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11778

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Halaman 211 / 236
Taliglucerase alfa Approved DB08876
biotech | CAS: 37228-64-1

Taliglucerase alfa is the recombinant active form of the human lysosomal enzyme, ?-glucocerebrosidase. It was approved in 2012 and is marketed under the name Elelyso for use in patients with type 1 Gaucher's disease.

Kategori:
Alimentary Tract and MetabolismEnzyme Replacement TherapyEnzymes +7
Target Protein:
Glucocerebroside
Waktu ParuhThe half life is be…
Vol. DistribusiThe steady state vo…
KlirensThe systemic cleara…
Genetik -
Talimogene laherparepvec Approved DB13896
biotech | CAS: 1187560-31-1

Talimogene laherparepvec is an oncolytic treatment used in local treatment of unresectable cutaneous, subcutaneous, and nodal lesions in patients with recurrent melanoma. It is a genetically administered herpes simplex virus 1 (HSV-1) that expresses human cyt…

Kategori:
AlphaherpesvirinaeAntineoplastic AgentsAntineoplastic Agents, Immunological +9
Target Protein:
Granulocyte-macrophage colony-stimulating factor
Waktu ParuhReadily accessible …
Vol. DistribusiTalimogene laherpar…
KlirensAlthough readily ac…
Genetik -
Talinolol DB11770
small molecule | CAS: 57460-41-0

Talinolol has been investigated for the basic science of Gastrointestinal Motility Disorder.

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-Antagonists +16
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TALL-104 DB17360
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Talnetant DB06429
small molecule | CAS: 174636-32-9

Talnetant (SB-223,412) is a neurokinin 3 receptor antagonist developed by GlaxoSmithKline, which is being researched for several different functions, primarily for irritable bowel syndrome and as a potential antipsychotic drug for the treatment of schizophren…

Kategori:
Heterocyclic Compounds, Fused-RingReceptors, Neurokinin-3, antagonists & inhibitors
Target Protein:
Neuromedin-K receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Talopram DB09190
small molecule | CAS: 7182-51-6

Talopram is a selective norepinephrine reuptake inhibitor (SNRI) that is structurally similar to citalopram and melitracen. It was researched in the 1960s and 1970s but never marketed.

Kategori:
Adrenergic Uptake InhibitorsAminesAntidepressive Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Talotrexin DB06178
small molecule | CAS: 113857-87-7

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +5
Target Protein:
Folate receptor alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Talquetamab Approved DB16678
biotech | CAS: 2226212-40-2

Talquetamab is a IgG4-PAA bispecific G protein-coupled receptor class C group 5 member D (GPRC5D)-directed CD3 T-cell engager. It consists of two arms - anti-GPRC5D and anti-CD3 arms - linked by two interchain disulfide bonds, each arm comprising a heavy and …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntineoplastic Agents +7
Target Protein:
T-cell surface glycoprotein CD3G-protein coupled receptor family C group 5 member D
Waktu ParuhThe mean (CV%) term…
Vol. DistribusiThe geometric mean …
KlirensTalquetamab clearan…
Genetik -
Talsaclidine DB12287
small molecule | CAS: 147025-53-4

Talsaclidine has been used in trials studying the treatment of Alzheimer Disease.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Talsupram DB09191
small molecule | CAS: 21489-20-3

Talsupram is a selective norepinephrine reuptake inhibitor (NRI). It was under research for the treatment of depression in 1960 and 1970 but it was never marketed. Talsupram presents a similar structure to [citalopram].

Kategori:
Sulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Talviraline DB07885
small molecule | CAS: 163451-80-7

Talviraline has been used in trials studying the treatment of HIV Infections.

Kategori:
Acquired Immunodeficiency SyndromeHeterocyclic Compounds, Fused-Ring
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tamarix gallica pollen Approved DB10725
biotech

Tamarix gallica pollen is the pollen of the Tamarix gallica plant. Tamarix gallica pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tamatinib DB07159
small molecule | CAS: 841290-80-0

Deskripsi belum tersedia.

Target Protein:
Tyrosine-protein kinase SYKProto-oncogene tyrosine-protein kinase receptor Ret
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tamibarotene DB04942
small molecule | CAS: 94497-51-5

Tamibarotene is a novel synthetic retinoid for acute promyelocytic leukaemia (APL). Tamibarotene is currently approved in Japan for treatment of recurrent APL, and is undergoing clinical trials in the United States.

Kategori:
Acids, CarbocyclicBenzene DerivativesNaphthalenes
Target Protein:
Retinoic acid receptor alphaRetinoic acid receptor beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Taminadenant DB18811
small molecule | CAS: 1337962-47-6

Deskripsi belum tersedia.

Target Protein:
Adenosine receptor A2a
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tamnorzatinib DB19201
small molecule | CAS: 1646839-59-9

Tamnorzatinib is under investigation in clinical trial NCT03176277 (A Study of ONO-7475 in Patients With Acute Leukemias).

Target Protein:
Tyrosine-protein kinase MerTyrosine-protein kinase receptor UFO
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tamoxifen Approved DB00675
small molecule | CAS: 10540-29-1

Tamoxifen is a non-steroidal antiestrogen used to treat estrogen receptor positive breast cancers as well as prevent the incidence of breast cancer in high risk populations.[A1025,L7799,L7802] Tamoxifen is used alone or as an adjuvant in these treatments.[L77…

Kategori:
Anti-EstrogensAntineoplastic AgentsAntineoplastic Agents, Hormonal +64
Target Protein:
Estrogen receptorEstrogen receptor betaProtein kinase C +7
Gen Terkait:
CYP2D6 F5
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of ta…
Genetik 2 Varian
biotech | CAS: 2148334-68-1

Tamrintamab pamozirine is an antibody-drug conjugate targeted against DPEP3.

Kategori:
Antibody-drug Conjugates
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tamsulosin Approved DB00706
small molecule | CAS: 106133-20-4

Tamsulosin is a selective alpha-1A and alpha-1B adrenoceptor antagonist that exerts its greatest effect in the prostate and bladder, where these receptors are most common.[Label] It is indicated for the treatment of signs and symptoms of benign prostatic hype…

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +22
Target Protein:
Alpha-1A adrenergic receptorAlpha-1D adrenergic receptorAlpha-1B adrenergic receptor
Waktu ParuhThe half life in fa…
Vol. Distribusi16L after intraveno…
Klirens2.88L/h.[Label]
Genetik -
biotech

Tanacetum cinerariifolium flower allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tanaproget DB04787
small molecule | CAS: 304853-42-7

Tanaproget (NSP-989) is an investigational non-steroidal progestin. It is a high affinity, high efficacy agonist of the progesterone receptor (PR) with a much more selective binding profile relative to most conventional progestins. Because of this tanaproget …

Kategori:
Heterocyclic Compounds, Fused-RingOxazinesReceptors, Progesterone, agonists +1
Target Protein:
Progesterone receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tandamine DB09192
small molecule | CAS: 42408-80-0

Tandamine was researched in 1970s as an antidepressant but was never commercialized. Tandamine is an analog of pirandamine and it acts as a selective serotonin reuptake inhibitor (SSRI).

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tandospirone DB12833
small molecule | CAS: 87760-53-0

Tandospirone has been used in trials studying the treatment of Schizophrenia.

Kategori:
Anti-Anxiety AgentsAntidepressive AgentsCentral Nervous System Agents +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tandutinib DB05465
small molecule | CAS: 387867-13-2

MLN518 is a novel, oral, small molecule designed to inhibit type III receptor tyrosine kinases, including FLT3, (platelet-derived growth-factor receptor) PDGFR and c-KIT. Tyrosine kinases are enzymes involved in several cellular processes and are known to be …

Kategori:
Heterocyclic Compounds, Fused-RingPotential QTc-Prolonging AgentsQTc Prolonging Agents +1
Target Protein:
Receptor-type tyrosine-protein kinase FLT3Platelet-derived growth factor D
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tanespimycin DB05134
small molecule | CAS: 75747-14-7

Tanespimycin, manufactured by Conforma Therapeutics is under development as a small molecule inhibitor of heat shock protein 90 (HSP90). It is developed for the treatment of several types of cancer, solid tumors or chronic myelogenous leukemia.

Kategori:
AmidesHSP90 Heat-Shock Proteins, antagonists & inhibitorsLactams +2
Target Protein:
Heat shock protein HSP 90-alphaHeat shock protein HSP 90-beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tanezumab DB12335
biotech | CAS: 880266-57-9

Tanezumab has been investigated for the treatment of Osteoarthritis, Knee and Neuralgia, Postherpetic.

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsAntibodies +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tanfanercept DB19142
biotech | CAS: 2119738-70-2

Tanfanercept is under investigation in clinical trial NCT06400589 (A Study to Evaluate the Efficacy and Safety of Tanfanercept (HL036) in Dry Eye Disease).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tangerine Approved DB10637
biotech

Tangerine allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Taniborbactam DB16338
small molecule | CAS: 1613267-49-4

Taniborbactam is under investigation in clinical trial NCT03840148 (Safety and Efficacy Study of Cefepime/vnrx-5133 in Patients With Complicated Urinary Tract Infections).

Kategori:
AcidsAcids, NoncarboxylicBoron Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Taniraleucel DB18311
biotech

Deskripsi belum tersedia.

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Vol. Distribusi-
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Genetik -
Tannic acid Approved DB09372
small molecule | CAS: 1401-55-4

Tannic acid is a polyphenolic compound. It is a type of the commercially available tannins. It acts as a weak acid. Tannic acid is found in the nutgalls formed by insects on twigs of certain oak trees (Quercus infectoria and other Quercus species). It is remo…

Kategori:
Benzene DerivativesBiopolymersCompounds used in a research, industrial, or household setting +4
Target Protein:
Anoctamin-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tanomastat DB06276
small molecule | CAS: 179545-77-8

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAntineoplastic AgentsBenzene Derivatives +1
Target Protein:
72 kDa type IV collagenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tanshinone I DB16886
small molecule | CAS: 568-73-0

Deskripsi belum tersedia.

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAnti-Infective Agents +16
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tantalum DB12859
small molecule | CAS: 7440-25-7

Tantalum has been investigated for the treatment and prevention of Osteoarthritis, Knee Osteoarthritis, Intraoperative Bleeding, and Adolescent Idiopathic Scoliosis.

Kategori:
ElementsMetalsMetals, Heavy +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tanzisertib DB11798
small molecule | CAS: 899805-25-5

Tanzisertib has been used in trials studying the treatment of Fibrosis, Discoid Lupus, Pulmonary Fibrosis, Interstitial Lung Disease, and Lung Diseases, Interstitial, among others.

Kategori:
AlcoholsCarbon RadioisotopesCyclohexanes +6
Target Protein:
Mitogen-activated protein kinase 8Mitogen-activated protein kinase 9Mitogen-activated protein kinase 10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tapencarium DB17821
small molecule

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingIndoles
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tapentadol Approved DB06204
small molecule | CAS: 175591-23-8

Tapentadol is a centrally-acting synthetic analgesic with a dual mechanism of action. It is a mu-opioid receptor agonist that also inhibits norepinephrine reuptake.[A260721, A36596] Tapentadol was first approved by the FDA on November 20, 2008. The extende…

Kategori:
Adrenergic AgentsAdrenergic Uptake InhibitorsAnalgesics +25
Target Protein:
Mu-type opioid receptorSodium-dependent noradrenaline transporterKappa-type opioid receptor +2
Waktu ParuhThe terminal half-l…
Vol. DistribusiTapentadol is widel…
KlirensThe total clearance…
Genetik -
Tapinarof Approved DB06083
small molecule | CAS: 79338-84-4

Tapinarof is a novel, first-in-class, small-molecule AhR agonist that is indicated for the treatment of adult psoriasis. It is available as a topical cream to be applied to the affected area once daily.[L41845, A248790] Tapiranof was first discovered as a met…

Kategori:
AntipsoriaticsAntipsoriatics for Topical UseAryl Hydrocarbon Receptor Agonist +11
Target Protein:
Aryl hydrocarbon receptor
Waktu ParuhDue to the insuffic…
Vol. DistribusiThe Vss of tapinaro…
Klirens-
Genetik -
Tapotoclax DB17166
small molecule | CAS: 1883727-34-1

Deskripsi belum tersedia.

Target Protein:
Induced myeloid leukemia cell differentiation protein Mcl-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Taprenepag DB12623
small molecule | CAS: 752187-80-7

Taprenepag has been used in trials studying the treatment of Ocular Hypertension and Glaucoma, Open-Angle.

Kategori:
Acids, AcyclicAmidesFatty Acids +5
Target Protein:
Prostaglandin E2 receptor EP2 subtype
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tarafenacin DB18810
small molecule | CAS: 385367-47-5

Deskripsi belum tersedia.

Target Protein:
Muscarinic acetylcholine receptor M3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Taranabant DB06624
small molecule | CAS: 701977-09-5

Deskripsi belum tersedia.

Kategori:
Cannabinoid Receptor AgonistsCannabinoids and similarsHormones +2
Target Protein:
Cannabinoid receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Taraxacum officinale pollen Approved DB10755
biotech

Taraxacum officinale pollen is the pollen of the Taraxacum officinale plant. Taraxacum officinale pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tarazepide DB06435
small molecule | CAS: 141374-81-4

Deskripsi belum tersedia.

Kategori:
BenzazepinesHeterocyclic Compounds, Fused-Ring
Target Protein:
Cholecystokinin receptor type A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2411896-53-0

Tarcocimab tedromer is under investigation in clinical trial NCT06270836 (A Study to Evaluate the Efficacy and Safety of Tarcocimab Tedromer Compared With Sham Treatment in Participants With Moderately Severe to Severe Non-proliferative Diabetic Retinopathy (…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Taribavirin DB06408
small molecule | CAS: 119567-79-2

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAntiviral AgentsNucleic Acids, Nucleotides, and Nucleosides +3
Target Protein:
Inosine-5'-monophosphate dehydrogenase 1DNARNA-directed RNA polymerase L +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tariquidar DB06240
small molecule | CAS: 206873-63-4

Deskripsi belum tersedia.

Kategori:
Drug Resistance, MultipleHeterocyclic Compounds, Fused-RingP-glycoprotein inhibitors
Target Protein:
ATP-dependent translocase ABCB1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tarlatamab Approved DB17256
biotech | CAS: 2307488-83-9

Tarlatamab is a first-in-class T-cell engager used to treat extensive-stage small cell lung cancer.[L50748] It is a bispecific monoclonal antibody that targets CD3 expressed on the surface of T-cells and delta-like ligand 3 (DLL3), an inhibitory ligand that s…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalBispecific Monoclonal Antibodies +5
Target Protein:
Delta-like protein 3T-cell surface glycoprotein CD3
Waktu ParuhThe median terminal…
Vol. DistribusiAt steady-state, th…
KlirensThe systemic cleara…
Genetik -
Tarloxotinib DB14944
small molecule | CAS: 1636938-13-0

Tarloxotinib is under investigation in clinical trial NCT03743350 (NSCLC Exon 20 or HER2-activating Mutations).

Target Protein:
Receptor tyrosine-protein kinase erbB-2Epidermal growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TAS-102 DB08937
small molecule | CAS: 733030-01-8

TAS-102 (Taiho Pharma USA, Inc.) is an anti-cancer drug under development and in stage 3 clinical trials for the treatment of colorectal cancer. It is composed of the thymidine phosphorylase inhibitor (TPI) tipiracil and the cytotoxin trifluridine. Trifluridi…

Kategori:
DeoxyribonucleosidesNucleic Acids, Nucleotides, and NucleosidesNucleosides +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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