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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
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12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 207 / 252
rhMBL DB05237
biotech

rhMBL is a protein therapeutic being developed by Enzon for the prevention and treatment of severe infections in individuals with low levels of Mannose-Binding Lectin (MBL). Over 10 percent of the general population is estimated to be MBL-deficient. Natural M…

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Rhodamine 6G DB03825
small molecule | CAS: 989-38-8

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsColoring AgentsCompounds used in a research, industrial, or household setting +7
Target Protein:
HTH-type transcriptional regulator QacRMultidrug efflux pump subunit AcrB
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Rhodamine B DB16853
small molecule | CAS: 81-88-9

Deskripsi belum tersedia.

Kategori:
Coloring AgentsCompounds used in a research, industrial, or household settingCosmetics +6
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Rhubarb Approved DB10651
biotech | CAS: 8016-55-5

Rhubarb allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract +1
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Rhus Glabra Pollen Approved DB13895
biotech

Rhus Glabra Pollen pollen is the pollen of the Rhus Glabra Pollen plant. The pollen is mainly used in allergenic testing.

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RI 624 DB05892
biotech

RI 624 is a novel humanized monoclonal antibody that blocks nerve growth factor (NGF), a key mediator of acute and chronic pain. RI 624 is being developed by Rinat and is currently in Phase I clinical trials.

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsAntibodies +11
Target Protein:
Beta-nerve growth factor
Waktu Paruh-
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Ribavirin Approved DB00811
small molecule | CAS: 36791-04-5

Producing a broad-spectrum activity against several RNA and DNA viruses, Ribavirin is a synthetic guanosine nucleoside and antiviral agent that interferes with the synthesis of viral mRNA. It is primarily indicated for use in treating hepatitis C and viral he…

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntimetabolites +13
Target Protein:
Inosine-5'-monophosphate dehydrogenase 1RNA-directed RNA polymerase LGenome polyprotein +2
Gen Terkait:
IFNL3
Waktu ParuhThe terminal half-l…
Vol. DistribusiRibavirin displays …
KlirensThe total apparent …
Genetik 1 Varian
small molecule | CAS: 1352921-29-9

Deskripsi belum tersedia.

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small molecule | CAS: 40925-28-8

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAntiviral AgentsCarbohydrates +3
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Ribaxamase DB16311
biotech | CAS: 1792207-66-9

Ribaxamase is under investigation in clinical trial NCT02563106 (A Study of SYN-004 for the Prevention of c.diff in Patients With a LRTI).

Kategori:
AmidohydrolasesAmino Acids, Peptides, and ProteinsEnzymes +3
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Ribitol DB14704
small molecule | CAS: 488-81-3

Deskripsi belum tersedia.

Kategori:
AlcoholsCarbohydratesSugar Alcohols
Waktu Paruh-
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Riboflavin Approved DB00140
small molecule | CAS: 83-88-5

Nutritional factor found in milk, eggs, malted barley, liver, kidney, heart, and leafy vegetables. The richest natural source is yeast. It occurs in the free form only in the retina of the eye, in whey, and in urine; its principal forms in tissues and cells a…

Kategori:
Alimentary Tract and MetabolismBiological FactorsCoenzymes +14
Target Protein:
Riboflavin kinaseRiboflavin synthaseFlavin reductase (NADPH)
Waktu Paruh66-84 minutes
Vol. Distribusi-
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Genetik -
small molecule | CAS: 752-56-7

Deskripsi belum tersedia.

Kategori:
Biological FactorsCoenzymesEnzymes and Coenzymes +4
Waktu Paruh-
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Ribose DB15073
small molecule | CAS: 50-69-1

Ribose is under investigation in clinical trial NCT01727479 (Ribose and Sport Performance).

Kategori:
CarbohydratesMonosaccharidesPentoses
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small molecule | CAS: 4151-19-3

Deskripsi belum tersedia.

Kategori:
CarbohydratesPentosephosphatesSugar Phosphates
Target Protein:
Ribose-5-phosphate isomerase A2-dehydro-3-deoxyphosphooctonate aldolaseADP-ribose pyrophosphatase
Waktu Paruh-
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Ribostamycin Approved DB03615
small molecule | CAS: 25546-65-0

Ribostamycin is an aminoglycoside antibiotic[A187166] isolated from _Streptomyces ribosidificus_[A187178] listed as one of the World Health Organization's critically important antimicrobials.[L9071]

Kategori:
Agents that produce neuromuscular block (indirect)Aminoglycoside AntibacterialsAnti-Bacterial Agents +9
Target Protein:
30S ribosomal protein S12Protein disulfide-isomeraseAminoglycoside N(6')-acetyltransferase type 1 +1
Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
3-keto-L-gulonate-6-phosphate decarboxylase UlaD
Waktu Paruh-
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Rice Approved DB10563
biotech

Rice allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
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Ricinoleic acid DB02955
small molecule | CAS: 141-22-0

Deskripsi belum tersedia.

Kategori:
Biological ProductsFatsFats, Unsaturated +6
Target Protein:
Cannabinoid receptor 1Cannabinoid receptor 2Transient receptor potential cation channel subfamily V member 1
Waktu Paruh-
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Ricolinostat DB12376
small molecule | CAS: 1316214-52-4

Ricolinostat is under investigation for the treatment of Breast Carcinoma and Metastatic Breast Cancer.

Kategori:
AminesAntineoplastic AgentsEnzyme Inhibitors +5
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Ridaforolimus DB06233
small molecule | CAS: 572924-54-0

Deskripsi belum tersedia.

Kategori:
Anti-Bacterial AgentsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +8
Target Protein:
Serine/threonine-protein kinase mTOR
Waktu Paruh-
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Ridinilazole DB15308
small molecule | CAS: 308362-25-6

Ridinilazole is under investigation in clinical trial NCT02092935 (A Study of SMT19969 Compared With Vancomycin for the Treatment of Clostridium Difficile-Associated Diarrhoea (CDAD)).

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsHeterocyclic Compounds, Fused-Ring
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Rifabutin Approved DB00615
small molecule | CAS: 72559-06-9

A broad-spectrum antibiotic that is being used as prophylaxis against disseminated Mycobacterium avium complex infection in HIV-positive patients.

Kategori:
Alimentary Tract and MetabolismAnti-Bacterial AgentsAnti-Infective Agents +27
Target Protein:
DNA-directed RNA polymerase subunit alphaDNA-directed RNA polymerase subunit betaDNA-directed RNA polymerase subunit beta' +2
Waktu Paruh45 (± 17) ho…
Vol. Distribusi-
Klirens* 0.69 +/- 0.32 L/h…
Genetik -
Rifalazil DB04934
small molecule | CAS: 129791-92-0

Rifalazil is a derivative of the antibiotic rifamycin. It is being investigated by ActivBiotics for the treatment of various bacterial infections.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibiotics, Antitubercular +7
Target Protein:
DNA-directed RNA polymerase subunit beta
Waktu Paruh-
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Rifampin Approved DB01045
small molecule | CAS: 13292-46-1

Rifampin, also known as rifampicin, is a broad-spectrum antimicrobial [A263748] that was first discovered in 1965 [A263753] and clinically used in 1968.[A263768] Rifampin is used to treat tuberculosis and works by inhibiting the microbial DNA-dependent RNA po…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +55
Target Protein:
DNA-directed RNA polymerase subunit betaNuclear receptor subfamily 1 group I member 2
Waktu ParuhIn healthy adults, …
Vol. DistribusiFollowing intraveno…
KlirensFollowing intraveno…
Genetik -
Rifamycin Approved DB11753
small molecule | CAS: 6998-60-3

Rifamycin is the prime member of the rifamycin family which are represented by drugs that are a product of fermentation from the gram-positive bacterium _Amycolatopsis mediterranei_, also known as _Streptomyces mediterranei_. The parent compound of rifamycin …

Kategori:
Alimentary Tract and MetabolismAnti-Bacterial AgentsAnti-Infective Agents +49
Target Protein:
DNA-directed RNA polymerase subunit betaDNA-directed RNA polymerase subunit beta'DNA-directed RNA polymerase subunit beta +2
Waktu ParuhThe reported half-l…
Vol. DistribusiThe reported volume…
KlirensThe reported cleara…
Genetik -
Rifapentine Approved DB01201
small molecule | CAS: 61379-65-5

Rifapentine is an antibiotic drug used in the treatment of tuberculosis. It inhibits DNA-dependent RNA polymerase activity in susceptible cells. Specifically, it interacts with bacterial RNA polymerase but does not inhibit the mammalian enzyme.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibiotics, Antitubercular +24
Target Protein:
DNA-directed RNA polymerase subunit beta'
Waktu Paruh-
Vol. Distribusi* 70.2 ± 9.1 L
Klirens* Apparent Oral cl=…
Genetik -
Rifasutenizol DB18981
small molecule | CAS: 1001314-13-1

Rifasutenizol is under investigation in clinical trial NCT05857163 (Efficacy and Safety of Rifasutenizol (TNP 2198) in Participants With H. Pylori Infection).

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Rifaximin Approved DB01220
small molecule | CAS: 80621-81-4

Rifaximin is a semisynthetic, rifamycin-based non-systemic antibiotic, meaning that the drug will not pass the gastrointestinal wall into the circulation as is common for other types of orally administered antibiotics. It has multiple indications and is used …

Kategori:
Alimentary Tract and MetabolismAnti-Bacterial AgentsAnti-Infective Agents +22
Target Protein:
DNA-directed RNA polymerase subunit betaNuclear receptor subfamily 1 group I member 2
Waktu ParuhApproximately 6 hou…
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1001859-46-6

Riferminogene pecaplasmid (non-viral fibroblast growth factor 1; NV1FGF) is a recombinant DNA plasmid in a pCOR backbone allowing expression of human FGF1.

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Rigosertib DB12146
small molecule | CAS: 592542-59-1

Rigosertib has been used in trials studying the treatment and basic science of MDS, RAEB, Cancer, Hepatoma, and Neoplasms, among others.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAntineoplastic Agents +3
Target Protein:
Serine/threonine-protein kinase PLK1Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
Waktu Paruh-
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Rilapladib DB05119
small molecule | CAS: 412950-08-4

Rilapladib is the third genomics-derived small molecule drug arising from the Human Genome Sciences-GlaxoSmithKline collaboration to enter clinical development. It is a lipoprotein-associated phospholipase A2 (Lp-PLA2) inhibitor. Lp-PLA2 is an enzyme associat…

Kategori:
AcetatesAcids, AcyclicAmides +2
Target Protein:
Thymidine kinase, cytosolicPhospholipase A2Platelet-activating factor acetylhydrolase
Waktu Paruh-
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Genetik -
Rilematovir DB15672
small molecule | CAS: 1383450-81-4

Rilematovir is under investigation in clinical trial NCT04056611 (Effects of JNJ-53718678 in Adult and Adolescent Participants Who Had a Hematopoietic Stem Cell Transplantation and Who Are Infected With Respiratory Syncytial Virus (RSV)).

Kategori:
Heterocyclic Compounds, Fused-RingImidazoles
Target Protein:
Fusion glycoprotein F0
Waktu Paruh-
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Genetik -
Riliprubart DB18355
biotech | CAS: 2756228-76-7

Deskripsi belum tersedia.

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Rilmenidine Approved DB11738
small molecule | CAS: 54187-04-1

Rilmenidine has been used in trials studying the treatment of Hypertension and Chronic Kidney Disease.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-2 Receptor Agonists +12
Target Protein:
Alpha-2C adrenergic receptorAlpha-2A adrenergic receptor
Waktu Paruh-
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Rilonacept Approved DB06372
biotech | CAS: 501081-76-1

Rilonacept is a dimeric fusion protein consisting of portions of IL-1R and the IL-1R accessory protein linked to the Fc portion of immunoglobulin G1. Rilonacept functions as an interleukin 1 inhibitor and is used in the treatment of CAPS, also known as cryopy…

Kategori:
Agents reducing cytokine levelsAmino Acids, Peptides, and ProteinsAnti-Inflammatory Agents +9
Target Protein:
Interleukin-1 betaInterleukin-1 alphaInterleukin-1 receptor antagonist protein
Waktu Paruh8.6 days
Vol. Distribusi-
Klirens-
Genetik -
Rilotumumab DB11972
biotech | CAS: 872514-65-3

Rilotumumab has been investigated for the treatment of Cancer, Lung Cancer, Solid Tumors, Gastric Cancer, and Prostate Cancer, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Waktu Paruh-
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Genetik -
Rilpivirine Approved DB08864
small molecule | CAS: 500287-72-9

Rilpivirine is non-nucleoside reverse transcriptase inhibitor (NNRTI) which is used for the treatment of HIV-1 infections in treatment-naive patients.[A31328] It is a diarylpyrimidine derivative.[A31329] The internal conformational flexibility of rilpivirine …

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +43
Target Protein:
Reverse transcriptase/RNaseHSodium channel protein type 10 subunit alphaGag-Pol polyprotein +1
Waktu ParuhRilpivirine has a t…
Vol. DistribusiIn HIV-1 patients, …
KlirensIn HIV-1 patients, …
Genetik -
Riltozinameran Approved DB17095
biotech | CAS: 2749948-25-0

The Omicron variant of SARS-CoV-2 is a variant of concern that was first reported in November 2021.[L43922] It tends to cause less severe disease but is significantly more virulent than both the original virus and earlier variants (e.g. Delta).[L43917] As of …

Kategori:
COVID-19 VaccinesmRNA VaccinesVaccines +1
Waktu Paruh-
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Riluzole Approved DB00740
small molecule | CAS: 1744-22-5

A glutamate antagonist (receptors, glutamate) used as an anticonvulsant (anticonvulsants) and to prolong the survival of patients with amyotrophic lateral sclerosis. Riluzole is marketed as Rilutek by Sanofi.

Kategori:
AnticonvulsantsBCRP/ABCG2 SubstratesBenzothiazoles +15
Target Protein:
Sodium channel protein type 5 subunit alphaSodium channel protein type 11 subunit alphaCystine/glutamate transporter
Waktu ParuhThe mean eliminatio…
Vol. Distribusi-
Klirens-
Genetik -
Rilvegostomig DB18991
biotech | CAS: 2640305-01-5

Rilvegostomig is under investigation in clinical trial NCT06109779 (Rilvegostomig + Chemotherapy as Adjuvant Therapy for Biliary Tract Cancer After Resection (Artemide-biliary01)).

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Rilzabrutinib DB17709
small molecule | CAS: 1575591-66-0

Rilzabrutinib is an oral, reversible covalent inhibitor of Bruton's tyrosine kinase being investigated for the treatment of immune disorders, such as immune thrombocytopenic purpura.[A259073, A259078]

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Rimacalib DB12571
small molecule | CAS: 215174-50-8

Rimacalib has been used in trials studying the treatment of Rheumatoid Arthritis (RA).

Kategori:
Enzyme InhibitorsOxazinesProtein Kinase Inhibitors
Target Protein:
Calcium/calmodulin-dependent protein kinase type II subunit alphaCalcium/calmodulin-dependent protein kinase type II subunit betaCalcium/calmodulin-dependent protein kinase type II subunit delta +1
Waktu Paruh-
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Rimazolium DB13289
small molecule | CAS: 35615-72-6

Rimazolium is an experimental analgesic drug [A176186].

Kategori:
AnalgesicsNervous SystemPyrimidines
Waktu Paruh-
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Rimegepant Approved DB12457
small molecule | CAS: 1289023-67-1

Rimegepant is an oral antagonist of the CGRP receptor developed by Biohaven Pharmaceuticals.[L11028] It received FDA approval on February 27, 2020 for the acute treatment migraine headache,[L11974] and was subsequently approved by the European Commission in A…

Kategori:
AnalgesicsAntimigraine PreparationsBCRP/ABCG2 Substrates +19
Target Protein:
Calcitonin gene-related peptide type 1 receptor
Waktu ParuhThe elimination hal…
Vol. DistribusiAt steady state, th…
Klirens-
Genetik -
Rimiducid DB04974
small molecule | CAS: 195514-63-7

Rimiducid is a lipid-permeable tacrolimus analogue and a protein dimerizer. It was designed to overcome limitations of current cellular immunotherapies used for cancer and other blood disorders by enhancing the control of the immune cell activity and function…

Kategori:
Cross-Linking Reagents
Target Protein:
Peptidyl-prolyl cis-trans isomerase FKBP1ASerine/threonine-protein kinase mTOR
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Rimiterol DB13559
small molecule | CAS: 32953-89-2

Deskripsi belum tersedia.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic beta-Agonists +8
Target Protein:
Beta-3 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rimonabant Approved DB06155
small molecule | CAS: 168273-06-1

Rimonabant is an anorectic anti-obesity drug produced and marketed by Sanofi-Aventis. It is an inverse agonist for the cannabinoid receptor CB1. Its main avenue of effect is reduction in appetite. Rimonabant is the first selective CB1 receptor blocker to be a…

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAnti-Obesity Agents +12
Target Protein:
Cannabinoid receptor 1G-protein coupled receptor 55
Waktu Paruh6 to 9 days with no…
Vol. Distribusi-
Klirens-
Genetik -
Rindopepimut DB05374
small molecule | CAS: 1108208-65-6

Rindopepimut (CDX-110) is an injectable peptide cancer vaccine which targets a mutant protein called EGFRvIII present in about 25% to 30% of glioblastoma cases. The vaccine consists of the EGFRv3-specific peptide (a 13-amino acid mutant vIII epitope) conjugat…

Kategori:
Antineoplastic AgentsAntineoplastic Agents, ImmunologicalBiological Products +2
Target Protein:
Epidermal growth factor receptor
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Rineterkib DB17560
small molecule | CAS: 1715025-32-3

Rineterkib is an inhibitor of extracellular signal-regulated kinase (ERK) being investigated in NCT04097821 (A Randomized, Open-label, Phase I/II Open Platform Study Evaluating Safety and Efficacy of Novel Ruxolitinib Combinations in Myelofibrosis Patients).

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Menampilkan 10301–10350 dari 12560
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