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13591

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10177 (74.9%)
Target
7625 (56.1%)
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104 (0.8%)
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13591 (100.0%)

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Halaman 210 / 272
Pimasertib DB14904
small molecule | CAS: 1236699-92-5

Pimasertib is under investigation in clinical trial NCT01378377 (Combination Trial of Pimasertib (MSC1936369B) With Temsirolimus).

Kategori:
Nicotinic AcidsProtein Kinase InhibitorsPyridines
Target Protein:
Mitogen-activated protein kinase kinase (MAPKK)
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pimavanserin Approved DB05316
small molecule | CAS: 706779-91-1

Pimavanserin is an atypical antipsychotic indicated for the treatment of psychiatric disorders.[L48236] Although the exact mechanism of action is unknown, it is thought that pimavanserin interacts with the serotonin receptors, particularly the 5-HT<sub>2A</su…

Kategori:
AmidesAntidepressive AgentsCentral Nervous System Agents +14
Target Protein:
5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 2CSigma non-opioid intracellular receptor 1
Waktu ParuhThe average plasma …
Vol. DistribusiFollowing administr…
Klirens-
Genetik -
Pimecrolimus Approved DB00337
small molecule | CAS: 137071-32-0

Pimecrolimus is an immunomodulating agent that was first marketed by Novartis under the trade name Elidel. It is now promoted in Canada by Galderma since early 2007. It is currently available as a topic cream used in the treatment of atopic dermatitis (eczema…

Kategori:
Agents for Dermatitis, Excluding CorticosteroidsAnalgesicsAnalgesics, Non-Narcotic +15
Target Protein:
Protein phosphatase 3 catalytic subunit alphaSerine/threonine-protein kinase mTORPeptidyl-prolyl cis-trans isomerase FKBP1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pimethixene Approved DB13292
small molecule | CAS: 314-03-4

Pimethixene is approved for use in Brazil and is marketed under the trade name Muricalm. It is an anticholinergic used in the treatment of bronchitis.

Kategori:
Antihistamines for Systemic UseHeterocyclic Compounds, Fused-RingSulfur Compounds +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pimicotinib DB18972
small molecule

Pimicotinib is under investigation in clinical trial NCT05804045 (Study of Pimicotinib (ABSK021) for Tenosynovial Giant Cell Tumor (MANEUVER)).

Waktu Paruh-
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Pimivalimab DB16667
biotech | CAS: 2293951-22-9

Pimivalimab is under investigation in clinical trial NCT04549025 (Study of PD-1 Inhibitor JTX-4014 Alone and in Combination With Vopratelimab in Biomarker-selected Subjects With Metastatic NSCLC After One Prior Platinum-containing Regimen).

Waktu Paruh-
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Pimodivir DB14974
small molecule | CAS: 1629869-44-8

Pimodivir is under investigation in clinical trial NCT02658825 (A Study to Evaluate the Effect of JNJ-63623872 on Cardiac Repolarization Interval in Healthy Participants).

Waktu Paruh-
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Pimonidazole DB12485
small molecule | CAS: 70132-50-2

Pimonidazole is under investigation for the diagnostic of Prostate Cancer and Head and Neck Cancer.

Kategori:
ImidazolesNitro CompoundsRadiation-Sensitizing Agents
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Pimozide Approved DB01100
small molecule | CAS: 2062-78-4

A diphenylbutylpiperidine that is effective as an antipsychotic agent and as an alternative to haloperidol for the suppression of vocal and motor tics in patients with Tourette syndrome. Although the precise mechanism of action is unknown, blockade of postsyn…

Kategori:
Agents that reduce seizure thresholdAnti-Dyskinesia AgentsAntipsychotic Agents +38
Target Protein:
D(2) dopamine receptorD(3) dopamine receptorVoltage-gated inwardly rectifying potassium channel KCNH2 +1
Waktu Paruh29 &plusmn; 10 hour…
Vol. Distribusi-
Klirens-
Genetik -
Pinacidil Approved DB06762
small molecule | CAS: 60560-33-0

Pinacidil is a cyanoguanidine drug that acts by opening ATP-sensitive potassium channels, leading to peripheral vasodilatation of arterioles and decreasing peripheral vascular resistance. The above processes result in reduced blood pressure. This drug has bee…

Kategori:
AmidinesAntihypertensive AgentsArteriolar Smooth Muscle, Agents Acting On +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1313706-14-7

Pinatuzumab vedotin is under investigation in clinical trial NCT01691898 (A Study of Pinatuzumab Vedotin (DCDT2980S) Combined With Rituximab or Polatuzumab Vedotin (DCDS4501A) Combined With Rituximab or Obinutuzumab in Participants With Relapsed or Refractory…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pinazepam DB13335
small molecule | CAS: 52463-83-9

Deskripsi belum tersedia.

Kategori:
Anti-Anxiety AgentsBenzazepinesBenzodiazepines and benzodiazepine derivatives +7
Target Protein:
GABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pindolol Approved DB00960
small molecule | CAS: 13523-86-9

Pindolol is a first generation non-selective beta blocker used in the treatment of hypertension.[L32353] Early research into the use of pindolol found it had chronotropic effects, and so further investigation focused on the treatment of arrhythmia.[A231059] R…

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-Antagonists +29
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptorBeta-3 adrenergic receptor +2
Waktu ParuhThe half life of pi…
Vol. DistribusiThe volume of distr…
KlirensIn otherwise health…
Genetik -
biotech | CAS: 8000-26-8

Pine needle oil is obtained from the needles of *Pinus mugo* tree via steam distillation. Major components of pine needle oil (pinus mugo) include ?-Pinene, ?-pinene, ?-3-carene, limonene, ?-phellandrene, (E)-caryophyllene, and germacrene D. It is present in …

Kategori:
Herbs and Natural Products
Waktu Paruh-
Vol. Distribusi-
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Pinometostat DB12920
small molecule | CAS: 1380288-87-8

Pinometostat has been used in trials studying the treatment of Leukemia, Acute Leukemias, Acute Myeloid Leukemia, Myelodysplastic Syndrome, and Acute Lymphocytic Leukemia, among others.

Kategori:
Antineoplastic AgentsHeterocyclic Compounds, Fused-Ring
Target Protein:
Histone-lysine N-methyltransferase, H3 lysine-79 specific
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pinus resinosa pollen Approved DB10923
biotech

Pinus resinosa pollen is the pollen of the Pinus resinosa plant. Pinus resinosa pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
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Genetik -
Pioglitazone Approved DB01132
small molecule | CAS: 111025-46-8

Pioglitazone is an antihyperglycemic used as an adjunct to diet, exercise, and other antidiabetic medications to manage type 2 diabetes mellitus.[L11416,L11419,L11422,L11425] It is administered as a racemic mixture, though there is no pharmacologic difference…

Kategori:
Alimentary Tract and MetabolismBlood Glucose Lowering AgentsCytochrome P-450 CYP2C8 Inhibitors +21
Target Protein:
Peroxisome proliferator-activated receptor gammaAmine oxidase [flavin-containing] B
Waktu ParuhThe mean serum half…
Vol. DistribusiThe average apparen…
KlirensThe apparent cleara…
Genetik -
Pipamperone DB09286
small molecule | CAS: 1893-33-0

Pipamperone is a typical antipsychotic of the _butyrophenone_ family used in the treatment of schizophrenia. It was developed by Janssen Pharmaceutica in 1961 and started its first round of clinical trials in 1963 [L1514, L1518]. In an effort to improve [h…

Kategori:
Antidepressive AgentsAntipsychotic AgentsButyrophenone Derivatives +15
Target Protein:
D(2) dopamine receptor5-hydroxytryptamine receptor 2AAlpha-1 adrenergic receptors +5
Waktu Paruh17-26h [L1522]
Vol. Distribusi-
Klirens-
Genetik -
Pipazethate DB08796
small molecule | CAS: 2167-85-3

A non-narcotic oral antitussive agent.

Kategori:
Antitussive AgentsCentral Nervous System AgentsCough and Cold Preparations +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pipecuronium Approved DB01338
small molecule | CAS: 68399-58-6

Pipecuronium is a piperazinyl androstane derivative which is a non-depolarizing neuromuscular blocking agent.

Kategori:
Agents producing tachycardiaAnticholinergic AgentsCentral Nervous System Depressants +13
Target Protein:
Neuronal acetylcholine receptor subunit alpha-2Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M3
Waktu ParuhPipecuronium has an…
Vol. Distribusi-
Klirens-
Genetik -
Pipemidic acid DB13823
small molecule | CAS: 51940-44-4

Deskripsi belum tersedia.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAnti-Infective Agents, Urinary +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pipendoxifene DB05414
small molecule | CAS: 198480-55-6

ER modulator, ERA-923(Pipendoxifene) is a estrogen receptor modulator being evaluated for the treatment of breast cancer. Pipendoxifene is a new 2-phenyl indole selective estrogen receptor modulators (SERM )that exhibits an excellent preclinical pharmacologic…

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Estrogen receptorEstrogen receptor betaIntegrase, catalytic core
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pipenzolate DB13844
small molecule | CAS: 13473-38-6

Deskripsi belum tersedia.

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAnticholinergic Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pipequaline DB13991
small molecule | CAS: 77472-98-1

Pipequaline is an anticonflict & anticonvulsant quinoline derivative. It is an anxiolytic drug that was never marketed. It presents a unique chemical structure that does not follow the structural properties of other drugs of its class. Pipequaline has a simil…

Kategori:
Central Nervous System AgentsHeterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Piperacetazine Approved DB06808
small molecule | CAS: 3819-00-9

Piperacetazine was an antipsychotic.

Kategori:
Heterocyclic Compounds, Fused-RingSulfur Compounds
Target Protein:
D(2) dopamine receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Piperacillin Approved DB00319
small molecule | CAS: 66258-76-2

Semisynthetic, broad-spectrum, ampicillin derived ureidopenicillin antibiotic proposed for pseudomonas infections. It is also used in combination with other antibiotics.

Kategori:
Agents that produce neuromuscular block (indirect)AmidesAnti-Bacterial Agents +15
Target Protein:
Penicillin-binding protein 3Penicillin-binding protein 2BPenicillin-binding protein 2a +1
Waktu Paruh36-72 minutes
Vol. Distribusi* 101 mL/kg [intrav…
Klirens* 32 - 41 mL/min/1.…
Genetik -
Piperaquine Approved DB13941
small molecule | CAS: 4085-31-8

Piperaquine is an antimalarial agent first synthesized in the 1960's and used throughout China [A31550]. Its use declined in the 1980's as piperaquine resistant strains of *Plasmodium falciparum* appeared and artemisinin derivatives became available. It has c…

Kategori:
Anti-Infective AgentsAntimalarialsAntiparasitic Agents +19
Waktu ParuhThe terminal elimin…
Vol. DistribusiPiperaquine is thou…
KlirensThe mean apparent t…
Genetik -
Piperazine Approved DB00592
small molecule | CAS: 110-85-0

Piperazine is an organic compound that consists of a six-membered ring containing two opposing nitrogen atoms. First used as a solvent for uric acid, the use of piperazine as an anthelmintic agent was first introduced in 1953. Upon entry into the systemic cir…

Kategori:
AnthelminticsAnti-Infective AgentsAntinematodal Agents +7
Target Protein:
Gamma-aminobutyric acid receptor subunit beta-3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Piperidione DB13224
small molecule | CAS: 77-03-2

Piperidione was cough medicine marketed by Roche under the trade name Sedulon.

Kategori:
Cough and Cold Preparations
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Piperidolate DB13351
small molecule | CAS: 82-98-4

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAgents producing tachycardiaAlimentary Tract and Metabolism +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Piperonyl butoxide Approved DB09350
small molecule | CAS: 51-03-6

Piperonyl butoxide (PBO) is an organic compound used as a component of pesticide formulations. It is used for the treatment of head, pubic (crab), and body lice. Piperonyl butoxide is a synergist. It has no pesticidal activity of its own, but acts to increase…

Kategori:
AgrochemicalsBenzodioxolesCompounds used in a research, industrial, or household setting +6
Waktu Paruh32 hours.
Vol. DistribusiPiperonyl butoxide …
KlirensClearance of pipero…
Genetik -
Pipethanate DB15888
small molecule | CAS: 4546-39-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Pipobroman Approved DB00236
small molecule | CAS: 54-91-1

An antineoplastic agent that acts by alkylation.

Kategori:
Alkylating DrugsAntineoplastic AgentsAntineoplastic Agents, Alkylating +4
Target Protein:
DNA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pipotiazine Approved DB01621
small molecule | CAS: 39860-99-6

Pipotiazine has actions similar to those of other phenothiazines. Among the different phenothiazine derivatives, it appears to be less sedating and to have a weak propensity for causing hypotension or potentiating the effects of CNS depressants and anesthetic…

Kategori:
Antidepressive AgentsAntipsychotic AgentsCentral Nervous System Depressants +26
Target Protein:
D(2) dopamine receptorD(1A) dopamine receptor5-hydroxytryptamine receptor 2A +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pipradrol Approved DB11584
small molecule | CAS: 467-60-7

Pipradrol (Meratran) [L2523] was initially developed in the 1950s as an antidepressant, however, the adverse effects associated with its use and its abuse potential led to its withdrawal and international regulation [L2524]. Pipradrol was made illegal in man…

Kategori:
Central Nervous System StimulantsNervous SystemPsychoanaleptics +1
Target Protein:
D(1) dopamine receptor
Waktu Paruh-
Vol. DistribusiDistributed in the …
KlirensRapidly cleared [T1…
Genetik -
Piprozolin DB13202
small molecule | CAS: 17243-64-0

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismBile and Liver TherapyBile Therapy +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Piracetam Approved DB09210
small molecule | CAS: 7491-74-9

Piracetam is a nootropic drug in the racetams group, with chemical name 2-oxo-1-pyrrolidine acetamide. It shares the same 2-oxo-pyrrolidone base structure with pyroglutamic acid and is a cyclic derivative of the neurotransmitter ?-aminobutyric acid (GABA). Ho…

Kategori:
AcetamidesAcetatesAcids, Acyclic +12
Waktu ParuhThe plasma half lif…
Vol. DistribusiVd is approximately…
KlirensThe apparent total …
Genetik -
Pirbuterol Approved DB01291
small molecule | CAS: 38677-81-5

Pirbuterol is a beta-2 adrenergic bronchodilator. In vitro studies and in vivo pharmacologic studies have demonstrated that pirbuterol has a preferential effect on beta-2 Adrenergic receptors compared with isoproterenol. While it is recognized that beta-2 adr…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic beta-2 Receptor Agonists +21
Target Protein:
Beta-2 adrenergic receptorBeta-1 adrenergic receptor
Waktu Paruh2 hours.
Vol. Distribusi-
Klirens-
Genetik -
Pirenoxine DB15945
small molecule | CAS: 1043-21-6

Deskripsi belum tersedia.

Kategori:
Cataract, drug therapy
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Pirenzepine Approved DB00670
small molecule | CAS: 28797-61-7

An antimuscarinic agent that inhibits gastric secretion at lower doses than are required to affect gastrointestinal motility, salivary, central nervous system, cardiovascular, ocular, and urinary function. It promotes the healing of duodenal ulcers and due to…

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAnti-Ulcer Agents +10
Target Protein:
Muscarinic acetylcholine receptor M1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pirepemat DB19165
small molecule | CAS: 1227638-29-0

Pirepemat is under investigation in clinical trial NCT05258071 (A Clinical Study Evaluating Efficacy of Pirepemat on Falls Frequency in Patients With Parkinson's Disease (PD)).

Waktu Paruh-
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Piretanide Approved DB02925
small molecule | CAS: 55837-27-9

Piretanide (INN, trade names Arelix, Eurelix, Tauliz) has been synthesized in 1973 at Hoechst AG (Germany) as a loop diuretic compound by using a then-new method for introducing cyclic amine residues in an aromatic nucleus in the presence of other aromaticall…

Kategori:
AmidesCardiovascular AgentsDiuretics +9
Target Protein:
Solute carrier family 12 member 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pirfenidone Approved DB04951
small molecule | CAS: 53179-13-8

Pirfenidone is a synthetic pyridone drug.[A251370] It is an antifibrotic agent with anti-inflammatory and antioxidant properties [A251370] that is used to treat idiopathic pulmonary fibrosis (IPF),[L26801] which is a chronic, progressive form of interstitial …

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAnti-Inflammatory Agents +29
Target Protein:
Transforming growth factor beta-1 proprotein
Waktu ParuhThe mean terminal h…
Vol. DistribusiMean apparent oral …
KlirensFollowing administr…
Genetik -
Piribedil DB12478
small molecule | CAS: 3605-01-4

Piribedil has been investigated in Parkinson's Disease.

Kategori:
Anti-Dyskinesia AgentsAnti-Parkinson Agents (Dopamine Agonist)Anti-Parkinson Drugs +7
Target Protein:
D(3) dopamine receptorAlpha-2C adrenergic receptor5-hydroxytryptamine receptor 1A +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pirisudanol DB13412
small molecule | CAS: 33605-94-6

Deskripsi belum tersedia.

Kategori:
Nervous SystemPsychoanalepticsPsychostimulants, Agents Used for ADHD and Nootropics
Waktu Paruh-
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Piritramide Approved DB12492
small molecule | CAS: 302-41-0

Piritramide is under investigation for the treatment of Colon Cancer and Minimal Residual Disease. Piritramide has been investigated for the supportive care of Pain, Postoperative and Postoperative Nausea and Vomiting.

Kategori:
AnalgesicsCentral Nervous System AgentsCentral Nervous System Depressants +9
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Piritrexim DB03695
small molecule | CAS: 72732-56-0

Piritrexim has been used in trials studying the treatment of Bladder Cancer, Urethral Cancer, and Transitional Cell Cancer of the Renal Pelvis and Ureter.

Kategori:
Antineoplastic AgentsEnzyme InhibitorsFolic Acid Antagonists
Target Protein:
Dihydrofolate reductase
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Pirlimycin DB11537
small molecule | CAS: 79548-73-5

Pirlimycin hydrochloride is an antibiotic belonging to the _lincosamide_ class. Often marketed as _Pirsue_, this drug is used to treat mastitis in cattle.

Kategori:
Anti-Bacterial AgentsCarbohydratesGlycosides +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pirlindole DB09244
small molecule | CAS: 60762-57-4

This drug is classified as a reversible inhibitor of monoamine oxidase A enzyme (also known as a RIMA drug). It was developed and is currently used as an antidepressant in Russia. Its chemical structure is similar to metralindole, and it also shares pharmacol…

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +14
Target Protein:
Amine oxidase [flavin-containing] A5-hydroxytryptamine receptor 1AAlpha-2A adrenergic receptor
Waktu Paruh0.7±0.3 in one stud…
Vol. Distribusi-
KlirensHigh plasma clearan…
Genetik -
Pirmitegravir DB18974
small molecule | CAS: 2245231-10-9

Pirmitegravir is under investigation in clinical trial NCT05869643 (A Clinical Trial of STP0404 in Treatment-naïve Adults With HIV-1 Infection).

Waktu Paruh-
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Menampilkan 10451–10500 dari 13591
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