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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

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Distribusi Wujud Zat

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Hasil Pencarian (14063)

Halaman 208 / 282
small molecule | CAS: 90736-23-5

p-Fluorofentanyl is an opioid analgesic being an analogue of fentanyl developed by Janssen Pharmaceutica in the 1960s. p-Fluorofentanyl was sold briefly on the US black market in the early 1980s, before the introduction of the Federal Analog Act which for the…

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small molecule | CAS: 123-08-0

Deskripsi belum tersedia.

Kategori:
Aldehydes
Target Protein:
4-aminobutyrate aminotransferase, mitochondrialAmine oxidase [flavin-containing] B
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small molecule | CAS: 1126-48-3

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicBenzene DerivativesBenzoates +9
Target Protein:
Carbonic anhydrase 2
Waktu Paruh-
Vol. Distribusi-
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p-Iodophenol DB03002
small molecule | CAS: 540-38-5

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesHydrocarbons, HalogenatedHydrocarbons, Iodinated
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P-nitrobiphenyl Approved DB12300
small molecule | CAS: 92-93-3

Pnb has been used in trials studying the treatment of Pelvic Organ Prolapse.

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P-Nitrophenol DB04417
small molecule | CAS: 100-02-7

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesNitro CompoundsPhenols
Target Protein:
Sulfotransferase 1A1Alpha-amylase 2B
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small molecule | CAS: 104-03-0

Deskripsi belum tersedia.

Kategori:
Acids, Carbocyclic
Target Protein:
Penicillin G acylase
Waktu Paruh-
Vol. Distribusi-
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p-Quaterphenyl DB12794
small molecule | CAS: 135-70-6

p-Quaterphenyl has been used in trials studying the treatment of Malaria.

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small molecule

p-tert-Butylphenol-formaldehyde resin is a widely used adhesive chemical used in a wide variety of commercially available products and a known dermatological sensitizer and allergen [A34290,A34291]. Sensitivity to p-tert-Butylphenol-formaldehyde resin may …

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseStandardized Chemical Allergen
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Genetik -
small molecule | CAS: 70-55-3

Deskripsi belum tersedia.

Kategori:
AmidesBenzene DerivativesSulfonamides +2
Target Protein:
Carbonic anhydrase 2Carbonic anhydrase 12Carbonic anhydrase 6 +1
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small molecule | CAS: 104-15-4

Deskripsi belum tersedia.

Kategori:
ArylsulfonatesArylsulfonic AcidsBenzene Derivatives +3
Target Protein:
Lysozyme CPro-cathepsin H
Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Thymidine kinase, cytosolicThymidylate kinaseThymidylate kinase +3
Waktu Paruh-
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Pabinafusp alfa DB15633
biotech | CAS: 2140211-48-7

Pabinafusp alfa is under investigation in clinical trial NCT03568175 (A Study of JR-141 in Patients With Mucopolysaccharidosis II).

Kategori:
Alimentary Tract and MetabolismEnzymesEnzymes and Coenzymes
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PAC-1 DB13048
small molecule | CAS: 315183-21-2

PAC-1 has been used in trials studying the treatment of Lymphoma, Melanoma, Solid Tumors, Breast Cancer, and Thoracic Cancers, among others.

Target Protein:
Caspase-3
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PAC-113 DB05756
small molecule

PAC-113 an anti-fungal, for the treatment of oral candidiasis infections. It is a 12 amino-acid antimicrobial peptide derived from a naturally occurring histatin protein found in saliva. In vitro studies demonstrate that it has potent anti-fungal activity aga…

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PAC-14028 DB12428
small molecule | CAS: 1005168-10-4

PAC-14028 has been used in trials studying the treatment of Skin Pruritus, Papulopustular Rosacea, and Erythematotelangiectatic Rosacea.

Kategori:
Acids, AcyclicAcrylatesAmides +1
Target Protein:
Transient receptor potential cation channel subfamily V member 1
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Pacanalotamab DB17254
biotech | CAS: 2251756-52-0

Deskripsi belum tersedia.

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Paclitaxel Approved DB01229
small molecule | CAS: 33069-62-4

Paclitaxel is a chemotherapeutic agent marketed under the brand name Taxol among others. Used as a treatment for various cancers, paclitaxel is a mitotic inhibitor that was first isolated in 1971 from the bark of the Pacific yew tree which contains endophytic…

Kategori:
Agents Causing Muscle ToxicityAlbuminsAmino Acids, Peptides, and Proteins +42
Target Protein:
Tubulin beta-1 chainApoptosis regulator Bcl-2Nuclear receptor subfamily 1 group I member 2
Waktu ParuhWhen a 24 hour infu…
Vol. Distribusi* 227 to 688 L/m^2 …
Klirens* 21.7 L/h/m2 [Dose…
Genetik -
small molecule | CAS: 186040-50-6

Deskripsi belum tersedia.

Kategori:
CyclodecanesCycloparaffinsDiterpenes +2
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small molecule | CAS: 199796-52-6

A combination of [docosahexaenoic Acid] (a natural fatty acid) and [paclitaxel] (an anticancer drug) being studied in the treatment of cancer. It is a type of mitotic inhibitor.

Kategori:
CyclodecanesCycloparaffinsDiterpenes +2
Target Protein:
Apoptosis regulator Bcl-2
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small molecule | CAS: 263351-82-2

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, AcidicAmino Acids, Dicarboxylic +11
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biotech | CAS: 1075214-55-9

Three paclitaxel molecules linked by a cleavable succinyl ester linkage to a brain peptide vector, Angiopep-2, conjugate named ANG1005.

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic AgentsCardiotoxic antineoplastic agents +5
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Pacmilimab DB18873
biotech | CAS: 2145091-51-4

Pacmilimab is under investigation in clinical trial NCT04596150 (Study to Evaluate the Safety and Antitumor Activity of CX-2009 Monotherapy and in Combination With CX-072 in Advanced Breast Cancer).

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Pacritinib Approved DB11697
small molecule | CAS: 937272-79-2

Myelofibrosis (MF) is a rare disorder characterized by hematopoietic abnormalities and fibrosis within the bone marrow.[L40793] The underlying cause of primary MF is unknown, but secondary MF can arise in patients with a history of polycythemia vera or essent…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Inhibitors +29
Target Protein:
Tyrosine-protein kinase JAK3Tyrosine-protein kinase JAK2Receptor-type tyrosine-protein kinase FLT3
Waktu ParuhThe mean effective …
Vol. DistribusiThe mean apparent v…
KlirensThe mean apparent c…
Genetik -
Pactimibe DB12971
small molecule | CAS: 189198-30-9

Pactimibe has been used in trials studying the treatment of Atherosclerosis and Coronary Heart Disease.

Kategori:
Heterocyclic Compounds, Fused-RingIndolesSterol O-Acyltransferase, antagonists & inhibitors
Target Protein:
Liver carboxylesterase 1
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Padeliporfin Approved DB15575
small molecule | CAS: 759457-82-4

Padeliporfin is a water-soluble chlorophyll derivative and cytotoxic photosensitizer used for vascular-targeted photodynamic therapy for malignancies.[A244559] Vascular-targeted photodynamic therapy (VTP), or vascular targeted photochemotherapy, is a focal tr…

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +9
Waktu ParuhThe estimated half-…
Vol. DistribusiIn healthy men rece…
KlirensFollowing administr…
Genetik -
Padimate A DB11229
small molecule

Padimate A is an ester derivative of PABA and an ingredient in some sunscreens. It absorbs ultraviolet rays thereby preventing sunburn, however, its chemical structure and behaviour is similar to an industrial free radical generator. In Europe this chemical w…

Kategori:
Acids, CarbocyclicAminobenzoatesBenzene Derivatives +1
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Padimate O Approved DB11570
small molecule | CAS: 21245-02-3

Padimate O is an active sunscreen agent in cosmetics and over-the-counter sunscreen drug products in concentrations up to 8%, as regulated by the FDA [L2153]. It is a structurally-related compound to [DB02362] that absorbs UV-B rays to prevent photodamage. It…

Kategori:
Acids, CarbocyclicAminobenzoatesBenzene Derivatives +7
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Padnarsertib DB19243
small molecule | CAS: 1643913-93-2

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAcrylatesAmides +2
Target Protein:
Serine/threonine-protein kinase PAK 4
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Vol. Distribusi-
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Padsevonil DB14977
small molecule | CAS: 1294000-61-5

Padsevonil is under investigation in clinical trial NCT03695094 (A Study in Participants With Epilepsy, to Evaluate the Pharmacokinetics, Safety and Tolerability of Oxcarbazepine on Padsevonil).

Kategori:
AnticonvulsantsCentral Nervous System AgentsCentral Nervous System Depressants +3
Target Protein:
Synaptic vesicle glycoprotein 2A
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Paecilomyces variotii Approved DB10822
biotech

Paecilomyces variotii is a fungus which can provoke allergic reactions. Paecilomyces variotii extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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Paeonol DB16830
small molecule | CAS: 552-41-0

Deskripsi belum tersedia.

Kategori:
Ketones
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Pafolacianine Approved DB15413
small molecule | CAS: 1628423-76-6

Pafolacianine, or OTL38, is a folate analogue conjugated with a fluorescent dye that absorbs light in the near-infrared (NIR) spectrum [A242572] within a range of 760 nm to 785 nm, with a peak absorption of 776 nm. It emits fluorescence within a range of 790 …

Kategori:
Compounds used in a research, industrial, or household settingDiagnostic AgentsDiagnostic Uses of Chemicals +10
Target Protein:
Folate receptor alpha
Waktu ParuhThe elimination hal…
Vol. DistribusiThe mean volume of …
KlirensThe mean plasma cle…
Genetik -
Pafuramidine DB06532
small molecule | CAS: 186953-56-0

Pafuramidine, a prodrug of furamidine, currently has orphan status for _Pneumocystis jiroveci_ pneumonia.

Kategori:
AmidinesAnti-Infective AgentsAntiparasitic Agents +2
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Pagoclone DB04903
small molecule | CAS: 133737-32-3

Pagoclone is an anxiolytic drug from the cyclopyrrolone family, which is related to other more well known drugs such as the sleeping medication zopiclone. It is one of a relatively recently developed class of medicines known as the nonbenzodiazepines, which h…

Kategori:
Central Nervous System DepressantsGABA AgentsHeterocyclic Compounds, Fused-Ring +2
Target Protein:
Gamma-aminobutyric acid receptor subunit gamma-3Gamma-aminobutyric acid receptor subunit alpha-2Gamma-aminobutyric acid receptor subunit alpha-3
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Palazestrant DB18971
small molecule | CAS: 2092925-89-6

Palazestrant is under investigation in clinical trial NCT06016738 (OP-1250 (Palazestrant) vs. Standard of Care for the Treatment of ER+/HER2- Advanced Breast Cancer).

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Palbociclib Approved DB09073
small molecule | CAS: 571190-30-2

Palbociclib is a piperazine pyridopyrimidine[A176792] that acts in the cell cycle machinery. It is a second generation cyclin-dependent kinase inhibitor[A176798] selected from a group of pyridopyrimidine compounds due to its favorable physical and pharmaceuti…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Inhibitors +21
Target Protein:
Cyclin-dependent kinase 4Cyclin-dependent kinase 6
Waktu ParuhThe mean plasma eli…
Vol. DistribusiThe mean apparent d…
KlirensThe mean apparent o…
Genetik -
Palifermin Approved DB00039
biotech | CAS: 162394-19-6

Palifermin is a recombinant human keratinocyte growth factor (KGF). It is 140 residues long, and is produced using E. coli. Palifermin was granted FDA approval on 15 December 2004.[L17933]

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsDetoxifying Agents for Antineoplastic Treatment +6
Target Protein:
Fibroblast growth factor receptor 2Fibroblast growth factor receptor 1Basement membrane-specific heparan sulfate proteoglycan core protein
Waktu ParuhElimination half-li…
Vol. Distribusi-
Klirens-
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Palifosfamide DB05668
small molecule | CAS: 31645-39-3

Palifosfamide (ZIO-201) is a proprietary stabilized metabolite of ifosfamide. Ifosfamide has been shown to be effective in high doses in treating testicular cancer, sarcoma and lymphoma.

Kategori:
Alkylating DrugsAmino AcidsAmino Acids, Basic +13
Target Protein:
DNA (cytosine-5)-methyltransferase 1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Paliperidone Approved DB01267
small molecule | CAS: 144598-75-4

Paliperidone is the primary active metabolite of risperidone. The mechanism of action is unknown but it is likely to act via a similar pathway to risperidone. It has been proposed that the drug's therapeutic activity in schizophrenia is mediated through a com…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +37
Target Protein:
5-hydroxytryptamine receptor 2AD(2) dopamine receptorD(4) dopamine receptor +12
Waktu ParuhThe terminal elimin…
Vol. Distribusi* 487 L
Klirens-
Genetik -
Paliroden DB05454
small molecule | CAS: 188396-77-2

Paliroden is an orally active neurotrophic, non-peptidic compound that activates synthesis of endogenous neurotrophines. Studies show that use of paliroden increased the rate of formation of both neural progenitors and mature neurons. It is indicated for use …

Target Protein:
Glutamate receptor 2
Waktu Paruh-
Vol. Distribusi-
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Palivizumab Approved DB00110
biotech | CAS: 188039-54-5

Humanized monoclonal antibody (IgG1k) produced by recombinant DNA technology, directed to an epitope in the A antigenic site of the F protein of respiratory syncytial virus (RSV). Synagis is a composite of human (95%) and murine (5%) antibody sequences. The h…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntibodies +15
Target Protein:
Fusion glycoprotein F0Low affinity immunoglobulin gamma Fc region receptor III-BComplement C1r subcomponent +6
Waktu Paruh18-20 days (in adul…
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 14967-68-1

Palladium Pd-103 is under investigation in clinical trial NCT00247312 (Pd-103 Dose De-Escalation for Early Stage Prostate Cancer: A Prospective Randomized Trial).

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Palm oil DB14377
biotech | CAS: 8002-75-3

Palm oil is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
Biological ProductsComplex MixturesDietary Fats +5
Waktu Paruh-
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Genetik -
Palmidrol DB14043
small molecule | CAS: 544-31-0

A cannabinoid receptor-inactive eCB-related molecule used as prophylactic in helping to prevent respiratory viral infection. Palmidrol is available for human use as a supplement (400 mg capsules) and as food for medical purposes In Italy and Spain (300 mg and…

Kategori:
Agents producing tachycardiaAlcoholsAmines +15
Target Protein:
Cannabinoid receptor 2Glucose-dependent insulinotropic receptorG-protein coupled receptor 55
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Genetik -
small molecule | CAS: 373-49-9

Deskripsi belum tersedia.

Kategori:
Fatty AcidsFatty Acids, UnsaturatedLipids
Target Protein:
UDP-3-O-[3-hydroxymyristoyl] N-acetylglucosamine deacetylaseFatty-acid peroxygenaseBifunctional cytochrome P450/NADPH--P450 reductase
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Genetik -
small molecule | CAS: 147732-56-7

Deskripsi belum tersedia.

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Genetik -
small molecule | CAS: 221227-05-0

Deskripsi belum tersedia.

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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Phosphatidylcholine transfer protein
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Palomid 529 DB12812
small molecule | CAS: 914913-88-5

Palomid 529 has been used in trials studying the treatment of Age-Related Macular Degeneration.

Kategori:
Heterocyclic Compounds, Fused-RingPyrans
Target Protein:
Target of rapamycin complex 2 subunit MAPKAP1
Waktu Paruh-
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Genetik -
Menampilkan 10351–10400 dari 14063
Sebelumnya Halaman 208 / 282 Berikutnya