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15718

Total database: 17430
Struktur (SMILES)
10762 (68.5%)
Target
7957 (50.6%)
Genomik
112 (0.7%)
Referensi
15718 (100.0%)

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Hasil Pencarian (15718)

Halaman 216 / 315
Nialamide Approved DB04820
small molecule | CAS: 51-12-7

Withdrawn from the Canadian, US, and UK markets in 1963 due to interactions with food products containing tyrosine.

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +11
Target Protein:
Amine oxidase [flavin-containing] BAmine oxidase [flavin-containing] ACatechol O-methyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Niaouli oil DB16618
biotech | CAS: 8014-68-4

Deskripsi belum tersedia.

Kategori:
Oils, Volatile
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Niaprazine DB13687
small molecule | CAS: 27367-90-4

Niaprazine is a selective brain catecholamine depletor.

Kategori:
Central Nervous System DepressantsHypnotics and SedativesNervous System +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nicarbazin DB11434
small molecule | CAS: 330-95-0

Deskripsi belum tersedia.

Kategori:
AmidesAminesAnilides +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nicergoline Approved DB00699
small molecule | CAS: 27848-84-6

An ergot derivative that has been used as a cerebral vasodilator and in peripheral vascular disease. It has been suggested to ameliorate cognitive deficits in cerebrovascular disease.

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +14
Target Protein:
Alpha-1A adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Niceritrol DB13441
small molecule | CAS: 5868-05-3

Deskripsi belum tersedia.

Kategori:
Hypolipidemic AgentsLipid Modifying AgentsLipid Modifying Agents, Plain +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nickel cation DB14204
small molecule | CAS: 14701-22-5

Deskripsi belum tersedia.

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Nickel sulfate Approved DB14180
small molecule | CAS: 7786-81-4

Nickel sulfate is used in allergenic testing.

Kategori:
Compounds used in a research, industrial, or household settingElementsIrritants +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Niclosamide Approved DB06803
small molecule | CAS: 50-65-7

Niclosamide is an antihelminthic used for the treatment of tapeworm infections. Helminths (worms) are multicellular organisms that infect very large numbers of humans and cause a broad range of diseases. Over 1 billion people are infected with intestinal nema…

Kategori:
AgrochemicalsAmidesAmines +22
Target Protein:
DNA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nicoboxil Approved DB12911
small molecule | CAS: 13912-80-6

Nicoboxil has been investigated for the treatment of Acute Low Back Pain, where it is typically considered an effective and safe therapeutic option. Nevertheless, it is predominantly found paired with nonivamide as a combination topical analgesic product wher…

Kategori:
Drugs that are Mainly Renally ExcretedPyridines
Waktu ParuhThe half-life of es…
Vol. DistribusiDespite the fact th…
KlirensThe elimination of …
Genetik -
Nicofetamide DB13531
small molecule | CAS: 553-06-0

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismDrugs for Functional Gastrointestinal DisordersSynthetic Antispasmodics, Amides With Tertiary Amines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nicofuranose DB13422
small molecule | CAS: 15351-13-0

Deskripsi belum tersedia.

Kategori:
Cardiovascular AgentsLipid Modifying AgentsLipid Modifying Agents, Plain +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nicomorphine DB13454
small molecule | CAS: 639-48-5

Deskripsi belum tersedia.

Kategori:
AlkaloidsAnalgesicsCentral Nervous System Agents +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nicorandil Approved DB09220
small molecule | CAS: 65141-46-0

Nicorandil is an orally efficacious vasodilatory drug and antianginal agent marketed in the UK, Australia, most of Europe, India, Philippines, Japan, South Korea, and Taiwan. It is not an approved drug by FDA. It is a niacinamide derivative that induces vasod…

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsAntihypertensive Agents +10
Target Protein:
ATP-binding cassette sub-family C member 9
Waktu ParuhThe elimination hal…
Vol. DistribusiAfter oral (and i.v…
KlirensThe total body clea…
Genetik -
Nicotinaldehyde DB15905
small molecule | CAS: 500-22-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Nicotinamide Approved DB02701
small molecule | CAS: 98-92-0

An important compound functioning as a component of the coenzyme NAD. Its primary significance is in the prevention and/or cure of blacktongue and pellagra. Most animals cannot manufacture this compound in amounts sufficient to prevent nutritional deficiency …

Kategori:
Alimentary Tract and MetabolismCytochrome P-450 CYP2D6 InhibitorsCytochrome P-450 CYP2D6 Inhibitors (strength unknown) +13
Target Protein:
ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 2Exotoxin APoly [ADP-ribose] polymerase 1 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

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small molecule | CAS: 53-59-8

Nicotinamide adenine dinucleotide phosphate. A coenzyme composed of ribosylnicotinamide 5'-phosphate (NMN) coupled by pyrophosphate linkage to the 5'-phosphate adenosine 2',5'-bisphosphate. It serves as an electron carrier in a number of react…

Kategori:
Adenine NucleotidesCoenzymesEnzymes and Coenzymes +6
Target Protein:
Isocitrate dehydrogenase [NADP]Aldo-keto reductase family 1 member B1Glucose-6-phosphate 1-dehydrogenase +57
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule

3-Carbamoyl-1-beta-D-ribofuranosyl pyridinium hydroxide-5'phosphate, inner salt. A nucleotide in which the nitrogenous base, nicotinamide, is in beta-N-glycosidic linkage with the C-1 position of D-ribose. Synonyms: Nicotinamide Ribonucleotide; NMN. [PubC…

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesRibonucleotides
Target Protein:
ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 2Nicotinamide/nicotinic acid mononucleotide adenylyltransferase 1Nicotinamide/nicotinic acid mononucleotide adenylyltransferase 3 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1341-23-7

Nicotinamide riboside is under investigation in clinical trial NCT03432871 (Nicotinamide Riboside and Mitochondrial Biogenesis).

Kategori:
Nicotinic AcidsPyridines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nicotine Approved DB00184
small molecule | CAS: 54-11-5

Nicotine is highly toxic alkaloid. It is the prototypical agonist at nicotinic cholinergic receptors where it dramatically stimulates neurons and ultimately blocks synaptic transmission. Nicotine is also important medically because of its presence in tobacco …

Kategori:
Agents producing tachycardiaAlkaloidsAutonomic Agents +40
Target Protein:
Neuronal acetylcholine receptor subunit alpha-4Neuronal acetylcholine receptor subunit alpha-7Neuronal acetylcholine receptor subunit beta-2 +10
Waktu ParuhCotinine has a half…
Vol. Distribusi* 2 to 3 L/kg
Klirens* 1.2 L/min [health…
Genetik -
small molecule | CAS: 100-55-0

A direct-acting peripheral vasodilator that causes flushing and may decrease blood pressure. It is used in vasospasm and threatened gangrene. [PubChem]

Kategori:
Cardiovascular AgentsLipid Modifying AgentsLipid Modifying Agents, Plain +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nidufexor DB16255
small molecule | CAS: 1773489-72-7

Nidufexor is under investigation in clinical trial NCT03804879 (Safety, Tolerability and Efficacy of LMB763 in Patients With Diabetic Nephropathy).

Target Protein:
Bile acid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nifedipine Approved DB01115
small molecule | CAS: 21829-25-4

Nifedipine, or BAY a 1040, is a first generation dihydropyridine L-type calcium channel blocker, similar to [nicardipine].[A190210,A190273,A175390,L11383] Nifedipine was developed by Bayer and first described in the literature, along with other dihydropyridin…

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsAntihypertensive Agents +57
Target Protein:
Voltage-dependent L-type calcium channel subunit alpha-1CVoltage-dependent L-type calcium channel subunit alpha-1DVoltage-dependent L-type calcium channel subunit beta-2 +5
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe steady state vo…
KlirensThe total body clea…
Genetik -
Nifekalant DB16008
small molecule | CAS: 130636-43-0

Nifekalant is under investigation in clinical trial NCT03855826 (Evaluation of the Efficacy and Safety of Nifekalant Hydrochloride (NIF) Injection).

Kategori:
Antiarrhythmic agentsCardiovascular AgentsPyrimidines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nifenazone DB13407
small molecule | CAS: 2139-47-1

Deskripsi belum tersedia.

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +16
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nifuratel DB13724
small molecule | CAS: 4936-47-4

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAntifungal AgentsAntiparasitic Agents +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nifuroxazide DB13855
small molecule | CAS: 965-52-6

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAlimentary Tract and MetabolismAnti-Infective Agents +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nifurpirinol DB11436
small molecule | CAS: 13411-16-0

Deskripsi belum tersedia.

Kategori:
FuransNitro Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nifurtimox Approved DB11820
small molecule | CAS: 23256-30-6

Chagas disease, caused by a parasite known as Trypanosoma cruzi (T.cruzi), is a vector-transmitted disease affecting animals and humans in the Americas. It is commonly known as American Trypanosomiasis.[L15366] The CDC estimates that approximately 8 millio…

Kategori:
Agents Against Leishmaniasis and TrypanosomiasisAnti-Infective AgentsAntiparasitic Agents +11
Target Protein:
NitroreductasesGlyceraldehyde-3-phosphate dehydrogenase, glycosomal
Waktu ParuhThe elimination hal…
Vol. DistribusiNifurtimox crosses …
KlirensOne pharmacokinetic…
Genetik -
Nifurtoinol DB13730
small molecule | CAS: 1088-92-2

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAnti-Infective Agents, UrinaryAntibacterials for Systemic Use +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nifurzide DB13325
small molecule | CAS: 39978-42-2

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismAntidiarrheals, Intestinal Antiinflammatory/antiinfective AgentsFurans +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nigericin DB14056
small molecule | CAS: 28380-24-7

A polyether antibiotic which affects ion transport and ATPase activity in mitochondria. It is produced by Streptomyces hygroscopicus. (From Merck Index, 11th ed)

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsCompounds used in a research, industrial, or household setting +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Niguldipine DB09239
small molecule | CAS: 113165-32-5

Niguldipine is a calcium channel blocker drug (CCB) with a1-adrenergic antagonist properties.

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +17
Target Protein:
Alpha-1A adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nikethamide DB13655
small molecule | CAS: 59-26-7

Deskripsi belum tersedia.

Kategori:
Central Nervous System AgentsCentral Nervous System StimulantsConvulsants +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nikkomycin Z DB12939
small molecule | CAS: 59456-70-1

Nikkomycin Z has been used in trials studying the treatment and basic science of Coccidioidomycosis.

Kategori:
Anti-Infective AgentsAntifungal AgentsCarbohydrates +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nilotinib Approved DB04868
small molecule | CAS: 641571-10-0

Nilotinib, also known as AMN107, is a tyrosine kinase inhibitor under investigation as a possible treatment for chronic myelogenous leukemia (CML). A Phase I clinical trial in 2006 showed that this drug was relatively safe and offered significant therapeutic …

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBcr-Abl Tyrosine Kinase Inhibitors +39
Target Protein:
Tyrosine-protein kinase ABL1Mast/stem cell growth factor receptor Kit
Gen Terkait:
UGT1A1
Waktu Paruh15 hours
Vol. Distribusi-
Klirens-
Genetik 1 Varian
Nilutamide Approved DB00665
small molecule | CAS: 63612-50-0

Nilutamide is an antineoplastic hormonal agent primarily used in the treatment of prostate cancer. Nilutamide is a pure, nonsteroidal anti-androgen with affinity for androgen receptors (but not for progestogen, estrogen, or glucocorticoid receptors). Conseque…

Kategori:
Androgen Receptor AntagonistsAndrogen Receptor InhibitorsAntiandrogens +18
Target Protein:
Androgen receptor
Waktu Paruh38.0-59.1 hours
Vol. Distribusi-
Klirens-
Genetik -
Nilvadipine Approved DB06712
small molecule | CAS: 75530-68-6

Nilvadipine is a calcium channel blocker (CCB) for the treatment of hypertension.

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsAntihypertensive Agents +27
Target Protein:
Voltage-dependent L-type calcium channel subunit alpha-1CVoltage-dependent calcium channel subunit alpha-2/delta-1Voltage-dependent L-type calcium channel subunit beta-2 +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nimacimab DB15115
biotech | CAS: 2098636-09-8

Nimacimab is under investigation in clinical trial NCT03261739 (Safety Tolerability, and PK of RYI-018 After Repeat Dosing in Subjects With Non-Alcoholic Fatty Liver Disease (NAFLD)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nimesulide Approved DB04743
small molecule | CAS: 51803-78-2

Nimesulide is a relatively COX-2 selective, non-steroidal anti-inflammatory drug (NSAID) with analgesic and antipyretic properties. Its approved indications are the treatment of acute pain, the symptomatic treatment of osteoarthritis and primary dysmenorrhoea…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAmides +25
Target Protein:
Prostaglandin G/H synthase 2Tumor necrosis factor ligand superfamily member 10Lactotransferrin +1
Waktu Paruh1.8–4.7 hours
Vol. Distribusi-
Klirens-
Genetik -
Nimodipine Approved DB00393
small molecule | CAS: 66085-59-4

Nimodipine is a 1,4-dihydropyridine calcium channel blocker. It acts primarily on vascular smooth muscle cells by stabilizing voltage-gated L-type calcium channels in their inactive conformation. By inhibiting the influx of calcium in smooth muscle cells, nim…

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsAntihypertensive Agents +19
Target Protein:
Voltage-dependent L-type calcium channel subunit alpha-1CVoltage-dependent L-type calcium channel subunit alpha-1DVoltage-dependent L-type calcium channel subunit alpha-1F +7
Waktu Paruh1.7-9 hours
Vol. Distribusi-
Klirens-
Genetik -
Nimorazole DB12172
small molecule | CAS: 6506-37-2

Nimorazole has been used in trials studying the treatment of Hypoxia, Radiotherapy, Hypoxic Modification, Gene Profile, Gene Signature, and Head and Neck Squamous Cell Carcinoma, among others.

Kategori:
Anti-Infective AgentsAntiparasitic AgentsAntiparasitic Products, Insecticides and Repellents +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nimotuzumab DB06192
biotech | CAS: 780758-10-3

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nimustine DB13069
small molecule | CAS: 42471-28-3

Nimustine has been used in trials studying the treatment of Glioblastoma.

Kategori:
Alkylating DrugsAmidesAntineoplastic Agents +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ningetinib DB16256
small molecule | CAS: 1394820-69-9

Ningetinib is under investigation in clinical trial NCT03758287 (Ningetinib (CT053PTSA) Plus Gefitinib in Stage IIIB or IV NSCLC Patients With EGFR Mutation and T790M Negative).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nintedanib Approved DB09079
small molecule | CAS: 656247-17-5

Nintedanib is a small molecule kinase inhibitor used in the treatment of pulmonary fibrosis, systemic sclerosis-associated interstitial lung disease, and non-small cell lung cancer (NSCLC).[L8453,L8459] It was first approved for use in the United States in 20…

Kategori:
Antifibrotic AgentsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +14
Target Protein:
Vascular endothelial growth factor receptor 1Vascular endothelial growth factor receptor 2Vascular endothelial growth factor receptor 3 +9
Waktu ParuhThe terminal elimin…
Vol. DistribusiNintedanib appears …
KlirensNintedanib is has a…
Genetik -
Niobium DB13031
small molecule | CAS: 7440-03-1

Niobium has been used in trials studying the treatment of Obesity and Overweight.

Kategori:
ElementsMetalsMetals, Heavy +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NIP-292 DB18055
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Menampilkan 10751–10800 dari 15718
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