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13591

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10177 (74.9%)
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7625 (56.1%)
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104 (0.8%)
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13591 (100.0%)

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Halaman 211 / 272
Pirnabine DB12840
small molecule | CAS: 19825-63-9

Pirnabine has been used in trials studying the treatment of Chronic Idiopathic Constipation.

Kategori:
Amino Acids, Peptides, and ProteinsEnzyme ActivatorsGastrointestinal Agents +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Piroctone DB15946
small molecule | CAS: 50650-76-5

Piroctone olamine is used in combination with other substances as a part of shampoo effectively reduced the amount of dandruff and, at the same time, provided hair conditioning advantages. Recently was shown, that piroctone olamine could induce apoptosis and …

Kategori:
AlcoholsAminesAmino Alcohols +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pirodavir DB08012
small molecule | CAS: 124436-59-5

Pirodavir is an antipicornavirus agent.

Kategori:
Antiviral Agents
Target Protein:
Genome polyproteinGenome polyproteinGenome polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Piromelatine DB12288
small molecule | CAS: 946846-83-9

Piromelatine has been used in trials studying the treatment of Alzheimer's Disease.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
5-hydroxytryptamine receptor 1A5-hydroxytryptamine receptor 1DMelatonin receptor type 1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Piromidic acid DB13744
small molecule | CAS: 19562-30-2

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAnti-Infective Agents, UrinaryAntibacterials for Systemic Use +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Piroxicam Approved DB00554
small molecule | CAS: 36322-90-4

A cyclooxygenase inhibiting, non-steroidal anti-inflammatory agent (NSAID) that is well established in treating rheumatoid arthritis and osteoarthritis and used for musculoskeletal disorders, dysmenorrhea, and postoperative pain. Its long half-life enables it…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +33
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu Paruh30 to 86 hours
Vol. Distribusi* 0.14 L/kg
Klirens-
Genetik -
small molecule | CAS: 87234-24-0

Deskripsi belum tersedia.

Kategori:
Anti-Inflammatory AgentsSulfur CompoundsThiazines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pirprofen DB13722
small molecule | CAS: 31793-07-4

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pirtobrutinib Approved DB17472
small molecule | CAS: 2101700-15-4

Pirtobrutinib is a small molecule and a highly selective non-covalent inhibitor of Bruton’s tyrosine kinase (BTK). Its high selectivity has been associated with lower discontinuation rates due to adverse events and a lower incidence of atrial fibrillation.[A2…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Inhibitors +42
Target Protein:
Tyrosine-protein kinase BTK
Waktu ParuhPirtobrutinib has a…
Vol. DistribusiPirtobrutinib has a…
KlirensPirtobrutinib has a…
Genetik -
Pitavastatin Approved DB08860
small molecule | CAS: 147511-69-1

Pitavastatin, also known as the brand name product Livalo, is a lipid-lowering drug belonging to the statin class of medications. By inhibiting the endogenous production of cholesterol within the liver, statins lower abnormal cholesterol and lipid levels and …

Kategori:
Agents Causing Muscle ToxicityAnticholesteremic AgentsBCRP/ABCG2 Substrates +20
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductaseIntegrin alpha-L
Waktu ParuhThe mean plasma eli…
Vol. DistribusiThe mean volume of …
KlirensFollowing a single …
Genetik -
Pitofenone DB15947
small molecule | CAS: 54063-52-4

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismBenzene DerivativesDrugs for Functional Gastrointestinal Disorders +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pitolisant Approved DB11642
small molecule | CAS: 362665-56-3

Pitolisant is a selective antagonist or inverse agonist of the histamine H3 receptor used to treat type 1 or 2 narcolepsy.[L8063] Narcolepsy is a chronic neurological disorder that affects 1 in 2,000 individuals and is characterized by excessive daytime sleep…

Kategori:
Cytochrome P-450 CYP1A2 InducersCytochrome P-450 CYP1A2 Inducers (strength unknown)Cytochrome P-450 CYP2B6 Inducers +25
Target Protein:
Histamine H3 receptorVoltage-gated inwardly rectifying potassium channel KCNH2
Waktu ParuhPitolisant has a pl…
Vol. DistribusiFollowing single an…
KlirensThe apparent oral c…
Genetik -
small molecule | CAS: 566170-04-5

Pittsburgh Compound B is under investigation in clinical trial NCT01723553 (Amyloid-related Imaging Abnormalities (Microbleeds) in Atypical AD).

Kategori:
AminesCarbon RadioisotopesSulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pivagabine DB12951
small molecule | CAS: 69542-93-4

Pivagabine has been used in trials studying the treatment of Stress and Anxiety.

Kategori:
Acids, AcyclicAmino AcidsAmino Acids, Peptides, and Proteins +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pivampicillin Approved DB01604
small molecule | CAS: 33817-20-8

Pivalate ester analog of ampicillin.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
Penicillin-binding protein 1A
Waktu ParuhApproximately 1 hou…
Vol. Distribusi-
Klirens-
Genetik -
Pivhydrazine DB09252
small molecule | CAS: 306-19-4

Pivhydrazine, also known as pivazide, is a member of the hydrazine family with irreversible and non-selective inhibitory activity against monoamine oxidases. In 1960, it was widely used as an antidepressant agent but it is now discontinued.

Kategori:
Acids, AcyclicAgents that produce hypertensionAgents that reduce seizure threshold +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pivmecillinam Approved DB01605
small molecule | CAS: 32886-97-8

Pivmecillinam is a mecillinam prodrug, a pivaloyloxymethyl ester of amdinocillin that is well absorbed orally, but broken down to amdinocillin in the intestinal mucosa. It is active against gram-negative organisms and used as for amdinocillin. [PubChem]

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
Penicillin-binding protein 1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pixantrone Approved DB06193
small molecule | CAS: 144510-96-3

Pixantrone is an aza-anthracenedione and DNA intercalator which inhibits topoisomerase II. It is similar in structure to anthracyclines such as mitoxantrone, but exerts fewer toxic effects on cardiac tissue. [2] The lower cardio-toxic effects of pixantrone ma…

Kategori:
Anthracyclines and Related SubstancesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +6
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-beta
Waktu ParuhHalf life ranges fr…
Vol. Distribusi9.7-29.7 L/kg. [2]
KlirensPlasma clearance is…
Genetik -
Pizotifen Approved DB06153
small molecule | CAS: 15574-96-6

Pizotifen belongs to the class of antamines and is related to [cyproheptadine].[A32532] It is a potent serotonin and tryptamine antagonist that has been used for migraine prevention for many years. It exhibits weak anticholinergic, antihistamine, and antikini…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +27
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M3 +12
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
Klirens-
Genetik -
PKI-179 DB13109
small molecule | CAS: 1197160-28-3

PKI-179 has been used in trials studying the treatment of Advanced Malignant Solid Tumors.

Kategori:
AmidesOxazines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PL-3994 DB15355
small molecule | CAS: 952295-80-6

PL-3994 is under investigation in clinical trial NCT01304628 (Cross-Over Study of Subcutaneous Study Drug for the Treatment of Patients With Mild to Moderate Asthma).

Kategori:
Amino Acids, Peptides, and ProteinsBronchodilator AgentsPeptides +1
Target Protein:
Atrial natriuretic peptide receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

The placenta serves many purposes, with one of the many being a bank of mesenchymal stem cells (MSCs). It can be obtained relatively easily as medical waste from which MSCs can be non-invasively extracted and without the ethical issues that come with embryoni…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Placulumab DB11983
biotech | CAS: 945781-29-3

Placulumab has been used in trials studying the treatment of Rheumatoid Arthritis.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Plamotamab DB18944
biotech | CAS: 2138442-31-4

Plamotamab is under investigation in clinical trial NCT05328102 (Phase 2 Study of Plamotamab Combined With Tafasitamab Plus Lenalidomide Versus Tafasitamab Plus Lenalidomide in Relapsed or Refractory (R/R) Diffuse Large-cell B-cell Lymphoma (DLBCL)).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech

The Covifenz COVID-19 vaccine (plant-based virus-like particles (VLP), recombinant, adjuvanted) is a plant-based vaccine developed in partnership by Medicago and GlaxoSmithKline which is approved in Canada for the prevention of COVID-19.[L40694] It is compose…

Kategori:
COVID-19 VaccinesVaccinesViral Vaccines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Plantago lanceolata pollen Approved DB10382
biotech

Plantago lanceolata pollen is the pollen of the Plantago lanceolata plant. Plantago lanceolata pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Plantago seed Approved DB11097
biotech | CAS: 8063-16-9

Platango seeds refer to the seeds collected from various species of plantago trees. It is found in some laxatives for treating occasional constipation and restoring regularity in bowel movements. Its potential benefit in maintaining remission in ulcerative co…

Kategori:
Biological ProductsBulk-Forming LaxativesComplex Mixtures +5
Waktu ParuhThe half-life of ps…
Vol. DistribusiPsyllium husk when …
KlirensPsyllium husk when …
Genetik -
biotech

The plasma protein fraction human (PPFh) is defined as a sterile solution of proteins composed mainly of albumin and globulin derived from human plasma.[A32512] It is already reviewed under the category of biologics by the FDA where the processing, required t…

Kategori:
AlbuminsAmino Acids, Peptides, and ProteinsBlood Derivatives +9
Waktu ParuhThe registered clea…
Vol. DistribusiThe registered volu…
KlirensThe registered clea…
Genetik -
PlasmaCord DB16363
biotech

PlasmaCord is platelet-poor plasma that is derived by fractionation from sterile umbilical cord and placental blood.[L27581] It is developed by Cellpraxis and is currently being investigated against severe acute respiratory syndrome (SARS).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Plasminogen Approved DB16701
biotech | CAS: 9001-91-6

Plasminogen is a pro-enzyme (i.e. a zymogen) which is cleaved to form plasmin - also known as [fibrinolysin] - as part of the fibrinolytic pathway that breaks down fibrin blood clots.[A236035] This pathway is activated when a clot is no longer needed or to pr…

Kategori:
Amino Acids, Peptides, and ProteinsAnticoagulantsBeta-Globulins +11
Waktu ParuhThe mean half-life …
Vol. DistribusiThe mean steady-sta…
KlirensThe clearance of Ry…
Genetik -
Platanus occidentalis pollen Approved DB10392
biotech

Platanus occidentalis pollen is the pollen of the Platanus occidentalis plant. Platanus occidentalis pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Platanus racemosa pollen Approved DB10393
biotech

Platanus racemosa pollen is the pollen of the Platanus racemosa plant. Platanus racemosa pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 74389-68-7

Deskripsi belum tersedia.

Kategori:
Adrenergic AgentsAlcoholsAmines +21
Target Protein:
Platelet-activating factor receptorGanglioside GM2 activator
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Platensimycin DB08407
small molecule | CAS: 835876-32-9

Deskripsi belum tersedia.

Kategori:
3-Oxoacyl-(Acyl-Carrier-Protein) SynthaseAcids, CarbocyclicAmides +10
Target Protein:
3-oxoacyl-[acyl-carrier-protein] synthase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Platycodon grandiflorus leaf is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Platycodon grandiflorus root is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
AngiospermsBiological ProductsCampanulaceae +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Plazomicin Approved DB12615
small molecule | CAS: 1154757-24-0

Developed by Achaogen biopharmaceuticals, plazomicin is a next-generation aminoglycoside synthetically derived from [DB12604]. The structure of plazomicin was established via appending hydroxylaminobutyric acid to [DB12604] at position 1 and 2-hydroxyethyl gr…

Kategori:
Agents that produce neuromuscular block (indirect)Aminoglycoside AntibacterialsAnti-Bacterial Agents +12
Target Protein:
rRNA methyltransferase 2, mitochondrial30S ribosomal protein S1130S ribosomal protein S14
Waktu ParuhThe mean (±SD) half…
Vol. DistribusiThe mean (±SD) volu…
KlirensFollowing administr…
Genetik -
Plecanatide Approved DB13170
small molecule | CAS: 467426-54-6

Plecanatide is a drug approved in January 2017 by the FDA for the treatment of chronic idiopathic constipation (CIC). It should not be used in children less than six years of age, and should be avoided in patients six years to 18 years of age

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsDrugs for Constipation +12
Target Protein:
Guanylyl cyclase CGuanylate cyclase soluble subunit alpha-2
Waktu Paruhhalf-life (t½) cann…
Vol. DistribusiConcentrations of p…
KlirensNo excretion studie…
Genetik -
Pleconaril DB05105
small molecule | CAS: 153168-05-9

Pleconaril is an antiviral drug from _viral capsid inhibitor_ class, manufactured by _Schering-Plough_ and intended for the prevention of acute asthma exacerbations and common cold symptoms in asthmatic patients who have had exposure to _picornavirus_. It act…

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +4
Target Protein:
Genome polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pleospora betae Approved DB10936
biotech

Pleospora betae is a fungus which can provoke allergic reactions. Pleospora betae extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pleospora tarda Approved DB10939
biotech

Pleospora tarda allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Plerixafor Approved DB06809
small molecule | CAS: 110078-46-1

Plerixafor is a small-molecule inhibitor of C-X-C chemokine receptor type 4 (CXCR4) that acts as a hematopoietic stem cell mobilizer.[A7117,L45678] It is used to stimulate the release of stem cells from the bone marrow into the blood in patients with non-Hodg…

Kategori:
Adjuvants, ImmunologicAminesAnti-HIV Agents +9
Target Protein:
C-X-C chemokine receptor type 4
Waktu ParuhPlerixafor has a di…
Vol. DistribusiPlerixafor has an a…
KlirensPlerixafor has a to…
Genetik -
Plevitrexed DB06163
small molecule | CAS: 153537-73-6

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsHeterocyclic Compounds, Fused-Ring
Target Protein:
Thymidylate synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PLG-0206 DB18116
biotech | CAS: 847061-43-2

PLG-0206 is a peptide antibiotic under investigation for the treatment of periprosthetic joint infections.[L48106]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Plicamycin Approved DB06810
small molecule | CAS: 18378-89-7

Plicamycin is an antineoplastic antibiotic produced by Streptomyces plicatus. It has been used in the treatment of testicular cancer, Paget's disease of bone, and, rarely, the management of hypercalcemia. The manufacturer discontinued plicamycin in 2000.

Kategori:
AnthracyclinesAntibiotics, AntineoplasticAntineoplastic Agents +15
Target Protein:
DNA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Plitidepsin DB04977
small molecule | CAS: 137219-37-5

Aplidine is a peptide found in tunicates which shows promise in shrinking tumors in pancreatic, stomach, bladder, and prostate cancers. The specific marine organism is _Aplidium albicans_. Aplidine is also of interest as a potential treatment for some leukemi…

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +7
Target Protein:
Palmitoyl-protein thioesterase 1Elongation factor 1-alpha 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PLN-74809 DB16515
small molecule

PLN-74809 is a small-molecule that dually inhibits both ?<sub>v</sub>?<sub>6</sub> and ?<sub>v</sub>?<sub>1</sub> to treat both idiopathic pulmonary fibrosis (IPF) and primary sclerosing cholangitis (PSC)[L31693]. The compound was granted orphan drug designat…

Kategori:
Experimental Unapproved Treatments for COVID-19
Target Protein:
Integrin alpha-VIntegrin beta-1Integrin beta-6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Plozasiran DB18997
biotech | CAS: 2379776-40-4

Plozasiran is under investigation in clinical trial NCT05089084 (Study of ARO-APOC3 (Plozasiran) in Adults With Familial Chylomicronemia Syndrome (FCS)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Plumbagin DB17048
small molecule | CAS: 481-42-5

Plumbagin is a compound investigated for its anticancer activity. It has been found that it inactivates the Akt/NF-kB, MMP-9 and VEGF pathways.[A253102]

Kategori:
Adjuvants, ImmunologicAdrenal Cortex HormonesAnthelmintics +17
Target Protein:
Dihydroorotate dehydrogenase (quinone), mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Plutavimab DB18856
biotech | CAS: 2529854-88-2

Plutavimab is under investigation in clinical trial NCT04900428 (Study to Evaluate a Single Intranasal Dose of STI-2099 (COVI-DROPS™) in Outpatient Adults With COVID-19 (UK)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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