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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
Referensi
12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 209 / 252
small molecule | CAS: 1673571-51-1

Deskripsi belum tersedia.

Target Protein:
Tryptophan 5-hydroxylase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rofecoxib Approved DB00533
small molecule | CAS: 162011-90-7

Rofecoxib is used for the treatment of osteoarthritis, rheumatoid arthritis, acute pain in adults, and primary dysmenorrhea, as well as acute treatment of migraine attacks with or without auras. Rofecoxib is a solid. This compound belongs to the stilbenes. Th…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +29
Target Protein:
Prostaglandin G/H synthase 2Elastin
Waktu Paruh17 hours
Vol. Distribusi-
Klirens-
Genetik -
Roflumilast Approved DB01656
small molecule | CAS: 162401-32-3

Roflumilast is a highly selective phosphodiesterase-4 (PDE4) inhibitor.[A251385] PDE4 is a major cyclic-3',5?-adenosinemonophosphate (cyclic AMP, cAMP)-metabolizing enzyme [L37564] expressed on nearly all immune and pro-inflammatory cells, in addition to stru…

Kategori:
Acids, CarbocyclicAgents to Treat Airway DiseaseAmides +17
Target Protein:
cAMP-specific 3',5'-cyclic phosphodiesterase 4 (PDE4)
Waktu ParuhFollowing oral admi…
Vol. DistribusiFollowing a single …
KlirensPlasma clearance of…
Genetik -
Rogaratinib DB15078
small molecule | CAS: 1443530-05-9

Rogaratinib is under investigation in clinical trial NCT03762122 (Rogaratinib in Patients With Advanced Pretreated Squamous-cell Non-small Cell Lung Cancer (SQCLC)).

Kategori:
Sulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Roginolisib DB18088
small molecule | CAS: 1305267-37-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rokitamycin DB13409
small molecule | CAS: 74014-51-0

Deskripsi belum tersedia.

Kategori:
Anti-Bacterial AgentsAntibacterials for Systemic UseAntiinfectives for Systemic Use +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rolapitant Approved DB09291
small molecule | CAS: 552292-08-7

Rolapitant is a potent, highly selective, long-acting Neurokinin-1 (NK-1) receptor antagonist approved for the prevention of delayed chemotherapy-induced nausea and vomiting (CINV) in adults. Delayed-phase CINV typically occurs >24 hours after chemotherapy tr…

Kategori:
Alimentary Tract and MetabolismAntiemetics and AntinauseantsBCRP/ABCG2 Inhibitors +11
Target Protein:
Substance-P receptor
Waktu ParuhMean terminal half …
Vol. Distribusi460 L
Klirens0.96 L/hour
Genetik -
Rolicyclidine DB01549
small molecule | CAS: 2201-39-0

Rolicyclidine (PCPy) is classified as a dissociative anesthetic agent. It also has hallucinogenic and sedative properties. Because of its pharmacodynamic similarity to the drug phencyclidine (PCP), rolicyclidine was added to the Schedule I list of illegal dr…

Kategori:
Piperidines
Target Protein:
Glutamate receptor ionotropic, NMDA 3AD(2) dopamine receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rolipram DB01954
small molecule | CAS: 61413-54-5

A phosphodiesterase inhibitor with antidepressant properties.

Kategori:
Antidepressive AgentsCentral Nervous System AgentsCentral Nervous System Depressants +6
Target Protein:
cGMP-specific 3',5'-cyclic phosphodiesterase3',5'-cyclic-AMP phosphodiesterase 4AcAMP-specific 3',5'-cyclic phosphodiesterase 4 (PDE4) +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rolitetracycline Approved DB01301
small molecule | CAS: 751-97-3

A pyrrolidinylmethyl tetracycline.

Kategori:
Agents that produce neuromuscular block (indirect)Anti-Bacterial AgentsAnti-Infective Agents +4
Target Protein:
30S ribosomal protein S916S ribosomal RNA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rolofylline DB12670
small molecule | CAS: 136199-02-5

Rolofylline is under clinical development by pharmaceutical company NovaCardia for the treatment of congestive heart failure.

Kategori:
AlkaloidsDiureticsHeterocyclic Compounds, Fused-Ring +3
Target Protein:
Adenosine receptor A1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Roluperidone DB13080
small molecule | CAS: 359625-79-9

Roluperidone has been used in trials studying the treatment of Schizophrenia.

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsHeterocyclic Compounds, Fused-Ring +4
Target Protein:
Sigma intracellular receptor 25-hydroxytryptamine receptor 2A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Romidepsin Approved DB06176
small molecule | CAS: 128517-07-7

Romidepsin is a selective inhibitor of histone deacetylase, approved in the US in 2009 for the treatment of cutaneous T-cell lymphoma (CTCL) in patients who have received at least one prior systemic therapy.

Kategori:
Amino Acids, Peptides, and ProteinsAntibiotics, AntineoplasticAntineoplastic Agents +30
Target Protein:
Histone deacetylase 1Histone deacetylase 2Histone deacetylase 4 +3
Waktu ParuhApproximately 3 hou…
Vol. Distribusi44.5L
Klirens8.4L/h
Genetik -
Romifidine DB11543
small molecule | CAS: 65896-16-4

Romifidine is a veterinary drug utilized as a sedative primarily in large animals, most frequently horses. It is also used less commonly in a wide variety of other animal species. This drug's chemical structure closely resembles that of clonidine, however, ro…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-2 Receptor Agonists +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Romilkimab DB16318
biotech | CAS: 1399584-78-1

Romilkimab is under investigation in clinical trial NCT02345070 (Efficacy and Safety of SAR156597 in the Treatment of Idiopathic Pulmonary Fibrosis).

Target Protein:
Interleukin-13Interleukin-4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Romiplostim Approved DB05332
biotech | CAS: 267639-76-9

Romiplostim is a thrombopoiesis stimulating dimer Fc-peptide fusion protein (peptibody) to increase platelet production through activation of the thrombopoietin receptor. The peptibody molecule has two identical single-chain subunits, each one is made up of 2…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood and Blood Forming Organs +17
Target Protein:
Thrombopoietin receptor
Waktu ParuhImmune thrombocytop…
Vol. DistribusiIn healthy voluntee…
Klirens-
Genetik -
Romlusevimab DB16494
biotech | CAS: 2509447-08-7

Romlusevimab (BRII-198) was under investigation in clinical trials (NCT04479644 and NCT04691180) to treat COVID-19, focusing on its safety, tolerability, and pharmacokinetics.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Romosozumab Approved DB11866
biotech | CAS: 909395-70-6

Romosozumab is a humanized monoclonal antibody indicated for the treatment of osteoperosis in postmenopausal women at high risk of fracture and patients who have failed in other treatments or are intolerant to other osteoperosis therapies[L9554]. Romosozumab …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +12
Target Protein:
Sclerostin
Waktu Paruh12.8 days[L9554].
Vol. Distribusi3.92L[L9554].
Klirens0.38mL/hr/kg[L9554].
Genetik -
Ronacaleret DB05255
small molecule | CAS: 753449-67-1

Ronacaleret is a calcium-sensing receptor antagonist.

Kategori:
Acids, CarbocyclicIndenes
Target Protein:
Extracellular calcium-sensing receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Roneparstat DB17153
biotech | CAS: 1407492-04-9

Deskripsi belum tersedia.

Kategori:
CarbohydratesGlycosaminoglycansPolysaccharides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ronifibrate DB13460
small molecule | CAS: 42597-57-9

Deskripsi belum tersedia.

Kategori:
Agents Causing Muscle ToxicityFibric AcidsLipid Modifying Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ronnel DB11456
small molecule | CAS: 299-84-3

Deskripsi belum tersedia.

Kategori:
Organophosphorus CompoundsSulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ronopterin DB12575
small molecule | CAS: 185243-78-1

Ronopterin has been used in trials studying the treatment of Traumatic Brain Injury.

Kategori:
CoenzymesEnzymes and CoenzymesHeterocyclic Compounds, Fused-Ring +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rontalizumab DB12844
biotech | CAS: 948570-30-7

Rontalizumab has been used in trials studying the treatment of Systemic Lupus Erythematosus.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ropanicant DB19134
small molecule | CAS: 2414674-70-5

Ropanicant is under investigation in clinical trial NCT06126497 (Study Evaluating Safety and Efficacy of Ropanicant in MDD Patients).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ropeginterferon alfa-2b Approved DB15119
biotech | CAS: 1335098-50-4

Polycythemia vera (PV) is the most common Philadelphia chromosome-negative myeloproliferative neoplasm (MPN), characterized by increased hematocrit and platelet/leukocyte counts, an increased risk for hemorrhage and thromboembolic events, and a long-term prop…

Kategori:
Adjuvants, ImmunologicAlfa InterferonsAntineoplastic and Immunomodulating Agents +12
Target Protein:
Interferon alpha/beta receptor (IFNAR)
Waktu ParuhRopeginterferon alf…
Vol. DistribusiRopeginterferon alf…
KlirensRopeginterferon alf…
Genetik -
Ropidoxuridine DB06485
small molecule | CAS: 93265-81-7

Ropidoxuridine is a novel, orally available, thymidine analogue and prodrug for IUdR, which demonstrated a survival advantage in Phase II studies in anaplastic astrocytoma, a type of brain tumor.

Kategori:
Antineoplastic AgentsNucleic Acids, Nucleotides, and NucleosidesNucleosides +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ropinirole Approved DB00268
small molecule | CAS: 91374-21-9

Ropinirole, also known as _ReQuip_, is a non-ergoline dopamine agonist used in Parkinson's disease and restless legs syndrome [FDA label], [A174547]. It is manufactured by GlaxoSmithKline Pharmaceuticals. Ropinirole was initially approved in 1997 by the FDA…

Kategori:
Anti-Dyskinesia AgentsAnti-Parkinson Agents (Dopamine Agonist)Anti-Parkinson Drugs +10
Target Protein:
D(3) dopamine receptorD(2) dopamine receptorD(4) dopamine receptor +1
Waktu ParuhApproximately 6 hou…
Vol. DistribusiRopinirole is found…
KlirensThe clearance of ro…
Genetik -
Ropivacaine Approved DB00296
small molecule | CAS: 84057-95-4

Ropivacaine is an aminoamide local anesthetic drug marketed by AstraZeneca under the trade name Naropin. It exists as a racemate of its S- and R-enantiomers, although the marketed form is supplied only as the purified S-enantiomer.[L42140]

Kategori:
AmidesAminesAnesthetics +19
Target Protein:
Sodium channel protein type 10 subunit alpha
Waktu ParuhThe mean terminal h…
Vol. DistribusiFollowing intravasc…
KlirensFollowing intraveno…
Genetik -
Ropsacitinib DB18709
small molecule | CAS: 2127109-84-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 4159-77-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rosemary oil Approved DB14689
biotech | CAS: 8000-25-7

Deskripsi belum tersedia.

Kategori:
Biological ProductsLipidsOils +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rosiglitazone Approved DB00412
small molecule | CAS: 122320-73-4

Rosiglitazone is an anti-diabetic drug in the thiazolidinedione class of drugs. It is marketed by the pharmaceutical company GlaxoSmithKline as a stand-alone drug (Avandia) and in combination with metformin (Avandamet) or with glimepiride (Avandaryl). Like ot…

Kategori:
Alimentary Tract and MetabolismBlood Glucose Lowering AgentsBSEP/ABCB11 Substrates +33
Target Protein:
Peroxisome proliferator-activated receptor gammaLong-chain-fatty-acid--CoA ligase 4Peroxisome proliferator-activated receptor alpha +4
Waktu Paruh3-4 hours (single o…
Vol. Distribusi* 17.6 L [oral volu…
Klirens* Oral clearance (C…
Genetik -
Rosin Approved DB11165
biotech | CAS: 8050-09-7

Rosin is a solid form of resin obtained from pines and other plants, mostly conifers. It is prepared from heating fresh liquid resin to vaporize the volatile liquid terpene components. Rosin is used in various commercial and industrial applications, including…

Kategori:
Biological ProductsBiopolymersCell-mediated Immunity +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rosmarinic acid DB16865
small molecule | CAS: 20283-92-5

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAldehyde Reductase, antagonists & inhibitorsAnalgesics +22
Target Protein:
TyrosinaseInduced myeloid leukemia cell differentiation protein Mcl-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rosnilimab DB18851
biotech | CAS: 2412764-40-8

Rosnilimab is under investigation in clinical trial NCT06041269 (A Study of Efficacy and Safety of Rosnilimab in Subjects With Moderate to Severe Rheumatoid Arthritis (RENOIR)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rosomidnar DB17154
biotech | CAS: 871597-03-4

Deskripsi belum tersedia.

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesOligonucleotides +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rostafuroxin DB12350
small molecule | CAS: 156722-18-8

Rostafuroxin has been used in trials studying the treatment of Essential Hypertension.

Kategori:
AndrostanesFused-Ring CompoundsSteroids
Target Protein:
Sodium/potassium-transporting ATPase subunit beta-1Sodium/potassium-transporting ATPase subunit beta-2Sodium/potassium-transporting ATPase subunit beta-3 +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rostaporfin DB06659
small molecule | CAS: 284041-10-7

Deskripsi belum tersedia.

Kategori:
Biological FactorsDermatologicalsHeterocyclic Compounds, Fused-Ring +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rosuvastatin Approved DB01098
small molecule | CAS: 287714-41-4

Rosuvastatin, also known as the brand name product Crestor, is a lipid-lowering drug that belongs to the statin class of medications, which are used to lower the risk of cardiovascular disease and manage elevated lipid levels by inhibiting the endogenous prod…

Kategori:
Agents Causing Muscle ToxicityAlimentary Tract and MetabolismAmides +32
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductaseIntegrin alpha-L
Gen Terkait:
KIF6 HMGCR ABCG2
Waktu ParuhThe elimination hal…
Vol. DistribusiRosuvastatin underg…
Klirens-
Genetik 3 Varian
Rotavirus vaccine Approved DB10276
biotech

Rotavirus commonly infects children and infants causing severe diarrhea and vomiting leading to potentially fatal dehydration.[L1117] Two rotavirus vaccines are available for the prevention of rotavirus gastroenteritis, Rotateq and Rotarix. Rotateq is a live …

Kategori:
Actively Acquired ImmunityAntiinfectives for Systemic UseBiological Products +6
Waktu ParuhThe median duration…
Vol. Distribusi-
Klirens-
Genetik -
Rotenone DB11457
small molecule | CAS: 83-79-4

Rotenone is an isoflavone compound that naturally occurs in the jicama vine plant as well as many Fabaceae plants. It has broad spectrum insecticide and pesticide activity and is also toxic to fish.

Kategori:
AgrochemicalsBenzopyransChromones +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rotigaptide DB13067
small molecule | CAS: 355151-12-1

Rotigaptide is under investigation for the basic science of Heart Disease and Vascular Disease.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rotigotine Approved DB05271
small molecule | CAS: 99755-59-6

Rotigotine (Neupro) is a non-ergoline dopamine agonist indicated for the treatment of Parkinson's disease (PD) and restless legs syndrome (RLS) in Europe and the United States. It is formulated as a once-daily transdermal patch which provides a slow and const…

Kategori:
Agents that produce hypertensionAnti-Parkinson Agents (Dopamine Agonist)Anti-Parkinson Drugs +23
Target Protein:
D(3) dopamine receptorD(4) dopamine receptorD(2) dopamine receptor +4
Waktu ParuhAfter removal of th…
Vol. DistribusiThe weight normaliz…
Klirens-
Genetik -
Rovanersen DB16982
biotech | CAS: 2072901-32-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rovatirelin DB15338
small molecule | CAS: 204386-76-5

Rovatirelin is under investigation in clinical trial NCT01384435 (A Phase II Double Blind Comparative Study of KPS-0373 in Patients With Spinocerebellar Degeneration (SCD)).

Kategori:
Oxazoles
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rovazolac DB16320
small molecule | CAS: 1454288-88-0

Rovazolac is under investigation in clinical trial NCT03175354 (A Study in Subjects With Moderate Atopic Dermatitis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ROX-888 DB05364
small molecule

ROX-888 is ROXRO's lead compound which is currently in Phase 3 trials for the treatment of acute pain, including post-operative pain.

Target Protein:
C-C motif chemokine 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Roxadustat Approved DB04847
small molecule | CAS: 808118-40-3

Roxadustat is a first-in-class hypoxia-inducible factor prolyl hydroxylase inhibitor used to treat anemia associated with chronic kidney disease. It works by reducing the breakdown of the hypoxia-inducible factor (HIF), which is a transcription factor that st…

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAntianemic Preparations +10
Target Protein:
Egl nine homolog 1Prolyl hydroxylase EGLN2Prolyl hydroxylase EGLN3
Waktu ParuhThe mean effective …
Vol. DistribusiThe blood-to-plasma…
KlirensThe apparent total …
Genetik -
Menampilkan 10401–10450 dari 12560
Sebelumnya Halaman 209 / 252 Berikutnya