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11778

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11778 (100.0%)

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Halaman 209 / 236
Sulopenem DB15284
small molecule | CAS: 120788-07-0

Sulopenem is a penem antibacterial. It is marketed as the prodrug [sulopenem etzadroxil] in combination with [probenecid].[L51768]

Kategori:
Amides
Waktu Paruh-
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Sulopenem etzadroxil Approved DB16335
small molecule | CAS: 1000296-70-7

Sulopenem etzadroxil is a prodrug of the penem antibacterial [sulopenem]. Like other beta-lactam antibacterials, it is a time-dependent inhibitor of bacterial cell wall synthesis.[L51768] Sulopenem etzadroxil was approved by the FDA in October 2024 for the…

Kategori:
OAT3/SLC22A8 SubstratesPenem Antibacterial
Target Protein:
Penicillin-binding protein 2Penicillin-binding protein 1APenicillin-binding protein 1B +4
Waktu ParuhIn the fasted state…
Vol. DistribusiIn the fasted state…
KlirensIn the fasted state…
Genetik -
Sulpiride Approved DB00391
small molecule | CAS: 15676-16-1

Sulpiride first appeared in published literature in 1967.[A229538] Clinical studies show a greater effect on treating the negative symptoms of schizophrenia rather than positive symptoms at low doses, though the effects are more equal at higher doses.[A229683…

Kategori:
Acids, CarbocyclicAmidesAntidepressive Agents +26
Target Protein:
D(2) dopamine receptorD(3) dopamine receptorCarbonic anhydrase 2 +2
Waktu ParuhReports of the half…
Vol. DistribusiThe average volume …
KlirensThe total systemic …
Genetik -
Sulprostone DB12708
small molecule | CAS: 60325-46-4

Sulprostone has been used in trials studying Abortion, Induced.

Kategori:
Abortifacient AgentsAbortifacient Agents, NonsteroidalAutacoids +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Sultamicillin Approved DB12127
small molecule | CAS: 76497-13-7

Sultamicillin has been used in trials studying the prevention and treatment of Ventilator Associated Pneumonia and Chronic Obstructive Pulmonary Disease (COPD).

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +9
Waktu Paruh-
Vol. Distribusi-
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Sultopride Approved DB13273
small molecule | CAS: 53583-79-2

Sultopride is used in Japan, Hong Kong, and Europe to treat schizophrenia. It is of the drug class atypical antipsychotics [L5626].

Kategori:
Acids, CarbocyclicAmidesAntidepressive Agents +17
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Sumanirole DB06477
small molecule | CAS: 179386-43-7

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
D(2) dopamine receptorD(3) dopamine receptorD(4) dopamine receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sumatriptan Approved DB00669
small molecule | CAS: 103628-46-2

Sumatriptan is a serotonin receptor agonist commonly used to treat migraines and sometimes cluster headaches.[L6793,L6796,L6799,L6805,L6808,L6811] Sumatriptan is the first of the triptans and was made available in Europe in 1991 to treat migraines.[A179761] S…

Kategori:
Agents that produce hypertensionAmidesAmines +33
Target Protein:
5-hydroxytryptamine receptor 1A5-hydroxytryptamine receptor 1D5-hydroxytryptamine receptor 1B +1
Gen Terkait:
GNB3
Waktu ParuhSubcutaneous sumatr…
Vol. DistribusiSumatriptan has a v…
KlirensSubcutaneous sumatr…
Genetik 1 Varian
SUN-101 DB17238
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
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Sunflower seed Approved DB10907
biotech

Sunflower seed allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
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Sunitinib Approved DB01268
small molecule | CAS: 557795-19-4

Sunitinib is a small-molecule multi-targeted receptor tyrosine kinase (RTK) inhibitor. On January 26, 2006, the agent was formally approved by the US FDA for the indications of treating renal cell carcinoma (RCC) and imatinib-resistant gastrointestinal stroma…

Kategori:
Angiogenesis InhibitorsAngiogenesis Modulating AgentsAntineoplastic Agents +31
Target Protein:
Platelet-derived growth factor receptor betaVascular endothelial growth factor receptor 1Mast/stem cell growth factor receptor Kit +6
Gen Terkait:
CYP3A4
Waktu ParuhFollowing administr…
Vol. Distribusi* 2230 L (apparent …
Klirens* 34 - 62 L/h [Tota…
Genetik 1 Varian
Sunobinop DB18955
small molecule | CAS: 1126793-40-5

Sunobinop is under investigation in clinical trial NCT04035200 (Safety, Tolerability and Efficacy Study of V117957 in Subjects With Insomnia Associated With Alcohol Cessation).

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Sunvozertinib DB18925
small molecule | CAS: 2370013-12-8

Sunvozertinib is under investigation in clinical trial NCT03974022 (Assessing an Oral EGFR Inhibitor, Sunvozertinib in Patients Who Have Advanced Non-small Cell Lung Cancer With EGFR or HER2 Mutation (WU-KONG1)).

Waktu Paruh-
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Supinoxin DB19010
small molecule | CAS: 888478-45-3

Supinoxin is under investigation in clinical trial NCT02003092 (RX-5902 Treatment of Subjects With Triple Negative Breast Cancer).

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Probable ATP-dependent RNA helicase DDX5
Waktu Paruh-
Vol. Distribusi-
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Suplatast DB19138
small molecule | CAS: 94055-75-1

Suplatast is under investigation in clinical trial NCT05983471 (Efficacy and Safety of ME-015 (Suplatast Tosilate) in Cough Related to Idiopathic Pulmonary Fibrosis (COSMIC-IPF)).

Kategori:
Anti-Allergic AgentsArylsulfonic AcidsHistamine Agents +6
Waktu Paruh-
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Suprofen Approved DB00870
small molecule | CAS: 40828-46-4

An ibuprofen-type anti-inflammatory analgesic and antipyretic. It inhibits prostaglandin synthesis and has been proposed as an anti-arthritic. It is no longer approved for use in the United States.

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAnalgesics +23
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2
Waktu Paruh-
Vol. Distribusi-
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Suptavumab DB12759
biotech | CAS: 1629615-23-1

Suptavumab has been used in trials studying the treatment and basic science of Respiratory Syncytial Virus Infections.

Waktu Paruh-
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Suramin DB04786
small molecule | CAS: 145-63-1

A polyanionic compound with an unknown mechanism of action. It is used parenterally in the treatment of African trypanosomiasis and it has been used clinically with diethylcarbamazine to kill the adult Onchocerca. (From AMA Drug Evaluations Annual, 1992, p164…

Kategori:
Agents Against Leishmaniasis and TrypanosomiasisAnti-Infective AgentsAntinematodal Agents +12
Target Protein:
HeparanaseP2Y purinoceptor 2NAD-dependent protein deacylase sirtuin-5, mitochondrial +5
Waktu ParuhApproximately 36 to…
Vol. Distribusi-
Klirens-
Genetik -
Suratadenoturev DB18672
biotech | CAS: 1268642-13-2

Suratadenoturev is a gene-modified oncolytic adenovirus expressing the telomerase reverse transcriptase gene.

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Surinabant DB13070
small molecule | CAS: 288104-79-0

Surinabant has been investigated for the treatment of Smoking Cessation.

Kategori:
Agents producing tachycardiaCannabinoid Receptor AntagonistsCannabinoids and similars +4
Target Protein:
Cannabinoid receptor 1
Waktu Paruh-
Vol. Distribusi-
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Surotomycin DB12076
small molecule | CAS: 1233389-51-9

Surotomycin has been used in trials studying the treatment of Diarrhea and Clostridium Difficile Infection. It is a benzenebutanoic acid derivative patented by Cubist Pharmaceuticals, Inc. as antibacterial agents for the treatment of Gram-positive infections.…

Kategori:
Amino Acids, Peptides, and ProteinsLipidsPeptides
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Surufatinib DB15106
small molecule | CAS: 1308672-74-3

Surufatinib is under investigation in clinical trial NCT02588170 (Phase III Study of Surufatinib in Treating Advanced Extrapancreatic Neuroendocrine Tumors).

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +4
Target Protein:
Fibroblast growth factor receptor 1Vascular endothelial growth factor receptor 2Vascular endothelial growth factor receptor 3 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
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SurVaxM DB17397
biotech | CAS: 2416847-76-0

Deskripsi belum tersedia.

Waktu Paruh-
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Survodutide DB18989
biotech | CAS: 2805997-46-8

Survodutide is under investigation in clinical trial NCT06077864 (A Study to Test the Effect of Survodutide (BI 456906) on Cardiovascular Safety in People With Overweight or Obesity (SYNCHRONIZE™ - CVOT)).

Kategori:
Amino Acids, Peptides, and Proteins
Waktu Paruh-
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Surzebiclimab DB16669
biotech | CAS: 2342597-90-2

Surzebiclimab is under investigation in clinical trial NCT03744468 (Study of BGB-A425 in Combination With Tislelizumab in Advanced Solid Tumors).

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Susoctocog alfa Approved DB11606
biotech | CAS: 1339940-90-7

Intravenous susoctocog alfa is a recombinant, B-domain deleted, porcine sequence antihaemophilic factor VIII (FVIII) product that has recently been approved for the treatment of bleeding episodes in adults with acquired haemophilia A (AHA). AHA is a rare blee…

Kategori:
Blood and Blood Forming OrgansBlood Coagulation FactorsHemostatics
Target Protein:
von Willebrand factor
Waktu ParuhThe terminal half-l…
Vol. DistribusiFollowing intraveno…
KlirensFollowing intraveno…
Genetik -
Sutetinib DB18841
small molecule | CAS: 1259519-20-4

Sutetinib is under investigation in clinical trial NCT05168566 (Study to Evaluate Sutetinib Maleate Capsule in Locally Advanced or Metastatic Non-small Cell Lung Cancer).

Waktu Paruh-
Vol. Distribusi-
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Sutilain Approved DB09379
biotech | CAS: 12211-28-8

Sutilain is a member of the keratase family which includes agents such as papain. It is able to dissolve the intercellular matrix which helps with desquamation. Sutilain contains proteolytic enzymes derived from _Bacillus subtilis_ and it is available as a cr…

Kategori:
EndopeptidasesEnzymesEnzymes and Coenzymes +4
Waktu ParuhThis pharmacokineti…
Vol. DistribusiThis pharmacokineti…
KlirensThis pharmacokineti…
Genetik -
Sutimlimab Approved DB14996
biotech | CAS: 2049079-64-1

Cold agglutinin disease (CAD) is a type of autoimmune hemolytic anemia (AIHA) in which autoantibodies directed against red blood cell surface antigens cause hemolysis at low (3-4°C) temperatures.[A245154,L40114] This cold subtype accounts for approximately 15…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +11
Target Protein:
Complement C1s subcomponent
Waktu ParuhAt the approved rec…
Vol. DistribusiAt steady-state, th…
KlirensAt the approved rec…
Genetik -
Suvecaltamide DB19139
small molecule | CAS: 953778-58-0

Suvecaltamide is under investigation in clinical trial NCT05122650 (A Study to Assess the Safety and Efficacy of JZP385 in the Treatment of Adults With Moderate to Severe Essential Tremor (ET)).

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SUVN-502 DB06140
small molecule | CAS: 701205-60-9

SUVN-502 is a novel, potent, safe, highly selective and orally active antagonist at a central nervous system serotonin receptor site 5-HT6 intended for treatment of cognitive disorders such as Alzheimer’s and Schizophrenia, an unmet medical need.

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsHeterocyclic Compounds, Fused-Ring +3
Target Protein:
5-hydroxytryptamine receptor 6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Suvodirsen DB17940
biotech | CAS: 2095270-67-8

Suvodirsen is an antisense oligonucleotide that has been investigated for the treatment of Duchenne muscular dystrophy.

Waktu Paruh-
Vol. Distribusi-
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Suvorexant Approved DB09034
small molecule | CAS: 1030377-33-3

Suvorexant is a selective dual antagonist of orexin receptors OX1R and OX2R that promotes sleep by reducing wakefulness and arousal. It has been approved for the treatment of insomnia.

Kategori:
Central Nervous System AgentsCentral Nervous System DepressantsCytochrome P-450 CYP3A Inhibitors +13
Target Protein:
Orexin/Hypocretin receptor type 1Orexin receptor type 2
Waktu ParuhMean half life is a…
Vol. DistribusiMean volume of dist…
Klirens-
Genetik -
Suvratoxumab DB15172
biotech | CAS: 1629620-18-3

Suvratoxumab is under investigation in clinical trial NCT02296320 (Study of the Efficacy and Safety of MEDI4893).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Suxibuzone DB13232
small molecule | CAS: 27470-51-5

Deskripsi belum tersedia.

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Suzetrigine DB18927
small molecule | CAS: 2649467-58-1

Suzetrigine is under investigation in clinical trial NCT05558410 (Evaluation of Efficacy and Safety of VX-548 for Acute Pain After an Abdominoplasty).

Waktu Paruh-
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SX-682 DB19210
small molecule | CAS: 1648843-04-2

SX-682 is under investigation in clinical trial NCT04574583 (Phase I/II Trial Investigating the Safety, Tolerability, Pharmacokinetics, Immune and Clinical Activity of SX-682 in Combination With Bintrafusp Alfa (M7824 or Tgf-beta "Trap"/pd-l1) With CV301 TRIC…

Target Protein:
C-X-C chemokine receptor type 2C-X-C chemokine receptor type 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SXR-1096 DB18119
small molecule | CAS: 1087624-28-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SY-5609 DB17099
small molecule | CAS: 2417302-07-7

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
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SYD-003 DB17106
small molecule | CAS: 249937-52-8

Deskripsi belum tersedia.

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SYNB1020 DB17667
biotech

SYNB1020 is an engineered strain of _Escherichia coli_ Nissle 1917 developed by Synlogic Inc. It was initially designed to convert ammonia to L-arginine [A258838] and granted orphan designation by the FDA for the treatment of urea cycle disorders in August 20…

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SYNB1353 DB17666
biotech

SYNB1353 is a strain of the probiotic bacteria _Escherichia coli_ (_E. coli_) type Nissle and an engineered probiotic drug.[A258833] Developed by Synlogic Operating Company, Inc., SYNB1353 is being investigated for the treatment of homocystinuria. It is desig…

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SYNB1891 DB17541
biotech

SYNB1891 is a live, modified strain of the probiotic _Escherichia coli_ Nissle engineered to produce cyclic di-AMP (CDA), a stimulator of the STING (STimulator of INterferon Genes) pathway.[A256733] SYNB1891 is under investigation in clinical trial NCT0416713…

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Synephrine DB09203
small molecule | CAS: 94-07-5

Synephrine, also referred to as, p-synephrine, is naturally occurring alkaloid. It is present in approved drug products as neo-synephrine, its m-substituted analog. p-synephrine and m-synephrine are known for their longer acting adrenergic effects compared to…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-Agonists +23
Target Protein:
Alpha-1 adrenergic receptors
Waktu Paruh-
Vol. Distribusi-
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SynKIR-110 DB17365
biotech

SynKIR-110 are autologous T cells genetically engineered to express an anti-mesothelin killer immunoglobulin-like receptor-chimeric antigen receptor (KIR-CAR).

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SynOV1.1 DB17539
biotech

SynOV1.1 is an investigational cancer immunotherapy developed by SyngenTech. It is a recombinant oncolytic adenovirus, controlled by synthetic gene circuit, encoding the human immunostimulating factor cytokine granulocyte-macrophage colony-stimulating factor …

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Genetik -
Synthetic camphor Approved DB14156
small molecule | CAS: 76-22-2

Deskripsi belum tersedia.

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Genetik -
small molecule

Synthetic conjugated estrogens A are composed of a blend of the following nine synthetic estrogenic substances: estrone sulfate, sodium equilin sulfate, sodium 17?-dihydroequilin sulfate, sodium 17?-estradiol sulfate, sodium 17?­ dihydroequilin sulfate, sodiu…

Kategori:
Cytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 SubstratesCytochrome P-450 Substrates +7
Target Protein:
Estrogen receptor
Waktu ParuhThe half life of ba…
Vol. DistribusiThe distribution of…
Klirens-
Genetik -
small molecule | CAS: 746658-13-9

Synthetic conjugated estrogens, B tablets contain a blend of ten synthetic estrogenic substances. The estrogenic substances are: sodium estrone sulfate, sodium equilin sulfate, sodium 17?-dihydroequilin sulfate, sodium 17?-estradiol sulfate, sodium 17?­ dihyd…

Kategori:
Cytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 SubstratesCytochrome P-450 Substrates +7
Target Protein:
Estrogen receptor
Waktu ParuhThe half life of ba…
Vol. DistribusiThe distribution of…
Klirens-
Genetik -
Syrosingopine Approved DB19379
small molecule | CAS: 84-36-6

Deskripsi belum tersedia.

Kategori:
AlkaloidsAntihypertensive AgentsHeterocyclic Compounds, Fused-Ring +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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