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17430

Total database: 17430
Struktur (SMILES)
12313 (70.6%)
Target
9368 (53.7%)
Genomik
112 (0.6%)
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17430 (100.0%)

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Halaman 208 / 349
Lorecivivint DB14883
small molecule | CAS: 1467093-03-3

Lorecivivint is under investigation in clinical trial NCT03246399 (A Study of the Safety, Tolerability, and Pharmacokinetics of SM04690 Injectable Suspension Following Single Intradiscal Injection in Subjects With Degenerative Disc Disease).

Kategori:
Anti-Inflammatory AgentsHeterocyclic Compounds, Fused-RingPyrazoles
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lorigerlimab DB18942
biotech | CAS: 2416595-46-3

Lorigerlimab is under investigation in clinical trial NCT05848011 (A Study of Lorigerlimab With Docetaxel or Docetaxel Alone in Participants With Metastatic Castration-resistant Prostate Cancer).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Lorlatinib Approved DB12130
small molecule | CAS: 1454846-35-5

Lorlatinib is a third-generation ALK tyrosine kinase inhibitor (TKI) for patients with ALK-positive metastatic non-small cell lung cancer[L39905] which was first approved by the US FDA in November of 2018. It was subsequently approved by the EMA in 2019 for t…

Kategori:
AmidesAminesAnaplastic lymphoma kinase (ALK) inhibitors +31
Target Protein:
Proto-oncogene tyrosine-protein kinase ROSALK tyrosine kinase receptor
Waktu ParuhThe mean plasma hal…
Vol. DistribusiThe mean (CV%) stea…
KlirensThe mean oral clear…
Genetik -
Lormetazepam Approved DB13872
small molecule | CAS: 848-75-9

Lormatazepam is an orally available benzodiazepine used in the UK for the treatment of short-term insomnia [L927]. It is marketed by Auden Mckenzie (Pharma Division) in 0.5 and 1 mg tablet formulations.

Kategori:
BenzazepinesBenzodiazepines and benzodiazepine derivativesBenzodiazepinones +6
Target Protein:
GABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site
Waktu ParuhThe terminal phase …
Vol. Distribusi-
Klirens-
Genetik -
Lornoxicam Approved DB06725
small molecule | CAS: 70374-39-9

Lornoxicam (chlortenoxicam) is a new nonsteroidal anti-inflammatory drug (NSAID) of the oxicam class with analgesic, anti-inflammatory and antipyretic properties. Lornoxicam differs from other oxicam compounds in its potent inhibition of prostaglandin biosynt…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +17
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2
Waktu Paruh3-5 hours
Vol. Distribusi-
Klirens-
Genetik -
Lorpiprazole Approved DB09195
small molecule | CAS: 108785-69-9

Lorpiprazole is a serotonin antagonist and reuptake inhibitor used for the treatment of major depressive disorder.[A31634] It is a piperazinyl-triazole derivative.[T83]

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsCytochrome P-450 CYP2D6 Substrates +10
Target Protein:
5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 2CAlpha-1 adrenergic receptors +3
Waktu ParuhThe estimated half-…
Vol. DistribusiThe serotonin antag…
Klirens-
Genetik -
Lortalamine DB09187
small molecule | CAS: 70384-91-7

Lortalamine (LM-1404) is a selective norepinephrine reuptake inhibitor developed in the 1980s. This drug never made it past clinical trials, likely due to ocular toxicity in animals, but has been used in positron emission tomography studies to label norepinep…

Kategori:
Adrenergic Uptake InhibitorsAntidepressive AgentsCentral Nervous System Depressants +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lorukafusp alfa DB15443
biotech | CAS: 2131168-99-3

Lorukafusp alfa is under investigation in clinical trial NCT01334515 (Biological Therapy, Sargramostim, and Isotretinoin in Treating Patients With Relapsed or Refractory Neuroblastoma).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBiological Factors +11
Waktu Paruh-
Vol. Distribusi-
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Lorundrostat DB18957
small molecule | CAS: 1820940-17-7

Lorundrostat is under investigation in clinical trial NCT06153693 (Efficacy and Safety of Lorundrostat in Subjects With Uncontrolled and Resistant Hypertension).

Waktu Paruh-
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biotech | CAS: 1008106-64-6

Lorvotuzumab mertansine has been used in trials studying the treatment of SCLC, Leukemia, Ovarian Cancer, Multiple Myeloma, and Merkel Cell Carcinoma, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAntibodies +29
Waktu Paruh-
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Klirens-
Genetik -
Losartan Approved DB00678
small molecule | CAS: 114798-26-4

Losartan is an angiotensin II receptor blocker (ARB) used to treat hypertension.[L7423] Angiotensin-converting enzyme (ACE) inhibitors are used for a similar indication but are associated with a cough.[L7423] When patients with ACE inhibitor associated coughs…

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing angioedemaAgents causing hyperkalemia +39
Target Protein:
Erythropoietin receptorType-1 angiotensin II receptor
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe volume of distr…
KlirensLosartan has a tota…
Genetik -
Losmapimod DB12270
small molecule | CAS: 585543-15-3

Losmapimod has been investigated for the prevention of Chronic Obstructive Pulmonary Disease.

Kategori:
Cycloparaffinsp38 Mitogen-Activated Protein KinasesProtein Kinase Inhibitors
Target Protein:
Mitogen-activated protein kinase 14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Loteprednol Approved DB00873
small molecule | CAS: 129260-79-3

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesAndrostadienesAndrostanes +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Loteprednol etabonate Approved DB14596
small molecule | CAS: 82034-46-6

Loteprednol Etabonate (LE) is a topical corticoid anti-inflammatory. It is used in ophthalmic solution for the treatment of steroid responsive inflammatory conditions of the eye such as allergic conjunctivitis, uveitis, acne rosacea, superficial punctate kera…

Kategori:
Adrenal Cortex HormonesAndrostadienesAndrostanes +9
Target Protein:
Steroid hormone receptor ERR1Steroid hormone receptor ERR2Estrogen-related receptor gamma +1
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe only data avail…
KlirensLoteprednol etabona…
Genetik -
Lotilaner Approved DB17992
small molecule | CAS: 1369852-71-0

Lotilaner is an ectoparasiticide that is a member of the isoxazoline family of compounds.[L47546] Lotilaner has largely been used for veterinary uses as an antiparasitic agent to treat flea and tick infestations in animals.[A260746, L47556] Lotilaner consists…

Kategori:
Antiparasitic AgentsEctoparasiticideEctoparasiticides, Incl. Scabicides +2
Target Protein:
Gaba-gated chloride channel, putative
Waktu ParuhThe effective half-…
Vol. DistribusiNo information is a…
KlirensNo information is a…
Genetik -
Lovastatin Approved DB00227
small molecule | CAS: 75330-75-5

Lovastatin, also known as the brand name product Mevacor, is a lipid-lowering drug and fungal metabolite derived synthetically from a fermentation product of _Aspergillus terreus_.[A174550] Originally named Mevinolin, lovastatin belongs to the statin class of…

Kategori:
Agents Causing Muscle ToxicityAnticholesteremic AgentsBSEP/ABCB11 Substrates +21
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductaseIntegrin alpha-LHistone deacetylase 2
Waktu ParuhLovastatin half-lif…
Vol. DistribusiLovastatin is able …
Klirens-
Genetik -
Lovotibeglogene autotemcel Approved DB18680
biotech

Lovotibeglogene autotemcel consists of autologous hematopoietic stem and progenitor cells transduced with the BB305 lentiviral vector encoding a modified ?-globin gene. Specifically, lovotibeglogene autotemcel provides a functional copy of a modified beta-glo…

Kategori:
Autologous Cultured CellAutologous Hematopoietic Stem Cell-Based Gene TherapyGenetic Therapy
Target Protein:
Hemoglobin subunit beta
Waktu ParuhLovotibeglogene aut…
Vol. DistribusiLovotibeglogene aut…
KlirensLovotibeglogene aut…
Genetik -
biotech

Ingredient used in over-the-counter medications.

Waktu Paruh-
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Genetik -
Loxapine Approved DB00408
small molecule | CAS: 1977-10-2

An antipsychotic agent used in schizophrenia. [PubChem]

Kategori:
Antidepressive AgentsAntipsychotic AgentsAntipsychotic Agents (First Generation [Typical]) +24
Target Protein:
5-hydroxytryptamine receptor 2AD(2) dopamine receptor5-hydroxytryptamine receptor 2C +30
Waktu ParuhOral-4 hours
Vol. Distribusi-
Klirens-
Genetik -
Loxicodegol DB14146
small molecule | CAS: 1211231-76-3

Loxicodegol was developed by Nektar Therapeutics as an opioid analgesic with low abuse potential for the treatment of chronic pain [L3263]. The lack of abuse potential is believed to be due to the drug's slow rate of entry into brain, a unique characteristic …

Kategori:
AlkaloidsHeterocyclic Compounds, Fused-RingOpiate Alkaloids +1
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorKappa-type opioid receptor
Waktu ParuhLoxicodegol has a h…
Vol. DistribusiLoxicodegol has a s…
KlirensLoxicodegol has a c…
Genetik -
Loxoprofen Approved DB09212
small molecule | CAS: 68767-14-6

Loxoprofen is a propionic acid derivative non-steroidal anti-inflammatory drug. It is marketed under the trade name Loxonin in Brazil, Mexico and Japan by Sankyo, as Loxomac in India, and as Oxeno in Argentina. A transdermal preparation was approved for use i…

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +13
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu ParuhThe elimination hal…
Vol. DistribusiLoxoprofen has a vo…
KlirensMost of the drug as…
Genetik -
Loxoribine DB17589
small molecule | CAS: 121288-39-9

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingNucleic Acids, Nucleotides, and NucleosidesNucleosides +3
Target Protein:
Toll-like receptor 7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LP-184 DB18215
small molecule | CAS: 924835-67-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
LP-2307 DB17470
biotech

LP-2307 is an investigational allogeneic large multivalent immunogen (LMI) vaccine developed by Avanir. It was investigated for melanoma.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
LP-284 DB18006
small molecule | CAS: 2412580-47-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lpc-Ether DB03633
small molecule

Deskripsi belum tersedia.

Target Protein:
Phospholipase A2Ganglioside GM2 activator
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LPT-99 DB17142
small molecule | CAS: 1263477-83-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LS11 DB05918
small molecule

LS11(talaporfin sodium) is an agent consisting of chlorin e6, derived from chlorophyll, and L-aspartic acid with photosensitizing activity. After intratumoral activation by light emitting diodes, taporfin sodium forms an extended high energy conformational st…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
LSALT Peptide DB16472
biotech

Deskripsi belum tersedia.

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LSP-GR3 DB16934
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
LSTA1 DB17346
biotech | CAS: 1392278-76-0

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
LSZ-102 DB15362
small molecule | CAS: 2135600-76-7

LSZ-102 is under investigation in clinical trial NCT02734615 (Phase I/Ib Trial of LSZ102 Single Agent or LSZ102 + LEE011 or LSZ102 + BYL719 in ER+ Breast Cancers).

Kategori:
Sulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LT2003 DB18359
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LTI-03 DB18491
biotech | CAS: 1504575-10-3

LTI-03 is a caveolin-1 Scaffolding Domain 7-Mer

Waktu Paruh-
Vol. Distribusi-
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Genetik -
LTX-109 DB12711
small molecule | CAS: 1166254-80-3

LTX-109 has been investigated for the treatment of Atopic Dermatitis, Mild Eczema/Dermatoses, and Gram-positive, Skin Infections.

Kategori:
Amino Acids, Peptides, and ProteinsPeptidesPeptidomimetics
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LTX-315 DB12748
small molecule | CAS: 1345407-05-7

LTX-315 has been used in trials studying the treatment of Cancer, Lymphoma, Melanoma, Carcinoma, and Breast Cancer, among others.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LU-31130 DB05828
small molecule

LU-31130 is a rapid acting therapy developed by H. Lundbeck A/S to treat Psychosis, Schizophrenia and Schizoaffective Disorders. It acts at the Dopamine D4 receptors in the cortex and has low affinity for D2 receptors, adrenoceptors, muscarinic and histaminer…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Lubazodone DB09196
small molecule | CAS: 161178-07-0

Lubazodone (YM-992, YM-35,995) is an arylpiperazine antidepressant which was being developed as a treatment for depression and obsessive compulsive disorder, and reached phase II clinical trials, but was discontinued. It acts as a serotonin reuptake inhibitor…

Kategori:
Oxazines
Target Protein:
5-hydroxytryptamine receptor 2ASodium-dependent serotonin transporter
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lubiprostone Approved DB01046
small molecule | CAS: 136790-76-6

Lubiprostone is a medication used in the management of idiopathic chronic constipation. A prostaglandin E1 derivative, lubiprostone is a bicyclic fatty acid that activates ClC-2 chloride channels located on the apical side of the gastrointestinal epithelial c…

Kategori:
Alimentary Tract and MetabolismChloride Channel AgonistsDrugs for Constipation +9
Target Protein:
Chloride channel protein 2
Waktu Paruh0.9 to 1.4 hours
Vol. Distribusi-
Klirens-
Genetik -
Lucanthone DB04967
small molecule | CAS: 479-50-5

One of the schistosomicides, it has been replaced largely by hycanthone and more recently praziquantel. (From Martindale The Extrapharmacopoeia, 30th ed., p46). It is currently being tested as a radiation sensitizer.

Kategori:
AnthelminticsAnti-Infective AgentsAntiparasitic Agents +7
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-betaDNA repair nuclease/redox regulator APEX1 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lucatumumab DB06360
biotech | CAS: 903512-50-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Target Protein:
Tumor necrosis factor receptor superfamily member 5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lucerastat DB14872
small molecule | CAS: 141206-42-0

Lucerastat is under investigation in clinical trial NCT03425539 (Efficacy and Safety of Lucerastat Oral Monotherapy in Adult Subjects With Fabry Disease).

Kategori:
AlkaloidsCarbohydratesImines +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lucinactant Approved DB04897
biotech | CAS: 825600-90-6

Lucinactant is a new synthetic peptide-containing surfactant for intratracheal use. It contains sinapultide, a novel, hydrophobic, 21-amino acid peptide (leucine and lysine repeating units, KL4 peptide) designed to mimic human surfactant protein-B (SB-P). Mor…

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsBiological Factors +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lucitanib DB11845
small molecule | CAS: 1058137-23-7

Lucitanib has been used in trials studying the treatment of ER+, MBC, SCLC, HER2+, and NSCLC, among others.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Fibroblast growth factor receptor 1Fibroblast growth factor receptor 2Vascular endothelial growth factor receptor 2 +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lufenuron DB11424
small molecule | CAS: 103055-07-8

Lufenuron is used in veterinary for the control of flea.

Kategori:
Acids, CarbocyclicAgrochemicalsAmides +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Luliconazole Approved DB08933
small molecule | CAS: 187164-19-8

Luliconazole is a topical antifungal agent that acts by unknown mechanisms but is postulated to involve altering the synthesis of fungi cell membranes. It was approved by the FDA (USA) in November 2013 and is marketed under the brand name Luzu. Luliconazole i…

Kategori:
Anti-Infective AgentsAntifungal AgentsAntifungals for Dermatological Use +10
Target Protein:
Lanosterol 14-alpha demethylase
Waktu ParuhThe half life of lu…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of lu…
Genetik -
Lulizumab pegol DB15441
biotech | CAS: 1421830-13-8

Lulizumab pegol is under investigation in clinical trial NCT02843659 (Proof of Concept Study to Evaluate the Efficacy and Safety of BMS-931699 (Lulizumab) or BMS-986142 in Primary Sjögren's Syndrome).

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsAntibodies, Monoclonal +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LuLym-T DB17405
biotech

LuLym-T is an investigational autologous immune cell therapy consisting of activated T Lymphocytes. Developed by Lukas Biomedical, Inc., it is currently being investigated in hepatocellular carcinoma.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Lumacaftor Approved DB09280
small molecule | CAS: 936727-05-8

Lumacaftor is a drug used in combination with [DB08820] as the fixed dose combination product Orkambi for the management of Cystic Fibrosis (CF) in patients aged 6 years and older. Cystic Fibrosis is an autosomal recessive disorder caused by one of several di…

Kategori:
AminesCytochrome P-450 CYP2B6 InducersCytochrome P-450 CYP2B6 Inducers (strength unknown) +21
Target Protein:
Cystic fibrosis transmembrane conductance regulator
Waktu ParuhThe half-life of lu…
Vol. DistribusiFollowing oral admi…
KlirensThe typical apparen…
Genetik -
Lumasiran Approved DB15935
biotech | CAS: 1834610-13-7

Lumasiran is a small interfering RNA used in the treatment of primary hyperoxaluria type 1 (PH1).[L23554] This condition, caused by a deficiency in the enzyme alanine-glyoxylate aminotransferase, leads to an accumulation of oxalate, causing calcium crystal fo…

Kategori:
Alimentary Tract and MetabolismAntisense Elements (Genetics)Cytochrome P-450 CYP2C8 Inhibitors +12
Target Protein:
2-Hydroxyacid oxidase 1
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe apparent centra…
KlirensThe apparent plasma…
Genetik -
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