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11778

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8554 (72.6%)
Target
6383 (54.2%)
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96 (0.8%)
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11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 213 / 236
small molecule | CAS: 165942-79-0

Technetium Tc-99m nofetumomab merpentan (Tc-99m nm) consists of a Fab fragment of an IgG2b of the pancarcinoma murine antibody NR-LU-10.[A32115] The NR-LU-10 antibody is directed against a 40 kDa glycoprotein antigen expressed in a variety of cancers and some…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Target Protein:
Epithelial cell adhesion moleculeB-lymphocyte antigen CD20
Waktu ParuhThe radioactive hal…
Vol. Distribusi-
Klirens-
Genetik -
Technetium Tc-99m oxidronate Approved DB09139
small molecule | CAS: 72945-61-0

Technetium Tc-99m oxidronate, also known as 99mTc-methylene diphosphonate, is a radiopharmaceutical agent. A radiopharmaceutical is defined as a medicinal formulation containing radioisotopes that are used in major clinical areas for diagnosis and/or therapy.…

Kategori:
Diagnostic RadiopharmaceuticalsDrugs that are Mainly Renally ExcretedOrganometallic Compounds +6
Waktu ParuhThe elimination of …
Vol. DistribusiThe distribution of…
KlirensDuring the first 24…
Genetik -
small molecule | CAS: 52997-54-3

A radionuclide imaging agent used primarily in scintigraphy or tomography of the heart to evaluate the extent of the necrotic myocardial process. It has also been used in noninvasive tests for the distribution of organ involvement in different types of amyloi…

Kategori:
AcidsAcids, NoncarboxylicCompounds used in a research, industrial, or household setting +17
Target Protein:
HydroxyapatiteAmorphous calcium phosphate
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Technetium Tc-99m red blood cells is a radiopharmaceutical diagnostic agent that is intravenously administered to be used in blood pool imaging, including cardiac first pass and gated equilibrium imaging and for detection of sites of gastrointestinal bleeding…

Kategori:
Radioactive Diagnostic AgentRadiopharmaceutical Activity
Waktu ParuhTechnetium Tc 99m d…
Vol. DistribusiFollowing intraveno…
Klirens-
Genetik -
Technetium Tc-99m sestamibi Approved DB09161
small molecule | CAS: 109581-73-9

Technetium Tc-99m sestamibi (commonly sestamibi) is a pharmaceutical agent used in nuclear medicine imaging. The drug is a coordination complex consisting of the radioisotope technetium-99m bound to six methoxyisobutylisonitrile (MIBI) ligands, hence the name…

Kategori:
Compounds used in a research, industrial, or household settingDiagnostic RadiopharmaceuticalsDiagnostic Uses of Chemicals +10
Waktu ParuhTechnetium Tc 99m d…
Vol. Distribusi-
KlirensThe effective half-…
Genetik -
Technetium Tc-99m succimer Approved DB09436
small molecule | CAS: 65438-08-6

Technetium Tc-99m (<sup>99m</sup>Tc) succimer, also known as technetium Tc-99m dimercaptosuccinic acid (DMSA),[A245643] is a radioactive diagnostic agent used to evaluate functional renal tissue and tubular function in patients with renal parenchymal disorder…

Kategori:
Acids, AcyclicCompounds used in a research, industrial, or household settingDiagnostic Radiopharmaceuticals +14
Waktu ParuhTechnetium Tc-99m d…
Vol. DistribusiThere is no informa…
KlirensThere is no informa…
Genetik -
small molecule

Technetium 99m sulfur colloid is a radiopharmaceutical diagnostic agent used in the evaluation of various conditions including lymph node metastases in breast cancer, detection of shunt patency, imaging of reticuloendothelial cells for assessment of liver fun…

Kategori:
Compounds used in a research, industrial, or household settingDiagnostic RadiopharmaceuticalsDiagnostic Uses of Chemicals +9
Waktu ParuhTechnetium Tc 99m d…
Vol. DistribusiFollowing oral inge…
Klirens-
Genetik -
small molecule | CAS: 127455-27-0

Technetium Tc-99m tetrofosmin is a drug used in nuclear myocardial perfusion imaging. The radioisotope, technetium-99m, is chelated by two 1,2-bis[di-(2-ethoxyethyl)phosphino]ethane ligands which belong to the group of diphosphines and which are referred to a…

Kategori:
Compounds used in a research, industrial, or household settingDiagnostic RadiopharmaceuticalsDiagnostic Uses of Chemicals +7
Waktu ParuhTechnetium-99m tetr…
Vol. DistribusiReports have shown …
KlirensTechnetium-99m tetr…
Genetik -
small molecule | CAS: 1262984-82-6

Technetium Tc-99m tilmanocept is a radiopharmaceutical diagnostic imaging agent approved by the U.S. Food and Drug Administration (FDA) for the imaging of lymph nodes with or without scintigraphic imaging. It is a macromolecule consisting of multiple units of…

Kategori:
Diagnostic RadiopharmaceuticalsRadioactive Diagnostic AgentRadiopharmaceutical Activity +2
Target Protein:
Macrophage mannose receptor 1
Waktu ParuhTechnetium Tc99m ti…
Vol. Distribusi-
KlirensIn dose-ranging cli…
Genetik -
small molecule | CAS: 1333204-77-5

Deskripsi belum tersedia.

Kategori:
Organometallic Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Teclistamab Approved DB16655
biotech | CAS: 2119595-80-9

Teclistamab is an IgG4-PAA bispecific antibody that targets the CD3 receptor expressed on the surface of T cells and B cell maturation antigen (BCMA) expressed on malignant multiple myeloma cells.[A253587] Teclistamab consists of an anti-BCMA arm and an anti-…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntineoplastic Agents +8
Target Protein:
T-cell surface glycoprotein CD3Tumor necrosis factor receptor superfamily member 17
Waktu ParuhBased on non-compar…
Vol. DistribusiThe mean (CV%) volu…
KlirensTeclistamab exhibit…
Genetik -
Teclozan DB13205
small molecule | CAS: 5560-78-1

Teclozan is an antiprotozoal agent employed typically as a therapy to treat protozoan infections.

Kategori:
AminesAntiparasitic Products, Insecticides and RepellentsAntiprotozoals +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tecovirimat Approved DB12020
small molecule | CAS: 869572-92-9

The World Health Organization declared smallpox, a contagious and sometimes fatal infectious disease, eradicated in 1980. However, there have been longstanding concerns that smallpox may be used as a bioweapon.[A35133,L3614] Tecovirimat is an antiviral drug t…

Kategori:
Acids, CarbocyclicAmidesAnti-Infective Agents +27
Target Protein:
Envelope protein F13
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe clearance rate …
Genetik -
Tedizolid Approved DB14569
small molecule | CAS: 856866-72-3

Drug-resistant bacteria, such as methicillin-resistant _Staphylococcus aureus_, vancomycin-resistant _Enterococcus faecium_, and penicillin-resistant _Streptococcus penumoniae_, represent a massive public health threat.[A199086, A199131] Tedizolid is a member…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibacterials for Systemic Use +5
Target Protein:
23S ribosomal RNA
Waktu ParuhTedizolid has a hal…
Vol. DistribusiThe volume of distr…
KlirensTedizolid has an ap…
Genetik -
Tedizolid phosphate Approved DB09042
small molecule | CAS: 856867-55-5

Drug-resistant bacteria, such as methicillin-resistant _Staphylococcus aureus_, vancomycin-resistant _Enterococcus faecium_, and penicillin-resistant _Streptococcus penumoniae_, represent a massive public health threat.[A199086, A199131] Tedizolid is a member…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntidepressive Agents +10
Target Protein:
23S ribosomal RNA
Waktu ParuhTedizolid has a hal…
Vol. DistribusiThe volume of distr…
KlirensTedizolid has an ap…
Genetik -
Teduglutide Approved DB08900
biotech | CAS: 197922-42-2

Teduglutide is a glucagon-like peptide-2 (GLP-2) analogue. It is made up of 33 amino acids and is manufactured using a strain of Escherichia coli modified by recombinant DNA technology. Teduglutide differs from GLP-2 by one amino acid (alanine is substituted …

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsAnalogs/Derivatives +15
Target Protein:
Glucagon-like peptide 2 receptor
Waktu ParuhTerminal half-life,…
Vol. DistribusiVd, healthy subject…
KlirensPlasma clearance, h…
Genetik -
Tefibazumab DB16378
biotech | CAS: 521079-87-8

Tefibazumab is under investigation in clinical trial NCT00198289 (Aurexis® in Cystic Fibrosis Subjects Chronically Colonized With Staphylococcus Aureus in Their Lungs).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2143580-10-1

Tefidsogene civaparvovec, formerly known as SB-913, is an investigational therapy for genome editing. It consists of an adeno-associated virus (AAV) type 2/6 vector and a zinc finger nuclease (ZFN) system that inserts a correct copy of the Iduronate 2-Sulfata…

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tefinostat DB15321
small molecule | CAS: 914382-60-8

Tefinostat is under investigation in clinical trial NCT02759601 (Dose Escalation Trial of Tefinostat for Cancer Associated Inflamation in Hepatocellular Carcinoma (HCC)).

Kategori:
AmidesAminesAniline Compounds +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tegafur Approved DB09256
small molecule | CAS: 17902-23-7

Tegafur (INN, BAN, USAN) is a prodrug of [DB00544] (5-FU), an antineoplastic agent used as the treatment of various cancers such as advanced gastric and colorectal cancers. It is a pyrimidine analogue used in combination therapies as an active chemotherapeuti…

Kategori:
AntimetabolitesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +22
Target Protein:
Thymidylate synthase
Gen Terkait:
DPYD DPYD DPYD +4
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensNo pharmacokinetic …
Genetik 7 Varian
Tegafur-uracil Approved DB09327
small molecule | CAS: 74578-38-4

Tegafur-uracil is an anti-tumor compound containing tegafur (1-(2-tetrahydrofuryl)-5-fluorouracil) and uracil in a molar ratio of 1:4. It was developed as an anti-cancer therapy by Taiho Pharmaceutical Co Ltd.[A32073] It is approved in different countries but…

Kategori:
Cytochrome P-450 CYP2A6 SubstratesCytochrome P-450 Substrates
Target Protein:
Dihydropyrimidine dehydrogenase [NADP(+)]Thymidylate synthaseRNA +1
Waktu ParuhThe presence of ura…
Vol. DistribusiThe volume of distr…
KlirensThe reported cleara…
Genetik -
Tegaserod Approved DB01079
small molecule | CAS: 145158-71-0

Novartis' brand name Zelnorm (tegaserod) had originally received approval from the US FDA in 2002 for the treatment of irritable bowel syndrome with constipation (IBS-C).[L5918,F4229] It was, however, voluntarily withdrawn from widespread use in the US market…

Kategori:
Alimentary Tract and MetabolismAntidepressive AgentsBCRP/ABCG2 Substrates +25
Target Protein:
5-hydroxytryptamine receptor 45-hydroxytryptamine receptor 2C5-hydroxytryptamine receptor 2A +1
Waktu ParuhThe mean terminal e…
Vol. DistribusiAlthough tegaserod …
KlirensAlthough tegaserod …
Genetik -
Tegavivint DB17109
small molecule | CAS: 1227637-23-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tegobuvir DB11852
small molecule | CAS: 1000787-75-6

Tegobuvir has been investigated for the treatment of Hepatitis C, Chronic.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Genome polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tegoprubart DB16974
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TEL540-548 DB17461
biotech

TEL540-548 is a recombinant peptide consisting of the amino acid residues 540 to 548 of the human telomerase reverse transcriptase (hTERT).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Telacebec DB17754
small molecule | CAS: 1334719-95-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Telaglenastat DB15232
small molecule | CAS: 1439399-58-2

Telaglenastat is under investigation in clinical trial NCT02071862 (Study of the Glutaminase Inhibitor CB-839 in Solid Tumors).

Kategori:
AcetamidesAmidesBenzene Derivatives +2
Target Protein:
Glutaminase kidney isoform, mitochondrialGlutaminase liver isoform, mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Telaprevir Approved DB05521
small molecule | CAS: 402957-28-2

Telaprevir is a direct acting antiviral medication used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV). HCV is a single-stranded RNA virus that is categorized into nine…

Kategori:
Amino Acids, Peptides, and ProteinsAntiinfectives for Systemic UseAntiviral Agents +21
Target Protein:
Genome polyproteinGenome polyproteinSolute carrier organic anion transporter family member 1B1 +1
Waktu ParuhTelaprevir has a ha…
Vol. DistribusiThe estimated appar…
KlirensTelaprevir has an e…
Genetik -
small molecule | CAS: 198414-31-2

Telapristone acetate, an orally-available, selective progesterone receptor modulator, is in development to alleviate symptoms associated with both uterine fibroids and endometriosis.

Kategori:
Fused-Ring CompoundsNorpregnanesNorsteroids +1
Target Protein:
Progesterone receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Telatinib DB15393
small molecule | CAS: 332012-40-5

Telatinib is under investigation in clinical trial NCT03817411 (Telatinib in Combination With Capecitabine/ Oxaliplatin in 1st Line Gastric or GEJ Cancer).

Target Protein:
Vascular endothelial growth factor receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Telavancin Approved DB06402
small molecule | CAS: 372151-71-8

Telavancin is a semi-synthetic derivative of vanocymycin that has bactericidal activity against Methicillin-resistant Staphylococcus aureus (MRSA) and other gram-positive bacteria. MRSA is an important pathogen capable of causing hospital-acquired pneumonia …

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +13
Target Protein:
Neuronal acetylcholine receptor subunit alpha-2Neuronal acetylcholine receptor subunit alpha-3Corticotropin-releasing factor receptor 1
Waktu ParuhTerminal eliminatio…
Vol. DistribusiVss, healthy subjec…
KlirensCl, healthy subject…
Genetik -
Telazorlimab DB16374
biotech | CAS: 2126777-87-3

Telazorlimab is under investigation in clinical trial NCT03568162 (Phase 2b Study to Evaluate the Efficacy and Safety of ISB 830 in Adults With Moderate to Severe Atopic Dermatitis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Telbermin DB12639
biotech | CAS: 205887-54-3

Telbermin has been used in trials studying the treatment of Foot Ulcer, Foot Ulcer, Diabetic, and Amyotrophic Lateral Sclerosis.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Telcagepant DB12228
small molecule | CAS: 781649-09-0

Telcagepant has been investigated for the treatment of Migraine. It is an antagonist of the receptor for calcitonin gene-related peptide (CGRP), a primary neuropeptide involved in the pathophysiology of migraine. CGRP and its receptors are found in areas of t…

Target Protein:
Calcitonin gene-related peptide type 1 receptorCalcitonin gene-related peptide 1Calcitonin gene-related peptide 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Telinavir DB12178
small molecule | CAS: 143224-34-4

Telinavir has been used in trials studying the treatment of HIV Infections.

Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Telisotuzumab DB14838
biotech | CAS: 1781223-80-0

Telisotuzumab is under investigation in clinical trial NCT01472016 (Study of ABT-700 in Subjects With Advanced Solid Tumors).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1714088-51-3

Telisotuzumab vedotin is under investigation in clinical trial NCT02099058 (A Study Evaluating the Safety, Pharmacokinetics (PK), and Preliminary Efficacy of ABBV-399 in Subjects With Advanced Solid Tumors.).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Telitacicept DB18312
biotech | CAS: 2136630-26-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsProteinsRecombinant Proteins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Telithromycin Approved DB00976
small molecule | CAS: 191114-48-4

Telithromycin, a semi-synthetic erythromycin derivative, belongs to a new chemical class of antibiotics called ketolides. Ketolides have been recently added to the macrolide-lincosamide-streptogramin class of antibiotics. Similar to the macrolide antibiotics,…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibacterials for Systemic Use +23
Target Protein:
23S ribosomal RNA
Waktu ParuhMain elimination ha…
Vol. Distribusi* 2.9 L/kg
Klirens-
Genetik -
Telmisartan Approved DB00966
small molecule | CAS: 144701-48-4

Telmisartan is an angiotensin II receptor antagonist (ARB) used in the management of hypertension. Generally, angiotensin II receptor blockers (ARBs) such as telmisartan bind to the angiotensin II type 1 (AT1) receptors with high affinity, causing inhibition …

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing angioedemaAgents causing hyperkalemia +24
Target Protein:
Peroxisome proliferator-activated receptor gammaType-1 angiotensin II receptor
Waktu ParuhTelmisartan display…
Vol. DistribusiTelmisartan has a v…
KlirensTelmisartan has a t…
Genetik -
Telotristat ethyl Approved DB12095
small molecule | CAS: 1033805-22-9

Telotristat ethyl is a prodrug of telotristat that was approved by the FDA in March 2017 as Xermelo.[L43342] It was previously referred to as telotristat etiprate, the hippurate salt form; however, the FDA recommends the use of the name of the neutral form ra…

Kategori:
AntidiarrhealsCytochrome P-450 CYP2B6 InducersCytochrome P-450 CYP2B6 Inducers (strength unknown) +20
Target Protein:
Tryptophan 5-hydroxylase 2Tryptophan 5-hydroxylase 1
Waktu ParuhFollowing a single …
Vol. DistribusiThe estimated appar…
KlirensThe apparent total …
Genetik -
Temazepam Approved DB00231
small molecule | CAS: 846-50-4

Temazepam, like many other similar and related benzodiazepines, acts as a gamma-aminobutyric acid (GABA) modulator and is capable of eliciting a variety of actions including sedation, hypnosis, skeletal muscle relaxation, anticonvulsant activity, and anxiolyt…

Kategori:
Anti-Anxiety AgentsBenzazepinesBenzodiazepine hypnotics and sedatives +18
Target Protein:
Translocator proteinGABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe volume of distr…
KlirensStudies regarding t…
Genetik -
small molecule | CAS: 18818-64-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Temelimab DB15634
biotech | CAS: 1393641-34-3

Temelimab is under investigation in clinical trial NCT02782858 (Clinical Trial Assessing the HERV-W Env Antagonist Gnbac1 for Efficacy in MS).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Temocapril DB08836
small molecule | CAS: 111902-57-9

Temocapril is a prodrug-type angiotensin-I converting enzyme (ACE) inhibitor not approved for use in the United States, but is approved in Japan and South Korea. Temocapril can also be used in hemodialysis patients without risk of serious accumulation.

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing angioedemaAgents causing hyperkalemia +9
Target Protein:
Angiotensin-converting enzyme
Waktu Paruh13.1 hours in patie…
Vol. Distribusi-
Klirens19.4% urinary recov…
Genetik -
Temocillin Approved DB12343
small molecule | CAS: 66148-78-5

Temocillin has been investigated in Infection, Liver Dysfunction, and Urinary Tract Infection.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Temozolomide Approved DB00853
small molecule | CAS: 85622-93-1

Refractory anaplastic astrocytoma (WHO grade III) and Glioblastoma multiforme (WHO grade IV) are primary malignant brain tumours with poor prognosis and limited treatment options. Despite considerable genetic heterogeneity, these tumours often have impaired D…

Kategori:
Alkylating ActivityAlkylating DrugsAntineoplastic Agents +13
Target Protein:
DNA
Waktu ParuhTemozolomide has a …
Vol. DistribusiTemozolomide has a …
KlirensTemozolomide has a …
Genetik -
Temsavir DB14675
small molecule | CAS: 701213-36-7

Deskripsi belum tersedia.

Kategori:
HIV Fusion Inhibitors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Temsirolimus Approved DB06287
small molecule | CAS: 162635-04-3

Temsirolimus is a derivative of sirolimus used in the treatment of renal cell carcinoma (RCC). It was developed by Wyeth Pharmaceuticals under the trade name Torisel. Temsirolimus was approved by the FDA in late May 2007 as well as the European Medicines Agen…

Kategori:
Agents causing angioedemaAnti-Bacterial AgentsAntineoplastic Agents +32
Target Protein:
Serine/threonine-protein kinase mTOR
Waktu ParuhTemsirolimus exhibi…
Vol. Distribusi172 L in whole bloo…
Klirens16.2 L/h (22%)
Genetik -
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