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14063

Total database: 17430
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10481 (74.5%)
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8038 (57.2%)
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107 (0.8%)
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14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 219 / 282
Pivmecillinam Approved DB01605
small molecule | CAS: 32886-97-8

Pivmecillinam is a mecillinam prodrug, a pivaloyloxymethyl ester of amdinocillin that is well absorbed orally, but broken down to amdinocillin in the intestinal mucosa. It is active against gram-negative organisms and used as for amdinocillin. [PubChem]

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
Penicillin-binding protein 1A
Waktu Paruh-
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Pixantrone Approved DB06193
small molecule | CAS: 144510-96-3

Pixantrone is an aza-anthracenedione and DNA intercalator which inhibits topoisomerase II. It is similar in structure to anthracyclines such as mitoxantrone, but exerts fewer toxic effects on cardiac tissue. [2] The lower cardio-toxic effects of pixantrone ma…

Kategori:
Anthracyclines and Related SubstancesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +6
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-beta
Waktu ParuhHalf life ranges fr…
Vol. Distribusi9.7-29.7 L/kg. [2]
KlirensPlasma clearance is…
Genetik -
Pixofisiran DB17294
biotech | CAS: 1152798-48-5

Deskripsi belum tersedia.

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Pizotifen Approved DB06153
small molecule | CAS: 15574-96-6

Pizotifen belongs to the class of antamines and is related to [cyproheptadine].[A32532] It is a potent serotonin and tryptamine antagonist that has been used for migraine prevention for many years. It exhibits weak anticholinergic, antihistamine, and antikini…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +27
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M3 +12
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
Klirens-
Genetik -
PKI-179 DB13109
small molecule | CAS: 1197160-28-3

PKI-179 has been used in trials studying the treatment of Advanced Malignant Solid Tumors.

Kategori:
AmidesOxazines
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PL-3994 DB15355
small molecule | CAS: 952295-80-6

PL-3994 is under investigation in clinical trial NCT01304628 (Cross-Over Study of Subcutaneous Study Drug for the Treatment of Patients With Mild to Moderate Asthma).

Kategori:
Amino Acids, Peptides, and ProteinsBronchodilator AgentsPeptides +1
Target Protein:
Atrial natriuretic peptide receptor 1
Waktu Paruh-
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Placulumab DB11983
biotech | CAS: 945781-29-3

Placulumab has been used in trials studying the treatment of Rheumatoid Arthritis.

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Plamotamab DB18944
biotech | CAS: 2138442-31-4

Plamotamab is under investigation in clinical trial NCT05328102 (Phase 2 Study of Plamotamab Combined With Tafasitamab Plus Lenalidomide Versus Tafasitamab Plus Lenalidomide in Relapsed or Refractory (R/R) Diffuse Large-cell B-cell Lymphoma (DLBCL)).

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biotech

The Covifenz COVID-19 vaccine (plant-based virus-like particles (VLP), recombinant, adjuvanted) is a plant-based vaccine developed in partnership by Medicago and GlaxoSmithKline which is approved in Canada for the prevention of COVID-19.[L40694] It is compose…

Kategori:
COVID-19 VaccinesVaccinesViral Vaccines
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Plantago lanceolata pollen Approved DB10382
biotech

Plantago lanceolata pollen is the pollen of the Plantago lanceolata plant. Plantago lanceolata pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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Plantago seed Approved DB11097
biotech | CAS: 8063-16-9

Platango seeds refer to the seeds collected from various species of plantago trees. It is found in some laxatives for treating occasional constipation and restoring regularity in bowel movements. Its potential benefit in maintaining remission in ulcerative co…

Kategori:
Biological ProductsBulk-Forming LaxativesComplex Mixtures +5
Waktu ParuhThe half-life of ps…
Vol. DistribusiPsyllium husk when …
KlirensPsyllium husk when …
Genetik -
biotech

The plasma protein fraction human (PPFh) is defined as a sterile solution of proteins composed mainly of albumin and globulin derived from human plasma.[A32512] It is already reviewed under the category of biologics by the FDA where the processing, required t…

Kategori:
AlbuminsAmino Acids, Peptides, and ProteinsBlood Derivatives +9
Waktu ParuhThe registered clea…
Vol. DistribusiThe registered volu…
KlirensThe registered clea…
Genetik -
PlasmaCord DB16363
biotech

PlasmaCord is platelet-poor plasma that is derived by fractionation from sterile umbilical cord and placental blood.[L27581] It is developed by Cellpraxis and is currently being investigated against severe acute respiratory syndrome (SARS).

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Plasminogen Approved DB16701
biotech | CAS: 9001-91-6

Plasminogen is a pro-enzyme (i.e. a zymogen) which is cleaved to form plasmin - also known as [fibrinolysin] - as part of the fibrinolytic pathway that breaks down fibrin blood clots.[A236035] This pathway is activated when a clot is no longer needed or to pr…

Kategori:
Amino Acids, Peptides, and ProteinsAnticoagulantsBeta-Globulins +11
Waktu ParuhThe mean half-life …
Vol. DistribusiThe mean steady-sta…
KlirensThe clearance of Ry…
Genetik -
Platanus occidentalis pollen Approved DB10392
biotech

Platanus occidentalis pollen is the pollen of the Platanus occidentalis plant. Platanus occidentalis pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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small molecule | CAS: 74389-68-7

Deskripsi belum tersedia.

Kategori:
Adrenergic AgentsAlcoholsAmines +21
Target Protein:
Platelet-activating factor receptorGanglioside GM2 activator
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Platelet Lysate DB15869
biotech

Platelet lysate is an acellular compound composed of platelet proteins while also being void of cellular debris, thus making the lysate rich with growth factors.[A220188] It is extracted through lysis of the plasma membrane of platelets. Because white cell an…

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biotech

Deskripsi belum tersedia.

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Platensimycin DB08407
small molecule | CAS: 835876-32-9

Deskripsi belum tersedia.

Kategori:
3-Oxoacyl-(Acyl-Carrier-Protein) SynthaseAcids, CarbocyclicAmides +10
Target Protein:
3-oxoacyl-[acyl-carrier-protein] synthase 2
Waktu Paruh-
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Platinum DB12257
small molecule | CAS: 7440-06-4

Platinum is under investigation for the treatment of Metastatic Breast Cancer, Non-small Cell Lung Cancer, Gastric Large Cell Neuroendocrine Carcinoma, Colorectal Large Cell Neuroendocrine Carcinoma, and Pancreatic Large Cell Neuroendocrine Carcinoma, among o…

Kategori:
Antineoplastic AgentsChlorine CompoundsCompounds used in a research, industrial, or household setting +9
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Plazomicin Approved DB12615
small molecule | CAS: 1154757-24-0

Developed by Achaogen biopharmaceuticals, plazomicin is a next-generation aminoglycoside synthetically derived from [DB12604]. The structure of plazomicin was established via appending hydroxylaminobutyric acid to [DB12604] at position 1 and 2-hydroxyethyl gr…

Kategori:
Agents that produce neuromuscular block (indirect)Aminoglycoside AntibacterialsAnti-Bacterial Agents +12
Target Protein:
rRNA methyltransferase 2, mitochondrial30S ribosomal protein S1130S ribosomal protein S14
Waktu ParuhThe mean (±SD) half…
Vol. DistribusiThe mean (±SD) volu…
KlirensFollowing administr…
Genetik -
Plecanatide Approved DB13170
small molecule | CAS: 467426-54-6

Plecanatide is a drug approved in January 2017 by the FDA for the treatment of chronic idiopathic constipation (CIC). It should not be used in children less than six years of age, and should be avoided in patients six years to 18 years of age

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsDrugs for Constipation +12
Target Protein:
Guanylyl cyclase CGuanylate cyclase soluble subunit alpha-2
Waktu Paruhhalf-life (t½) cann…
Vol. DistribusiConcentrations of p…
KlirensNo excretion studie…
Genetik -
Pleospora herbarum Approved DB10825
biotech

Pleospora herbarum is a fungus which can provoke allergic reactions. Pleospora herbarum extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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Plerixafor Approved DB06809
small molecule | CAS: 110078-46-1

Plerixafor is a small-molecule inhibitor of C-X-C chemokine receptor type 4 (CXCR4) that acts as a hematopoietic stem cell mobilizer.[A7117,L45678] It is used to stimulate the release of stem cells from the bone marrow into the blood in patients with non-Hodg…

Kategori:
Adjuvants, ImmunologicAminesAnti-HIV Agents +9
Target Protein:
C-X-C chemokine receptor type 4
Waktu ParuhPlerixafor has a di…
Vol. DistribusiPlerixafor has an a…
KlirensPlerixafor has a to…
Genetik -
PLG-0206 DB18116
biotech | CAS: 847061-43-2

PLG-0206 is a peptide antibiotic under investigation for the treatment of periprosthetic joint infections.[L48106]

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Plicamycin Approved DB06810
small molecule | CAS: 18378-89-7

Plicamycin is an antineoplastic antibiotic produced by Streptomyces plicatus. It has been used in the treatment of testicular cancer, Paget's disease of bone, and, rarely, the management of hypercalcemia. The manufacturer discontinued plicamycin in 2000.

Kategori:
AnthracyclinesAntibiotics, AntineoplasticAntineoplastic Agents +15
Target Protein:
DNA
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Plinabulin DB05992
small molecule | CAS: 714272-27-2

Deskripsi belum tersedia.

Kategori:
DeuteriumPiperazines
Target Protein:
Translation initiation factor eIF2B subunit alphaTranslation initiation factor eIF2B subunit betaTumor necrosis factor
Waktu Paruh-
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Plitidepsin DB04977
small molecule | CAS: 137219-37-5

Aplidine is a peptide found in tunicates which shows promise in shrinking tumors in pancreatic, stomach, bladder, and prostate cancers. The specific marine organism is _Aplidium albicans_. Aplidine is also of interest as a potential treatment for some leukemi…

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +7
Target Protein:
Palmitoyl-protein thioesterase 1Elongation factor 1-alpha 2
Waktu Paruh-
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PLN-74809 DB16515
small molecule

PLN-74809 is a small-molecule that dually inhibits both ?<sub>v</sub>?<sub>6</sub> and ?<sub>v</sub>?<sub>1</sub> to treat both idiopathic pulmonary fibrosis (IPF) and primary sclerosing cholangitis (PSC)[L31693]. The compound was granted orphan drug designat…

Kategori:
Experimental Unapproved Treatments for COVID-19
Target Protein:
Integrin alpha-VIntegrin beta-1Integrin beta-6
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Plozalizumab DB12520
biotech | CAS: 1610761-46-0

Plozalizumab has been investigated for the treatment of Atherosclerosis. Plozalizumab, a novel humanized monoclonal antibody, specifically targets CCR2 chemokine receptors found on the surface of certain white blood cells including macrophages and monocytes. …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Target Protein:
C-C chemokine receptor type 2
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Plozasiran DB18997
biotech | CAS: 2379776-40-4

Plozasiran is under investigation in clinical trial NCT05089084 (Study of ARO-APOC3 (Plozasiran) in Adults With Familial Chylomicronemia Syndrome (FCS)).

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Plumbagin DB17048
small molecule | CAS: 481-42-5

Plumbagin is a compound investigated for its anticancer activity. It has been found that it inactivates the Akt/NF-kB, MMP-9 and VEGF pathways.[A253102]

Kategori:
Adjuvants, ImmunologicAdrenal Cortex HormonesAnthelmintics +17
Target Protein:
Dihydroorotate dehydrogenase (quinone), mitochondrial
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Plutavimab DB18856
biotech | CAS: 2529854-88-2

Plutavimab is under investigation in clinical trial NCT04900428 (Study to Evaluate a Single Intranasal Dose of STI-2099 (COVI-DROPS™) in Outpatient Adults With COVID-19 (UK)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
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PLX-4720 DB06999
small molecule | CAS: 918505-84-7

Deskripsi belum tersedia.

Kategori:
AmidesHeterocyclic Compounds, Fused-RingSulfones +1
Target Protein:
Vascular endothelial growth factor receptor 2Serine/threonine-protein kinase B-raf
Waktu Paruh-
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PLX51107 DB17543
small molecule | CAS: 1627929-55-8

PLX51107 is a potent and selective inhibitor of the bromodomain and extraterminal (BET) protein family.[A257246,A257251] PLX51107 is under investigation in clinical trial NCT04022785 (PLX51107 and Azacitidine in Treating Patients With Acute Myeloid Leukemia o…

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PLX8394 DB16038
small molecule | CAS: 1393466-87-9

PLX8394 is under investigation in clinical trial NCT02428712 (A Study of PLX8394 as a Single Agent in Patients With Advanced Unresectable Solid Tumors).

Kategori:
AmidesHeterocyclic Compounds, Fused-RingSulfones +1
Target Protein:
Serine/threonine-protein kinase B-raf
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PM-060184 DB13137
small molecule | CAS: 960210-99-5

PM060184 has been used in trials studying Solid Tumors.

Kategori:
LactonesPyrans
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pM-81 DB17432
biotech

Deskripsi belum tersedia.

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PM02734 DB05158
small molecule

PM02734 is a marine derived compound. PM02734 as a new antiproliferative drug demonstrating activity against a broad spectrum of tumor types: breast, colon, pancreas, lung and prostate, among others.

Kategori:
Amino Acids, Peptides, and ProteinsPeptidesPeptides, Cyclic
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PMC-403 DB18132
biotech

PMC-403 is a novel Tie2-activating antibody being investigated for the treatment of systemic capillary leak syndrome.

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PMI-001 DB05730
small molecule

PMI-001 is a stand-alone, disease-modifying, anti-rheumatic drug (DMARD) being developed by Phytomedics Inc. It is an extract of the roots of an undisclosed perennial shrub which interferes with the production of IL-2 and COX-2 proteins, for the potential tre…

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PMX-205 DB17938
small molecule | CAS: 514814-49-4

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsPeptidesReceptor, Anaphylatoxin C5a, antagonists & inhibitors
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PN0621 DB05218
biotech

PN0621 is an anti-TNF, domain antibody (dAb) based therapeutic. It targets tumour necrosis factor (TNF) to treat auto-immune inflammatory diseases such as rheumatoid arthritis. It is being developed by Peptech.

Target Protein:
Tumor necrosis factor
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PNT001 DB18375
biotech

PNT001 is a humanized IgG4 S228P monoclonal antibody targeting the cis conformation of the phosphorylated Thr231-Pro232 motif in tau.

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PNU-142721 DB08414
small molecule | CAS: 185220-03-5

Deskripsi belum tersedia.

Target Protein:
Gag-Pol polyprotein
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PNU177836 DB02977
small molecule

Deskripsi belum tersedia.

Target Protein:
Tyrosine-protein phosphatase non-receptor type 1
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Pocapavir DB17736
small molecule | CAS: 146949-21-5

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAntiviral AgentsBenzene Derivatives +2
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Pociredir DB18070
small molecule | CAS: 2490676-18-9

Deskripsi belum tersedia.

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Podofilox Approved DB01179
small molecule | CAS: 518-28-5

A lignan found in podophyllin resin from the roots of podophyllum plants. It is a potent spindle poison, toxic if taken internally, and has been used as a cathartic. It is very irritating to skin and mucous membranes, has keratolytic actions, has been used to…

Kategori:
Antimitotic AgentsAntineoplastic Agents, PhytogenicAntiviral Agents +11
Target Protein:
DNA topoisomerase 2-betaTubulin alpha-4A chainTubulin beta chain +1
Waktu Paruh1.0 to 4.5 hours.
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Polaprezinc DB09221
small molecule | CAS: 107667-60-7

Polaprezinc is a chelated form of zinc and L-carnosine. It is a zinc-related medicine approved for the first time in Japan, which has been clinically used to treat gastric ulcers [L1307, L1308]. It was determined that polaprezinc may be effective in pressure…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Ulcer AgentsDipeptides +10
Target Protein:
Tumor necrosis factorInterleukin-6Interleukin-3 +5
Waktu ParuhThe half-life of po…
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Menampilkan 10901–10950 dari 14063
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