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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 217 / 236
Thymectacin DB05116
small molecule | CAS: 232925-18-7

Thymectacin, a phosphoramidate derivative of (E)-5-(2-bromovinyl)-2'-deoxyuridine, is a novel small molecule anticancer agent. Thymectacin is selectively active against tumor cells expressing high levels of thymidylate synthase (TS), a critical enzyme in DNA …

Kategori:
DeoxyribonucleosidesDeoxyuridineNucleic Acids, Nucleotides, and Nucleosides +4
Target Protein:
Thymidylate synthaseThymidylate synthase
Waktu Paruh-
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small molecule | CAS: 365-07-1

5-Thymidylic acid. A thymine nucleotide containing one phosphate group esterified to the deoxyribose moiety.

Kategori:
DeoxyribonucleotidesNucleic Acids, Nucleotides, and NucleosidesNucleotides +3
Target Protein:
Thymidylate synthaseThymidine kinase, cytosolicThymidylate kinase +7
Waktu Paruh-
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Thymine DB03462
small molecule | CAS: 65-71-4

Deskripsi belum tersedia.

Kategori:
PyrimidinesPyrimidinones
Target Protein:
Thymidine phosphorylaseDeoxyribodipyrimidine photo-lyaseThymidine phosphorylase
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Thymoquinone DB16447
small molecule | CAS: 490-91-5

Thymoquinone is a natural compound with widespread protective effects, including anti-oxidative, anti-inflammatory, immunomodulatory, anti-cancer, and anti-microbial.

Kategori:
Experimental Unapproved Treatments for COVID-19Quinones
Target Protein:
Cellular tumor antigen p53Apoptosis regulator Bcl-2Apoptosis regulator BAX
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Thymosin beta-4 DB12003
biotech | CAS: 77642-24-1

Thymosin Beta 4 has been investigated for the treatment of STEMI, Dry Eye, Diabetes, Pressure Ulcers, and Dry Eye Syndrome, among others.

Kategori:
Amino Acids, Peptides, and ProteinsHormonesHormones, Hormone Substitutes, and Hormone Antagonists +5
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Thyroid, porcine Approved DB09100
biotech

Thyroid extract is dried and powdered thyroid glands from pigs containing tiiodothyronine (T3) and thyroxine (T4) used to supplement low or absent thyroid activity.[A190831,L11755] Thyroid extract has been described in literature to treat hypothyroidism since…

Kategori:
Agents used to treat hypothyroidismThyroid Products
Target Protein:
Thyroid hormone receptor alphaThyroid hormone receptor beta
Waktu ParuhData regarding the …
Vol. DistribusiData regarding the …
KlirensData regarding the …
Genetik -
Thyrotropin DB15263
biotech | CAS: 9002-71-5

Thyrotropin is under investigation in clinical trial NCT01348191 (Detection of Thyrotrophin Receptor in Human Myometrium).

Kategori:
Amino Acids, Peptides, and ProteinsDiagnostic AgentsHormones +7
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Tiamulin DB11468
small molecule | CAS: 55297-95-5

Tiamulin is a pleuromutilin antibiotic drug that is used in veterinary medicine particularly for pigs and poultry.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsTerpenes
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Tianeptine DB09289
small molecule | CAS: 72797-41-2

Tianeptine is a drug used primarily in the treatment of major depressive disorder and has been studied in the treatment of irritable bowel syndrome (IBS) [A31983]. Structurally, it is classified as a tricyclic antidepressant (TCA), however, it possesses diffe…

Kategori:
Agents Causing Muscle ToxicityAgents that produce hypertensionAgents that reduce seizure threshold +20
Target Protein:
Mu-type opioid receptorSodium-dependent serotonin transporterGlutamate receptor 1 +2
Waktu ParuhApproximately 2.5 h…
Vol. Distribusi0.8 L/kg (0.77 +/- …
KlirensRapidly cleared by …
Genetik -
Tiaprofenic acid Approved DB01600
small molecule | CAS: 33005-95-7

Tiaprofenic acid is a non-steroidal anti-inflammatory drug employed in the treatment of pain, particularly arthritis pain. It belongs to the _arylpropionic acid_ (profen) group of nonsteroidal anti-inflammatory drugs (NSAIDs).

Kategori:
Acids, AcyclicAgents causing hyperkalemiaAgents that produce hypertension +20
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2
Waktu Paruh1.5-2.5 hours
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Tiazofurine DB13243
small molecule | CAS: 60084-10-8

Tiazofurine has potential clinical use in cancer treatment as it is a potential inhibitor of Inosine- 5’-monophosphate (IMP) dehydrogenase [A174991].

Kategori:
AntimetabolitesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +5
Target Protein:
Inosine-5'-monophosphate dehydrogenase 1
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small molecule | CAS: 54663-47-7

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismAntiinfectives and Antiseptics for Local Oral TreatmentStomatological Preparations
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Tibolone Approved DB09070
small molecule | CAS: 5630-53-5

Tibolone is a synthetic steroid hormone drug, which is mainly non-selective in its binding profile, acting as an agonist primarily at estrogen receptors (ER), with a preference for ER alpha [L1874]. Tibolone (Livial, Org OD 14), produced by Organon (West O…

Kategori:
Anabolic AgentsAntineoplastic Agents, HormonalCardiovascular Agents +12
Target Protein:
Estrogen receptor
Waktu ParuhThe elimination hal…
Vol. Distribusi-
KlirensElimination of tibo…
Genetik -
Tibulizumab DB14848
biotech | CAS: 1849636-24-3

Tibulizumab is under investigation in clinical trial NCT03736772 (A Study of LY3090106 in Japanese and Caucasian Healthy Participants).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
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Ticagrelor Approved DB08816
small molecule | CAS: 274693-27-5

Ticagrelor, or AZD6140, was first described in the literature in 2003.[A204170,A2903] Ticagrelor is an ADP derivative developed for its P2Y<sub>12</sub> receptor antagonism.[A2903] Unlike [clopidogrel], ticagrelor is not a prodrug.[A2903] It is marketed by As…

Kategori:
AnticoagulantsAntiplatelet agentsBlood and Blood Forming Organs +37
Target Protein:
P2Y purinoceptor 12
Waktu ParuhTicagrelor has a pl…
Vol. DistribusiThe steady state vo…
KlirensThe renal clearance…
Genetik -
Ticarcillin Approved DB01607
small molecule | CAS: 34787-01-4

An antibiotic derived from penicillin similar to carbenicillin in action.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +9
Target Protein:
Penicillin binding protein 2a
Waktu Paruh1.1 hours
Vol. Distribusi-
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biotech

Tick-borne encephalitis (TBE) is a disease caused by the TBE virus (TBEV), transmitted by ticks from the genus _Ixodes_. The disease course is variable. Some patients will be asymptomatic or experience a mild febrile illness, while others will experience the …

Kategori:
VaccinesViral Vaccines
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Ticlatone DB13613
small molecule | CAS: 70-10-0

Deskripsi belum tersedia.

Kategori:
Antifungals for Dermatological UseAntifungals for Topical UseDermatologicals +1
Waktu Paruh-
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small molecule | CAS: 30986-62-0

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismBile and Liver TherapyLiver Therapy +1
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Tidutamab DB18839
biotech | CAS: 2148354-90-7

Tidutamab is under investigation in clinical trial NCT04590781 (Safety and Efficacy of Xmab18087 ± Pembrolizumab in Advanced Merkel Cell Carcinoma or Extensive-stage Small Cell Lung Cancer).

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small molecule | CAS: 144-12-7

Deskripsi belum tersedia.

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAnticholinergic Agents +4
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Tifacogin DB06437
small molecule | CAS: 148883-56-1

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and Proteins
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Tigatuzumab DB15101
biotech | CAS: 918127-53-4

Tigatuzumab is under investigation in clinical trial NCT00991796 (CS-1008 With Carboplatin/Paclitaxel in Chemotherapy naïve Subjects With Metastatic or Unresectable Non-small Cell Lung Cancer (NSCLC)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
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Tigecycline Approved DB00560
small molecule | CAS: 220620-09-7

Tigecycline is a glycylcycline antibiotic developed and marketed by Wyeth under the brand name Tygacil. It was developed in response to the growing prevalence of antibiotic resistance in bacteria such as Staphylococcus aureus. It was granted fast-track approv…

Kategori:
Agents that produce neuromuscular block (indirect)Anti-Bacterial AgentsAnti-Infective Agents +7
Target Protein:
16S ribosomal RNA30S ribosomal protein S930S ribosomal protein S12 +3
Waktu Paruh27-43 hours
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small molecule | CAS: 943001-56-7

Deskripsi belum tersedia.

Kategori:
Terpenes
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Tigozertinib DB19239
small molecule | CAS: 2660250-10-0

Tigozertinib (BLU-945) is currently under investigation in clinical trial NCT04862780 (Phase 1/?2 Study Targeting EGFR Resistance Mechanisms in NSCLC) for the treatment of NSCLC.

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Tigulixostat DB18799
small molecule | CAS: 1287766-55-5

Deskripsi belum tersedia.

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TIK-301 DB16909
small molecule | CAS: 118702-11-7

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingHormonesHormones, Hormone Substitutes, and Hormone Antagonists +2
Target Protein:
Melatonin receptor type 1A
Waktu Paruh-
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Tilactase Approved DB13761
biotech | CAS: 9031-11-2

Tilactase is a beta-D-galactosidase obtained from _Aspergillus oryzae_. It is produced as a chewable tablet that has to be taken before the consumption of a lactose-containing meal.[A27172] The beta-D-galactosidase us a large monomeric multi-domain enzyme of …

Kategori:
Alimentary Tract and MetabolismAntifoaming Agentsbeta-Galactosidase +8
Target Protein:
Lactose
Waktu ParuhTilactase half-life…
Vol. DistribusiTilactase is not ab…
KlirensTilactase is not ab…
Genetik -
Tilarginine Approved DB11815
small molecule | CAS: 17035-90-4

Tilarginine has been investigated for the basic science, treatment, and diagnostic of Obesity, Type 2 Diabetes, Ocular Physiology, and Regional Blood Flow.

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +4
Target Protein:
Nitric oxide synthase 3
Waktu Paruh-
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Tilavonemab DB17014
biotech | CAS: 2096513-89-0

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
Waktu Paruh-
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Tilbroquinol Approved DB13222
small molecule | CAS: 7175-09-9

Tilbroquinol was approved in France, Morocco, and Saudi Arabia but it has been withdrawn in France and Saudi Arabia markets mainly due to its hepatotoxicity risk outweighing the drug benefit [L5467]. In Morocco, the drug has been limited to use in the treatme…

Kategori:
Antiparasitic Products, Insecticides and RepellentsAntiprotozoalsHeterocyclic Compounds, Fused-Ring +3
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Tildacerfont DB18545
small molecule | CAS: 1014983-00-6

Tildacerfont is a corticotropin-releasing factor receptor-1 antagonist containing an unfused thiazole ring

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Tildipirosin DB11470
small molecule | CAS: 328898-40-4

Tildipirosin is a veterinary antibiotic.

Kategori:
Anti-Bacterial AgentsCytochrome P-450 CYP3A InhibitorsCytochrome P-450 CYP3A4 Inhibitors +4
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Tildrakizumab Approved DB14004
biotech | CAS: 1326244-10-3

Tildrakizumab is a high-affinity, humanized, IgG1 ? antibody targeting interleukin 23 p19 that shows promise in the evolution of treatment strategy in chronic plaque psoriasis [A32255]. The Food and Drug Administration (FDA) approved ILUMYA (tildrakizumab-…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +11
Target Protein:
Interleukin-23
Waktu ParuhThe half-life is ap…
Vol. DistribusiThe geometric mean …
KlirensThe mean (CV%) syst…
Genetik -
Tiletamine DB11549
small molecule | CAS: 14176-49-9

This drug is a dissociative anesthetic agent that falls under the drug category of _NMDA receptor antagonists_. Tiletamine is chemically similar to another dissociative anesthetic, ketamine. Tiletamine hydrochloride, the salt form, exists as odorless white cr…

Kategori:
AnestheticsAnesthetics, DissociativeAnesthetics, General +10
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Tilia americana pollen Approved DB10732
biotech

Tilia americana pollen is the pollen of the Tilia americana plant. Tilia americana pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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Tilidine DB13787
small molecule | CAS: 51931-66-9

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAnalgesicsCentral Nervous System Agents +8
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Tilletia caries Approved DB10705
biotech

Tilletia caries allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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Tilmanocept Approved DB15373
small molecule | CAS: 1185986-76-8

Tilmanocept is under investigation in clinical trial NCT03241446 (Pharmacokinetics and Dosimetry of Tc 99m Tilmanocept Following a Single Intravenous Dose Administration in Male and Female Subjects Diagnosed With Rheumatoid Arthritis (RA)).

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Tilmicosin DB11471
small molecule | CAS: 108050-54-0

Tilmicosin is a macrolide antibiotic. It is used in veterinary medicine for the treatment of bovine respiratory disease and ovine respiratory disease associated with _Mannheimia haemolytica_.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsLactones +1
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Tilorone DB17965
small molecule | CAS: 27591-97-5

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAnti-Inflammatory AgentsAntiinfectives for Systemic Use +7
Waktu Paruh-
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Tilpisertib DB18798
small molecule | CAS: 2065153-41-3

Deskripsi belum tersedia.

Waktu Paruh-
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small molecule | CAS: 2567459-64-5

Deskripsi belum tersedia.

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Tilsotolimod DB16341
biotech | CAS: 1948266-37-2

Tilsotolimod is under investigation in clinical trial NCT03865082 (Study of Tilsotolimod in Combination With Nivolumab and Ipilimumab for the Treatment of Solid Tumors (ILLUMINATE-206)).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Target Protein:
Toll-like receptor 9
Waktu Paruh-
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TILT-123 DB17519
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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Tiludronic acid Approved DB01133
small molecule | CAS: 89987-06-4

Tiludronate, or (4-chlorophenyl)thio-methylene-1,1-bisphosphonate, is a first generation bisphosphonate similar to [etidronic acid] and [clodronic acid].[A1923,A203111] These drugs were developed to mimic the action of pyrophosphate, a regulator of calcificat…

Kategori:
BisphosphonatesBone Density Conservation AgentsDrugs Affecting Bone Structure and Mineralization +6
Target Protein:
HydroxylapatiteAdenosine triphosphate (ATP)Tyrosine-protein phosphatase non-receptor type 12 +3
Waktu ParuhThe mean plasma eli…
Vol. DistribusiThe volume of distr…
KlirensTiludronic acid has…
Genetik -
Timbetasin DB19119
biotech | CAS: 77591-33-4

Timbetasin is under investigation in clinical trial NCT05555589 (Assessment of the Safety and Efficacy of 0.1% RGN-259 Ophthalmic Solution for the Treatment of NK: SEER-2).

Kategori:
Amino Acids, Peptides, and ProteinsHormonesHormones, Hormone Substitutes, and Hormone Antagonists +5
Waktu Paruh-
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Timcodar DB12761
small molecule | CAS: 179033-51-3

Timcodar has been used in trials studying the treatment of Unspecified Adult Solid Tumor, Protocol Specific.

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Timdarpacept DB17544
biotech | CAS: 2749520-17-8

IMM01 is a recombinant human signal regulatory protein ? (SIRP?) IgG 1 fusion protein.[A257261] IMM01 is under investigation in clinical trial NCT05140811 (A Study of IMM01 Combined With Azacitidine in Patients With Acute Myeloid Leukemia and Myelodysplastic …

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