Hasil Filter

14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (14063)

Halaman 209 / 282
Palonosetron Approved DB00377
small molecule | CAS: 135729-56-5

Palonosetron (INN, trade name Aloxi) is an antagonist of 5-HT3 receptors that is indicated for the prevention and treatment of chemotherapy-induced nausea and vomiting (CINV). It is the most effective of the 5-HT3 antagonists in controlling delayed CINV nause…

Kategori:
Alimentary Tract and MetabolismAntidepressive AgentsAntiemetic Serotonin 5-HT3 Receptor Antagonists +22
Target Protein:
5-hydroxytryptamine receptor 3A
Waktu ParuhApproximately 40 ho…
Vol. Distribusi* 8.3 ± 2.5 L/kg
Klirens* 160 +/- 35 mL/h/kg
Genetik -
Palopegteriparatide Approved DB18676
biotech | CAS: 2222514-07-8

Palopegteriparatide is a parathyroid hormone (PTH) analog. Palopegteriparatide is a prodrug consisting of PTH(1-34) conjugated to a methoxy polyethylene glycol carrier (mPEG) via a proprietary TransCon Linker.[L51134] PTH(1-34) contains the N-terminal part of…

Kategori:
Calcium HomeostasisParathyroid Hormones and AnaloguesSystemic Hormonal Preparations, Excl. Sex Hormones and Insulins +1
Target Protein:
Parathyroid hormone/parathyroid hormone-related peptide receptor
Waktu ParuhThe apparent half-l…
Vol. DistribusiThe estimated appar…
KlirensThe estimated clear…
Genetik -
Palovarotene Approved DB05467
small molecule | CAS: 410528-02-8

Fibrodysplasia Ossificans Progressiva (FOP), with an estimated worldwide prevalence of one in 2 million individuals, is an exceptionally rare genetic disorder.[A244920] FOP is caused by a gain-of-function mutation in the ACVR1/ALK2 gene which results in progr…

Kategori:
BCRP/ABCG2 InhibitorsBenzene DerivativesBenzylidene Compounds +17
Target Protein:
Retinoic acid receptor gamma
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe mean (SD) appar…
KlirensThe apparent total …
Genetik -
Paltusotine DB16277
small molecule | CAS: 2172870-89-0

Paltusotine is under investigation in clinical trial NCT04261712 (A Study to Evaluate the Long-term Safety and Efficacy of Paltusotine for the Treatment of Acromegaly (ACROBAT Advance)).

Target Protein:
Somatostatin receptor type 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pam2csk4 DB16474
small molecule | CAS: 574741-81-4

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsDNA-Binding ProteinsExperimental Unapproved Treatments for COVID-19 +5
Target Protein:
Toll-like receptor 6Toll-like receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pamapimod DB19169
small molecule | CAS: 449811-01-2

Pamapimod is under investigation in clinical trial NCT05659459 (The KIN-FAST Trial (KIN001 for Accelerated Symptoms Termination) in Non Hospitalized Patients Infected With Sars-cov-2).

Kategori:
p38 Mitogen-Activated Protein Kinases, antagonists & inhibitorsPyridines
Target Protein:
Mitogen-activated protein kinase 14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pamidronic acid Approved DB00282
small molecule | CAS: 40391-99-9

Pamidronic acid is a second generation, nitrogen containing bisphosphonate similar to [neridronic acid] and [alendronic acid].[A203111] Pamidronic acid was first described in the literature in 1977.[A203267] The second generation bisphosphonates are less comm…

Kategori:
Agents Causing Muscle ToxicityAntineoplastic AgentsBisphosphonates +7
Target Protein:
Farnesyl pyrophosphate synthaseHydroxylapatiteGeranylgeranyl pyrophosphate synthase +2
Waktu ParuhThe mean eliminatio…
Vol. Distribusi-
KlirensThe mean total clea…
Genetik -
Pamiparib DB14769
small molecule | CAS: 1446261-44-4

Pamiparib is under investigation in clinical trial NCT03933761 (Pamiparib in Fusion Positive, Reversion Negative High Grade Serous Ovarian Cancer or Carcinosarcoma With BRCA1/2 Gene Mutations If Progression on Substrate Poly ADP Ribose Polymerase Inhibitbor (…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsEnzyme Inhibitors +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pamrevlumab DB14952
biotech | CAS: 946415-13-0

Pamrevlumab is under investigation in clinical trial NCT00913393 (Study of FibroGen (FG)-3019 in Subjects With Type 2 Diabetes Mellitus and Kidney Disease on ACEi and/or ARB Therapy).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Panax ginseng fruit is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
Biological ProductsGinseng & Ginseng ExtractsPlant Preparations
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Panax ginseng root oil is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
Biological ProductsGinseng & Ginseng ExtractsPlant Preparations
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Panax ginseng whole is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
AngiospermsAraliaceaeBiological Products +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Panax quinquefolius whole is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
Biological ProductsGinseng & Ginseng ExtractsPlant Preparations
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 59763-91-6

Pancreatic Polypeptide has been investigated for the treatment of Diabetes Mellitus, Type 1.

Kategori:
Amino Acids, Peptides, and ProteinsGastrointestinal AgentsHormones +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pancrelipase Approved DB00085
biotech | CAS: 53608-75-6

Pancrelipase, in general, is composed of a mixture of pancreatic enzymes which include amylases, lipases, and proteases. These enzymes are extracted from porcine pancreatic glands.[L2509] The pancrelipase mixture was developed by Ortho-McNeil-Janssen Pharmace…

Kategori:
Alimentary Tract and MetabolismCarboxylic Ester HydrolasesComplex Mixtures +10
Target Protein:
Dietary fatDietary proteinDietary starch
Waktu ParuhPancrelipase acts l…
Vol. DistribusiPancrelipase acts l…
KlirensPancrelipase acts l…
Genetik -
Pancrelipase amylase Approved DB11065
biotech | CAS: 9000-90-2

Pancrelipase, in general, is composed of a mixture of pancreatic enzymes which include amylases, lipases, and proteases. These enzymes are extracted from porcine pancreatic glands.[L2509] The amylases are enzymes that help in the chemical process of digestion…

Kategori:
AmylasesAmylases, antagonists & inhibitorsEnzymes +3
Target Protein:
Dietary starch
Waktu ParuhPlease refer to [DB…
Vol. DistribusiPlease refer to [DB…
KlirensPlease refer to [DB…
Genetik -
Pancrelipase lipase Approved DB13147
biotech | CAS: 9001-62-1

Pancrelipase, in general, is composed of a mixture of pancreatic enzymes which include amylases, lipases, and proteases. These enzymes are extracted from porcine pancreatic glands.[L2509] The pancrelipase lipase is an enzyme secreted by the pancreas that is r…

Kategori:
Carboxylic Ester HydrolasesEnzymesEnzymes and Coenzymes +4
Target Protein:
Dietary fat
Waktu ParuhPlease refer to [DB…
Vol. DistribusiPlease refer to [DB…
KlirensPlease refer to [DB…
Genetik -
Pancrelipase protease Approved DB11066
biotech | CAS: 9001-94-9

Pancrelipase, in general, is composed of a mixture of pancreatic enzymes which include amylases, lipases, and proteases. These enzymes are extracted from porcine pancreatic glands.[L2509] The pancrelipase protease is a mix of enzymes, formed by trypsin and ch…

Kategori:
EnzymesEnzymes and CoenzymesHydrolases +1
Target Protein:
Dietary protein
Waktu ParuhPlease refer to [DB…
Vol. DistribusiPlease refer to [DB…
KlirensPlease refer to [DB…
Genetik -
Panitumumab Approved DB01269
biotech | CAS: 339177-26-3

Panitumumab (ABX-EGF) is a recombinant human IgG2 monoclonal antibody that binds specifically to the human epidermal growth factor receptor (EGFR). This drug is an antineoplastic agent. Panitumumab was granted FDA approval on 27 September 2006.[L17663]

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +16
Target Protein:
Epidermal growth factor receptor
Waktu Paruh7.5 days (range: 4-…
Vol. Distribusi-
Klirens* 4.9+/- 1.4 mL/kg/…
Genetik -
Panobacumab DB15342
biotech | CAS: 885053-97-4

Panobacumab is under investigation in clinical trial NCT00851435 (Safety and Pharmacokinetics of KBPA-101 in Hospital Acquired Pneumonia Caused by O11 Pseudomonas Aeruginosa).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Panobinostat Approved DB06603
small molecule | CAS: 404950-80-7

Panobinostat is an oral deacetylace (DAC) inhibitor approved on February 23, 2015 by the FDA for the treatment of multiple myeloma. The approval was accelerated based on progression-free survival, therefore confirmatory trials by the sponsor to demonstrate cl…

Kategori:
AminesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +21
Target Protein:
Histone deacetylase 1Histone deacetylase
Waktu Paruh30 hours
Vol. Distribusi-
Klirens-
Genetik -
Pantethine Approved DB11190
small molecule | CAS: 16816-67-4

Pantethine is a naturally occurring compound synthesized in the body from pantothenic acid (vitamin B5) via addition of cysteamine. It consists of two molecules of pantetheine that form a dimer via disufide linkages, and acts as an intermediate in the product…

Kategori:
Alimentary Tract and MetabolismSulfhydryl CompoundsSulfur Compounds +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Panthenol Approved DB11204
small molecule | CAS: 16485-10-2

Panthenol is an alcohol derivative of pantothenic acid, a component of the B complex vitamins and an essential component of a normally functioning epithelium. Panthenol exists as a racemic mixture containing both the dextrorotatory form (dexpanthenol) and the…

Kategori:
AlanineAmino AcidsAmino Acids, Peptides, and Proteins +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pantoprazole Approved DB00213
small molecule | CAS: 102625-70-7

Pantoprazole is a first-generation proton pump inhibitor (PPI) used for the management of gastroesophageal reflux disease (GERD), for gastric protection to prevent recurrence of stomach ulcers or gastric damage from chronic use of NSAIDs, and for the treatmen…

Kategori:
2-PyridinylmethylsulfinylbenzimidazolesAcid ReducersAlimentary Tract and Metabolism +27
Target Protein:
Potassium-transporting ATPase alpha chain 1Potassium-transporting ATPase subunit betaN(G),N(G)-dimethylarginine dimethylaminohydrolase 1
Waktu ParuhAbout 1 hour[F3202]
Vol. DistribusiThe apparent volume…
Klirens**Adults**: With in…
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Phosphopantothenoylcysteine decarboxylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Acetyl-CoA acetyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Pantothenate synthetase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Papain Approved DB11193
biotech | CAS: 9001-73-4

Papain, also known as papaya proteinase I, is a cysteine protease (EC 3.4.22.2) enzyme that is found in species of papaya, _Carica papaya_ and _Vasconcellea cundinamarcensis_. The enzyme is found to be localized in the skin of papaya, and is collected from sl…

Kategori:
Cysteine EndopeptidasesCysteine ProteasesEndopeptidases +6
Target Protein:
Toll-like receptor 4
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Papaverine Approved DB01113
small molecule | CAS: 58-74-2

An alkaloid found in opium but not closely related to the other opium alkaloids in its structure or pharmacological actions. It is a direct-acting smooth muscle relaxant used in the treatment of impotence and as a vasodilator, especially for cerebral vasodila…

Kategori:
Alimentary Tract and MetabolismAlkaloidsBenzylisoquinolines +18
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4DcGMP-specific 3',5'-cyclic phosphodiesterase3',5'-cyclic-AMP phosphodiesterase 4B +2
Waktu Paruh0.5-2 hours
Vol. Distribusi-
Klirens-
Genetik -
Paquinimod DB13118
small molecule | CAS: 248282-01-1

Paquinimod is developed for the treatment of SLE (Systemic Lupus Erythematosus), which is an autoimmune disease. The disease affects mainly women of fertile age and progresses in flares with relatively symptom free periods in between. Current treatments of SL…

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Protein S100-A9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 873-75-6

Deskripsi belum tersedia.

Kategori:
AlcoholsBenzene DerivativesBenzyl Compounds
Target Protein:
Alcohol dehydrogenase 1C
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Estrogen receptor betaGalectin-10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Paraldehyde Approved DB09117
small molecule | CAS: 123-63-7

Paraldehyde was initially introduced into medical practice in the United Kingdom in 1882 by the Italian physician Vincenzo Cervello. It is classified as a central nervous system (CNS) depressant and has also been found to be an effective anticonvulsant, hypno…

Kategori:
AcetaldehydeAnticonvulsantsCentral Nervous System Agents +4
Waktu ParuhThe mean half life …
Vol. Distribusi-
Klirens-
Genetik -
Paramethasone acetate Approved DB14657
small molecule | CAS: 1597-82-6

Deskripsi belum tersedia.

Kategori:
Fused-Ring CompoundsPregnadienesPregnadienetriols +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Parasorbic acid DB14121
small molecule | CAS: 10048-32-5

Sole constituent of "Vogelbeerol" oil obtained by steam distillation of the acidified juice of the ripe berries of the mountain ash.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Parathiazine DB15978
small molecule | CAS: 84-08-2

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingSulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Parathyroid hormone Approved DB05829
biotech | CAS: 9002-64-6

Parathyroid hormone (PTH) is a single-chain polypeptide composed of 84 amino acids. Available as Preotact, it is an identical form of human recombinant hormome which produced as a fusion protein undergoeing post-translational processing involving the cleava…

Kategori:
Amino Acids, Peptides, and ProteinsCalcium HomeostasisCalcium-Regulating Hormones and Agents +7
Target Protein:
Parathyroid hormone 2 receptorParathyroid hormone/parathyroid hormone-related peptide receptor
Waktu Paruh1.5 hours.
Vol. DistribusiThe volume of distr…
Klirens-
Genetik -
biotech | CAS: 172867-62-8

Parathyroid Hormone-Related Protein 1-36 is under investigation in clinical trial NCT00853723 (Comparison Study of Pthrp and PTH to Treat Osteoporosis).

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsHormones +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pardoprunox DB12061
small molecule | CAS: 269718-84-5

Pardoprunox has been used in trials studying the treatment of Early Stage Parkinson's Disease and Advanced Stage Parkinson's Disease. Pardoprunox is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
D(2) dopamine receptorD(3) dopamine receptorD(4) dopamine receptor +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Parecoxib Approved DB08439
small molecule | CAS: 198470-84-7

Parecoxib is a water-soluble and injectable prodrug of valdecoxib. It is marketed as Dynastat in the European Union. Parecoxib is a COX2 selective inhibitor in the same category as celecoxib (Celebrex) and rofecoxib (Vioxx). As it is injectable, it can be use…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +18
Target Protein:
Prostaglandin G/H synthase 2Lactotransferrin
Waktu Paruh22 minutes (parecox…
Vol. Distribusi-
Klirens-
Genetik -
Parethoxycaine DB19380
small molecule | CAS: 94-23-5

Parethoxycaine is a local anesthetic that was previously approved in the US.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pargyline Approved DB01626
small molecule | CAS: 555-57-7

Pargyline is a monoamine oxidase inhibitor with antihypertensive properties.

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAmines +12
Target Protein:
Amine oxidase [flavin-containing] BAmine oxidase [flavin-containing] A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Paricalcitol Approved DB00910
small molecule | CAS: 131918-61-1

Paricalcitol is a synthetic vitamin D analog. Paricalcitol has been used to reduce parathyroid hormone levels. Paricalcitol is indicated for the prevention and treatment of secondary hyperparathyroidism associated with chronic renal failure.

Kategori:
Anti-Parathyroid AgentsBone Density Conservation AgentsCalcium Homeostasis +16
Target Protein:
Vitamin D3 receptor
Waktu Paruh4 to 6 hours
Vol. Distribusi* 30.8 ± 7.5 L [CKD…
Klirens* 1.49 +/- 0.60 L/h…
Genetik -
biotech | CAS: 2259927-72-3

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Paritaprevir Approved DB09297
small molecule | CAS: 1216941-48-8

Paritaprevir is a direct acting antiviral medication used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV). HCV is a single-stranded RNA virus that is categorized into ni…

Kategori:
AmidesAmino AcidsAmino Acids, Cyclic +27
Target Protein:
Genome polyproteinGag-Pol polyprotein
Waktu Paruh5.5 hr [FDA Label]
Vol. DistribusiVolume of distribut…
Klirens-
Genetik -
Parnaparin Approved DB09260
small molecule | CAS: 9005-49-6

Parnaparin is an heparin of low molecular weight with antithrombotic effects.

Kategori:
Agents causing hyperkalemiaAnticoagulantsBlood and Blood Forming Organs +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Paromomycin Approved DB01421
small molecule | CAS: 7542-37-2

An oligosaccharide antibiotic produced by various streptomyces. [PubChem]

Kategori:
Agents that produce neuromuscular block (indirect)Alimentary Tract and MetabolismAmebicides +10
Target Protein:
30S ribosomal protein S1016S ribosomal RNASmall ribosomal subunit protein uS2 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Paroxetine Approved DB00715
small molecule | CAS: 61869-08-7

Paroxetine is a selective serotonin reuptake inhibitor (SSRI) drug commonly known as Paxil. It has a variety of uses, including the treatment of anxiety disorders, major depression, posttraumatic stress disorder, and symptoms of menopause, among others.[T653]…

Kategori:
Agents producing tachycardiaAnticholinergic AgentsAntidepressive Agents +39
Target Protein:
Sodium-dependent serotonin transporterSodium-dependent noradrenaline transporter5-hydroxytryptamine receptor 2A +9
Gen Terkait:
ABCB1 CYP2D6 CYP2D6 +4
Waktu ParuhThe mean eliminatio…
Vol. DistribusiParoxetine has a la…
KlirensThe apparent oral c…
Genetik 7 Varian
PARPI F-18 DB18657
small molecule | CAS: 1883580-48-0

PARPI F-18 is a diagnostic agent under investigation for use in the management of glioblastoma multiforme.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Parsaclisib DB14867
small molecule | CAS: 1426698-88-5

Parsaclisib is under investigation in clinical trial NCT03126019 (An Open-Label Study of Parsaclisib in Relapsed or Refractory Follicular Lymphoma (CITADEL-203)).

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsPhosphatidylinositol-3-kinase (Pi3K) inhibitors +1
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 10401–10450 dari 14063
Sebelumnya Halaman 209 / 282 Berikutnya