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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 216 / 236
Thallium Tl-201 DB15361
small molecule | CAS: 15064-65-0

Thallium Tl-201 is under investigation in clinical trial NCT02697760 (The CZT Dynamic Myocardial Perfusion Imaging).

Kategori:
IsotopesRadioisotopes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Radioactive Diagnostic AgentRadiopharmaceutical Activity
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thallous chloride Approved DB09316
small molecule | CAS: 7791-12-0

Thallous chloride (also known as Thallium(I) chloride) is a colourless solid intermediate in the isolation of thallium from its ores. It is created from the treatment of thallium(I) sulfate with hydrochloric acid. This solid crystallizes in the caesium chlori…

Kategori:
ElementsMetalsMetals, Heavy +1
Waktu Paruh91% of the blood ra…
Vol. Distribusi3–10 L/kg
KlirensApproximately 4-8% …
Genetik -
Thallous chloride Tl-201 Approved DB16624
small molecule | CAS: 55172-29-7

Deskripsi belum tersedia.

Kategori:
Diagnostic Radiopharmaceuticals
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
THE-630 DB16750
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Theanine DB12444
small molecule | CAS: 3081-61-6

Theanine, a precursor of ethylamine, is found in green tea. It is under investigation in clinical trial NCT00291070 (Effects of L-Theanine in Boys With ADHD).

Kategori:
Amino AcidsAmino Acids, AcidicAmino Acids, Dicarboxylic +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 326-91-0

Thenoyltrifluoroacetone is a chelating agent and inhibitor of cellular respiration.

Kategori:
ButanonesChelating AgentsCompounds used in a research, industrial, or household setting +4
Target Protein:
Liver carboxylesterase 1Succinate dehydrogenase [ubiquinone] flavoprotein subunit, mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thenyldiamine Approved DB16022
small molecule | CAS: 91-79-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Theobromine DB01412
small molecule | CAS: 83-67-0

Theobromine (3,7-dimethylxanthine) is the principle alkaloid in Theobroma cacao (the cacao bean) and other plants. A xanthine alkaloid that is used as a bronchodilator and as a vasodilator. It has a weaker diuretic activity than theophylline and is also a les…

Kategori:
AlkaloidsAnti-Asthmatic AgentsAutonomic Agents +15
Target Protein:
Adenosine receptor A15'-nucleotidaseAdenosine receptor A2a +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Theodrenaline DB12927
small molecule | CAS: 13460-98-5

Theodrenaline is under investigation in clinical trial NCT01311414 (Effect of Cafedrine/Theodrenaline and Urapidil on Cerebral Oxygenation).

Kategori:
Adrenergic and Dopaminergic AgentsAgents that produce hypertensionAlcohols +20
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Theophylline Approved DB00277
small molecule | CAS: 58-55-9

A methylxanthine derivative from tea with diuretic, smooth muscle relaxant, bronchial dilation, cardiac and central nervous system stimulant activities. Mechanistically, theophylline acts as a phosphodiesterase inhibitor, adenosine receptor blocker, and histo…

Kategori:
Agents that reduce seizure thresholdAlkaloidsAnti-Asthmatic Agents +32
Target Protein:
Adenosine receptor A15'-nucleotidaseAdenosine receptor A2a +12
Gen Terkait:
CYP1A2
Waktu Paruh8 hours
Vol. Distribusi* 0.3 to 0.7 L/kg
Klirens* 0.29 mL/kg/min [P…
Genetik 1 Varian
Theralizumab DB15717
biotech | CAS: 906068-56-2

Theralizumab is a humanized anti-CD28 monoclonal antibody designed for treating autoimmune diseases and cancer. After the first human trial, it was withdrawn due to severe toxicity (likely due to lymphopenia and human cytokine release).[A216527,A216532]

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

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Genetik -
Thermomyces lanuginosus Approved DB10973
biotech

Thermomyces lanuginosus allergenic extract is used in allergenic testing.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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Thiabendazole Approved DB00730
small molecule | CAS: 148-79-8

2-Substituted benzimidazole first introduced in 1962. It is active against a variety of nematodes and is the drug of choice for strongyloidiasis. It has CNS side effects and hepatototoxic potential. (From Smith and Reynard, Textbook of Pharmacology, 1992, p91…

Kategori:
AnthelminticsAnti-Infective AgentsAntifungals for Dermatological Use +18
Target Protein:
Fumarate reductase flavoprotein subunit
Waktu ParuhThe half-life for t…
Vol. Distribusi-
Klirens-
Genetik -
Thiamine Approved DB00152
small molecule | CAS: 70-16-6

Thiamine or thiamin, also known as vitamin B1, is a colorless compound with the chemical formula C12H17N4OS. It is soluble in water and insoluble in alcohol. Thiamine decomposes if heated. Thiamine was first discovered by Umetaro Suzuki in Japan when research…

Kategori:
Alimentary Tract and MetabolismDiet, Food, and NutritionFood +10
Target Protein:
Thiamine pyrophosphokinase 1Pyruvate dehydrogenase E1 component
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 67-16-3

Deskripsi belum tersedia.

Kategori:
PyrimidinesSulfur CompoundsThiazoles
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thiamylal Approved DB01154
small molecule | CAS: 77-27-0

A barbiturate that is administered intravenously for the production of complete anesthesia of short duration, for the induction of general anesthesia, or for inducing a hypnotic state. (From Martindale, The Extra Pharmacopoeia, 30th ed, p919)

Kategori:
AnestheticsAnesthetics, GeneralAnesthetics, Intravenous +22
Target Protein:
Gamma-aminobutyric acid receptor subunit gamma-3ATP-sensitive inward rectifier potassium channel 8ATP-sensitive inward rectifier potassium channel 11 +1
Waktu ParuhAlthough no studies…
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Urokinase-type plasminogen activatorSerine protease 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Coagulation factor X
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thiethylperazine Approved DB00372
small molecule | CAS: 1420-55-9

A dopamine antagonist that is particularly useful in treating the nausea and vomiting associated with anesthesia, mildly emetic cancer chemotherapy agents, radiation therapy, and toxins. This piperazine phenothiazine does not prevent vertigo or motion sicknes…

Kategori:
AntiemeticsAntihistamines for Systemic UseAntipsychotic Agents +16
Target Protein:
D(2) dopamine receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thimerosal Approved DB11590
small molecule | CAS: 54-64-8

Thiomersal (INN), commonly known in the U.S. as thimerosal, is an organomercury compound. This compound is a well-established and widely used antiseptic and antifungal agent. Developed in 1927, thimerosal has been and is still being used as a preservative…

Kategori:
Alkylmercury CompoundsAntiseptics and DisinfectantsCell-mediated Immunity +11
Target Protein:
Methionine synthaseCystine/glutamate transporterSodium/potassium-transporting ATPase subunit gamma
Waktu ParuhA study was done to…
Vol. Distribusi266 L in one study …
KlirensThe high concentrat…
Genetik -
THIO-ATPA DB04798
small molecule

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsSulfur Compounds
Target Protein:
Glutamate receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Cyclomaltodextrin glucanotransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thiocamphor DB02851
small molecule | CAS: 7519-74-6

Deskripsi belum tersedia.

Kategori:
Bicyclic MonoterpenesBornanesBridged-Ring Compounds +4
Target Protein:
Camphor 5-monooxygenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thiocitrulline DB03953
small molecule | CAS: 156719-37-8

Deskripsi belum tersedia.

Kategori:
AmidesAmino AcidsAmino Acids, Diamino +4
Target Protein:
Nitric oxide synthase, inducible
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 137314-40-0

A salt of alpha-lipoic acid and tromethamine; may be useful in treating vascular stress in patients with diabetes.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 51555-87-4

Thiodigalactoside is a solid. This compound belongs to the dihexoses. These are disaccharides containing two hexose carbohydrates. This medication is known to target galectin-1, heat-labile enterotoxin b chain, neurocan core protein, and lactose permease.

Kategori:
CarbohydratesGalactosidesGlycosides +2
Target Protein:
Heat-labile enterotoxin B chainLactose permeaseNeurocan core protein +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thiopental Approved DB00599
small molecule | CAS: 76-75-5

A barbiturate that is administered intravenously for the induction of general anesthesia or for the production of complete anesthesia of short duration. It is also used for hypnosis and for the control of convulsive states. It has been used in neurosurgical p…

Kategori:
AnestheticsAnesthetics, GeneralAnesthetics, Intravenous +27
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1Gamma-aminobutyric acid receptor subunit alpha-2Gamma-aminobutyric acid receptor subunit alpha-3 +9
Waktu Paruh3-8 hours
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Carbonic anhydrase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thiopropazate DB13557
small molecule | CAS: 84-06-0

Deskripsi belum tersedia.

Kategori:
Antipsychotic AgentsCentral Nervous System DepressantsHeterocyclic Compounds, Fused-Ring +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 68488-87-9

Deskripsi belum tersedia.

Kategori:
AcidsAcids, NoncarboxylicAnions +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thioridazine Approved DB00679
small molecule | CAS: 50-52-2

A phenothiazine antipsychotic used in the management of psychoses, including schizophrenia, and in the control of severely disturbed or agitated behavior. It has little antiemetic activity. Thioridazine has a higher incidence of antimuscarinic effects, but a …

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +37
Target Protein:
D(2) dopamine receptorD(1A) dopamine receptorAlpha-1A adrenergic receptor +3
Waktu Paruh21-25 hours
Vol. Distribusi-
Klirens-
Genetik -
Thiorphan DB08626
small molecule | CAS: 76721-89-6

A potent inhibitor of membrane metalloendopeptidase (enkephalinase). Thiorphan potentiates morphine-induced analgesia and attenuates naloxone-precipitated withdrawal symptoms.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAmino Acids, Sulfur +4
Target Protein:
Neprilysin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 147-93-3

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAlkylmercury CompoundsAnalgesics +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thiostrepton DB11467
small molecule

Thiostrepton is a natural cyclic oligopeptide antibiotic, derived from several strains of streptomycetes including Streptomyces azureus and Streptomyces laurentii. Thiostrepton is a natural product of the ribosomally synthesized and post-translationally modif…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thiosulfuric acid Approved DB09499
small molecule | CAS: 13686-28-7

Thiosulfuric acid is available in its salt forms sodium thiosulfate and sodium thiosulfate pentahydrate. Sodium thiosulfate is part of the World Health Organization’s list of essential medicines, and it has a variety of industrial uses, including food preserv…

Kategori:
AcidsAnti-Infective AgentsAntidotes +14
Waktu ParuhThe half-life of th…
Vol. DistribusiThiosulfate has a m…
KlirensIn patients with fu…
Genetik -
Thiotepa Approved DB04572
small molecule | CAS: 52-24-4

N,N'N'-triethylenethiophosphoramide (ThioTEPA) is a cancer chemotherapeutic member of the alkylating agent group, now in use for over 50 years. It is a stable derivative of N,N',N''- triethylenephosphoramide (TEPA). It is mostly used to treat breast cancer, o…

Kategori:
Alkylating ActivityAlkylating DrugsAntineoplastic Agents +23
Target Protein:
DNA
Waktu Paruh1.5 to 4.1 hours
Vol. Distribusi-
Klirens* 446 +/- 63 mL/min…
Genetik -
Thiram Approved DB13245
small molecule | CAS: 137-26-8

Thiram may be used in dermatology as a scabicide [T436]. Thiram is mainly used as a fungicide for plants and treatment for seeds, however, this use is being investigated for safety in many markets including Canada [L5425].

Kategori:
Acids, AcyclicAgrochemicalsAntiparasitic Products, Insecticides and Repellents +16
Target Protein:
Tyrosine-protein kinase JAK2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
THK-5351 DB19222
small molecule | CAS: 1707147-26-9

Deskripsi belum tersedia.

Kategori:
AminesFluorine RadioisotopesHeterocyclic Compounds, Fused-Ring +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
THK-5351 F-18 DB19223
small molecule | CAS: 1707148-68-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thonzylamine Approved DB11235
small molecule | CAS: 91-85-0

Thonzylamine is an antihistamine and anticholinergic drug. It is available as combination products with [DB04837] or [DB00388] for temporary relief of symptoms of common cold, hay fever (allergic rhinitis) or other upper respiratory allergies.

Kategori:
Agents producing tachycardiaAntiallergic Agents, Excl. CorticosteroidsAnticholinergic Agents +11
Target Protein:
Histamine H1 receptorMuscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2 +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
THR-184 DB19097
biotech | CAS: 930274-80-9

THR-184 is under investigation in clinical trial NCT01830920 (A Study of THR-184 in Patients at Risk of Developing Cardiac Surgery Associated-acute Kidney Injury (CSA-AKI)).

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Threonine Approved DB00156
small molecule | CAS: 72-19-5

An essential amino acid occurring naturally in the L-form, which is the active form. It is found in eggs, milk, gelatin, and other proteins.

Kategori:
Amino AcidsAmino Acids, EssentialAmino Acids, Neutral +5
Target Protein:
Threonine--tRNA ligase 1, cytoplasmicThreonine--tRNA ligase, mitochondrialBeta-lactamase Toho-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
L-asparaginase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Thrombin alfa Approved DB11572
biotech | CAS: 869858-13-9

Thrombin Alfa is a human coagulation protein produced via recombinant DNA technology from a genetically modified CHO cell line. Thrombin Alfa is identical in amino acid sequence and structurally similar to naturally occurring human thrombin. Thrombin Alfa pre…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +12
Target Protein:
Coagulation factor VCoagulation factor VIIIFibrinogen alpha chain +2
Waktu ParuhFollowing intraveno…
Vol. DistribusiTraditional absorpt…
KlirensTraditional absorpt…
Genetik -
Thrombomodulin Alfa Approved DB05777
biotech | CAS: 120313-91-9

Thrombomodulin Alfa is a novel, recombinant and soluble thrombomodulin (ART-123). It is a human protein with both thrombin inhibiting and protein C stimulating activities, for the potential treatment of thromboembolism and blood clotting disorders, such as di…

Kategori:
Amino Acids, Peptides, and ProteinsCarbohydratesGlycoconjugates +7
Target Protein:
ProthrombinCoagulation factor V
Waktu Paruh2–3 days after sc i…
Vol. Distribusi-
Klirens7-10 days
Genetik -
Thymalfasin DB04900
biotech | CAS: 62304-98-7

Thymalfasin is a chemically synthesized version of thymosin alpha 1 that is identical to human thymosin alpha 1. Thymosin alpha 1 is an acetylated polypeptide. Thymosin alpha 1 is now approved in 35 developing countries for the treatment of Hepatitis B and C.…

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAntineoplastic Agents +7
Waktu ParuhApproximately 2 hou…
Vol. Distribusi-
Klirens-
Genetik -
Thyme oil DB16610
biotech | CAS: 8007-46-3

Deskripsi belum tersedia.

Kategori:
AngiospermsBenzene DerivativesBiological Products +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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