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17430

Total database: 17430
Struktur (SMILES)
12313 (70.6%)
Target
9368 (53.7%)
Genomik
112 (0.6%)
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17430 (100.0%)

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Halaman 207 / 349
LJP-538 DB17810
biotech

Deskripsi belum tersedia.

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LJP-539 DB17811
biotech

Deskripsi belum tersedia.

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LL-37 DB16532
biotech

LL-37 is a human cathelicidin that inhibits viral replication and while also playing a role in host defense against infection.

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LLL-3348 DB05771
biotech

The botanical drug product LLL-3348 is a once-daily oral formulation for treatment of chronic stable plaque type psoriasis.

Kategori:
Biological ProductsComplex MixturesPharmaceutical Preparations +1
Target Protein:
Interleukin-10
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LM-030 DB18283
small molecule | CAS: 1122484-55-2

Deskripsi belum tersedia.

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LM-609 DB05787
biotech

LM-609 (Vitaxin) is an artificial antibody that targets a protein on the surface of newly forming blood vessels, as well as on certain tumors. In addition to cancer, the protein has been implicated in bone destruction in rheumatoid arthritis and the inflammat…

Target Protein:
Integrin beta-3
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LMB-100 DB18591
biotech | CAS: 1841500-93-3

LMB-100 is a is an antibody-toxin conjugate with an antimesothelin Fab linked to a 24-kilodalton portion of Pseudomonas exotoxin A with mutations that decrease immunogenicity.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
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biotech

LNP-nCoVsaRNA is a purified, synthetic mRNA vaccine candidate encoding the S glycoprotein of SARS-CoV-2, which is used primarily by the virus to attach to and invade human cells. The vaccine was developed in and tested by the Medical Research Council Clinical…

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LNS-8801 DB18091
small molecule | CAS: 881639-98-1

Deskripsi belum tersedia.

Target Protein:
G-protein coupled estrogen receptor 1
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Lobaplatin DB13049
small molecule | CAS: 135558-11-1

Lobaplatin has been used in trials studying the treatment of Breast Cancer, Hepatocellular Carcinoma, and Lobaplatin and Gemcitabine in Combination, Second-line Treatments on Advanced Osteosarcoma.

Kategori:
CycloparaffinsOrganometallic Compounds
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Lobeglitazone DB09198
small molecule | CAS: 607723-33-1

Lobeglitazone is an antidiabetic medication from the thiazolidinedione class of drugs. It primarily functions as an insulin sensitizer by binding and activating Peroxisome Proliferator-Activated Receptors (PPAR) gamma within fat cells. By activating PPAR-gamm…

Kategori:
Alimentary Tract and MetabolismBlood Glucose Lowering AgentsCytochrome P-450 CYP1A2 Inhibitors +19
Target Protein:
Peroxisome proliferator-activated receptor alphaPeroxisome proliferator-activated receptor gamma
Waktu ParuhFollowing an intrav…
Vol. DistribusiThe steady state vo…
KlirensIn rat studies, sys…
Genetik -
Lobeline DB05137
small molecule | CAS: 90-69-7

An alkaloid that has actions similar to nicotine on nicotinic cholinergic receptors but is less potent. It has been proposed for a variety of therapeutic uses including in respiratory disorders, peripheral vascular disorders, insomnia, and smoking cessation. …

Kategori:
AlkaloidsAutonomic AgentsCholinergic Agents +7
Target Protein:
Synaptic vesicular amine transporterNeuronal acetylcholine receptor subunit alpha-7Neuronal acetylcholine receptor subunit alpha-9 +1
Waktu Paruh-
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Lobster Approved DB10541
biotech

Lobster allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
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Lobucavir DB12531
small molecule | CAS: 127759-89-1

Lobucavir has been used in trials studying the treatment of HIV Infections and Cytomegalovirus Infections.

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +10
Target Protein:
Gag-Pol polyprotein
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small molecule | CAS: 398507-55-6

Lodenafil carbonate has been used in trials studying the treatment of Coronaropathy and Erectile Dysfunction.

Kategori:
AlkaliesAnionsCarbon Compounds, Inorganic +3
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Lodoxamide Approved DB06794
small molecule | CAS: 53882-12-5

Lodoxamide is a mast-cell stabilizer for topical administration into the eye. Mast-cell stabilizers, first one approved being cromolyn sodium, are used in treatment of ocular hypersensitivity reactions such as vernal conjunctivitis. These conditions often req…

Kategori:
Acids, AldehydicAlcoholsAmino Acids +13
Waktu ParuhElimination half-li…
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Lofentanil DB09174
small molecule | CAS: 61380-40-3

Lofentanil is an analog of fentanyl and is one of the most potent opioids available today. It displays most similarity to carfentanil (4-carbomethoxyfentanyl) and is considered to be slightly more potent than this drug.

Kategori:
AnalgesicsCentral Nervous System AgentsCentral Nervous System Depressants +6
Target Protein:
Mu-type opioid receptorKappa-type opioid receptorDelta-type opioid receptor
Waktu Paruh-
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Lofepramine DB13411
small molecule | CAS: 23047-25-8

Deskripsi belum tersedia.

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +11
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Lofexidine Approved DB04948
small molecule | CAS: 31036-80-3

Lofexidine is a non-opioid centrally acting alpha2-adrenergic receptor agonist that was first approved for the treatment of opioid withdrawal in the United Kingdom in 1992.[A33084] It was first studied for use as an antihypertensive in 1980, but its researche…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-2 Receptor Agonists +31
Target Protein:
Alpha-2A adrenergic receptorAlpha-1A adrenergic receptor5-hydroxytryptamine receptor 1A +3
Waktu ParuhThe reported elimin…
Vol. DistribusiLofexidine has a vo…
KlirensThe total eliminati…
Genetik -
Lolium perenne pollen Approved DB10389
biotech

Lolium perenne pollen is the pollen of the Lolium perenne plant. Lolium perenne pollen is mainly used in allergenic testing.

Kategori:
Allergenic ExtractsCell-mediated ImmunityGrass Pollen Allergen Extracts +3
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biotech

Lolium perenne subsp. multiflorum pollen is the pollen of the Lolium perenne subsp. multiflorum plant. Lolium perenne subsp. multiflorum pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityGrass Pollen Allergen ExtractsIncreased Histamine Release +2
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Lomefloxacin Approved DB00978
small molecule | CAS: 98079-51-7

Lomefloxacin is a fluoroquinolone antibiotic, used to treat bacterial infections including bronchitis and urinary tract infections (UTIs). Additionally, it has been employed for the prophylaxis of UTIs prior to surgery as well.

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +22
Target Protein:
DNA gyrase subunit ADNA topoisomerase 2-betaDNA topoisomerase 4 subunit A +1
Waktu Paruh8 hours
Vol. Distribusi-
Klirens* 271 mL/min/1.73 m…
Genetik -
Lomerizine DB14065
small molecule | CAS: 101477-55-8

Lomerizine is a diphenylmethylpiperazine calcium channel blocker[A245378, A245383] with relatively selective central nervous system (CNS) effects.[A245383] This drug is used to prophylactically treat migraines[A245368, A245373] and is also being investigated…

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsBradycardia-Causing Agents +8
Target Protein:
Sodium channel protein type 5 subunit alphaVoltage-dependent N-type calcium channel subunit alpha-1BATP-dependent translocase ABCB1
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Lometrexol DB12769
small molecule | CAS: 106400-81-1

Lometrexol has been used in trials studying the treatment of Lung Cancer, Drug/Agent Toxicity by Tissue/Organ, and Unspecified Adult Solid Tumor, Protocol Specific.

Kategori:
AntimetabolitesAntineoplastic AgentsCoenzymes +9
Target Protein:
Dihydrofolate reductase
Waktu Paruh-
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Lomibuvir DB11954
small molecule | CAS: 1026785-55-6

Lomibuvir has been used in trials studying the treatment of Chronic Hepatitis C Virus and Chronic Hepatitis C Virus Infection.

Kategori:
AlcoholsCyclohexanesCycloparaffins +4
Target Protein:
Genome polyprotein
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Lomifylline Approved DB18002
small molecule | CAS: 10226-54-7

Deskripsi belum tersedia.

Kategori:
AlkaloidsDrugs for Obstructive Airway DiseasesHeterocyclic Compounds, Fused-Ring +3
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Lomitapide Approved DB08827
small molecule | CAS: 182431-12-5

Lomitapide is a microsomal triglyceride transfer protein (MTP) inhibitor used in homozygous familial hypercholesterolemia (HoFH) patients. It is marketed under the name Juxtapid (R).

Kategori:
Cytochrome P-450 CYP3A InhibitorsCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Inhibitors +17
Target Protein:
Microsomal triglyceride transfer protein large subunit
Waktu ParuhLomitapide half-lif…
Vol. DistribusiThe steady state vo…
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Lomustine Approved DB01206
small molecule | CAS: 13010-47-4

An alkylating agent of value against both hematologic malignancies and solid tumors.

Kategori:
Alkylating ActivityAlkylating DrugsAmides +17
Target Protein:
DNAStathmin-4
Waktu ParuhApproximately 94 mi…
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Lomvastomig DB19060
biotech | CAS: 2648840-52-0

Lomvastomig is under investigation in clinical trial NCT04785820 (A Study of Lomvastomig (RO7121661) and Tobemstomig (RO7247669) Compared With Nivolumab in Participants With Advanced or Metastatic Squamous Cell Carcinoma of the Esophagus).

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Lonafarnib Approved DB06448
small molecule | CAS: 193275-84-2

Hutchinson-Gilford progeria syndrome (HGPS) is a rare autosomal dominant disorder estimated to affect approximately one in 20 million individuals resulting in adverse symptoms associated with premature ageing: skeletal dysplasia, joint contractures, atheroscl…

Kategori:
Alimentary Tract and MetabolismBCRP/ABCG2 InhibitorsBenzocycloheptenes +30
Target Protein:
Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alphaProtein farnesyltransferase subunit beta
Waktu ParuhLonafarnib has a me…
Vol. DistribusiIn healthy patients…
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Lonapegsomatropin Approved DB16220
biotech | CAS: 1934255-39-6

Lonapegsomatropin, also known as TransCon hGH or ACP 001, is a methoxypegylated prodrug of human growth hormone ([somatropin]) indicated for the treatment of children 1 year and older, weighing at least 11.5 kg, with growth failure due to insufficient growth …

Kategori:
Amino Acids, Peptides, and ProteinsAnterior Pituitary Lobe Hormones and AnaloguesCytochrome P-450 CYP1A2 Inducers +18
Target Protein:
Growth hormone receptorProlactin receptor
Waktu ParuhThe half life of lo…
Vol. DistribusiLonapegsomatropin-t…
KlirensIn pediatric patien…
Genetik -
Lonaprisan DB16221
small molecule | CAS: 211254-73-8

Lonaprisan is under investigation in clinical trial NCT00555919 (ZK 230211 in Postmenopausal Woman With Metastatic Breast Cancer).

Kategori:
EstranesFused-Ring CompoundsHydrocarbons, Fluorinated +2
Target Protein:
Progesterone receptorGlucocorticoid receptorAndrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Lonazolac DB13432
small molecule | CAS: 53808-88-1

Deskripsi belum tersedia.

Kategori:
Acetic Acid Derivatives and Related SubstancesAgents causing hyperkalemiaAgents that produce hypertension +13
Waktu Paruh-
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Loncastuximab tesirine Approved DB16222
biotech | CAS: 1879918-31-6

Relapsed and refractory B-cell acute lymphoblastic leukemia (B-ALL) are a therapeutic challenge for patients who have undergone prior systemic therapies with limited success.[A234439] Prognosis is poor and more effective therapies are needed to treat relapsed…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +19
Target Protein:
B-lymphocyte antigen CD19
Waktu ParuhThe half-life of lo…
Vol. DistribusiIn clinical studies…
KlirensIn pharmacokinetic …
Genetik -
Londamocitinib DB19190
small molecule | CAS: 2241039-81-4

Londamocitinib is under investigation in clinical trial NCT06020014 (Phase 2a Study to Assess the Efficacy and Safety of AZD4604 in Adult Patients With Moderate-to-severe Asthma Uncontrolled on Medium-high Dose ICS-LABA).

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Lonicera caprifolium flower Approved DB14280
biotech

Lonicera caprifolium flower is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

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biotech

Lonicera confusa flower is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

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Lonidamine DB06266
small molecule | CAS: 50264-69-2

Lonidamine (LND) is a drug that interferes with energy metabolism of cancer cells, principally inhibiting aerobic glycolytic activity, by its effect on mitochondrially-bound hexokinase (HK). In such way LND could impair energy-requiring processes, as recovery…

Kategori:
Adrenal Cortex HormonesAnti-Infective AgentsAntineoplastic Agents +11
Target Protein:
Cystic fibrosis transmembrane conductance regulatorHexokinase-1
Waktu Paruh-
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Lonigutamab DB18940
biotech | CAS: 2362015-67-4

Lonigutamab is under investigation in clinical trial NCT05683496 (Efficacy and Safety of Lonigutamab in Subjects With Thyroid Eye Disease (TED)).

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Lonoctocog alfa Approved DB13998
biotech | CAS: 1388129-63-2

Deskripsi belum tersedia.

Kategori:
Hemostatics
Target Protein:
Coagulation factor XCoagulation factor IXvon Willebrand factor +8
Waktu Paruh8.4-19.3 hrs
Vol. Distribusi-
Klirens* 4.1 mL/h•kg [Prev…
Genetik -
Loperamide Approved DB00836
small molecule | CAS: 53179-11-6

Loperamide is an anti-diarrheal agent that is available as an over-the-counter product for treating diarrhea.[L42785] The drug was first synthesized in 1969 and used medically in 1976.[A251610] It is a highly lipophilic synthetic phenylpiperidine opioid that …

Kategori:
Agents causing hyperkalemiaAlimentary Tract and MetabolismAntiarrhythmic agents +20
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorKappa-type opioid receptor +4
Waktu ParuhThe apparent elimin…
Vol. DistribusiLoperamide has a la…
Klirens-
Genetik -
small molecule | CAS: 106900-12-3

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismAntidiarrhealsAntidiarrheals, Intestinal Antiinflammatory/antiinfective Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lopinavir Approved DB01601
small molecule | CAS: 192725-17-0

Lopinavir is an antiretroviral protease inhibitor used in combination with other antiretrovirals in the treatment of HIV-1 infection.[L11163] Lopinavir is marketed and administered exclusively in combination with [ritonavir] - this combination, first marketed…

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +42
Target Protein:
Pol polyprotein
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe estimated appar…
Genetik -
Loprazolam DB13643
small molecule | CAS: 61197-73-7

Loprazolam is an imidazobenzodiazepine with anxiolytic, anticonvulsant, hypnotic, sedative and skeletal muscle relaxant properties. It is indicated for the short-term treatment of insomnia including difficulty in falling asleep and/or frequent nocturnal awake…

Kategori:
Anti-Anxiety AgentsBenzazepinesBenzodiazepine hypnotics and sedatives +9
Target Protein:
GABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Loracarbef Approved DB00447
small molecule | CAS: 76470-66-1

Loracarbef is a carbacephem antibiotic sometimes grouped together with the second-generation cephalosporin antibiotics. It is marketed under the trade name Lorabid.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
Penicillin-binding protein 3Penicillin-binding protein 1A
Waktu Paruh1 hour. In subjects…
Vol. Distribusi-
Klirens-
Genetik -
Lorajmine DB13651
small molecule | CAS: 47562-08-3

Deskripsi belum tersedia.

Kategori:
AlkaloidsAntiarrhythmic agentsAntiarrhythmics, Class I +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Loratadine Approved DB00455
small molecule | CAS: 79794-75-5

Loratadine is a second generation antihistamine used to manage symptoms of allergic rhinitis.[A176435] A lack of sedative and CNS adverse effects make loratadine, along with other second generation antihistamines, preferable over their 1st generation counterp…

Kategori:
Anti-Allergic AgentsAntihistamines for Systemic UseAntipruritics +34
Target Protein:
Histamine H1 receptorVoltage-gated inwardly rectifying potassium channel KCNH2
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of lo…
Genetik -
Lorazepam Approved DB00186
small molecule | CAS: 846-49-1

Lorazepam is a short-acting and rapidly cleared benzodiazepine used commonly as a sedative and anxiolytic.[A957] It was developed by DJ Richards, presented and marketed initially by Wyeth Pharmaceuticals in the USA in 1977. The first historic FDA label approv…

Kategori:
Anti-Anxiety AgentsAnticonvulsantsAntiemetics +21
Target Protein:
Translocator proteinGABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site
Waktu ParuhWhen administered p…
Vol. DistribusiThe reported volume…
Klirens_In vivo_ studies w…
Genetik -
Lorcainide DB13653
small molecule | CAS: 59729-31-6

Deskripsi belum tersedia.

Kategori:
AcetamidesAmidesAntiarrhythmic agents +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lorcaserin Approved DB04871
small molecule | CAS: 616202-92-7

Lorcaserin (previously APD-356), a highly selective 5HT2C receptor agonist, is used for the treatment of obesity. It has been shown to reduce body weight and food intake in animal models of obesity, and it is thought that targeting the 5HT2C receptor may alte…

Kategori:
Alimentary Tract and MetabolismAntidepressive AgentsAntiobesity Preparations, Excl. Diet Products +22
Target Protein:
5-hydroxytryptamine receptor 2C
Waktu ParuhThe plasma half lif…
Vol. DistribusiThe volume of distr…
KlirensThe clearance value…
Genetik -
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