Hasil Filter

14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (14063)

Halaman 218 / 282
Pinus banksiana pollen Approved DB10922
biotech

Pinus banksiana pollen is the pollen of the Pinus banksiana plant. Pinus banksiana pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pinus nigra pollen Approved DB10924
biotech

Pinus nigra pollen is the pollen of the Pinus nigra plant. Pinus nigra pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pinus resinosa pollen Approved DB10923
biotech

Pinus resinosa pollen is the pollen of the Pinus resinosa plant. Pinus resinosa pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pinus thunbergii pollen Approved DB10925
biotech

Pinus thunbergii pollen is the pollen of the Pinus thunbergii plant. Pinus thunbergii pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pioglitazone Approved DB01132
small molecule | CAS: 111025-46-8

Pioglitazone is an antihyperglycemic used as an adjunct to diet, exercise, and other antidiabetic medications to manage type 2 diabetes mellitus.[L11416,L11419,L11422,L11425] It is administered as a racemic mixture, though there is no pharmacologic difference…

Kategori:
Alimentary Tract and MetabolismBlood Glucose Lowering AgentsCytochrome P-450 CYP2C8 Inhibitors +21
Target Protein:
Peroxisome proliferator-activated receptor gammaAmine oxidase [flavin-containing] B
Waktu ParuhThe mean serum half…
Vol. DistribusiThe average apparen…
KlirensThe apparent cleara…
Genetik -
Pipamperone DB09286
small molecule | CAS: 1893-33-0

Pipamperone is a typical antipsychotic of the _butyrophenone_ family used in the treatment of schizophrenia. It was developed by Janssen Pharmaceutica in 1961 and started its first round of clinical trials in 1963 [L1514, L1518]. In an effort to improve [h…

Kategori:
Antidepressive AgentsAntipsychotic AgentsButyrophenone Derivatives +15
Target Protein:
D(2) dopamine receptor5-hydroxytryptamine receptor 2AAlpha-1 adrenergic receptors +5
Waktu Paruh17-26h [L1522]
Vol. Distribusi-
Klirens-
Genetik -
Pipazethate DB08796
small molecule | CAS: 2167-85-3

A non-narcotic oral antitussive agent.

Kategori:
Antitussive AgentsCentral Nervous System AgentsCough and Cold Preparations +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pipemidic acid DB13823
small molecule | CAS: 51940-44-4

Deskripsi belum tersedia.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAnti-Infective Agents, Urinary +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pipendoxifene DB05414
small molecule | CAS: 198480-55-6

ER modulator, ERA-923(Pipendoxifene) is a estrogen receptor modulator being evaluated for the treatment of breast cancer. Pipendoxifene is a new 2-phenyl indole selective estrogen receptor modulators (SERM )that exhibits an excellent preclinical pharmacologic…

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Estrogen receptorEstrogen receptor betaIntegrase, catalytic core
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pipequaline DB13991
small molecule | CAS: 77472-98-1

Pipequaline is an anticonflict & anticonvulsant quinoline derivative. It is an anxiolytic drug that was never marketed. It presents a unique chemical structure that does not follow the structural properties of other drugs of its class. Pipequaline has a simil…

Kategori:
Central Nervous System AgentsHeterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Piperacillin Approved DB00319
small molecule | CAS: 66258-76-2

Semisynthetic, broad-spectrum, ampicillin derived ureidopenicillin antibiotic proposed for pseudomonas infections. It is also used in combination with other antibiotics.

Kategori:
Agents that produce neuromuscular block (indirect)AmidesAnti-Bacterial Agents +15
Target Protein:
Penicillin-binding protein 3Penicillin-binding protein 2BPenicillin-binding protein 2a +1
Waktu Paruh36-72 minutes
Vol. Distribusi* 101 mL/kg [intrav…
Klirens* 32 - 41 mL/min/1.…
Genetik -
Piperaquine Approved DB13941
small molecule | CAS: 4085-31-8

Piperaquine is an antimalarial agent first synthesized in the 1960's and used throughout China [A31550]. Its use declined in the 1980's as piperaquine resistant strains of *Plasmodium falciparum* appeared and artemisinin derivatives became available. It has c…

Kategori:
Anti-Infective AgentsAntimalarialsAntiparasitic Agents +19
Waktu ParuhThe terminal elimin…
Vol. DistribusiPiperaquine is thou…
KlirensThe mean apparent t…
Genetik -
Piperazine Approved DB00592
small molecule | CAS: 110-85-0

Piperazine is an organic compound that consists of a six-membered ring containing two opposing nitrogen atoms. First used as a solvent for uric acid, the use of piperazine as an anthelmintic agent was first introduced in 1953. Upon entry into the systemic cir…

Kategori:
AnthelminticsAnti-Infective AgentsAntinematodal Agents +7
Target Protein:
Gamma-aminobutyric acid receptor subunit beta-3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Piperidione DB13224
small molecule | CAS: 77-03-2

Piperidione was cough medicine marketed by Roche under the trade name Sedulon.

Kategori:
Cough and Cold Preparations
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Piperidolate DB13351
small molecule | CAS: 82-98-4

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAgents producing tachycardiaAlimentary Tract and Metabolism +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Piperine DB12582
small molecule | CAS: 94-62-2

Bioperine has been used in trials studying the treatment of Multiple Myeloma and Deglutition Disorders.

Kategori:
AlkenesAlkynesAmides +11
Target Protein:
Amine oxidase [flavin-containing] AAmine oxidase [flavin-containing] BNuclear receptor subfamily 1 group I member 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pipobroman Approved DB00236
small molecule | CAS: 54-91-1

An antineoplastic agent that acts by alkylation.

Kategori:
Alkylating DrugsAntineoplastic AgentsAntineoplastic Agents, Alkylating +4
Target Protein:
DNA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pipotiazine Approved DB01621
small molecule | CAS: 39860-99-6

Pipotiazine has actions similar to those of other phenothiazines. Among the different phenothiazine derivatives, it appears to be less sedating and to have a weak propensity for causing hypotension or potentiating the effects of CNS depressants and anesthetic…

Kategori:
Antidepressive AgentsAntipsychotic AgentsCentral Nervous System Depressants +26
Target Protein:
D(2) dopamine receptorD(1A) dopamine receptor5-hydroxytryptamine receptor 2A +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pipradrol Approved DB11584
small molecule | CAS: 467-60-7

Pipradrol (Meratran) [L2523] was initially developed in the 1950s as an antidepressant, however, the adverse effects associated with its use and its abuse potential led to its withdrawal and international regulation [L2524]. Pipradrol was made illegal in man…

Kategori:
Central Nervous System StimulantsNervous SystemPsychoanaleptics +1
Target Protein:
D(1) dopamine receptor
Waktu Paruh-
Vol. DistribusiDistributed in the …
KlirensRapidly cleared [T1…
Genetik -
Piprozolin DB13202
small molecule | CAS: 17243-64-0

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismBile and Liver TherapyBile Therapy +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Piracetam Approved DB09210
small molecule | CAS: 7491-74-9

Piracetam is a nootropic drug in the racetams group, with chemical name 2-oxo-1-pyrrolidine acetamide. It shares the same 2-oxo-pyrrolidone base structure with pyroglutamic acid and is a cyclic derivative of the neurotransmitter ?-aminobutyric acid (GABA). Ho…

Kategori:
AcetamidesAcetatesAcids, Acyclic +12
Waktu ParuhThe plasma half lif…
Vol. DistribusiVd is approximately…
KlirensThe apparent total …
Genetik -
Pirarubicin DB11616
small molecule | CAS: 72496-41-4

Deskripsi belum tersedia.

Kategori:
AnthracyclinesAnthracyclines and Related SubstancesAntineoplastic Agents +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pirbuterol Approved DB01291
small molecule | CAS: 38677-81-5

Pirbuterol is a beta-2 adrenergic bronchodilator. In vitro studies and in vivo pharmacologic studies have demonstrated that pirbuterol has a preferential effect on beta-2 Adrenergic receptors compared with isoproterenol. While it is recognized that beta-2 adr…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic beta-2 Receptor Agonists +21
Target Protein:
Beta-2 adrenergic receptorBeta-1 adrenergic receptor
Waktu Paruh2 hours.
Vol. Distribusi-
Klirens-
Genetik -
Pirenoxine DB15945
small molecule | CAS: 1043-21-6

Deskripsi belum tersedia.

Kategori:
Cataract, drug therapy
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pirenzepine Approved DB00670
small molecule | CAS: 28797-61-7

An antimuscarinic agent that inhibits gastric secretion at lower doses than are required to affect gastrointestinal motility, salivary, central nervous system, cardiovascular, ocular, and urinary function. It promotes the healing of duodenal ulcers and due to…

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAnti-Ulcer Agents +10
Target Protein:
Muscarinic acetylcholine receptor M1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pirepemat DB19165
small molecule | CAS: 1227638-29-0

Pirepemat is under investigation in clinical trial NCT05258071 (A Clinical Study Evaluating Efficacy of Pirepemat on Falls Frequency in Patients With Parkinson's Disease (PD)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Piretanide Approved DB02925
small molecule | CAS: 55837-27-9

Piretanide (INN, trade names Arelix, Eurelix, Tauliz) has been synthesized in 1973 at Hoechst AG (Germany) as a loop diuretic compound by using a then-new method for introducing cyclic amine residues in an aromatic nucleus in the presence of other aromaticall…

Kategori:
AmidesCardiovascular AgentsDiuretics +9
Target Protein:
Solute carrier family 12 member 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pirfenidone Approved DB04951
small molecule | CAS: 53179-13-8

Pirfenidone is a synthetic pyridone drug.[A251370] It is an antifibrotic agent with anti-inflammatory and antioxidant properties [A251370] that is used to treat idiopathic pulmonary fibrosis (IPF),[L26801] which is a chronic, progressive form of interstitial …

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAnti-Inflammatory Agents +29
Target Protein:
Transforming growth factor beta-1 proprotein
Waktu ParuhThe mean terminal h…
Vol. DistribusiMean apparent oral …
KlirensFollowing administr…
Genetik -
Piribedil DB12478
small molecule | CAS: 3605-01-4

Piribedil has been investigated in Parkinson's Disease.

Kategori:
Anti-Dyskinesia AgentsAnti-Parkinson Agents (Dopamine Agonist)Anti-Parkinson Drugs +7
Target Protein:
D(3) dopamine receptorAlpha-2C adrenergic receptor5-hydroxytryptamine receptor 1A +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pirisudanol DB13412
small molecule | CAS: 33605-94-6

Deskripsi belum tersedia.

Kategori:
Nervous SystemPsychoanalepticsPsychostimulants, Agents Used for ADHD and Nootropics
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Piritramide Approved DB12492
small molecule | CAS: 302-41-0

Piritramide is under investigation for the treatment of Colon Cancer and Minimal Residual Disease. Piritramide has been investigated for the supportive care of Pain, Postoperative and Postoperative Nausea and Vomiting.

Kategori:
AnalgesicsCentral Nervous System AgentsCentral Nervous System Depressants +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Piritrexim DB03695
small molecule | CAS: 72732-56-0

Piritrexim has been used in trials studying the treatment of Bladder Cancer, Urethral Cancer, and Transitional Cell Cancer of the Renal Pelvis and Ureter.

Kategori:
Antineoplastic AgentsEnzyme InhibitorsFolic Acid Antagonists
Target Protein:
Dihydrofolate reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pirlindole DB09244
small molecule | CAS: 60762-57-4

This drug is classified as a reversible inhibitor of monoamine oxidase A enzyme (also known as a RIMA drug). It was developed and is currently used as an antidepressant in Russia. Its chemical structure is similar to metralindole, and it also shares pharmacol…

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +14
Target Protein:
Amine oxidase [flavin-containing] A5-hydroxytryptamine receptor 1AAlpha-2A adrenergic receptor
Waktu Paruh0.7±0.3 in one stud…
Vol. Distribusi-
KlirensHigh plasma clearan…
Genetik -
Pirmitegravir DB18974
small molecule | CAS: 2245231-10-9

Pirmitegravir is under investigation in clinical trial NCT05869643 (A Clinical Trial of STP0404 in Treatment-naïve Adults With HIV-1 Infection).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pirnabine DB12840
small molecule | CAS: 19825-63-9

Pirnabine has been used in trials studying the treatment of Chronic Idiopathic Constipation.

Kategori:
Amino Acids, Peptides, and ProteinsEnzyme ActivatorsGastrointestinal Agents +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pirodavir DB08012
small molecule | CAS: 124436-59-5

Pirodavir is an antipicornavirus agent.

Kategori:
Antiviral Agents
Target Protein:
Genome polyproteinGenome polyproteinGenome polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Piromelatine DB12288
small molecule | CAS: 946846-83-9

Piromelatine has been used in trials studying the treatment of Alzheimer's Disease.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
5-hydroxytryptamine receptor 1A5-hydroxytryptamine receptor 1DMelatonin receptor type 1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Piromidic acid DB13744
small molecule | CAS: 19562-30-2

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAnti-Infective Agents, UrinaryAntibacterials for Systemic Use +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Piroxicam Approved DB00554
small molecule | CAS: 36322-90-4

A cyclooxygenase inhibiting, non-steroidal anti-inflammatory agent (NSAID) that is well established in treating rheumatoid arthritis and osteoarthritis and used for musculoskeletal disorders, dysmenorrhea, and postoperative pain. Its long half-life enables it…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +33
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu Paruh30 to 86 hours
Vol. Distribusi* 0.14 L/kg
Klirens-
Genetik -
small molecule | CAS: 87234-24-0

Deskripsi belum tersedia.

Kategori:
Anti-Inflammatory AgentsSulfur CompoundsThiazines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pirprofen DB13722
small molecule | CAS: 31793-07-4

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pirtobrutinib Approved DB17472
small molecule | CAS: 2101700-15-4

Pirtobrutinib is a small molecule and a highly selective non-covalent inhibitor of Bruton’s tyrosine kinase (BTK). Its high selectivity has been associated with lower discontinuation rates due to adverse events and a lower incidence of atrial fibrillation.[A2…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Inhibitors +42
Target Protein:
Tyrosine-protein kinase BTK
Waktu ParuhPirtobrutinib has a…
Vol. DistribusiPirtobrutinib has a…
KlirensPirtobrutinib has a…
Genetik -
Pitavastatin Approved DB08860
small molecule | CAS: 147511-69-1

Pitavastatin, also known as the brand name product Livalo, is a lipid-lowering drug belonging to the statin class of medications. By inhibiting the endogenous production of cholesterol within the liver, statins lower abnormal cholesterol and lipid levels and …

Kategori:
Agents Causing Muscle ToxicityAnticholesteremic AgentsBCRP/ABCG2 Substrates +20
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductaseIntegrin alpha-L
Waktu ParuhThe mean plasma eli…
Vol. DistribusiThe mean volume of …
KlirensFollowing a single …
Genetik -
Pitofenone DB15947
small molecule | CAS: 54063-52-4

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismBenzene DerivativesDrugs for Functional Gastrointestinal Disorders +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pitolisant Approved DB11642
small molecule | CAS: 362665-56-3

Pitolisant is a selective antagonist or inverse agonist of the histamine H3 receptor used to treat type 1 or 2 narcolepsy.[L8063] Narcolepsy is a chronic neurological disorder that affects 1 in 2,000 individuals and is characterized by excessive daytime sleep…

Kategori:
Cytochrome P-450 CYP1A2 InducersCytochrome P-450 CYP1A2 Inducers (strength unknown)Cytochrome P-450 CYP2B6 Inducers +25
Target Protein:
Histamine H3 receptorVoltage-gated inwardly rectifying potassium channel KCNH2
Waktu ParuhPitolisant has a pl…
Vol. DistribusiFollowing single an…
KlirensThe apparent oral c…
Genetik -
small molecule | CAS: 566170-04-5

Pittsburgh Compound B is under investigation in clinical trial NCT01723553 (Amyloid-related Imaging Abnormalities (Microbleeds) in Atypical AD).

Kategori:
AminesCarbon RadioisotopesSulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pivagabine DB12951
small molecule | CAS: 69542-93-4

Pivagabine has been used in trials studying the treatment of Stress and Anxiety.

Kategori:
Acids, AcyclicAmino AcidsAmino Acids, Peptides, and Proteins +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pivampicillin Approved DB01604
small molecule | CAS: 33817-20-8

Pivalate ester analog of ampicillin.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
Penicillin-binding protein 1A
Waktu ParuhApproximately 1 hou…
Vol. Distribusi-
Klirens-
Genetik -
Pivhydrazine DB09252
small molecule | CAS: 306-19-4

Pivhydrazine, also known as pivazide, is a member of the hydrazine family with irreversible and non-selective inhibitory activity against monoamine oxidases. In 1960, it was widely used as an antidepressant agent but it is now discontinued.

Kategori:
Acids, AcyclicAgents that produce hypertensionAgents that reduce seizure threshold +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 10851–10900 dari 14063
Sebelumnya Halaman 218 / 282 Berikutnya