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12560

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Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
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109 (0.9%)
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12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 217 / 252
Sirolimus Approved DB00877
small molecule | CAS: 53123-88-9

Sirolimus, also known as rapamycin, is a macrocyclic lactone antibiotic produced by bacteria _Streptomyces hygroscopicus_, which was isolated from the soil of the Vai Atari region of Rapa Nui (Easter Island).[A242412] It was first isolated and identified as a…

Kategori:
Agents causing angioedemaAnti-Bacterial AgentsAnti-Infective Agents +35
Target Protein:
Serine/threonine-protein kinase mTOR
Waktu ParuhThe mean ± SD termi…
Vol. DistribusiThe mean (± SD) blo…
KlirensIn adult renal tran…
Genetik -
Sirpiglenastat DB17536
small molecule | CAS: 2079939-05-0

Sirpiglenastat, also known as DRP-104, is a prodrug of [6-diazo-5-oxo-L-norleucine] (DON), which is a broad-acting glutamine antagonist. It is under investigation in clinical trial NCT04471415 (Study to Investigate DRP-104 in Adults With Advanced Solid Tumors…

Kategori:
AcetatesAcids, AcyclicAmides +1
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Sirukumab DB11803
biotech | CAS: 1194585-53-9

Sirukumab has been used in trials studying the treatment and basic science of Giant Cell Arteritis and Arthritis, Rheumatoid.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
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SIS-101-ADO DB18085
biotech

SIS-101-ADO is a siRNA therapeutic under investigation for the treatment of Autosomal Dominant Osteopetrosis Type 2 (ADO2).[L48091]

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Sisomicin DB12604
small molecule | CAS: 32385-11-8

Sisomicin has been used in trials studying the treatment of Pyoderma.

Kategori:
Agents that produce neuromuscular block (indirect)Aminoglycoside AntibacterialsAnti-Bacterial Agents +12
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Sisunatovir DB15674
small molecule | CAS: 1903763-82-5

Sisunatovir is under investigation in clinical trial NCT04267822 (Study of RV521 in the Treatment of Adult Subjects Who Have Undergone HCT With an URTI With RSV).

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Fusion glycoprotein F0
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Sitafloxacin DB13261
small molecule | CAS: 163253-35-8

Deskripsi belum tersedia.

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +14
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Sitagliptin Approved DB01261
small molecule | CAS: 486460-32-6

Sitagliptin is an oral dipeptidyl peptidase-4 (DPP-4) inhibitor used in conjunction with diet and exercise to improve glycemic control in patients with type 2 diabetes mellitus[FDA label,A2260,A2255,A2256]. The effect of this medication leads to glucose depen…

Kategori:
Agents causing angioedemaAlimentary Tract and MetabolismBlood Glucose Lowering Agents +17
Target Protein:
Dipeptidyl peptidase 4
Waktu ParuhApproximately 12.4 …
Vol. Distribusi198L[FDA label,A226…
Klirens350mL/min[FDA label…
Genetik -
Sitamaquine DB04909
small molecule | CAS: 57695-04-2

Sitamaquine (WR-6026) is an orally active 8-aminoquinoline analog in development by the Walter Reed Army Institute, in collaboration with GlaxoSmithKline (formerly SmithKline Beecham), for the potential treatment of visceral leishmaniasis.

Kategori:
Heterocyclic Compounds, Fused-RingQuinolines
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biotech | CAS: 898830-54-1

Sitimagene ceradenovec is a novel gene-based product for the treatment of patients with operable high grade glioma, a type of malignant brain tumour, given in addition to standard surgery and radiotherapy/chemotherapy. It is being developed by Ark Therapeutic…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsAntineoplastic cell and gene therapy +6
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Sitravatinib DB15036
small molecule | CAS: 1123837-84-2

Sitravatinib is under investigation in clinical trial NCT03680521 (Neoadjuvant Sitravatinib in Combination With Nivolumab in Patients With Clear Cell Renal Cell Carcinoma).

Kategori:
AmidesAminesAniline Compounds +3
Target Protein:
Hepatocyte growth factor receptorVascular endothelial growth factor receptor 3Vascular endothelial growth factor receptor 2 +1
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Sivifene DB05686
small molecule | CAS: 2675-35-6

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesHydrazines
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Sivopixant DB18816
small molecule | CAS: 2414285-40-6

Deskripsi belum tersedia.

Kategori:
Amines
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Sizofiran DB13128
small molecule | CAS: 9050-67-3

A beta-D-glucan obtained from the Aphyllophoral fungus Schizophyllum commune. It is used as an immunoadjuvant in the treatment of neoplasms, especially tumors found in the stomach. Sizofiran has been used in trials studying the treatment of Cervical Cancer.

Kategori:
Adjuvants, ImmunologicAntineoplastic AgentsAntineoplastic Agents, Phytogenic +6
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SJ-733 DB12659
small molecule | CAS: 1424799-20-1

SJ-733 has been used in trials studying Malaria.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
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SJG-136 DB11965
small molecule | CAS: 232931-57-6

SJG-136 has been used in trials studying the treatment of Recurrent Fallopian Tube Cancer, Secondary Acute Myeloid Leukemia, de Novo Myelodysplastic Syndromes, Recurrent Ovarian Epithelial Cancer, and Secondary Myelodysplastic Syndromes, among others.

Kategori:
BenzazepinesHeterocyclic Compounds, Fused-Ring
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Skf 107457 DB04191
small molecule | CAS: 144285-77-8

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
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small molecule | CAS: 162849-90-3

SKF-96365 is a receptor-mediated calcium entry (RMCE) inhibitor structurally different from other calcium antagonists.[A253132]

Kategori:
Antiarrhythmic agentsAntiplatelet agentsCalcium Channel Blockers +4
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Skim milk Approved DB15546
biotech

Skim milk allergenic extract is used in allergenic testing.

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biotech

Skin-derived ABCB5-positive Mesenchymal Stem cells are under investigation in clinical trial NCT04971161 (Allogeneic Abcb5-positive Dermal Mesenchymal Stromal Cells for Treatment of CVU (Phase Iib)).

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SL017 DB05156
small molecule

SL017 formulated as a topical gel, has been combined with a widely available light source for permanent removal of unwanted hair and for treatment of actinic keratosis

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SLC-0111 DB18815
small molecule | CAS: 178606-66-1

Deskripsi belum tersedia.

Kategori:
AmidesAntineoplastic AgentsBenzene Derivatives +2
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SLC-391 DB18814
small molecule | CAS: 1783825-18-2

Deskripsi belum tersedia.

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SLN500 DB18636
biotech

SLN500 is a synthetic double-strand small interfering ribonucleic acid (siRNA) oligonucleotide drug directed against C3 messenger RNA

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SLV-334 DB15356
small molecule | CAS: 182821-33-6

SLV-334 is under investigation in clinical trial NCT00735085 (A Phase 2a Dose Escalation Study With SLV334 in Patients With Traumatic Brain Injury.).

Target Protein:
Neprilysin
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SLV319 DB05077
small molecule

SLV319 belongs to a novel class of agents called CB1 antagonists, which work by blocking the cannabinoid type 1 (CB1) receptor. It is developed for the treatment of obesity and other metabolic disorders.

Kategori:
Agents producing tachycardiaAmidesCannabinoid Receptor Antagonists +4
Target Protein:
Cannabinoid receptor 1
Waktu Paruh-
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SLx-2101 DB05615
small molecule

SLx-2101 is an oral, long-acting PDE5 inhibitor developed by Surface Logix Inc. to treat Hypertension.

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SLx-4090 DB05678
small molecule | CAS: 913541-47-6

SLx-4090 is a microsomal triglyceride transfer protein (MTTP) inhibitor potentially for the treatment of type 2 diabetes. [A33218]

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +2
Target Protein:
Microsomal triglyceride transfer protein large subunit
Waktu Paruh-
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Genetik -
biotech

The New York City Board of Health strain of _Vaccinia_ is a viral strain used as a component of some smallpox vaccinations.[L12747] ACAM2000, a percutaneously administered smallpox vaccine that was approved by the FDA in 2007, contains live antigens of this s…

Kategori:
Actively Acquired ImmunityBiological ProductsComplex Mixtures +4
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biotech

Deskripsi belum tersedia.

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Smilagenin DB05450
small molecule | CAS: 126-18-1

Smilagenin is a novel non-peptide, orally bioavailable neurotrophic factor inducer that readily reverses free radical neurotoxicity produced by 1-ethyl-4- phenylpyridium (MPP+) in dopaminergic neurones and reverses the decrease of neuronal growth factors and …

Kategori:
CholestanesDrugs, Chinese HerbalFused-Ring Compounds +4
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SN-38 DB05482
small molecule | CAS: 86639-52-3

7-ethyl-10-hydroxycamptothecin (SN 38) is a liposomal formulation of the active metabolite of Irinotecan [DB00762], a chemotherapeutic pro-drug approved for the treatment of advanced colorectal cancer. SN 38 has been used in trials studying the treatment of …

Kategori:
AlkaloidsAntineoplastic AgentsCytochrome P-450 CYP3A Inhibitors +9
Target Protein:
DNA topoisomerase 1
Waktu Paruh-
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small molecule | CAS: 59734-15-5

Deskripsi belum tersedia.

Kategori:
GlycerophosphatesGlycerophospholipidsLipids +3
Target Protein:
Annexin A5
Waktu Paruh-
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small molecule | CAS: 17989-41-2

Deskripsi belum tersedia.

Target Protein:
Fructose-bisphosphate aldolase BPyridoxine 5'-phosphate synthaseTriosephosphate isomerase +1
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Snail, unspecified Approved DB14245
biotech

Snail, unspecified is an animal extract used in some OTC (over-the-counter) products. It is not an approved drug.

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SNP-ACTH (1-39) DB18544
biotech

SNP-ACTH (1-39) is a synthetic porcine Corticotropin (ACTH)

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SNS-032 DB05969
small molecule | CAS: 345627-80-7

Deskripsi belum tersedia.

Kategori:
Sulfur Compounds
Target Protein:
Cyclin-dependent kinase 9Cyclin-dependent kinase 2Cyclin-dependent kinase 7 +1
Waktu Paruh-
Vol. Distribusi-
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SNS-314 DB06134
small molecule | CAS: 1057249-41-8

SNS-314 is a potent and selective inhibitor of Aurora kinases A, B, and C. Proliferating cells treated with SNS-314 bypass the mitotic spindle checkpoint and fail to undergo cytokinesis, leading to multiple rounds of endoreduplication and eventually cell deat…

Kategori:
AmidesBenzene DerivativesProtein Kinase Inhibitors +1
Target Protein:
Aurora kinase BAurora kinase CAurora kinase A
Waktu Paruh-
Vol. Distribusi-
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SNS01-T DB17302
biotech

SNS01-T is a gene therapy nanoparticle. It is composed of three components: a B cell-specific plasmid expressing eIF5AK50R; an siRNA that targets the native eIF5A that promotes growth/anti-apoptosis of cancer cells; and polyethylenimine.[A254706]

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small molecule | CAS: 1226795-18-1

Snubh-nm-333 F-18 is under investigation in clinical trial NCT02149017 (Phase 1 and Phase 2 Clinical Trials of SNUBH-NM-333(18F)).

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SNX-2112 DB17055
small molecule | CAS: 908112-43-6

SNX-2112 is a heat shock protein 90 (Hsp90) inhibitor.[A253137]

Kategori:
Heterocyclic Compounds, Fused-RingHSP90 Heat-Shock Proteins, antagonists & inhibitors
Target Protein:
Heat shock protein HSP 90-alpha
Waktu Paruh-
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SNX-5422 DB06070
small molecule | CAS: 908115-27-5

SNX-5422 is a synthetic, novel, small molecule Hsp90 Inhibitor. As an oral formulation that demonstrates strong efficacy and tolerability, SNX-5422 is positioned as a breakthrough therapy with broad applicability across a wide range of cancers.

Kategori:
Acids, CarbocyclicAmidesAmino Acids +5
Target Protein:
Heat shock protein HSP 90-alphaHeat shock protein HSP 90-beta
Waktu Paruh-
Vol. Distribusi-
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Genetik -
SO-101 DB05345
small molecule

SO-101(Silenor) is a low-dose oral tablet formulation of doxepin hydrochloride that is patent protected for its use in insomnia. Doxepin has been prescribed for more than 40 years for the treatment of depression and anxiety at dosages typically ranging from 7…

Target Protein:
Histamine H1 receptor
Waktu Paruh-
Vol. Distribusi-
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Sobetirome DB07425
small molecule | CAS: 211110-63-3

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicBenzene DerivativesFatty Acids +2
Target Protein:
Muscarinic acetylcholine receptor M1Thyroid hormone receptor, alpha isoform 1 variantThyroid hormone receptor beta
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SOBI-003 DB15451
biotech

SOBI-003 is a chemically modified variant of a recombinant human sulfamidase. It is under investigation in clinical trial NCT03811028 (A Study to Assess the Safety, Tolerability, and Efficacy of Long-term SOBI003 Treatment in Pediatric MPS IIIA Patients).

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Sobrerol DB13315
small molecule | CAS: 42370-41-2

Deskripsi belum tersedia.

Kategori:
Cough and Cold PreparationsExpectorantsRespiratory System Agents
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Socazolimab DB18845
biotech | CAS: 2305043-30-3

Socazolimab is under investigation in clinical trial NCT04878016 (A Study of Carboplatin Plus Etoposide With or Without ZKAB001 (Anti-pd-l1 Antibody) in Patients With ES-SCLC).

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small molecule | CAS: 200880-41-7

Deskripsi belum tersedia.

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Sodium acetate Approved DB09395
small molecule | CAS: 127-09-3

Sodium Acetate is chemically designated CH3COONa, a hygroscopic powder very soluble in water. Sodium acetate could be used as additives in food, industry, concrete manufacture, heating pads and in buffer solutions. Medically, sodium acetate is important compo…

Kategori:
AcetatesAcids, AcyclicBlood and Blood Forming Organs +5
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small molecule | CAS: 1344-00-9

Deskripsi belum tersedia.

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