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12560

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9109 (72.5%)
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6912 (55.0%)
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109 (0.9%)
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12560 (100.0%)

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Halaman 219 / 252
Solriamfetol Approved DB14754
small molecule | CAS: 178429-62-4

Solriamfetol marketed under the brand name Sunosi by Jazz Pharmaceuticals in the United States is a dopamine and norepinephrine reuptake inhibitor (DNRI) indicated in treating daytime sleepiness associated with narcolepsy or obstructive sleep apnea[FDA Label]…

Kategori:
Acids, AcyclicAdrenergic AgentsAdrenergic Uptake Inhibitors +22
Target Protein:
Sodium-dependent dopamine transporterSodium-dependent noradrenaline transporter
Waktu Paruh7.1 hours[FDA Label…
Vol. Distribusi199L[FDA Label]. Ot…
KlirensRenal clearance is …
Genetik -
Somapacitan Approved DB15093
biotech | CAS: 1338578-34-9

Somapacitan, also known as NNC0195-0092,[A219136] is a growth hormone analog indicated to treat adults with growth hormone deficiency.[A219126,L15661] This human growth hormone analog differs by the creation of an albumin binding site, and prolonging the effe…

Kategori:
AlcoholsAmino AcidsAmino Acids, Cyclic +25
Target Protein:
Growth hormone receptor
Waktu ParuhThe elimination hal…
Vol. DistribusiThe approximate vol…
KlirensThe apparent maximu…
Genetik -
Somatorelin DB12656
biotech | CAS: 83930-13-6

Somatorelin has been used in trials studying the treatment of Aging, Elderly, Sleep Disorders, Hormone Deficiency, and Mild Cognitive Impairment.

Kategori:
Amino Acids, Peptides, and ProteinsDiagnostic AgentsGrowth Hormone-Releasing Hormone, agonists +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Somatotropin Approved DB00052
biotech | CAS: 12629-01-5

Human growth hormone (HGH), also known as somatotropin, is a peptide hormone that is synthesized and secreted by the somatotropic cells of the anterior pituitary gland.[A228183] Growth hormone plays an essential role in growth regulation during childhood as w…

Kategori:
Agents Causing Muscle ToxicityAmino Acids, Peptides, and ProteinsAnterior Pituitary Lobe Hormones and Analogues +23
Target Protein:
Growth hormone receptorProlactin receptor
Waktu ParuhWhen somatotropin w…
Vol. DistribusiInformation is unav…
KlirensFollowing intraveno…
Genetik -
Somatrogon Approved DB14960
biotech | CAS: 1663481-09-1

Somatrogon is a long-acting recombinant human growth hormone. Growth hormone is a peptide hormone secreted by the pituitary gland that plays a crucial role in promoting longitudinal growth during childhood and adolescence and regulating metabolic function in …

Kategori:
Amino Acids, Peptides, and ProteinsAnterior Pituitary Lobe Hormones and AnaloguesGrowth Hormone +10
Target Protein:
Growth hormone receptor
Waktu ParuhFollowing subcutane…
Vol. DistribusiFollowing subcutane…
KlirensFollowing subcutane…
Genetik -
biotech | CAS: 1088845-67-3

Somatropin pegol is under investigation in clinical trial NCT00715689 (Dose Study in Growth Hormone Deficient Adults Investigating Safety, Pharmacokinetics and Pharmacodynamics of NNC126-0083).

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsEthylene Glycols +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Somavaratan DB12421
biotech | CAS: 1448335-08-7

Somavaratan has been used in trials studying the treatment of Growth Disorders and Adult Growth Hormone Deficiency.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Soneclosan DB04393
small molecule | CAS: 3380-30-1

Deskripsi belum tersedia.

Target Protein:
Enoyl-[acyl-carrier-protein] reductase [NADH]Enoyl-[acyl-carrier-protein] reductase [NADH] FabI
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sonedenoson DB12443
small molecule | CAS: 131865-88-8

Sonedenoson has been used in trials studying the treatment of Foot Ulcer, Diabetic and Diabetes Complications.

Kategori:
Heterocyclic Compounds, Fused-RingNucleic Acids, Nucleotides, and NucleosidesNucleosides +3
Target Protein:
Adenosine receptor A2a
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sonelokimab DB18843
biotech | CAS: 1414386-05-2

Sonelokimab is under investigation in clinical trial NCT06411379 (Study to Evaluate the Efficacy and Safety of Subcutaneous Sonelokimab Compared With Placebo in Adult Participants With Moderate to Severe Hidradenitis Suppurativa).

Kategori:
Amino Acids, Peptides, and ProteinsBlood ProteinsGlobulins +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sonepcizumab DB06305
biotech | CAS: 1031360-18-5

A humanized monoclonal antibody directed against sphingosine 1-phosphate (S1P) with potential antiangiogenic and antineoplastic activities. Upon administration, sonepcizumab binds S1P, which may result in the inhibition of tumor angiogenesis. S1P is the extra…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sonidegib Approved DB09143
small molecule | CAS: 956697-53-3

Sonidegib is a Hedgehog signaling pathway inhibitor (via smoothened antagonism) developed as an anticancer agent by Novartis. It was FDA approved in 2015 for the treatment of basal cell carcinoma.

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBenzene Derivatives +8
Target Protein:
Protein smoothened
Waktu ParuhHalf-life ~ 28 days…
Vol. DistribusiEstimated volume of…
Klirens-
Genetik -
Sonlicromanol DB16333
small molecule | CAS: 1541170-75-5

Sonlicromanol is under investigation in clinical trial NCT04165239 (The KHENERGYZE Study).

Kategori:
AntioxidantsBenzopyransBiological Factors +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sonolisib DB12601
small molecule | CAS: 502632-66-8

Sonolisib has been used in trials studying the treatment of Glioblastoma, Prostate Cancer, Advanced Solid Tumors, Advanced BRAF-mutant Cancers, and Non Small Cell Lung Cancer (NSCLC), among others.

Kategori:
Fused-Ring CompoundsSteroids
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sonrotoclax DB18753
small molecule | CAS: 2383086-06-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Kategori:
Biological ProductsComplex MixturesPharmaceutical Preparations +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Soquelitinib DB18749
small molecule | CAS: 2226636-04-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SOR-C13 DB15366
biotech | CAS: 1187852-48-7

SOR-C13 is under investigation in clinical trial NCT01578564 (Safety and Tolerability Study of SOR-C13 in Subjects With Advanced Cancers Commonly Known to Express the TRPV6 Channel).

Kategori:
Amino Acids, Peptides, and ProteinsAntiarrhythmic agentsAntineoplastic Agents +9
Target Protein:
Transient receptor potential cation channel subfamily V member 6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sorafenib Approved DB00398
small molecule | CAS: 284461-73-0

Sorafenib is a bi-aryl urea and an oral multikinase inhibitor. It targets cell surface tyrosine kinase receptors and downstream intracellular kinases that are implicated in tumour cell proliferation and tumour angiogenesis.[A255852] First approved by the FDA …

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +51
Target Protein:
Serine/threonine-protein kinase B-rafEpidermal growth factor receptorRAF proto-oncogene serine/threonine-protein kinase +8
Waktu ParuhThe mean eliminatio…
Vol. DistribusiSorafenib is widely…
Klirens-
Genetik -
Soraphen A DB02859
small molecule | CAS: 122547-72-2

Deskripsi belum tersedia.

Kategori:
LactonesPolyketides
Target Protein:
Acetyl-CoA carboxylase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Soraprazan DB17856
small molecule | CAS: 261944-46-1

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Potassium-transporting ATPase alpha chain 1Potassium-transporting ATPase subunit beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sorbinil DB02712
small molecule | CAS: 68367-52-2

Deskripsi belum tersedia.

Kategori:
Aldehyde Reductase, antagonists & inhibitorsImidazoles
Target Protein:
Aldo-keto reductase family 1 member B1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sorbitol Approved DB01638
small molecule | CAS: 50-70-4

A polyhydric alcohol with about half the sweetness of sucrose. Sorbitol occurs naturally and is also produced synthetically from glucose. It was formerly used as a diuretic and may still be used as a laxative and in irrigating solutions for some surgical proc…

Kategori:
AlcoholsAlimentary Tract and MetabolismBlood and Blood Forming Organs +22
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Sorghum bicolor subsp. bicolor pollen is the pollen of the Sorghum bicolor subsp. bicolor plant. Sorghum bicolor subsp. bicolor pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sorghum halepense pollen Approved DB10365
biotech

Sorghum halepense pollen is the pollen of the Sorghum halepense plant. Sorghum halepense pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityGrass Pollen Allergen ExtractsIncreased Histamine Release +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SOT-107 DB05337
biotech

SOT-107 is a drug that is a combination of a protein called transferrin and a poison called diphtheria toxin. This drug treat for a type of brain cancer called a high grade glioma brain tumour. About half of all brain tumours are gliomas.

Kategori:
ADP Ribose TransferasesBacterial ToxinsBiological Factors +6
Target Protein:
Glioma pathogenesis-related protein 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sotagliflozin Approved DB12713
small molecule | CAS: 1018899-04-1

Sotagliflozin is a dual inhibitor of SGLT1 and SGLT2, the first of its kind,[A244499] which is approved for use in the EU, in combination with insulin, to improve glycemic control in patients with type 1 diabetes mellitus (T1DM) and a BMI ?27 kg/m<sup>2</sup>…

Kategori:
Alimentary Tract and MetabolismBCRP/ABCG2 InhibitorsBlood Glucose Lowering Agents +24
Target Protein:
Sodium/glucose cotransporter 2Sodium/glucose cotransporter 1
Waktu ParuhThe mean terminal h…
Vol. DistribusiSotagliflozin has a…
KlirensIn healthy voluntee…
Genetik -
Sotalol Approved DB00489
small molecule | CAS: 3930-20-9

Sotalol is a methanesulfonanilide developed in 1960.[A178579] It was the first of the class III anti arrhythmic drugs.[A178579] Sotalol was first approved as an oral tablet on 30 October 1992.[L6334] A racemic mixture of sotalol is currently formulated as a t…

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-Antagonists +23
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptorVoltage-gated inwardly rectifying potassium channel KCNH2
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe apparent volume…
KlirensIn patients with a …
Genetik -
Sotatercept Approved DB12118
biotech | CAS: 1001080-50-7

Sotatercept is an activin signalling inhibitor. It is a homodimeric recombinant fusion protein consisting of the extracellular domain of the human activin receptor type IIA (ActRIIA) linked to the human IgG1 Fc domain.[L50351] On March 26, 2024, sotatercep…

Kategori:
Amino Acids, Peptides, and ProteinsBlood ProteinsImmunoglobulin G +5
Target Protein:
Activin receptor type-2AActivin receptor type-1BGrowth/differentiation factor 8 +1
Waktu ParuhThe effective half-…
Vol. DistribusiThe population PK m…
KlirensClearance is approx…
Genetik -
Sotevtamab DB19120
biotech | CAS: 2411526-47-9

Sotevtamab is under investigation in clinical trial NCT06225843 (Sotevtamab (AB-16B5) Combined With FOLFOX as Neoadjuvant Treatment Prior to Resection of Colorectal Cancer Liver Metastasis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Soticlestat DB16987
small molecule | CAS: 1429505-03-2

Deskripsi belum tersedia.

Kategori:
Cholesterol 24S-Hydroxylase Inhibitor
Target Protein:
Cholesterol 24-hydroxylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sotigalimab DB16413
biotech | CAS: 2305607-45-6

Sotigalimab is under investigation in clinical trial NCT03123783 (CD40 Agonistic Antibody APX005M in Combination With Nivolumab).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sotirimod DB05680
small molecule | CAS: 227318-75-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sotorasib Approved DB15569
small molecule | CAS: 2252403-56-6

Sotorasib, also known as AMG-510, is an acrylamide-derived KRAS inhibitor developed by Amgen.[A187547,A187556] It is indicated in the treatment of adult patients with KRAS G12C mutant non-small cell lung cancer.[L34288] This mutation makes up >50% of all KRAS…

Kategori:
Antineoplastic AgentsAntineoplastic Agents, ImmunologicalAntineoplastic and Immunomodulating Agents +13
Target Protein:
GTPase KRas
Waktu ParuhSotorasib has a ter…
Vol. DistribusiThe volume of distr…
KlirensSotorasib has an ap…
Genetik -
Sotrastaurin DB12369
small molecule | CAS: 425637-18-9

Sotrastaurin has been used in trials studying the basic science and treatment of Uveal Melanoma, Richter Syndrome, Prolymphocytic Leukemia, Recurrent Mantle Cell Lymphoma, and Recurrent Small Lymphocytic Lymphoma, among others.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Protein kinase C theta typeProtein kinase C beta typeProtein kinase C alpha type
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sotrovimab Approved DB16355
biotech | CAS: 2423014-07-5

Sotrovimab (VIR-7831), also known as GSK4182136, is a monoclonal antibody that can neutralize the SARS-CoV-2 virus.[L34440] Sotrovimab was initially been granted emergency use authorization (EUA) to treat mild-to-moderate COVID-19 on May 26, 2021, based on in…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntibodies +13
Target Protein:
Spike glycoprotein
Waktu ParuhThis antibody has u…
Vol. DistribusiSotrovimab is an Fc…
Klirens-
Genetik -
Sovesudil DB18812
small molecule | CAS: 1333400-14-8

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicBenzene Derivatives
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sovleplenib DB17557
small molecule | CAS: 1415792-84-5

Sovleplenib is a novel, investigational, selective small molecule inhibitor for oral administration targeting spleen tyrosine kinase (Syk). It is under investigation in clinical trial NCT03483948 (Phase I Study of Hmpl-523+azacitidine in Elderly Patients With…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Soy sterol DB11325
biotech | CAS: 129311-52-0

Deskripsi belum tersedia.

Kategori:
Biological FactorsCholestanesFused-Ring Compounds +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Soybean Approved DB10568
biotech

Soybean allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Soybean oil Approved DB09422
biotech | CAS: 8001-22-7

Derived from soybeans, soybean oil is a common vegetable oil and a source of polyunsaturated and saturated fatty acids. It is a complex mixture of triglycerides where per 100 g, soybean oil has 16 g of saturated fat, 23 g of monounsaturated fat, and 58 g of p…

Kategori:
Biological ProductsCaloric AgentsComplex Mixtures +12
Target Protein:
Peroxisome proliferator-activated receptor alpha
Waktu Paruh-
Vol. DistribusiAfter triglycerides…
KlirensThe elimination rat…
Genetik -
SP-420 DB16069
small molecule | CAS: 911714-45-9

SP-420 is under investigation in clinical trial NCT03801889 (SP-420 in Subjects With Transfusion-dependent Beta-thalassemia or Other Rare Anemias).

Kategori:
CyclohexanesCycloparaffinsKetones +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sp-722 DB04503
small molecule

Deskripsi belum tersedia.

Target Protein:
Thymidylate synthaseThymidylate synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SP-8203 DB11670
small molecule | CAS: 1176758-04-5

SP-8203 has been used in trials studying the treatment of Ischemic Stroke.

Kategori:
AcetatesAcids, AcyclicAmides +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SP-876 DB03558
small molecule

Deskripsi belum tersedia.

Target Protein:
Thymidylate synthaseThymidylate synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SP2456 DB03957
small molecule

Deskripsi belum tersedia.

Target Protein:
Interleukin-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SP4160 DB02555
small molecule

Deskripsi belum tersedia.

Target Protein:
Interleukin-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Spaglumic acid DB08835
small molecule | CAS: 4910-46-7

Spaglumic acid is the ?-aspartyl isoform of N-Acetyl-l-aspartylglutamate (isospaglumic Acid is N-(N-Acetyl-l-?-aspartyl)-l-glutamic acid). In eye drops, spaglumic acid is either a magnesium or sodium salt of N-Acetyl-l-aspartylglutamate. Spaglumic acid is a m…

Kategori:
Antiallergic Agents, Excl. CorticosteroidsDecongestants and AntiallergicsMast Cell Stabilizers +3
Target Protein:
Glutamate carboxypeptidase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sparfloxacin Approved DB01208
small molecule | CAS: 110871-86-8

Sparfloxacin is a fluoroquinolone antibiotic indicated for bacterial infections. Sparfloxacin exerts its antibacterial activity by inhibiting DNA gyrase, a bacterial topoisomerase. DNA gyrase is an essential enzyme which controls DNA topology and assists in D…

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +16
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA gyrase subunit A +2
Waktu ParuhMean terminal elimi…
Vol. Distribusi-
Klirens-
Genetik -
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