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17430

Total database: 17430
Struktur (SMILES)
12313 (70.6%)
Target
9368 (53.7%)
Genomik
112 (0.6%)
Referensi
17430 (100.0%)

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Hasil Pencarian (17430)

Halaman 217 / 349
Mericitabine DB12045
small molecule | CAS: 940908-79-2

Mericitabine has been investigated for the treatment of Hepatitis C, Chronic. Mericitabine is a polymerase inhibitor being developed for the treatment of chronic hepatitis C. Mericitabine is a prodrug of PSI-6130, which demonstrated excellent potency in p…

Kategori:
DeoxyribonucleosidesNucleic Acids, Nucleotides, and NucleosidesNucleosides +2
Target Protein:
Genome polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Merimepodib DB04862
small molecule | CAS: 198821-22-6

Merimepodib (VX-497) is a novel noncompetitive inhibitor of IMPDH. Merimepodib is orally bioavailable and inhibits the proliferation of primary human, mouse, rat, and dog lymphocytes at concentrations of approximately 100 nM.

Kategori:
Acids, AcyclicAmidesBenzene Derivatives +1
Target Protein:
Inosine-5'-monophosphate dehydrogenase 1Receptor tyrosine-protein kinase erbB-2Epidermal growth factor receptor +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Meriones unguiculatus skin Approved DB10603
biotech

Meriones unguiculatus skin or pelt is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Meropenem Approved DB00760
small molecule | CAS: 96036-03-2

Meropenem is a broad-spectrum carbapenem antibiotic. It is active against Gram-positive and Gram-negative bacteria. Meropenem exerts its action by penetrating bacterial cells readily and interfering with the synthesis of vital cell wall components, which lead…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
D-alanyl-D-alanine carboxypeptidase DacB
Waktu ParuhApproximately 1 hou…
Vol. Distribusi-
Klirens-
Genetik -
Merotocin DB12932
biotech | CAS: 1190083-57-8

Merotocin has been used in trials studying the treatment of Preterm Delivery.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mersalyl DB09338
small molecule | CAS: 486-67-9

Mersalyl is the sodium salt form of mersalyl acid, a mercurial diuretic. It is an outdated drug, and its approval has been discontinued by the FDA. Mersalyl acid is currently replaced by less toxic non-mercury containing diuretics [L1575, L1577]. The sodium s…

Kategori:
Alkylmercury CompoundsDiureticsDrugs that are Mainly Renally Excreted +5
Target Protein:
Alkaline phosphatase, tissue-nonspecific isozymeAquaporin-1Monocarboxylate transporter 1
Waktu Paruh-
Vol. Distribusi-
KlirensThe hepatobiliary e…
Genetik -
Mertiatide DB15780
small molecule | CAS: 66516-09-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mesalazine Approved DB00244
small molecule | CAS: 89-57-6

An anti-inflammatory agent, structurally related to the salicylates and non-steroidal anti-inflammatory drugs like acetylsalicylic acid, which is active in inflammatory bowel disease [A174022]. Although demonstrably effective in treating and maintaining remis…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAminosalicylate +13
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1Polyunsaturated fatty acid 5-lipoxygenase +4
Waktu ParuhFor the delayed-rel…
Vol. DistribusiFor the extended-re…
KlirensThe mean (SD) renal…
Genetik -
Mescaline DB19083
small molecule | CAS: 54-04-6

Mescaline is under investigation in clinical trial NCT05933213 (Comparing Mescaline Sodium Enteric-coated Tablets vs Morte-mescaline in the Treatment of Adult Lupus Nephritis).

Kategori:
AlkaloidsAminesAntidepressive Agents +9
Target Protein:
5-hydroxytryptamine receptor 2A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mesdopetam DB16229
small molecule | CAS: 1403894-72-3

Mesdopetam is under investigation in clinical trial NCT04435431 (A Clinical Study of Mesdopetam in Patients With Parkinson's Disease Experiencing Levodopa Induced Dyskinesia).

Kategori:
AminesBenzene DerivativesDopamine Agents +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 147-73-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Flavin reductase (NADPH)
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mesocricetus auratus skin Approved DB10605
biotech

Mesocricetus auratus skin or pelt is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mesoheme DB02577
small molecule

The color-furnishing portion of hemoglobin. It is found free in tissues and as the prosthetic group in many hemeproteins.

Kategori:
Biological FactorsHeterocyclic Compounds, Fused-RingPigments, Biological +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mesoridazine Approved DB00933
small molecule | CAS: 5588-33-0

A phenothiazine antipsychotic with effects similar to chlorpromazine.

Kategori:
Antidepressive AgentsAntipsychotic AgentsAntipsychotic Agents (First Generation [Typical]) +23
Target Protein:
D(2) dopamine receptor5-hydroxytryptamine receptor 2A
Waktu Paruh24 to 48 hours
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 208465-21-8

Mesosulfuron-methyl is under investigation in clinical trial NCT01118117 (A Multi-center Clinical Trial of the Misago™ Self-Expanding Stent System for Superficial Femoral Artery).

Kategori:
AmidesSulfonesSulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mesoxalic acid DB03589
small molecule | CAS: 473-90-5

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicDicarboxylic Acids
Target Protein:
NAD-dependent malic enzyme, mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mesterolone DB13587
small molecule | CAS: 1424-00-6

Mesterolone is a synthetic anabolic-androgenic steroid (AAS) and derivative of dihydrotestosterone (DHT). It is inactivated by 3?-hydroxysteroid dehydrogenase in skeleta muscules so it is considered a weak androgen. It is not a substrate for aromatase so it i…

Kategori:
5-Androstanon (3) DerivativesAnabolic AgentsAndrogens +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mestranol Approved DB01357
small molecule | CAS: 72-33-3

The 3-methyl ether of ethinyl estradiol. It must be demethylated to be biologically active. It is used as the estrogen component of many combination ORAL contraceptives.

Kategori:
Adrenal Cortex HormonesContraceptive Agents, FemaleContraceptive Agents, Hormonal +25
Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mesulfen DB13356
small molecule | CAS: 135-58-0

Deskripsi belum tersedia.

Kategori:
AnionsAnti-Acne PreparationsAnti-Acne Preparations for Topical Use +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metabutethamine DB13578
small molecule | CAS: 4439-25-2

Deskripsi belum tersedia.

Kategori:
AnestheticsAnesthetics, LocalEsters of Aminobenzoic Acid +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metacavir DB19084
small molecule | CAS: 120503-45-9

Metacavir is under investigation in clinical trial NCT02965859 (The Safety and Dose-range Study of Metacavir Enteric-coated Capsules in Patients With Chronic Hepatitis B).

Kategori:
Heterocyclic Compounds, Fused-RingNucleic Acids, Nucleotides, and NucleosidesNucleosides +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metacycline Approved DB00931
small molecule | CAS: 914-00-1

A broad-spectrum semisynthetic antibiotic related to tetracycline but excreted more slowly and maintaining effective blood levels for a more extended period.

Kategori:
Agents that produce neuromuscular block (indirect)Anti-Bacterial AgentsAnti-Infective Agents +4
Target Protein:
16S ribosomal RNA
Waktu Paruh14 hours
Vol. Distribusi-
Klirens-
Genetik -
Metadoxine DB16554
small molecule | CAS: 74536-44-0

Deskripsi belum tersedia.

Kategori:
Alcohol DeterrentsAlimentary Tract and MetabolismAmino Acids +16
Target Protein:
Sodium- and chloride-dependent GABA transporter 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metahexamide DB13675
small molecule | CAS: 565-33-3

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismAmidesBlood Glucose Lowering Agents +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metamfetamine Approved DB01577
small molecule | CAS: 537-46-2

Metamfetamine (methamphetamine) is a psychostimulant and sympathomimetic drug, and a member of the amphetamine group of sympathomimetic amines. Methamphetamine can induce effects such as euphoria, increased alertness and energy, and enhanced self-esteem. It i…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-2 Receptor Agonists +33
Target Protein:
D(2) dopamine receptorAlpha-1B adrenergic receptorSodium-dependent dopamine transporter +10
Gen Terkait:
PICK1
Waktu ParuhThe biological half…
Vol. Distribusi-
Klirens-
Genetik 1 Varian
Metamizole Approved DB04817
small molecule | CAS: 50567-35-6

Metamizole (dipyrone) is a pyrazolone derivative that belongs to the group of nonacid nonopioids. It is considered a potent analgesic and antipyretic with favourable gastrointestinal tolerability.[A251885] Metamizole was formerly marketed in the US as Dimetho…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAminopyrine +16
Target Protein:
Prostaglandin G/H synthase 1
Waktu Paruh_In vitro_, the hal…
Vol. DistribusiMetamizole is quick…
KlirensThe clearance of 4-…
Genetik -
Metampicillin DB13836
small molecule | CAS: 6489-97-0

Metampicillin is a penicillin antibiotic prepared by the reaction of ampicillin with formaldehyde. It is hydrolysed in aqueous solution to form ampicillin. Hydrolysis is rapid under acid conditions like the stomach.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metandienone DB13586
small molecule | CAS: 72-63-9

Metandienone is an orally active anabolic androgenic steroid. It was introduced to the market in the 1960s but later discontinued and withdrawn from the market. Although it is prohibited in and outside competition by the World Anti-Doping Agency, metandienone…

Kategori:
Alimentary Tract and MetabolismAnabolic AgentsAnabolic Agents for Systemic Use +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Heat-labile enterotoxin B chainCholera enterotoxin subunit B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metaraminol Approved DB00610
small molecule | CAS: 54-49-9

An adrenergic agonist that acts predominantly at alpha adrenergic receptors and also stimulates the release of norepinephrine. It has been used primarily as a vasoconstrictor in the treatment of hypotension.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-1 Receptor Agonists +17
Target Protein:
D(2) dopamine receptorAlpha-1A adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metavert DB17306
small molecule | CAS: 1841125-91-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metaxalone Approved DB00660
small molecule | CAS: 1665-48-1

Metaxalone is a moderate to strong muscle relaxant used in the symptomatic treatment of musculoskeletal pain caused by strains, sprains, and other musculoskeletal conditions. It is marketed by King Pharmaceuticals under the brand name Skelaxin®. Its main mech…

Kategori:
Central Nervous System DepressantsCentrally-mediated Muscle RelaxationDrugs that are Mainly Renally Excreted +5
Waktu Paruh9.2 (+/- 4.8) hours
Vol. Distribusi* 800 L
Klirens* 68 +/- 50 L/h [Su…
Genetik -
Metelimumab DB18695
biotech | CAS: 272780-74-2

Metelimumab (CAT-192) is a monoclonal antibody targeted against transforming growth factor (TGF) beta-1.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metenkefalin DB12668
small molecule | CAS: 58569-55-4

Metenkefalin is an endogenous opioid and beta-endorphin.[A203225] It has been shown to reduce chromosomal abberations in patients with multiple sclerosis.[A203210] Metenkefalin, along with [tridecactide], are under investigation as an immunomodulatory therap…

Kategori:
Amino Acids, Peptides, and ProteinsEnkephalin, MethionineEnkephalins +9
Target Protein:
Delta-type opioid receptorMu-type opioid receptor
Waktu ParuhThe half life of me…
Vol. Distribusi-
Klirens-
Genetik -
Metenolone DB13710
small molecule | CAS: 153-00-4

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismAnabolic AgentsAnabolic Agents for Systemic Use +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metergoline Approved DB13520
small molecule | CAS: 17692-51-2

Metergoline is an ergot-derived psychoactive drug that acts as a ligand for serotonin and dopamine receptors. Metergoline is an antagonist at various 5-HT receptor subtypes at a relatively low concentration and agonist at dopamine receptors.[A27181] Its use h…

Kategori:
Agents that produce hypertensionAlkaloidsAntidepressive Agents +18
Target Protein:
5-hydroxytryptamine receptor 2C5-hydroxytryptamine receptor 1B5-hydroxytryptamine receptor 1E +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metformin Approved DB00331
small molecule | CAS: 657-24-9

Metformin is a biguanide antihyperglycemic agent and first-line pharmacotherapy used in the management of type II diabetes.[L12207,A176173] Metformin is considered an antihyperglycemic drug because it lowers blood glucose concentrations in type II diabete…

Kategori:
Alimentary Tract and MetabolismAmidinesBiguanides +11
Target Protein:
Multidrug and toxin extrusion protein 1Acetyl-CoA carboxylase 2Electron transfer flavoprotein-ubiquinone oxidoreductase, mitochondrial +2
Waktu ParuhThe plasma eliminat…
Vol. DistribusiThe apparent volume…
KlirensRenal clearance is …
Genetik -
Metformin C-11 DB15181
small molecule

Metformin c-11 is under investigation in clinical trial NCT03122769 (Cardiac Uptake of Metformin, Visualized by Positron Emission Tomography).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 72156-70-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Methacholine Approved DB06709
small molecule | CAS: 55-92-5

Asthma is a complex condition associated with phenomena such as airway hyperresponsiveness (AHR), in which the smooth muscle in the airways (ASM) excessively contracts in response to stimuli, reducing pulmonary function and causing symptoms such as difficulty…

Kategori:
AminesAmmonium CompoundsAutonomic Agents +17
Target Protein:
Muscarinic acetylcholine receptor M3Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M1 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 6008-91-9

Deskripsi belum tersedia.

Kategori:
Adenine NucleotidesCoenzymesEnzymes and Coenzymes +6
Target Protein:
Isobutyryl-CoA dehydrogenase, mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methadone Approved DB00333
small molecule | CAS: 76-99-3

Methadone is a potent synthetic analgesic that works as a full µ-opioid receptor (MOR) agonist and N-methyl-d-aspartate (NMDA) receptor antagonist. As a full MOR agonist, methadone mimics the natural effects of the body's opioids, endorphins, and enkephalins …

Kategori:
AnalgesicsAnticholinergic AgentsAntidepressive Agents +50
Target Protein:
Mu-type opioid receptorNMDA receptorDelta-type opioid receptor +5
Waktu ParuhDue to interindivid…
Vol. DistribusiDue to interindivid…
KlirensDue to interindivid…
Genetik -
small molecule | CAS: 509-74-0

A narcotic analgesic with a long onset and duration of action. It is used mainly in the treatment of narcotic dependence.

Kategori:
AnalgesicsCentral Nervous System AgentsCentral Nervous System Depressants +6
Target Protein:
Mu-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methallenestril DB13143
small molecule | CAS: 517-18-0

Deskripsi belum tersedia.

Kategori:
EstrogensGenito Urinary System and Sex HormonesSex Hormones and Modulators of the Genital System +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methamidophos DB14972
small molecule | CAS: 10265-92-6

Methamidophos is under investigation in clinical trial NCT03223753 (Web-Based Physical Activity Intervention in Improving Long Term Health in Children and Adolescents With Newly Diagnosed Acute Lymphoblastic Leukemia in First Remission).

Kategori:
AgrochemicalsCompounds used in a research, industrial, or household settingInsecticides +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methane DB15994
small molecule | CAS: 74-82-8

Deskripsi belum tersedia.

Kategori:
AlkanesHydrocarbons, Acyclic
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 558-25-8

Methanesulfonyl Fluoride has been used in trials studying the treatment of Safety.

Kategori:
Cholinergic AgentsCholinesterase InhibitorsEnzyme Inhibitors +2
Target Protein:
Acetylcholinesterase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methantheline Approved DB00940
small molecule | CAS: 5818-17-7

Methantheline is a synthetic antispasmodic. Antispasmodics are used to relieve cramps or spasms of the stomach, intestines, and bladder. Methantheline is used to treat intestine or stomach ulcers (peptic ulcer disease), intestine problems (irritable bowel syn…

Kategori:
Acid ReducersAgents producing tachycardiaAlimentary Tract and Metabolism +12
Target Protein:
Histamine H2 receptorMuscarinic acetylcholine receptor M5Muscarinic acetylcholine receptor M2 +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methapyrilene DB04819
small molecule | CAS: 91-80-5

Methapyrilene, formerly marketed in many drug products, was shown to be a potent carcinogen. Manufacturers voluntarily withdrew methapyriline drug products from the market in May and June 1979.

Kategori:
AminesAminopyridinesAnti-Allergic Agents +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 10801–10850 dari 17430
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