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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
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14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 212 / 282
Pelitrexol DB12757
small molecule | CAS: 446022-33-9

Pelitrexol has been used in trials studying the treatment of Unspecified Adult Solid Tumor, Protocol Specific.

Kategori:
Sulfur Compounds
Target Protein:
Trifunctional purine biosynthetic protein adenosine-3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pelubiprofen DB12150
small molecule | CAS: 69956-77-0

Pelubiprofen has been investigated for the treatment of Chronic Back Pain.

Kategori:
Acids, Carbocyclic
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pemafibrate DB15212
small molecule | CAS: 848259-27-8

Pemafibrate is under investigation in clinical trial NCT03350165 (A Study of Pemafibrate in Patients With Nonalcoholic Fatty Liver Disease (NAFLD)).

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +6
Target Protein:
Peroxisome proliferator-activated receptor alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pembrolizumab Approved DB09037
biotech | CAS: 1374853-91-4

Pembrolizumab is a highly selective IgG4-kappa humanized monoclonal antibody against PD-1 receptors. It was generated by grafting the variable sequences of a very high-affinity mouse antihuman PD-1 antibody onto a human IgG4-kappa isotype containing a stabili…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +18
Target Protein:
Programmed cell death protein 1Programmed cell death 1 ligand 1
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe steady-state vo…
KlirensClearance is modera…
Genetik -
Pemetrexed Approved DB00642
small molecule | CAS: 137281-23-3

Pemetrexed is a chemotherapy drug that is manufactured and marketed by Eli Lilly and Company under the brand name Alimta. It is indicated for use in combination with cisplatin for the treatment of patients with malignant pleural mesothelioma whose disease is …

Kategori:
Amino AcidsAmino Acids, AcidicAmino Acids, Dicarboxylic +19
Target Protein:
Thymidylate synthaseThymidylate synthaseBifunctional purine biosynthesis protein ATIC +2
Waktu ParuhThe elimination hal…
Vol. DistribusiPemetrexed has a st…
KlirensThe total systemic …
Genetik -
Pemigatinib Approved DB15102
small molecule | CAS: 1513857-77-6

Pemigatinib is a small molecule kinase inhibitor with antitumour activity. It works by inhibiting fibroblast growth factor receptors (FGFRs), which are receptor tyrosine kinases that activate signalling pathways in tumour cells.[A193719] FGFRs gained attentio…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Substrates +16
Target Protein:
Fibroblast growth factor receptor 1Fibroblast growth factor receptor 2Fibroblast growth factor receptor 3 +1
Waktu ParuhFollowing administr…
Vol. DistribusiThe apparent volume…
KlirensFollowing administr…
Genetik -
Pemirolast Approved DB00885
small molecule | CAS: 69372-19-6

Pemirolast potassium is a slightly yellow powder that is soluble in water. It is a mast cell stabilizer that acts as an antiallergic agent. As an ophthalmic aqueous sterile solution, pemirolast is used for the prevention of itching of the eyes caused by aller…

Kategori:
Decreased Histamine ReleaseHistamine AgentsMast Cell Stabilizers +3
Target Protein:
Histamine H1 receptor
Waktu Paruh4.5 hours (Ophthalm…
Vol. Distribusi-
Klirens-
Genetik -
Pemivibart DB18720
biotech | CAS: 2858673-18-2

Pemivibart (Pemgarda) is a human IgG1 monoclonal antibody targeting the SARS-CoV-2 spike protein receptor binding domain.[L50326] It received emergency use authorization (EUA) from the FDA in March 2024 for pre-exposure prophylaxis (PrEP) of COVID-19 in certa…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalApproved Treatments for COVID-19 +4
Target Protein:
Spike glycoprotein
Waktu ParuhPemivibart has an e…
Vol. DistribusiFollowing the admin…
KlirensFollowing the admin…
Genetik -
biotech

Pemlimogene merolisbac is under investigation in clinical trial NCT03371381 (An Efficacy and Safety Study of JNJ-64041757, a Live Attenuated Listeria Monocytogenes Immunotherapy, in Combination With Nivolumab Versus Nivolumab Monotherapy in Participants With …

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pemoline Approved DB01230
small molecule | CAS: 2152-34-3

In 2005, the Food and Drug Administration (FDA) withdrew approval for pemoline. In March 2005, Abbott Laboratories (Cylert marketer) had discontinued the production of Cylert arguing economic reasons.

Kategori:
Central Nervous System AgentsCentral Nervous System StimulantsCentrally Acting Sympathomimetics +4
Waktu ParuhThe serum half-life…
Vol. Distribusi-
Klirens-
Genetik -
Pemrametostat DB19170
small molecule | CAS: 1616392-22-3

Pemrametostat is under investigation in clinical trial NCT03614728 (Study to Investigate the Safety and Clinical Activity of GSK3326595 and Other Agents to Treat Myelodysplastic Syndrome (MDS) and Acute Myeloid Leukemia (AML)).

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-Ring
Target Protein:
Protein arginine N-methyltransferase 5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pemvidutide DB18998
biotech | CAS: 2538014-94-5

Pemvidutide is under investigation in clinical trial NCT05989711 (Efficacy and Safety of Pemvidutide in Subjects With Nonalcoholic Steatohepatitis (NASH) (IMPACT Trial)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PEN-866 DB16186
small molecule | CAS: 1472614-83-7

PEN-866 is under investigation in clinical trial NCT03221400 (PEN-866 in Patients With Advanced Solid Malignancies).

Target Protein:
DNA topoisomerase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Penbutolol Approved DB01359
small molecule | CAS: 38363-40-5

Penbutolol is a drug in the beta-blocker class used to treat hypertension. Penbutolol binds both beta-1 and beta-2 adrenergic receptors, rendering it a non-selective beta-blocker. Penbutolol can act as a partial agonist at beta adrenergic receptors, since it …

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-Antagonists +23
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptor5-hydroxytryptamine receptor 1A +1
Waktu ParuhPlasma= approximate…
Vol. Distribusi-
KlirensApproximately 90% o…
Genetik -
Penciclovir Approved DB00299
small molecule | CAS: 39809-25-1

Penciclovir is a synthetic acyclic guanine derivative with antiviral activity used for the treatment of various herpes simplex virus (HSV) infections. Displaying low toxicity and good selectivity, penciclovir is a nucleoside analogue.

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +12
Target Protein:
Thymidine kinase, cytosolicDNA polymerase catalytic subunitThymidine kinase
Waktu Paruh2 hours
Vol. Distribusi-
Klirens-
Genetik -
Penclomedine DB12987
small molecule | CAS: 108030-77-9

Penclomedine has been used in trials studying the treatment of Lymphoma and Unspecified Adult Solid Tumor, Protocol Specific.

Kategori:
Antineoplastic AgentsPyridines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 87827-02-9

Penequinine, Penehyclidine is under investigation in clinical trial NCT02644876 (Preventive Effects of Penehyclidine Hydrochloride Inhalation on Postoperative Pulmonary Complications).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Penfluridol DB13791
small molecule | CAS: 26864-56-2

Deskripsi belum tersedia.

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsAntipsychotic Agents +20
Target Protein:
Voltage-dependent T-type calcium channel subunit alpha-1G
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Penicillamine Approved DB00859
small molecule | CAS: 52-67-5

Penicillamine is a pharmaceutical of the chelator class. The pharmaceutical form is D-penicillamine, as L-penicillamine is toxic (it inhibits the action of pyridoxine). It is an ?-amino acid metabolite of penicillin, although it has no antibiotic properties.

Kategori:
Agents Causing Muscle ToxicityAmino AcidsAmino Acids, Peptides, and Proteins +16
Target Protein:
Copper
Waktu Paruh1 hour
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Agents causing hyperkalemia
Target Protein:
Regulatory protein BlaR1Beta-lactam-inducible penicillin-binding protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Penicillium digitatum Approved DB11023
biotech

Penicillium digitatum allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Penicillium roqueforti Approved DB10812
biotech

Penicillium roqueforti is a fungus which can provoke allergic reactions. Penicillium roqueforti extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Penimepicycline DB13264
small molecule | CAS: 4599-60-4

Penimepicycline is a tetracycline-class antibiotic. It is mentioned on List A produced by the Government of Canada, which is a list of antimicrobial active pharmaceutical ingredients [L2791]. In the classification of the active ingredients included on this li…

Kategori:
Agents that produce neuromuscular block (indirect)AmidesAnti-Bacterial Agents +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Penpulimab DB16747
biotech | CAS: 2350298-92-7

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pentaerithrityl DB13526
small molecule | CAS: 115-77-5

Deskripsi belum tersedia.

Kategori:
AlcoholsAlimentary Tract and MetabolismDrugs for Constipation +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pentaerythritol tetranitrate Approved DB06154
small molecule | CAS: 78-11-5

Pentaerythritol tetranitrate is the nitrate ester of pentaerythritol that possesses explosive properties. When mixed with a plasticizer, this chemical forms a plastic explosive. It is recognized by the FDA to be a coronary vasodilator in the treatment of hear…

Kategori:
AlcoholsAntianginal AgentsCarbohydrates +11
Target Protein:
Hemoglobin subunit alphaHemoglobin subunit betaFree radicals
Waktu ParuhThe elimination hal…
Vol. DistribusiThe steady-state vo…
KlirensIn a pharmacokineti…
Genetik -
Pentagastrin Approved DB00183
small molecule | CAS: 5534-95-2

A synthetic pentapeptide that mimics the actions of endogenous gastrin when given parenterally. It works by stimulating the secretion of gastric acid, pepsin, and intrinsic factor. It has also been used as a diagnostic aid.

Kategori:
Amino Acids, Peptides, and ProteinsDiagnostic AgentsGastrins +8
Target Protein:
Gastrin/cholecystokinin type B receptor
Waktu Paruh10 minutes or less
Vol. Distribusi-
Klirens-
Genetik -
Pentaglobin DB15865
biotech | CAS: 97794-27-9

Pentaglobin, also known as IgM-enriched immunoglobulin, falls under a group of polyclonal immunoglobulin preparations.[A220173] It is comprised of [immunoglobulin G (IgG)](https://www.drugbank.ca/drugs/DB00028) and immunoglobulin A (IgA) while also being enri…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pentaglyme DB02580
small molecule | CAS: 1191-87-3

Deskripsi belum tersedia.

Target Protein:
Profilin-2Restriction endonuclease R.BpuJICytochrome c-552 +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pentanal DB01919
small molecule | CAS: 110-62-3

Pentanal is a solid. This compound belongs to the polyamines. These are compounds containing more than one amine group. This drug targets the protein cAMP-dependent protein kinase catalytic subunit alpha.

Target Protein:
cAMP-dependent protein kinase catalytic subunit alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pentapiperium DB19383
small molecule | CAS: 26372-86-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pentastarch Approved DB09111
small molecule | CAS: 9005-27-0

Pentastarch is an artificial colloid (hydroxyethyl starch derivative). Pentastarch is characterized by presenting five hydroxyethyl groups, which signifies an approximate 50% hydroxyethylation. It is sold under the name Pentaspan by Bristol-Myers Squibb and i…

Kategori:
Blood SubstitutesCarbohydratesCompounds used in a research, industrial, or household setting +9
Waktu Paruh~2.5 hours.
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Sulfide dehydrogenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 22537-51-5

Pentavalent Antimony has been investigated for the treatment of Cutaneous Leishmaniasis.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pentazocine Approved DB00652
small molecule | CAS: 359-83-1

The first mixed agonist-antagonist analgesic to be marketed. It is an agonist at the kappa and sigma opioid receptors and has a weak antagonist action at the mu receptor. (From AMA Drug Evaluations Annual, 1991, p97)

Kategori:
Adjuvants, AnesthesiaAgents that reduce seizure thresholdAlkaloids +20
Target Protein:
Sigma non-opioid intracellular receptor 1Mu-type opioid receptorKappa-type opioid receptor
Waktu Paruh2 to 3 hours
Vol. Distribusi-
Klirens-
Genetik -
Pentetic acid Approved DB14007
small molecule | CAS: 67-43-6

Pentetic acid, also known as diethylenetriaminepentaacetic acid (DTPA), is a synthetic polyamino carboxylic acid with eight coordinate bond forming sites that can sequester metal ions and form highly stable DTPA-metal ion complexes. DTPA, along with its calci…

Kategori:
AcetatesAcids, AcyclicAmines +10
Target Protein:
Transuranium elements
Waktu ParuhIn preclinical stud…
Vol. DistribusiThe volume of distr…
KlirensPentetic acid prese…
Genetik -
Pentetrazol DB13415
small molecule | CAS: 54-95-5

Pentetrazol, also known as pentylenetetrazole, is a gamma-aminobutyric acid type A (GABA<sub>A</sub>) receptor antagonist that was approved by the FDA until 1982.[A254437]

Kategori:
AzepinesCentral Nervous System AgentsCentral Nervous System Stimulants +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pentetreotide Approved DB12602
small molecule | CAS: 138661-02-6

Pentetreotide has been used in trials studying the diagnosis of Cushing's syndrome.

Kategori:
AcetatesAcids, AcyclicAmines +20
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Penthienate DB13695
small molecule | CAS: 22064-27-3

Deskripsi belum tersedia.

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAmines +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pentifylline DB13634
small molecule | CAS: 1028-33-7

Deskripsi belum tersedia.

Kategori:
AlkaloidsCytochrome P-450 CYP1A2 SubstratesCytochrome P-450 Substrates +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pentobarbital Approved DB00312
small molecule | CAS: 76-74-4

A short-acting barbiturate that is effective as a sedative and hypnotic (but not as an anti-anxiety) agent and is usually given orally. It is prescribed more frequently for sleep induction than for sedation but, like similar agents, may lose its effectiveness…

Kategori:
Adjuvants, AnesthesiaAnticholinergic AgentsAnticonvulsants +23
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1Gamma-aminobutyric acid receptor subunit alpha-2Gamma-aminobutyric acid receptor subunit alpha-3 +10
Waktu Paruh5 to 50 hours (dose…
Vol. Distribusi-
Klirens-
Genetik -
Pentosan polysulfate Approved DB00686
small molecule | CAS: 37300-21-3

Pentosan polysulfate is a sulfated pentosyl polysaccharide with heparin-like properties.

Kategori:
AnticoagulantsAntivaricose TherapyCarbohydrates +12
Target Protein:
Fibroblast growth factor 2Fibroblast growth factor 1Fibroblast growth factor 4
Waktu Paruh4.8 hours
Vol. Distribusi-
Klirens-
Genetik -
Pentostatin Approved DB00552
small molecule | CAS: 53910-25-1

A potent inhibitor of adenosine deaminase. The drug is effective in the treatment of many lymphoproliferative malignancies, particularly hairy-cell leukemia. It is also synergistic with some other antineoplastic agents and has immunosuppressive activity.

Kategori:
Adenosine Deaminase InhibitorsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +18
Target Protein:
Adenosine deaminase
Waktu Paruh5.7 hours (with a r…
Vol. Distribusi-
Klirens* 68 mL/min/m2
Genetik -
Pentoxifylline Approved DB00806
small molecule | CAS: 6493-05-6

Pentoxifylline (PTX) is a synthetic dimethylxanthine derivative that modulates the rheological properties of blood and also has both anti-oxidant and anti-inflammatory properties.[A226415, L30300] Although originally developed to treat intermittent claudicati…

Kategori:
AlkaloidsAntioxidantsAntiplatelet agents +23
Target Protein:
Adenosine receptor A2aTumor necrosis factorPhosphodiesterase enzymes +2
Waktu ParuhOverall, pentoxifyl…
Vol. DistribusiPentoxifylline has …
KlirensPentoxifylline give…
Genetik -
Pentoxyverine Approved DB11186
small molecule | CAS: 77-23-6

Pentoxyverine, also referred to as carbetapentane, is a non-opioid central acting antitussive with antimuscarinic, anticonvulsant [A32717], and local anesthetic properties. It is an active ingredient in over-the-counter cough suppressants in combination with …

Kategori:
Antitussive AgentsCentral Nervous System AgentsCough and Cold Preparations +2
Target Protein:
Sigma non-opioid intracellular receptor 1Voltage-gated inwardly rectifying potassium channel KCNH2Voltage-gated sodium channel alpha subunit +2
Waktu ParuhThe half-life is 2.…
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Peoniflorin DB16288
small molecule | CAS: 23180-57-6

Peoniflorin is under investigation in clinical trial NCT02878863 (Paeoniflorin Combination of Hepatoprotective Drugs Versus Hepatoprotective Drugs Only for Auto-immune Hepatitis).

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAnti-Inflammatory Agents +8
Target Protein:
Adenosine receptor A1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PEP0101 DB18572
biotech

PEP0101 is a nanocomplex consisting of elastin-like polypeptides and a small interfering RNA (siRNA) designed to down-regulate the expression of EVI1 oncogene in cancer cells.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pepinemab DB15155
biotech | CAS: 2097151-87-4

Pepinemab is under investigation in clinical trial NCT03769155 (VX15/2503 With or Without Ipilimumab and/or Nivolumab in Patients With Resectable Stage IIIB-D Melanoma).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Peppermint oil Approved DB11198
biotech | CAS: 8006-90-4

Extracted from the stem, leaves, and flowers of _Mentha piperita_ L. plant, peppermint oil (Mentha piperita) is a popular essential oil used in aromatherapy for both external and internal use. Mentha piperita is a hybrid of spearmint (Mentha spicata) and wate…

Kategori:
Alimentary Tract and MetabolismAngiospermsAntiemetics +31
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
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