestheticsAnesthetics, GeneralNervous System +2
Target Protein:
Mu-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aniline DB06728
small molecule | CAS: 62-53-3

Aniline, phenylamine or aminobenzene is an organic compound with the formula C6H5NH2. Consisting of an amine attached to a benzene ring, aniline is the prototypical aromatic amine. Being a precursor to many industrial chemicals, its main use is in the manufac…

Kategori:
AminesCarcinogensCytochrome P-450 CYP2E1 Substrates +3
Target Protein:
Kallikrein-1Albumin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anisomycin DB07374
small molecule | CAS: 22862-76-6

Anisomycin (sometimes known as flagecidin), is an antibiotic retrieved from the bacteria _Streptomyces griseolus_. This drug acts to inhibit bacterial protein and DNA synthesis.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntiparasitic Agents +5
Target Protein:
Ribosomal protein uL16-likeLarge ribosomal subunit protein uL13Large ribosomal subunit protein uL14 +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anisotropine methylbromide Approved DB00517
small molecule | CAS: 80-50-2

Anisotropine methylbromide is a quaternary ammonium compound. Its use as treatment adjunct in peptic ulcer has been replaced by the use of more effective agents. Depending on the dose, anisotropine methylbromide may reduce the motility and secretory activity …

Kategori:
Agents producing tachycardiaAlkaloidsAnticholinergic Agents +5
Target Protein:
Muscarinic acetylcholine receptor M5Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2 +1
Waktu ParuhNot Known
Vol. Distribusi-
Klirens-
Genetik -
Anivamersen DB16089
biotech | CAS: 959716-29-1

Anivamersen is under investigation in clinical trial NCT01848106 (A Study to Determine the Efficacy and Safety of REG1 Compared to Bivalirudin in Patients Undergoing PCI).

Kategori:
CoagulantsNucleic Acids, Nucleotides, and NucleosidesNucleotides +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Annamycin DB06420
small molecule | CAS: 92689-49-1

Deskripsi belum tersedia.

Kategori:
AnthracyclinesAntibiotics, AntineoplasticAntineoplastic Agents +4
Target Protein:
DNA topoisomerase 2-alphaDNA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anpocogin DB06552
biotech

Recombinant nematode anticoagulant protein c2 (rNAPc2) is a specific inhibitor of tissue factor (TF)/factor VIIa complex with novel antithrombotic activity. [A175642]

Target Protein:
Coagulation factor VIITissue factorCoagulation factor X
Waktu ParuhOver 50 hours
Vol. Distribusi-
Klirens-
Genetik -
Anthoxanthum odoratum Approved DB14163
biotech

Anthoxanthum odoratum allergenic extract is used in allergenic testing.

Kategori:
Allergenic ExtractsNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anthralin Approved DB11157
small molecule | CAS: 1143-38-0

Anthralin (1,8?dihydroxy?9anthrone, dithranol) is an older anti-psoriatic agent that was first synthesized as a derivative of chrysarobin, obtained from the araroba tree in Brazil over 100 years ago. Adverse effects of anthralin include irritation and discolo…

Kategori:
AnthracenesAntipsoriaticsAntipsoriatics for Topical Use +2
Target Protein:
Keratin, type II cytoskeletal 2 epidermalKeratin, type I cytoskeletal 12C-Jun-amino-terminal kinase-interacting protein 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 118-92-3

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAminobenzoatesBenzene Derivatives +2
Target Protein:
L-amino-acid oxidaseD-amino-acid oxidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Anthrax immune globulin is a human antibody given with antibiotics for the treatment of anthrax. It is derived from the plasma of humans immunized with BioThrax (adsorbed anthrax vaccine), which is then further purified. Available as the product Anthrasil (FD…

Kategori:
Amino Acids, Peptides, and ProteinsBlood ProteinsHuman Immunoglobulin +5
Target Protein:
Protective antigen
Waktu Paruh24.3 days
Vol. Distribusi5714.8 mL
Klirens174.2 mL/day
Genetik -
Anthrax vaccine Approved DB11003
biotech

Anthrax vaccine is a vaccine used for the pre- or post-exposure prophylaxis of disease in those at high risk of, suspected or confirmed exposure to *Bacillus anthracis*. It is subcutaneously or intramuscularly administered. It is derived from cell-free filtra…

Kategori:
Actively Acquired ImmunityAnthrax VaccinesBacterial Vaccines +6
Waktu ParuhLimited information…
Vol. DistribusiLimited information…
KlirensLimited information…
Genetik -
biotech

Anti-SARS-COV-2 REGN-COV2 is a combination of novel antibodies designed by Regeneron for both the prevention and treatment of SARS-COV-2, the virus that causes COVID-19. This drug is a combination of the antibodies REGN10933 and REGN10987, derived from human…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntibodies +10
Target Protein:
Spike glycoprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1628187-15-4

Antihemophilic Factor (Recombinant), PEGylated, was approved by the FDA in December 2016 as the product _Adynovate_ [FDA label]. Antihemophilic Factor (Recombinant), PEGylated, is a recombinant full-length human coagulation factor VIII (2,332 amino acids w…

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsBiological Factors +14
Target Protein:
von Willebrand factor
Waktu Paruh14.69 ± 3.79h for a…
Vol. DistribusiAt steady state: 0.…
Klirens2.27 ± 0.84 for adu…
Genetik -
Antihemophilic factor human Approved DB13192
biotech

Antihemophilic factor human, also known as Coagulation Factor VIII or Anti-Hemophilic Factor (AHF), is a non-recombinant, lyophilized concentrate of coagulation factor VIII, an endogenous protein and essential component of the coagulation cascade. Antihemophi…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood and Blood Forming Organs +11
Target Protein:
Coagulation factor IXCoagulation factor X
Waktu ParuhThe mean half-life …
Vol. DistribusiThe pharmacokinetic…
KlirensThe reported cleara…
Genetik -
biotech

Equine anti-thymocyte globulin is composed of purified gamma globulin containing primarily IgG against human thymus lymphocytes. It is formed by inoculating a horse with an antigen (human thymoyctes) which then induces the horse immune system's B-lymphocytes …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibody-Surface Protein Interactions +22
Waktu ParuhThe half-life of eq…
Vol. DistribusiDuring infusion of …
Klirens-
Genetik -
Antimonous acid DB02453
small molecule

Deskripsi belum tersedia.

Target Protein:
Arsenical pump-driving ATPase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 28300-74-5

Antimony potassium tartrate is a schistosomicide possibly useful against other parasites. It has irritant emetic properties and may cause lethal cardiac toxicity among other adverse effects.

Kategori:
AnthelminticsAnti-Infective AgentsAntiparasitic Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Antithrombin Alfa Approved DB11166
biotech | CAS: 84720-88-7

Antithrombin Alfa is a recombinant antithrombin , an anticoagulant, that is used for the prevention of thromboembolic events in patients that have hereditary deficiency of antithrombin in high risk situations.

Kategori:
AnticoagulantsDecreased Coagulation Factor ActivityFactor Xa Inhibitors +2
Target Protein:
ProthrombinCoagulation factor X
Waktu ParuhDose of: 50IU/kg: …
Vol. DistribusiDose of: 50IU/kg: …
KlirensDose of: 50IU/kg: …
Genetik -
ANX-510 DB05308
small molecule

ANX-510 (CoFactor) is a folate-based biomodulator drug being developed to enhance the activity and reduce associated toxicity of the widely used cancer chemotherapy, 5-fluorouracil (5-FU). CoFactor use with 5-FU is being evaluated in clinical trials in first …

Target Protein:
Thymidylate synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AOC 1001 DB18620
biotech | CAS: 2653183-66-3

Delpacibart (AOC 1001) is being investigated in a global study for the treatment of Myotonic Dystrophy type 1 (DM1) in clinical trial NCT06411288

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AP-001 DB18511
small molecule | CAS: 660430-03-5

Deskripsi belum tersedia.

Kategori:
Dietary FatsDietary Fats, UnsaturatedFats +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apadamtase alfa Approved DB15164
biotech | CAS: 2086325-24-6

Thrombotic thrombocytopenic purpura (TTP) is a rare blood clotting disorder characterized by thrombocytopenia, microangiopathic hemolytic anemia, and various degrees of organ damage.[A262076] It may be inherited (congenital TTP; cTTP) or acquired due to autoa…

Kategori:
ADAM ProteinsADAMTS ProteinsAmino Acids, Peptides, and Proteins +12
Target Protein:
von Willebrand factor
Waktu ParuhFollowing the intra…
Vol. Distribusi-
Klirens-
Genetik -
Apalutamide Approved DB11901
small molecule | CAS: 956104-40-8

Apalutamide is a potent androgen receptor (AR) antagonist that selectively binds to the ligand-binding domain of AR and blocks AR nuclear translocation or binding to androgen response elements [A31846]. It has been used in trials studying the treatment of Pro…

Kategori:
Androgen Receptor InhibitorsAntiandrogensAntineoplastic Agents +28
Target Protein:
Androgen receptorGABA(A) Receptor
Waktu ParuhThe mean effective …
Vol. DistribusiThe mean apparent v…
KlirensThe CL/F of apaluta…
Genetik -
APD-209 DB18759
small molecule | CAS: 1261156-82-4

Deskripsi belum tersedia.

Target Protein:
Beta-2 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
APD668 DB05166
small molecule

APD668 is a novel, highly potent and orally active glucose-dependent insulinotropic receptor (GDIR) agonist intended to more efficiently stimulate insulin release by beta cells in response to elevated blood glucose levels, and to also avoid hypoglycemia.

Target Protein:
Glucose-dependent insulinotropic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
APD791 DB05227
small molecule

APD791 is an oral anti-thrombotic drug candidate being evaluated in a Phase 1 clinical trial by Arena. APD791 is intended to lower the risk of arterial thrombosis by reducing the amplification of platelet aggregation, arterial constriction and intimal hyperpl…

Kategori:
Acids, CarbocyclicAmidesAntidepressive Agents +8
Target Protein:
5-hydroxytryptamine receptor 2A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apitolisib DB12180
small molecule | CAS: 1032754-93-0

Apitolisib has been used in trials studying the treatment of Solid Cancers, Breast Cancer, Prostate Cancer, Renal Cell Carcinoma, and Endometrial Carcinoma, among others.

Kategori:
Phosphatidylinositol 3-Kinases, antagonists & inhibitors
Target Protein:
Serine/threonine-protein kinase mTORPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apomab DB15022
biotech | CAS: 1108170-71-3

Apomab is under investigation in clinical trial NCT00851136 (A Study of PRO95780 Administered in Combination With the FOLFOX Regimen and Bevacizumab in Patients With Previously Untreated, Locally Advanced, Recurrent, and Metastatic Colorectal Cancer (APM4566g…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apomine DB12276
small molecule | CAS: 126411-13-0

Apomine has been used in trials studying the treatment of Osteoporosis and Unspecified Adult Solid Tumor, Protocol Specific.

Kategori:
OrganophosphonatesOrganophosphorus Compounds
Target Protein:
Bile acid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apomorphine Approved DB00714
small molecule | CAS: 58-00-4

Apomorphine is a non-ergoline dopamine D2 agonist indicated to treat hypomobility associated with Parkinson's. It was first synthesized in 1845 and first used in Parkinson's disease in 1884.[A203618] Apomorphine has also been investigated as an emetic, a seda…

Kategori:
AlkaloidsAnti-Parkinson Agents (Dopamine Agonist)Anti-Parkinson Drugs +32
Target Protein:
D(4) dopamine receptorD(2) dopamine receptorD(3) dopamine receptor +11
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe apparent volume…
KlirensThe clearance of a …
Genetik -
small molecule | CAS: 42337-33-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apramycin DB04626
small molecule | CAS: 37321-09-8

Apramycin is an aminoglycoside antibiotic and has a bactericidal action against many gram-negative bacteria. Apramycin is a structurally unique antibiotic that contains a bicyclic sugar moiety and a monosubstituted deoxystreptamine. It is not approved for use…

Kategori:
Agents that produce neuromuscular block (indirect)Aminoglycoside AntibacterialsAnti-Bacterial Agents +4
Target Protein:
16S ribosomal RNA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apremilast Approved DB05676
small molecule | CAS: 608141-41-9

Apremilast, also known as Otezla, is a phosphodiesterase 4 (PDE4) inhibitor used to treat various types of symptoms resulting from certain inflammatory autoimmune diseases. It belongs to the same drug class as [Roflumilast] and [Crisaborole].[A181244,L7495] I…

Kategori:
Agents reducing cytokine levelsAnti-Inflammatory AgentsAntineoplastic and Immunomodulating Agents +17
Target Protein:
Phosphodiesterase isozyme 4Cyclin-dependent kinase 4Cyclin-dependent kinase 6
Waktu ParuhThe average elimina…
Vol. DistribusiThe average apparen…
KlirensIn healthy patients…
Genetik -
Aprepitant Approved DB00673
small molecule | CAS: 170729-80-3

Aprepitant, an antiemetic, is a substance P/neurokinin 1 (NK1) receptor antagonist which, in combination with other antiemetic agents, is indicated for the prevention of acute and delayed nausea and vomiting associated with initial and repeat courses of highl…

Kategori:
Alimentary Tract and MetabolismAntiemeticsAntiemetics and Antinauseants +36
Target Protein:
Substance-P receptor
Waktu Paruh9-13 hours
Vol. Distribusi* 70 L
Klirens* Apparent plasma c…
Genetik -
Apricitabine DB12855
small molecule | CAS: 160707-69-7

Apricitabine has been used in trials studying the treatment of HIV Infections.

Kategori:
DeoxyribonucleosidesNucleic Acids, Nucleotides, and NucleosidesNucleosides +2
Target Protein:
Gag-Pol polyproteinReverse transcriptase/RNaseH
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aprinocarsen DB06451
biotech | CAS: 151879-73-1

Aprinocarsen is a specific antisense oligonucleotide inhibitor of protein kinase C-alpha.

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesOligonucleotides +3
Target Protein:
Protein kinase C alpha type
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aprobarbital DB01352
small molecule | CAS: 77-02-1

Aprobarbital is a barbiturate derivative synthesized in the 1920s by Ernst Preiswerk. It was determined that the substance was capable of demonstrating sedative, hypnotic, and anticonvulsant effects. A primary treatment indicated for the use of aprobarbital w…

Kategori:
Anticholinergic AgentsBarbiturates, PlainCentral Nervous System Depressants +10
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1Gamma-aminobutyric acid receptor subunit alpha-2Gamma-aminobutyric acid receptor subunit alpha-3 +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aprocitentan Approved DB15059
small molecule | CAS: 1103522-45-7

Aprocitentan is a dual antagonist of endothelin receptors A and B used for treatment-resistant hypertension. It is the active metabolite of [macitentan]. Approximately 10-15% of patients with hypertension have resistant hypertension, defined as uncontrolle…

Kategori:
AmidesAntihypertensive AgentsBCRP/ABCG2 Inhibitors +26
Target Protein:
Endothelin-1 receptorEndothelin receptor type B
Waktu ParuhThe effective half-…
Vol. DistribusiThe apparent volume…
KlirensThe apparent cleara…
Genetik -
Aprotinin Approved DB06692
biotech | CAS: 9087-70-1

Aprotinin is a protein-based drug that is also known as bovine pancreatic trypsin inhibitor (BPTI). Since it demonstrates the capacity to slow fibrinolysis, it has been employed to reduce bleeding during complex surgery such as heart and liver surgery. For th…

Kategori:
Amino Acids, Peptides, and ProteinsAntifibrinolytic AgentsBlood and Blood Forming Organs +11
Target Protein:
Serine protease 1Chymotrypsinogen BPlasminogen +1
Waktu ParuhFollowing this dist…
Vol. Distribusi-
Klirens-
Genetik -
APT-101 DB18003
small molecule | CAS: 2100848-01-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aptazapine DB09305
small molecule | CAS: 71576-40-4

Aptazapine (CGS-7525A) was a tetracyclic antidepressant developed in the 1980s. Aptazapine had noradrenergic and specific serotonergic activity. It antagonised ?2 adrenergic receptors approximately 10 times more effectively than mianserin, antagonised 5-HT2 r…

Kategori:
Antidepressive Agents, TetracyclicBenzazepinesHeterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
APX-3330 DB18786
small molecule | CAS: 136164-66-4

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +2
Target Protein:
DNA repair nuclease/redox regulator APEX1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Ribonuclease pancreatic
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 506-32-1

An unsaturated, essential fatty acid. It is found in animal and human fat as well as in the liver, brain, and glandular organs, and is a constituent of animal phosphatides. It is formed by the synthesis from dietary linoleic acid and is a precursor in the bio…

Kategori:
Arachidonic AcidsCytochrome P-450 CYP2C9 SubstratesCytochrome P-450 Substrates +5
Target Protein:
Prostaglandin G/H synthase 1Peroxisome proliferator-activated receptor alphaBile acid receptor +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 1051–1100 dari 6694
Sebelumnya Halaman 22 / 134 Berikutnya