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13591

Total database: 17430
Struktur (SMILES)
10177 (74.9%)
Target
7625 (56.1%)
Genomik
104 (0.8%)
Referensi
13591 (100.0%)

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Hasil Pencarian (13591)

Halaman 207 / 272
PF-06700841 DB15003
small molecule | CAS: 1883299-62-4

PF-06700841 is under investigation in clinical trial NCT03236493 (Safety and Pharmacokinetic Study of PF-06700841 in Japanese Healthy Volunteers).

Kategori:
Enzyme InhibitorsProtein Kinase Inhibitors
Target Protein:
Non-receptor tyrosine-protein kinase TYK2Tyrosine-protein kinase JAK1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PF-06751979 DB15105
small molecule | CAS: 1818339-66-0

PF-06751979 is under investigation in clinical trial NCT03126721 (The Study is to Evaluate the Effect of Multiple Doses PF-06751979 on the Pharmacokinetics of Midazolam in Healthy Adults).

Kategori:
Sulfur Compounds
Waktu Paruh-
Vol. Distribusi-
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Genetik -
PF-06815345 DB14862
small molecule | CAS: 1900686-46-5

PF-06815345 is under investigation in clinical trial NCT02654899 (Single Dose Study of PF-06815345 in Healthy Subjects).

Waktu Paruh-
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PF-06821497 DB14799
small molecule | CAS: 1844849-10-0

PF-06821497 is under investigation in clinical trial NCT03460977 (PF-06821497 Treatment Of Relapsed/Refractory SCLC, Castration Resistant Prostate Cancer, and Follicular Lymphoma).

Target Protein:
Histone-lysine N-methyltransferase EZH2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PF-06835919 DB19163
small molecule | CAS: 2102501-84-6

PF-06835919 is under investigation in clinical trial NCT05463575 (Ketohexokinase Inhibition in NAFLD).

Kategori:
Aza Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PF-06842874 DB18039
small molecule | CAS: 2516247-98-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
PF-06882961 DB16043
small molecule | CAS: 2230198-02-2

PF-06882961 is under investigation in clinical trial NCT03985293 (A 16 Week Study to Evaluate the Efficacy and Safety of PF-06882961 in Adults With Type 2 Diabetes Mellitus).

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Glucagon-like peptide 1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PF-07038124 DB19143
small molecule | CAS: 2415085-44-6

PF-07038124 is under investigation in clinical trial NCT05298033 (Study of Efficacy, Safety and Tolerability of Crisaborole and PF-07038124 With and Without NBUVB in Vitiligo).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PF-07059013 DB18122
small molecule | CAS: 2435610-93-6

Deskripsi belum tersedia.

Target Protein:
Hemoglobin subunit beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PF-07304814 DB16514
small molecule

PF-07304814 is a small molecule prodrug that targets the 3CL<sup>pro</sup> protease (M<sup>pro)</sup>, which is used by viruses like SARS-CoV-2 to assemble and multiply[L31718]. Once administered through intravenous infusion, the compound is cleaved into PF-0…

Kategori:
Amino AcidsAmino Acids, Branched-ChainAmino Acids, Essential +4
Target Protein:
Replicase polyprotein 1ab
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PF-07799933 DB17489
small molecule

PF-07799933 is a BRAF class 2 inhibitor developed by Pfizer.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PF-232798 DB14813
small molecule | CAS: 849753-15-7

PF-232798 is under investigation in clinical trial NCT01140425 (Study To Evaluate The Effect Of A Multiple Oral Dose Of PF-00232798 On QT Intervals In Healthy Subjects).

Kategori:
AlkaloidsAnti-HIV AgentsAnti-Infective Agents +5
Target Protein:
C-C chemokine receptor type 5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PF-4136309 DB17200
small molecule | CAS: 1341224-83-6

Deskripsi belum tersedia.

Waktu Paruh-
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PF-4191834 DB11645
small molecule | CAS: 1029317-21-2

PF-4191834 has been investigated for the basic science of Asthma.

Kategori:
AnionsElectrolytesHydrogen Sulfide +2
Target Protein:
Polyunsaturated fatty acid 5-lipoxygenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PF-477736 DB12611
small molecule | CAS: 952021-60-2

PF-00477736 has been used in trials studying the treatment of Neoplasms.

Kategori:
BenzazepinesEnzyme InhibitorsHeterocyclic Compounds, Fused-Ring +1
Target Protein:
Serine/threonine-protein kinase Chk1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PF-5190457 DB14870
small molecule | CAS: 1334782-79-4

PF-5190457 is under investigation in clinical trial NCT01522807 (A Study Of Three PF-05190457 Formulations In Healthy Volunteers).

Kategori:
Azetines
Target Protein:
Growth hormone secretagogue receptor type 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PF-5212372 DB19212
small molecule | CAS: 916136-25-9

PF-5212372 is under investigation in clinical trial NCT02795832 (A Study to Determine the Safety & Efficacy of ZPL-5212372 in Healthy Subjects and in Subjects With Atopic Dermatitis).

Kategori:
Acids, CarbocyclicAmidesEnzyme Inhibitors +3
Waktu Paruh-
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Genetik -
PG-530742 DB05495
small molecule | CAS: 291533-11-4

PG-530742 selectively inhibits certain matrix metalloproteinases that have been implicated in the cartilage degradation that occurs in osteoarthritis. By inhibiting these MMPs, it potentially limits cartilage degradation and disease progression. Studies are c…

Kategori:
AminesHydroxy AcidsHydroxylamines
Target Protein:
Stromelysin-1Matrix metalloproteinase-9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PG-701 DB12252
small molecule | CAS: 583028-68-6

Hydroxytriptolide has been investigated for the treatment of Rheumatoid Arthritis.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PH-797804 DB07941
small molecule | CAS: 586379-66-0

PH-797804 has been investigated for the treatment of Osteoarthritis.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +3
Target Protein:
Mitogen-activated protein kinase 14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PHA-767491 DB17043
small molecule | CAS: 845714-00-3

PHA-767491 is a Cdc7/CDK9 inhibitor.[A253077]

Kategori:
Piperidines
Target Protein:
Cell division cycle 7-related protein kinase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PHA-793887 DB12686
small molecule | CAS: 718630-59-2

PHA-793887 has been used in trials studying the treatment of Advanced/Metastatic Solid Tumors.

Kategori:
Cyclin-Dependent Kinases, antagonists & inhibitors
Target Protein:
Cyclin-dependent kinase 2Cyclin-dependent kinase 4Cyclin-dependent kinase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Phalaris minor pollen Approved DB10963
biotech

Phalaris minor pollen is the pollen of the Phalaris minor plant. Phalaris minor pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityGrass Pollen Allergen ExtractsIncreased Histamine Release +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Phanquinone DB13469
small molecule | CAS: 84-12-8

Deskripsi belum tersedia.

Kategori:
Antiparasitic Products, Insecticides and RepellentsAntiprotozoalsHeterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PHE885 DB18123
biotech

PHE885 is an investigational, autologous B-cell Maturation Antigen (BCMA)-directed chimeric antigen receptor (CAR)-T cell therapy.

Waktu Paruh-
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Phelimin DB18332
small molecule

Phelemin (PHE-MIP) is a methacrylic acid-based copolymer purified to bind to L-phenylalanine and L-phenylalanine-containing peptides.[L48151] It is under investigation for the treatment of hyperphenylalaninemia.

Waktu Paruh-
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Genetik -
biotech

Phellodendron amurense bark is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
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Phenacemide Approved DB01121
small molecule | CAS: 63-98-9

Phenacemide is used to control certain seizures in the treatment of epilepsy. This medicine acts on the central nervous system (CNS) to reduce the number and severity of seizures.

Kategori:
AcetamidesAmidesAnticonvulsants +3
Target Protein:
Sodium channel protein type 1 subunit alpha
Waktu Paruh22-25 hours.
Vol. Distribusi-
Klirens-
Genetik -
Phenacetin DB03783
small molecule | CAS: 62-44-2

Phenacetin was withdrawn from the Canadian market in June 1973 due to concerns regarding nephropathy (damage to or disease of the kidney).

Kategori:
AcetanilidesAmidesAmines +18
Target Protein:
Prostaglandin G/H synthase 1Inosine-5'-monophosphate dehydrogenase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Phenaglycodol DB19373
small molecule | CAS: 79-93-6

Deskripsi belum tersedia.

Kategori:
AlcoholsGlycols
Waktu Paruh-
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Genetik -
Phenazepam DB19164
small molecule | CAS: 51753-57-2

Phenazepam is under investigation in clinical trial NCT03017430 (Pregabalin for Opiate Withdrawal Syndrome).

Kategori:
Adjuvants, ImmunologicAntiarrhythmic agentsAnticonvulsants +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Phenazocine DB13606
small molecule | CAS: 58073-76-0

Deskripsi belum tersedia.

Kategori:
AlkaloidsAnalgesicsBenzomorphan Derivatives +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Phenazopyridine Approved DB01438
small molecule | CAS: 94-78-0

Phenazopyridine, also known as Pyridium, is a urinary tract analgesic used for the short-term management of urinary tract irritation and its associated unpleasant symptoms such as burning and pain during urination. In the USA, this drug was previously marked …

Kategori:
AminesAminopyridinesAntipruritics and Local Anesthetics +6
Target Protein:
Sodium channel protein type 1 subunit alphaGroup A nerve fibers
Waktu ParuhThe mean eliminatio…
Vol. DistribusiSmall, trace quanti…
KlirensThis drug is rapidl…
Genetik -
Phencyclidine DB03575
small molecule | CAS: 77-10-1

A hallucinogen formerly used as a veterinary anesthetic, and briefly as a general anesthetic for humans. Phencyclidine is similar to ketamine in structure and in many of its effects. Like ketamine, it can produce a dissociative state. It exerts its pharmacolo…

Kategori:
Central Nervous System AgentsCentral Nervous System DepressantsCytochrome P-450 CYP2B6 Inhibitors +11
Target Protein:
Glutamate receptor ionotropic, NMDA 3AGlutamate receptor ionotropic, NMDA 2BGlutamate receptor ionotropic, NMDA 2A +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Phendimetrazine Approved DB01579
small molecule | CAS: 634-03-7

Phendimetrazine is a weight loss medication. Phendimetrazine is chemically related to amphetamines and is a Schedule III drug under the Convention on Psychotropic Substances and in the US since 1970.

Kategori:
Adrenergic AgonistsAdrenergic alpha-1 Receptor AgonistsAdrenergic alpha-Agonists +10
Target Protein:
Alpha-1A adrenergic receptorSodium-dependent noradrenaline transporterAlpha-1B adrenergic receptor
Waktu Paruh19-24 hours
Vol. Distribusi-
Klirens-
Genetik -
Phenelzine Approved DB00780
small molecule | CAS: 51-71-8

Phenelzine, with the formula ?-phenylethylhydrazine, is a monoamine oxidase inhibiting antidepressant that is effective in the treatment of panic disorder and social anxiety disorder.[A15753] It was developed by Parke Davis and originally FDA approved on June…

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +33
Target Protein:
Amine oxidase [flavin-containing] AAmine oxidase [flavin-containing] BAmine oxidase [copper-containing] 3 +4
Waktu ParuhAfter administratio…
Vol. DistribusiThe volume of distr…
Klirens-
Genetik -
Phenethylamine DB04325
small molecule | CAS: 64-04-0

Deskripsi belum tersedia.

Kategori:
AminesCentral Nervous System AgentsCentral Nervous System Depressants +2
Target Protein:
5-hydroxytryptamine receptor 2APrimary amine oxidaseSerine protease 1 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pheneticillin Approved DB13337
small molecule | CAS: 147-55-7

Pheneticillin (or phenethicillin) is a penicillin antibiotic which is approved for use internationally.

Kategori:
Anti-Bacterial AgentsAntibacterials for Systemic UseAntiinfectives for Systemic Use +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pheneturide DB13362
small molecule | CAS: 90-49-3

Deskripsi belum tersedia.

Kategori:
AmidesAnticonvulsantsCentral Nervous System Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Phenformin Approved DB00914
small molecule | CAS: 114-86-3

A biguanide hypoglycemic agent with actions and uses similar to those of metformin. Although it is generally considered to be associated with an unacceptably high incidence of lactic acidosis, often fatal, it is still available in some countries. (From Martin…

Kategori:
Alimentary Tract and MetabolismAmidinesBiguanides +9
Target Protein:
5'-AMP-activated protein kinase catalytic subunit alpha-15'-AMP-activated protein kinase subunit gamma-15'-AMP-activated protein kinase subunit beta-1 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Phenglutarimide DB13413
small molecule | CAS: 1156-05-4

Deskripsi belum tersedia.

Kategori:
Agents producing tachycardiaAnti-Parkinson DrugsAnticholinergic Agents +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Phenibut DB13455
small molecule | CAS: 1078-21-3

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAmino AcidsAmino Acids, Peptides, and Proteins +16
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Phenindione Approved DB00498
small molecule | CAS: 83-12-5

An indandione that has been used as an anticoagulant. Phenindione has actions similar to warfarin, but it is now rarely employed because of its higher incidence of severe adverse effects. (From Martindale, The Extra Pharmacopoeia, 30th ed, p234)

Kategori:
AnticoagulantsBlood and Blood Forming OrgansHematologic Agents +4
Target Protein:
Vitamin K epoxide reductase complex subunit 1
Waktu Paruh5-10 hours
Vol. Distribusi-
Klirens-
Genetik -
Phenmetrazine Approved DB00830
small molecule | CAS: 134-49-6

A sympathomimetic drug used primarily as an appetite depressant. Its actions and mechanisms are similar to dextroamphetamine.

Kategori:
Agents producing tachycardiaAgents that produce hypertensionAnti-Obesity Agents +8
Target Protein:
Sodium-dependent noradrenaline transporterSodium-dependent dopamine transporter
Waktu Paruh16 to 31 hours
Vol. Distribusi-
Klirens-
Genetik -
Phenobarbital Approved DB01174
small molecule | CAS: 50-06-6

A barbituric acid derivative that acts as a nonselective central nervous system depressant. It promotes binding to inhibitory gamma-aminobutyric acid subtype receptors, and modulates chloride currents through receptor channels. It also inhibits glutamate indu…

Kategori:
Anticholinergic AgentsAnticonvulsantsBarbiturates +57
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1Neuronal acetylcholine receptor subunit alpha-4Neuronal acetylcholine receptor subunit alpha-7 +4
Waktu Paruh53 to 118 hours (me…
Vol. Distribusi-
Klirens-
Genetik -
Phenol Approved DB03255
small molecule | CAS: 108-95-2

Phenol is an antiseptic and disinfectant. It is active against a wide range of micro-organisms including some fungi and viruses, but is only slowly effective against spores. Phenol has been used to disinfect skin and to relieve itching. Phenol is also used as…

Kategori:
AnestheticsAnesthetics, LocalAnti-Infective Agents +19
Target Protein:
Carbonic anhydrase 1Carbonic anhydrase 4Carbonic anhydrase 12 +5
Waktu Paruh-
Vol. DistribusiAt I5 min after exp…
KlirensIn rabbits, 72% is …
Genetik -
Phenolphthalein Approved DB04824
small molecule | CAS: 77-09-8

Phenolphthalein was withdrawn in Canada due to concerns with carcinogenicity in 1997.

Kategori:
Alimentary Tract and MetabolismBenzene DerivativesCompounds used in a research, industrial, or household setting +7
Target Protein:
UDP-glucuronosyltransferase 1A9Nuclear receptor subfamily 1 group I member 2Nuclear receptor subfamily 1 group I member 3 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 98-67-9

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
small molecule | CAS: 143-74-8

Phenolsulfonphthalein or otherwise called phenol red is a pH indicator commonly used in cell biology laboratories. Phenolsulfonphthalein is being investigated for use clinically due to its weak estrogen mimicking actions [A174964].

Kategori:
Benzene DerivativesColoring AgentsCompounds used in a research, industrial, or household setting +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Phenoperidine DB13605
small molecule | CAS: 562-26-5

Deskripsi belum tersedia.

Kategori:
AnalgesicsAnestheticsAnesthetics, General +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 10301–10350 dari 13591
Sebelumnya Halaman 207 / 272 Berikutnya