Hasil Filter

11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (11778)

Halaman 210 / 236
T-2000 DB11654
small molecule | CAS: 97846-21-4

T2000 has been used in trials studying the treatment of Myoclonus and Essential Tremor.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
T-5224 DB05998
small molecule | CAS: 530141-72-1

T-5224 is an investigational drug developed to treat Sepsis-induced Acute Kidney Injury. It's mechanism of action is to inhibit c-Fos/activator protein-1.

Kategori:
Benzene DerivativesKetones
Target Protein:
Transcription factor Jun
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
T-900607 DB12068
small molecule | CAS: 261944-52-9

T900607 has been used in trials studying the treatment of Liver Cancer and Gastric Cancer.

Kategori:
AmidesSulfonesSulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1948-33-0

Deskripsi belum tersedia.

Kategori:
AntioxidantsBenzene DerivativesBiological Factors +5
Target Protein:
HemagglutininHemagglutinin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
T-Guard DB18357
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
T487 DB05474
small molecule

T487 is a small molecule chemokine receptor antagonist to correct or modify immune system responses. It binds selectively and potently to CXCR3. The formulation is administered orally and has anti-inflammatory effects in conditions such as rheumatoid arthriti…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TA-CIN DB05809
biotech

TA-CIN is a subunit vaccine comprising L2/E6/E7 proteins from Human Papillomavirus (HPV16), designed to generate a strong cellular immune response against HPV-infected cells.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tabalumab DB11657
biotech | CAS: 1143503-67-6

Tabalumab has been used in trials studying the treatment of Autoimmune Disease, Rheumatoid Arthritis, Kidney Failure, Chronic, Connective Tissue Disease, and Systemic Lupus Erythematosus, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tabelecleucel Approved DB17072
biotech

Tabelecleucel is an innovative therapy that uses Epstein-Barr virus (EBV)-specific allogeneic cytotoxic T cells (CTLs). It is produced by mixing T-cells with B-cells that have been infected with the Epstein-Barr virus (EBV). Both T-cells and B-cells are obtai…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsAntineoplastic cell and gene therapy
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 943980-47-0

Taberminogene vadenovec (EG004) is a novel product consisting of a local delivery device and a gene-based medicine, being developed to prevent the blocking of veins and arteries that frequently occurs after vascular surgery. The initial target market is haemo…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 2412170-98-8

Tabirafusp tedromer is under investigation in clinical trial NCT06556368 (A Study to Evaluate the Efficacy and Safety of Tarcocimab Tedromer and Tabirafusp Tedromer Compared to Aflibercept in Participants With Neovascular (Wet) Age-related Macular Degeneratio…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1612758-88-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

A version of [tabituximab barzuxetan] radiolabeled with yttrium-90.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tacalcitol DB13689
small molecule | CAS: 57333-96-7

Deskripsi belum tersedia.

Kategori:
Anti-Inflammatory AgentsAntipsoriaticsAntipsoriatics for Topical Use +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tacrine Approved DB00382
small molecule | CAS: 321-64-2

A centerally active cholinesterase inhibitor that has been used to counter the effects of muscle relaxants, as a respiratory stimulant, and in the treatment of Alzheimer's disease and other central nervous system disorders. Tacrine has been discontinued for t…

Kategori:
AcridinesAgents Causing Muscle ToxicityAminoacridines +16
Target Protein:
CholinesteraseAcetylcholinesteraseLiver carboxylesterase 1
Waktu Paruh2 to 4 hours
Vol. Distribusi* 349 ± 193 L
Klirens-
Genetik -
Tacrolimus Approved DB00864
small molecule | CAS: 104987-11-3

Tacrolimus (also FK-506 or Fujimycin) is an immunosuppressive drug whose main use is after organ transplant to reduce the activity of the patient's immune system and so the risk of organ rejection. It is also used in a topical preparation in the treatment of …

Kategori:
Agents causing hyperkalemiaAgents Causing Muscle ToxicityAgents for Dermatitis, Excluding Corticosteroids +33
Target Protein:
Protein phosphatase 3 catalytic subunit alphaPeptidyl-prolyl cis-trans isomerase FKBP1A
Gen Terkait:
CYP3A5 ABCB1
Waktu ParuhThe elimination hal…
Vol. Distribusi* 2.6 ± 2.1 L/kg [p…
Klirens* 0.040 L/hr/kg [he…
Genetik 2 Varian
Tadalafil Approved DB00820
small molecule | CAS: 171596-29-5

Tadalafil is a selective phosphodiesterase-5 inhibitor that is used in the treatment of erectile dysfunction (ED), pulmonary arterial hypertension (PAH), and benign prostatic hypertrophy.[L39100, L39105] It was first approved in 2003 by the FDA for use in ED …

Kategori:
5-alpha Reductase InhibitorsAntihypertensive AgentsAntihypertensives for Pulmonary Arterial Hypertension +20
Target Protein:
cGMP-specific 3',5'-cyclic phosphodiesteraseDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11ARetinal rod rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit gamma
Waktu ParuhThe mean half-life …
Vol. DistribusiTadalafil has a mea…
KlirensThe mean apparent o…
Genetik -
Tadekinig alfa DB14858
biotech | CAS: 220712-29-8

Tadekinig alfa is under investigation in clinical trial NCT03113760 (Therapeutic Use of Tadekinig Alfa in NLRC4 Mutation and XIAP Deficiency).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TAFA-93 DB05887
small molecule

TAFA93 is a novel prodrug of the mTOR inhibitor rapamycin which has successfully completed Phase 1 clinical development. mTOR inhibitors are currently used in the prevention of organ rejection in transplantation, the treatment of autoimmune and oncological di…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tafamidis Approved DB11644
small molecule | CAS: 594839-88-0

Tafamidis and tafamidis meglumine (FX-1006A) are benzoxazole derivatives[A27206] developed by FoldRX.[A189717] Tafamidis is structurally similar to diflusinal.[A189717] Tafamidis was granted an EMA market authorisation on 16 November 2011[L6247] and FDA ap…

Kategori:
Anti-Inflammatory AgentsBCRP/ABCG2 InhibitorsFused-Ring Compounds +8
Target Protein:
Transthyretin
Waktu ParuhThe half life of ta…
Vol. DistribusiThe apparent volume…
KlirensThe oral clearance …
Genetik -
Tafasitamab Approved DB15044
biotech | CAS: 1422527-84-1

Tafasitamab is a humanized, CD19-directed cytolytic monoclonal antibody intended for the treatment of B-cell malignancies.[L15302] It is produced using recombinant DNA technology in Chinese hamster ovary cells, and contains an IgG1/2 hybrid Fc-domain which ha…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +13
Target Protein:
B-lymphocyte antigen CD19
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe total volume of…
KlirensThe clearance of ta…
Genetik -
Tafenoquine Approved DB06608
small molecule | CAS: 106635-80-7

Tafenoquine is an 8-aminoquinoline analogue of primaquine which varies only on the presence of a 5-phenoxy group.[A35671, A35690] It was discovered by the scientists at the Walter Reed Army Institute of Research in 1978 as a substitute for primaquine that wou…

Kategori:
AminoquinolinesAnti-Infective AgentsAntimalarials +11
Waktu ParuhTafenoquine present…
Vol. DistribusiTafenoquine present…
KlirensTafenoquine present…
Genetik -
Tafluprost Approved DB08819
small molecule | CAS: 209860-87-7

A prostaglandin analogue ester prodrug used topically (as eye drops) to control the progression of glaucoma and in the management of ocular hypertension. Chemically, tafluprost is a fluorinated analog of prostaglandin F2-alpha. Tafluprost was approved for use…

Kategori:
Antiglaucoma Preparations and MioticsAutacoidsBiological Factors +13
Target Protein:
Prostaglandin F2-alpha receptor
Waktu Paruh-
Vol. DistribusiThe highest concent…
Klirens-
Genetik -
Tafolecimab DB16336
biotech | CAS: 2225109-03-3

Tafolecimab is under investigation in clinical trial NCT04031742 (A Study to Evaluate Safety and Efficacy of IBI306, a PCSK9 Monoclonal Antibody in Chinese Subjects With Homozygous Familial Hypercholesterolemia).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tagatose DB04936
small molecule | CAS: 87-81-0

Tagatose is a functional sweetener. It is a naturally occurring monosaccharide, specifically a hexose. It is commonly found in dairy with a similar texture and sweetened capacity to sucrose but with only a third of the calories. It is approved as a food addit…

Kategori:
CarbohydratesChelating AgentsCompounds used in a research, industrial, or household setting +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tagetitoxin DB04788
small molecule | CAS: 87913-21-1

Tagetitoxin is a bacterial phytotoxin. It preferentially inhibits eukaryotic RNA polymerase.

Kategori:
Acids, AcyclicBacterial Toxins
Target Protein:
DNA-directed RNA polymerase subunit betaDNA-directed RNA polymerase subunit beta'
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tagitanlimab DB18221
biotech | CAS: 2417649-97-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tagraxofusp Approved DB14731
biotech | CAS: 2055491-00-2

Tagraxofusp is a CD123-directed cytotoxin. It is a fusion protein composed of a human interleukin-3 (IL-3) that is genetically fused to the catalytic and translocation domains of truncated diphtheria toxin (DT) produced in _Escherichia coli_.[A253762, A253887…

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +7
Target Protein:
Interleukin-3 receptor subunit alpha
Waktu ParuhThe mean (SD) termi…
Vol. DistribusiFollowing administr…
KlirensMean clearance (SD)…
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TAK-071 DB18954
small molecule | CAS: 1820812-16-5

TAK-071 is under investigation in clinical trial NCT04334317 (A Study of TAK-071 in People With Parkinson Disease).

Kategori:
Cholinergic AgentsCholinergic AgonistsHeterocyclic Compounds, Fused-Ring +2
Target Protein:
Muscarinic acetylcholine receptor M1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 667931-25-1

Deskripsi belum tersedia.

Kategori:
Receptors, Calcium-Sensing, antagonists & inhibitors
Target Protein:
Extracellular calcium-sensing receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TAK-448 DB11975
biotech | CAS: 1234319-68-6

TAK-448 has been used in trials studying the treatment of Prostate Cancer, Low Testosterone, Prostatic Neoplasms, and Hypogonadotropic Hypogonadism.

Kategori:
Amino Acids, Peptides, and ProteinsIntercellular Signaling Peptides and ProteinsNeoplasm Proteins +4
Target Protein:
Metastasis-suppressor KiSS-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TAK-475 DB05317
small molecule

TAK-475 is a "squalene synthase inhibitor", a type of cholesterol-lowering drug that has not yet been brought to market.

Kategori:
AzepinesFarnesyl-Diphosphate Farnesyltransferase, antagonists & inhibitors
Target Protein:
Squalene synthase3-hydroxy-3-methylglutaryl-coenzyme A reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TAK-593 DB13093
small molecule | CAS: 1005780-62-0

TAK-593 has been used in trials studying the treatment of Solid Tumors.

Kategori:
Aza CompoundsReceptors, Platelet-Derived Growth Factor, antagonists & inhibitors
Target Protein:
Vascular endothelial growth factor receptor 2Platelet-derived growth factor receptor beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TAK-603 DB17892
small molecule | CAS: 158146-85-1

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Interferon gamma
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TAK-611 DB17644
biotech

TAK-611, formerly known as SHP611, is a recombinant human arylsulfatase A. First developed by Takeda, it is being investigated for the treatment of metachromatic leukodystrophy.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TAK-653 DB16304
small molecule | CAS: 1358751-06-0

TAK-653 is under investigation in clinical trial NCT03312894 (Efficacy and Safety of TAK-653 in Treatment-resistant Depression).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TAK-715 DB16108
small molecule | CAS: 303162-79-0

TAK-715 is under investigation in clinical trial NCT00760864 (Safety and Efficacy of TAK-715 in Subjects With Rheumatoid Arthritis).

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TAK-733 DB12241
small molecule | CAS: 1035555-63-5

TAK-733 has been used in trials studying the treatment of Advanced Metastatic Melanoma, Advanced Nonhematologic Malignancies, and Advanced Non-hematologic Malignancies.

Kategori:
PyridinesPyrimidines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TAK-751S DB06432
small molecule

TAK-751S is a synthetic analog of Shiga toxin (Stx) receptor, Gb3, produced by enterohemorrhagic _Escherichia coli_.[A260296]

Kategori:
CarbohydratesOligosaccharidesPolysaccharides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TAK-754 DB17850
biotech

TAK-754 is an adeno-associated virus serotype 8 vector (AAV8) expressing B domain deleted codon optimized factor VIII. Developed by Takeda, it is being investigated for the treatment of hemophilia A.[A259831]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TAK-901 DB12756
small molecule | CAS: 934541-31-8

TAK-901 has been used in trials studying the treatment of Lymphoma, Myelofibrosis, Multiple Myeloma, Myeloid Metaplasia, and Advanced Solid Tumors, among others.

Kategori:
Heterocyclic Compounds, Fused-RingIndole AlkaloidsIndoles +3
Target Protein:
Aurora kinase BApoptosis regulator BAX
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Talabostat DB06182
small molecule | CAS: 149682-77-9

Deskripsi belum tersedia.

Kategori:
AcidsAcids, NoncarboxylicAmino Acids, Peptides, and Proteins +4
Target Protein:
Prolyl endopeptidase FAPDipeptidyl peptidase 9Dipeptidyl peptidase 8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Talacotuzumab DB14796
biotech | CAS: 1826831-79-1

Talacotuzumab is an IgG1 monoclonal antibody directed toward the IL3 receptor ?–subunit, also known as CD123. It is under investigation in clinical trial NCT01632852 (A Study of CSL362 in Patients With CD123+ Acute Myeloid Leukemia Currently in Remission).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Talampicillin DB13814
small molecule | CAS: 47747-56-8

Deskripsi belum tersedia.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Talastine DB13349
small molecule | CAS: 16188-61-7

Deskripsi belum tersedia.

Kategori:
Antihistamines for Systemic UsePyridazinesSubstituted Alkylamines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Talazoparib Approved DB11760
small molecule | CAS: 1207456-01-6

Talazoparib is an inhibitor of mammalian polyadenosine 5’-diphosphoribose polymerases (PARPs), enzymes responsible for regulating essential cellular functions, such as DNA transcription and DNA repair.[L47236] Developed by Pfizer, talazoparib was first app…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Substrates +7
Target Protein:
Poly [ADP-ribose] polymerase 1Poly [ADP-ribose] polymerase 2
Waktu ParuhThe mean terminal p…
Vol. DistribusiThe mean apparent v…
KlirensThe mean apparent o…
Genetik -
Talc Approved DB09511
small molecule | CAS: 14807-96-6

Talc is a mineral composed primarily of magnesium, silicon and oxygen. It is a substance often found in cosmetic and personal hygiene products including baby powder, adult body powders and facial powders. Talc helps absorb moisture, freshen materials, and red…

Kategori:
AntiperspirantsCompounds used in a research, industrial, or household settingCosmetics +6
Waktu ParuhIntended for local …
Vol. DistribusiIntended for local …
KlirensIntended for local …
Genetik -
biotech | CAS: 1580555-26-5

Talditercept alfa is under investigation in clinical trial NCT03039686 (Clinical Trial to Evaluate the Efficacy, Safety, and Tolerability of RO7239361 in Ambulatory Boys With Duchenne Muscular Dystrophy).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
taletrectinib DB18711
small molecule | CAS: 1505515-69-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 10451–10500 dari 11778
Sebelumnya Halaman 210 / 236 Berikutnya