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12560

Total database: 17430
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9109 (72.5%)
Target
6912 (55.0%)
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109 (0.9%)
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12560 (100.0%)

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Halaman 216 / 252
SGN-30 DB05471
biotech

SGN-30 is an engineered monoclonal antibody (mAb) that reacts with significant affinity to the CD30 antigen, which is highly expressed on a variety of hematologic malignancies as compared to on normal cells. SGN-30 has been shown to induce direct anti-cancer…

Target Protein:
Nuclear factor NF-kappa-B p105 subunitNuclear factor NF-kappa-B p100 subunit
Waktu Paruh-
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Genetik -
SGS-742 DB05010
small molecule | CAS: 123690-78-8

SGS-742 has been used in trials studying the treatment of Seizures and Metabolic Disease.

Kategori:
Central Nervous System AgentsCompounds used in a research, industrial, or household settingGABA Agents +4
Target Protein:
Gamma-aminobutyric acid type B receptor subunit 1Gamma-aminobutyric acid type B receptor subunit 2
Waktu Paruh4 hours
Vol. Distribusi-
Klirens-
Genetik -
SGS518 DB05042
small molecule

SGS518, a novel antagonist for the 5HT6 subtype of the serotonin receptor, is being developed as a treatment for Cognitive Impairment Associated with Schizophrenia (CIAS).

Target Protein:
5-hydroxytryptamine receptor 6
Waktu Paruh-
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SGX-523 DB06314
small molecule | CAS: 1022150-57-7

A MET receptor tyrosine kinase inhibitor.

Target Protein:
Hepatocyte growth factor receptor
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Shark liver oil DB11088
biotech | CAS: 68990-63-6

Shark oil is extracted from the livers of sharks, which can account for up to 25% of their total body weight. The 3 main targeted species are the deep sea shark (Centrophorus squamosus), the dogfish (Sqaulus acanthias), and the basking shark (Cetorhinus maxim…

Waktu Paruh-
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Genetik -
biotech

Deskripsi belum tersedia.

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Shrimp Approved DB10567
biotech

Shrimp allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
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Siagoside DB12351
small molecule | CAS: 100345-64-0

Siagoside (Sygen, AGF 2) has been investigated for the treatment of Parkinson Disease. It is a naturally occurring substance in the nerve cell’s membrane that is thought to play a role in cell growth, development, and repair. Siagoside completed phase 2 trial…

Kategori:
Acidic GlycosphingolipidsCarbohydratesGangliosides +7
Waktu Paruh-
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Sibeprenlimab DB18919
biotech | CAS: 2382896-07-1

Sibeprenlimab is under investigation in clinical trial NCT05248659 (Phase 2/3 Open-label Trial of Sibeprenlimab in the Treatment of Immunoglobulin a Nephropathy).

Waktu Paruh-
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Sibofimloc DB16400
small molecule | CAS: 1616113-45-1

Sibofimloc is under investigation in clinical trial NCT03943446 (TAK-018 for Prevention of the Recurrence of Postoperative Crohn's Disease (CD)).

Waktu Paruh-
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Sibutramine Approved DB01105
small molecule | CAS: 106650-56-0

Sibutramine (trade name Meridia in the USA, Reductil in Europe and other countries), usually as sibutramide hydrochloride monohydrate, is an orally administered agent for the treatment of obesity. It is a centrally acting stimulant chemically related to amphe…

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAnti-Obesity Agents +23
Target Protein:
Sodium-dependent dopamine transporterSodium-dependent serotonin transporterSodium-dependent noradrenaline transporter
Gen Terkait:
GNB3
Waktu Paruh1.1 hours
Vol. Distribusi-
Klirens* Oral cl=1750 L/h …
Genetik 1 Varian
SIG-007 DB17710
biotech

SIG-007 is a gene therapy that consists of cells that are genetically modified with a non-viral vector to express human alpha-galactosidase A. Developed by Sigilon Therapeutics, t is being investigated for the treatment of Fabry Disease.[L46153]

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SIG-205 DB18548
biotech

SIG-205 is a Cultured human retinal pigment epithelial cells (ARPE-19) genetically modified with a non-viral vector to express human native alpha-L-iduronidase enzyme (hIDUA), encapsulated within two-layer modified alginate spheres

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SIG-207 DB18547
biotech

SIG-207 is a Cultured human retinal pigment epithelial cells (ARPE-19) genetically modified with a non-viral vector to express Human alpha-galactosidase A (alpha-Gal A), encapsulated within two-layer modified alginate spheres

Waktu Paruh-
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siG12D LODER DB16329
biotech

siG12D LODER is under investigation in clinical trial NCT01676259 (A Phase 2 Study of Sig12d LODER in Combination With Chemotherapy in Patients With Locally Advanced Pancreatic Cancer).

Waktu Paruh-
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Sildenafil Approved DB00203
small molecule | CAS: 139755-83-2

In eliciting its mechanism of action, sildenafil ultimately prevents or minimizes the breakdown of cyclic guanosine monophosphate (cGMP) by inhibiting cGMP specific phosphodiesterase type 5 (PDE5) [F3850, F3853, F3856, F3859, F3883, F3886, L5611, L5614]. The …

Kategori:
Agents Causing Muscle ToxicityAmidesCardiovascular Agents +33
Target Protein:
Plasma protease C1 inhibitorcGMP-specific 3',5'-cyclic phosphodiesteraseRetinal rod rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit gamma +3
Gen Terkait:
ACE GNB3
Waktu ParuhThe terminal phase …
Vol. DistribusiThe mean steady-sta…
KlirensThe total body clea…
Genetik 2 Varian
Silk sericin DB15531
biotech | CAS: 1190590-38-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsArthropod ProteinsBiopolymers +4
Waktu Paruh-
Vol. Distribusi-
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Silmitasertib DB15408
small molecule | CAS: 1009820-21-6

Silmitasertib is under investigation in clinical trial NCT03904862 (Testing the Safety and Tolerability of CX-4945 in Patients With Recurrent Medulloblastoma Who May or May Not Have Surgery).

Kategori:
Casein Kinase II, antagonists & inhibitorsHeterocyclic Compounds, Fused-Ring
Target Protein:
Casein kinase II subunit alpha
Waktu Paruh-
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Silodosin Approved DB06207
small molecule | CAS: 160970-54-7

Silodosin is a selective antagonist of alpha(?)-1 adrenergic receptors that binds to the ?<sub>1A</sub> subtype with the highest affinity. ?1-adrenergic receptors regulate smooth muscle tone in the bladder neck, prostate, and prostatic urethra: the ?<sub>1A</…

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +15
Target Protein:
Alpha-1A adrenergic receptorAlpha-1D adrenergic receptorAlpha-1B adrenergic receptor +1
Waktu ParuhThe elimination hal…
Vol. DistribusiSilodosin has an ap…
KlirensAfter intravenous a…
Genetik -
Siltuximab Approved DB09036
biotech | CAS: 541502-14-1

Siltuximab is a chimeric (human-mouse) monoclonal immunoglobulin G1-kappa antibody produced in a Chinese hamster ovary (CHO) cell line by recombinant DNA technology. Siltuximab prevents the binding of IL-6 to soluble and membrane-bound IL-6 receptors by formi…

Kategori:
Agents reducing cytokine levelsAmino Acids, Peptides, and ProteinsAntibodies +20
Target Protein:
Interleukin-6
Waktu ParuhThe mean terminal h…
Vol. DistribusiBased on population…
KlirensBody weight was ide…
Genetik -
Silver Approved DB12965
small molecule | CAS: 7440-22-4

Silver (Ag) is a chemical element that belongs in the family of transition metals in the periodic table. It has a high electrical conductivity, thermal conductivity, and reflectivity. Silver exists as a pure elemental form, alloy with other metals, and minera…

Kategori:
Antiseptics and DisinfectantsDermatologicalsElements +4
Target Protein:
MetallothioneinCeruloplasminAlbumin +1
Waktu ParuhThe biological half…
Vol. DistribusiFollowing exposure …
Klirens-
Genetik -
Silver cation DB14521
small molecule | CAS: 14701-21-4

Deskripsi belum tersedia.

Waktu Paruh-
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Silver citrate DB11233
small molecule | CAS: 126-45-4

Deskripsi belum tersedia.

Waktu Paruh-
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Silver oxide DB15668
small molecule | CAS: 20667-12-3

Deskripsi belum tersedia.

Kategori:
AnionsAnti-Infective AgentsElectrolytes +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 9015-51-4

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAnti-Infective Agents, Local +1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Silver sulfadiazine Approved DB05245
small molecule | CAS: 22199-08-2

Silver sulfadiazine is a sulfa derivative topical antibacterial used primarily on second- and third-degree burns.

Kategori:
AmidesAminesAniline Compounds +14
Target Protein:
DNADihydropteroate synthase
Waktu Paruh-
Vol. Distribusi-
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Simendan DB12286
small molecule | CAS: 131741-08-7

Simendan is under investigation in clinical trial NCT00527059 (Renal Effects of Levosimendan in Patients Admitted With Acute Decompensated Heart Failure).

Kategori:
Antiarrhythmic agentsCardiotonic AgentsCardiovascular Agents +11
Waktu Paruh-
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Genetik -
small molecule | CAS: 910562-13-9

Simenepag isopropyl has been used in trials studying the treatment of Ocular Hypertension and Glaucoma, Open-Angle.

Waktu Paruh-
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Simeprevir Approved DB06290
small molecule | CAS: 923604-59-5

Simeprevir is a hepatitis C virus (HCV) NS3/4A protease inhibitor indicated in patient's with HCV genotype 1 for the treatment of chronic hepatitis C virus (HCV) infection. HCV is a single-stranded RNA virus that is categorized into nine distinct genotypes, w…

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +37
Target Protein:
Genome polyproteinNS3 proteaseGenome polyprotein
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of si…
Genetik -
Simethicone Approved DB09512
small molecule | CAS: 8050-81-5

Simethicone is a silicon based surfactant that decreases the surface tension of gastrointestinal gas bubbles to facilitate their elimination.[A228308] It has a favourable safety profile as it is not systemically absorbed.[A228308] Simethicone has been in u…

Kategori:
Antifoaming AgentsCompounds used in a research, industrial, or household settingDermatologicals +9
Waktu ParuhSimethicone is not …
Vol. DistribusiSimethicone is not …
KlirensSimethicone is not …
Genetik -
Simoctocog alfa Approved DB09108
biotech | CAS: 1219013-68-9

Simoctocog alfa is a recombinant B-domain deleted (BDD) rFVIII produced in genetically modified human embryonic kidney (HEK) 293F cells. The harvested product is concentrated and purified by a series of chromatography steps. It is an antihemorrhagic agent use…

Kategori:
Amino Acids, Peptides, and ProteinsCarbohydratesGlycoconjugates +1
Target Protein:
von Willebrand factor
Waktu ParuhAt initial assessme…
Vol. DistribusiIt is observed that…
KlirensAt initial assessme…
Genetik -
Simotaxel DB15384
small molecule | CAS: 791635-59-1

Simotaxel is under investigation in clinical trial NCT00088647 (Study Evaluating MST-997 in Advanced Malignant Solid Tumors).

Kategori:
CyclodecanesCycloparaffinsDiterpenes +1
Waktu Paruh-
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Genetik -
Simpinicline DB17065
small molecule | CAS: 753015-44-0

Deskripsi belum tersedia.

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Simtuzumab DB12152
biotech | CAS: 1318075-13-6

Simtuzumab has been used in trials studying the treatment and basic science of Myelofibrosis, Pancreatic Cancer, Colorectal Cancer, and Idiopathic Pulmonary Fibrosis.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Simufilam DB18817
small molecule | CAS: 1224591-33-6

Deskripsi belum tersedia.

Target Protein:
Filamin-A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Simvastatin Approved DB00641
small molecule | CAS: 79902-63-9

Simvastatin, also known as the brand name product Zocor, is a lipid-lowering drug derived synthetically from a fermentation product of _Aspergillus terreus_. It belongs to the statin class of medications, which are used to lower the risk of cardiovascular dis…

Kategori:
Agents Causing Muscle ToxicityAnticholesteremic AgentsBSEP/ABCB11 Substrates +37
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductaseIntegrin alpha-LHistone deacetylase 2
Gen Terkait:
KIF6 HMGCR SLCO1B1
Waktu Paruh4.85 hours[A181571]
Vol. DistribusiRat studies indicat…
Klirens-
Genetik 3 Varian
Sinapic acid DB08587
small molecule | CAS: 7362-37-0

Sinapic acid is a matrix for matrix-assisted laser desorption technique for protein MW determination. It is also a constituent of propolis.

Kategori:
Acids, CarbocyclicCinnamatesCompounds used in a research, industrial, or household setting +2
Target Protein:
Endo-1,4-beta-xylanase Y
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sinapultide Approved DB11332
small molecule | CAS: 138531-07-4

Sinapultide (also known as KL4 peptide) is a synthetic protein used to mimic human lung surfactant protein B.[L2502] This protein has a weight of 2469.40.[L2502] Sinapultide is a 21-residue peptide made up of lysine (K) and leucine (L) residues with the se…

Kategori:
Amino Acids, Peptides, and ProteinsPulmonary Surfactants
Target Protein:
Lung epithelial cells
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sinbaglustat DB17619
small molecule | CAS: 441061-33-2

Deskripsi belum tersedia.

Kategori:
CarbohydratesImines
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Sincalide Approved DB09142
biotech | CAS: 25126-32-3

Sincalide is a medication given by injection to assist in the diagnosis of gallbladder and pancreas disorders. It is identified as the 8-amino acid C-terminal segment of cholecystokinin and is also known as _CCK-8_. Naturally occurring cholecystokinin is a ga…

Kategori:
Amino Acids, Peptides, and ProteinsCholecystokinin AnalogDiagnostic Agents +7
Target Protein:
Cholecystokinin receptor type AGastrin/cholecystokinin type B receptor
Waktu ParuhLimited information…
Vol. DistribusiLimited information…
Klirens-
Genetik -
Sinecatechins Approved DB01266
small molecule | CAS: 188265-33-0

Sinecatechins is a botanical drug product for topical use. It is a partially purified fraction of the water extract of green tea leaves from Camellia sinensis, and is a mixture of catechins and other green tea components. Catechins constitute 85 to 95% (by we…

Kategori:
Antiviral AgentsBenzopyransChromans +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sinefungin DB01910
small molecule | CAS: 58944-73-3

Sinefungin is a solid. This compound belongs to the purine nucleosides and analogues. These are compounds comprising a purine base attached to a sugar. The proteins that adenosyl-ornithine target include RdmB, modification methylase TaqI, rRNA (adenine-N6-)-m…

Kategori:
Anti-Infective AgentsAntifungal AgentsAntiparasitic Agents +7
Target Protein:
Modification methylase RsrIAclacinomycin 10-hydroxylase RdmBrRNA adenine N-6-methyltransferase +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sinomenine DB16892
small molecule | CAS: 115-53-7

Deskripsi belum tersedia.

Kategori:
AlkaloidsAntirheumatic AgentsHeterocyclic Compounds, Fused-Ring +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sintilimab DB15765
biotech | CAS: 2072873-06-2

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Target Protein:
Programmed cell death protein 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Siponimod Approved DB12371
small molecule | CAS: 1230487-00-9

Siponimod, also known as _Mayzent_, by Novartis, is a new drug formulated for the management of Multiple Sclerosis (MS). It was approved by the FDA on March 26, 2019 [L5792] and by Health Canada on February 20, 2020.[L12171] This drug is considered a _sphingo…

Kategori:
Agents that produce hypertensionAntineoplastic and Immunomodulating AgentsAzetines +18
Target Protein:
Sphingosine 1-phosphate receptor 1Sphingosine 1-phosphate receptor 5
Waktu ParuhThe apparent elimin…
Vol. DistribusiSiponimod distribut…
KlirensApparent systemic c…
Genetik -
Sipuleucel-T Approved DB06688
biotech | CAS: 917381-47-6

Sipuleucel-T is a personalized, autologous, cellular immunotherapy. Sipuleucel-T is a therapeutic cancer vaccine for prostate cancer. Sipuleucel-T selectively targets the prostate-specific antigen (PSA) known as prostatic acid phosphatase (PAP) that is expres…

Kategori:
Adjuvants, ImmunologicAntineoplastic and Immunomodulating AgentsAutologous Cellular Immunotherapy +6
Target Protein:
Prostatic acid phosphatase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Siramesine DB06555
small molecule | CAS: 147817-50-3

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Alpha-1A adrenergic receptorAlpha-1D adrenergic receptorAlpha-1B adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sirexatamab DB17515
biotech | CAS: 2414962-49-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sirna-027 DB05896
small molecule

Sirna-027 is a chemically modified short interfering RNA(siRNA) targeting Vascular Endothelial Growth Factor Receptor-1(VEGFR-1). VEGFR-1 is a key component of the clinically validated vascular endothelial growth factor (VEGF) pathway. Sirna-027 is developed …

Waktu Paruh-
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Genetik -
Siroheme DB02832
small molecule | CAS: 52553-42-1

Deskripsi belum tersedia.

Kategori:
Biological FactorsHeterocyclic Compounds, Fused-RingMetalloporphyrins +2
Target Protein:
Sulfite reductase [NADPH] hemoprotein beta-component
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 10751–10800 dari 12560
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